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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)phenyl]-N-(2,6-dichlorophenyl)piperazine-1-carboxamide 1092480-55-1 C23H25Cl2N5O2
4-[4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)phenyl]-N-(2,6-dichlorophenyl)piperazine-1-carboxamide
—— 4-[4-(1-tert-butyl-1,2,4-triazol-3-yl)phenyl]-N-(2,6-dichlorophenyl)piperazine-1-carboxamide 1092480-57-3 C23H26Cl2N6O
4-[4-(1-tert-butyl-1,2,4-triazol-3-yl)phenyl]-N-(2,6-dichlorophenyl)piperazine-1-carboxamide
—— 3-Methyl-6-α-furyl-4,5,6,7-tetrahydro-indazol-4-on 19933-34-7 C12H12N2O2
3-Methyl-6-α-furyl-4,5,6,7-tetrahydro-indazol-4-on
—— 3-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-N-phenyl-N-(piperidin-4-yl)propionamide 1186213-33-1 C24H39N5O
3-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]-N-phenyl-N-(piperidin-4-yl)propionamide
—— tert-butyl 4-(5-nitro-1-trityl-1H-indazol-3-yl)-1H-pyrazole-1-carboxylate 1093064-71-1 C34H29N5O4
tert-butyl 4-(5-nitro-1-trityl-1H-indazol-3-yl)-1H-pyrazole-1-carboxylate
—— 4-[2-(3-diethylaminophenoxy)phenylsulfamoyl]-N-(3-piperidin-4-ylpropyl)benzamide hydrochloride 1021362-98-0 C31H40N4O4S*ClH
4-[2-(3-diethylaminophenoxy)phenylsulfamoyl]-N-(3-piperidin-4-ylpropyl)benzamide hydrochloride
—— 7-({[3-(7,8-dimethoxy-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-3-oxopropyl]amino}methyl)bicyclo[4.2.0]octa-1,3,5-trien-3-yl 4,4-difluoro-1-piperidinecarboxylate 1132075-22-9 C30H37F2N3O5
7-({[3-(7,8-dimethoxy-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-3-oxopropyl]amino}methyl)bicyclo[4.2.0]octa-1,3,5-trien-3-yl 4,4-difluoro-1-piperidinecarboxylate
—— methyl 3-[(3,3-diphenylpropyl){3-[3-(2-ethoxy-2-oxoethoxy)phenyl]propyl}carbamoyl]benzoate 1034021-02-7 C37H39NO6
methyl 3-[(3,3-diphenylpropyl){3-[3-(2-ethoxy-2-oxoethoxy)phenyl]propyl}carbamoyl]benzoate
—— 1-benzyl-3-thien-2-ylpyrrolidin-3-ol 1092573-99-3 C15H17NOS
1-benzyl-3-thien-2-ylpyrrolidin-3-ol
—— [3-(3-chloro-4'-methoxybiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1035926-92-1 C21H22ClN3O2S
[3-(3-chloro-4'-methoxybiphenyl-4-yl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— ethyl 3-[(5-isobutyl-2-thienylsulfonyl)amino]-2-(4-nitrobenzyl)-3-oxopropionate 1094201-75-8 C20H24N2O7S2
ethyl 3-[(5-isobutyl-2-thienylsulfonyl)amino]-2-(4-nitrobenzyl)-3-oxopropionate
—— N-cyclopropyl-4-[2-(4-fluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl]-2-aminopyrimidine 1161075-13-3 C20H20FN5
N-cyclopropyl-4-[2-(4-fluorophenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl]-2-aminopyrimidine
—— Ethyl 11-(1-methylpiperidin-4-ylidene)-6,11-dihydrodibenz[b,e]oxepin-4-carboxylate 1017796-13-2 C23H25NO3
Ethyl 11-(1-methylpiperidin-4-ylidene)-6,11-dihydrodibenz[b,e]oxepin-4-carboxylate
—— 1-benzyl-3-(2,3-difluorophenyl)-3-fluoropyrrolidine 1092573-96-0 C17H16F3N
1-benzyl-3-(2,3-difluorophenyl)-3-fluoropyrrolidine
—— 3-(4-methylpiperazin-1-yl)-N-phenyl-N-(piperidin-4-yl)propionamide 1186213-31-9 C19H30N4O
3-(4-methylpiperazin-1-yl)-N-phenyl-N-(piperidin-4-yl)propionamide
—— 3-ethyl-5-isopropyl-7-methyl-2-[2-methyl-4-(trifluoromethoxy)phenyl]pyrrolo[2,1-f] [1,2,4]triazin-4(3H)-one 1079361-37-7 C20H22F3N3O2
3-ethyl-5-isopropyl-7-methyl-2-[2-methyl-4-(trifluoromethoxy)phenyl]pyrrolo[2,1-f] [1,2,4]triazin-4(3H)-one
—— 3-((((2R)-1-acetyl-2-pyrrolidinyl)-methyl)-oxy)-5-(trifluoromethyl)-phenylamine 1135497-32-3 C14H17F3N2O2
3-((((2R)-1-acetyl-2-pyrrolidinyl)-methyl)-oxy)-5-(trifluoromethyl)-phenylamine
—— 2-[4-(benzoylamino)benzyl]-N, N-dimethyl-N'-(2-naphthylsulfonyl)malonamide 1094196-97-0 C29H27N3O5S
2-[4-(benzoylamino)benzyl]-N, N-dimethyl-N'-(2-naphthylsulfonyl)malonamide
—— Dinonyl-<2-hydroxy-1,1-bis-hydroxymethyl-ethyl>-amin 102547-32-0 C22H47NO3
Dinonyl-<2-hydroxy-1,1-bis-hydroxymethyl-ethyl>-amin
—— 3-(2-fluoro-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-1-(2-hydroxyethyl)-1-(pyridin-3-yl)urea 1219727-87-3 C21H19FN6O2
3-(2-fluoro-4-(5-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-1-(2-hydroxyethyl)-1-(pyridin-3-yl)urea
—— 5,6-dimethyl-2-phenyl-1-((1-tosyl-indole-3-yl)methyl)benzimidazole 1234802-28-8 C31H27N3O2S
5,6-dimethyl-2-phenyl-1-((1-tosyl-indole-3-yl)methyl)benzimidazole
—— 2-chloro-4-(morpholin-4-yl)benzoic acid hydrazide 1035929-36-2 C11H14ClN3O2
2-chloro-4-(morpholin-4-yl)benzoic acid hydrazide
—— ethyl 3-{1-[4-(difluoromethoxy)phenyl]-3-(2-pyridin-2-ylethyl)-1H-indol-5-yl}propanoate 1069044-98-9 C27H26F2N2O3
ethyl 3-{1-[4-(difluoromethoxy)phenyl]-3-(2-pyridin-2-ylethyl)-1H-indol-5-yl}propanoate
—— ethyl 3-[1-(3-cyanophenyl)-3-(2-phenylethyl)-1H-indol-5-yl]propanoate 1069043-94-2 C28H26N2O2
ethyl 3-[1-(3-cyanophenyl)-3-(2-phenylethyl)-1H-indol-5-yl]propanoate
—— N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-4-pyridin-4-ylbenzamide 1127308-24-0 C24H22N4O2
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-4-pyridin-4-ylbenzamide
—— 3-(4-bromo-2-chlorophenyl)-8-({[t-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1035928-14-3 C20H29BrClN3OSSi
3-(4-bromo-2-chlorophenyl)-8-({[t-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 2-Aminooxazole-4-carbonitrile 1240598-27-9 C4H3N3O
2-Aminooxazole-4-carbonitrile
—— (2S,5S)-2-tert-butyl-5-(2-fluoro-5-hydroxymethyl-benzyl)-3-methyl-4-oxoimidazoline-1-carboxylic acid tert-butyl ester 1159894-77-5 C21H31FN2O4
(2S,5S)-2-tert-butyl-5-(2-fluoro-5-hydroxymethyl-benzyl)-3-methyl-4-oxoimidazoline-1-carboxylic acid tert-butyl ester
—— 2-[4-(2,3-difluoro-phenyl)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-piperidin-1-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one 1082988-87-1 C31H32F2N4O2
2-[4-(2,3-difluoro-phenyl)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-piperidin-1-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one
—— 6-(isopropylamino)-9-(2-fluorobenzyl)-2-(trifluoromethyl)purine 1082247-76-4 C16H15F4N5
6-(isopropylamino)-9-(2-fluorobenzyl)-2-(trifluoromethyl)purine
—— cyclopropanecarboxylic acid 4-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)benzylamide 1031747-47-3 C17H24BNO3
cyclopropanecarboxylic acid 4-(4,4,5,5-tetramethyl[1,3,2]dioxaborolan-2-yl)benzylamide
—— 5-isopropyl-2-(2-isopropyl-4-methoxyphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079354-04-3 C21H27N3O2
5-isopropyl-2-(2-isopropyl-4-methoxyphenyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 5-chloro-N-[3-fluoro-4-(piperidin-4-ylamino)phenyl]-2-hydroxybenzamide 1000048-34-9 C18H19ClFN3O2
5-chloro-N-[3-fluoro-4-(piperidin-4-ylamino)phenyl]-2-hydroxybenzamide
—— methyl (2S)-2-(3-{3-[5-(diphenylmethyl)-2-oxopyridin-1(2H)-yl]propyl}phenoxy)propanoate 1034020-43-3 C31H31NO4
methyl (2S)-2-(3-{3-[5-(diphenylmethyl)-2-oxopyridin-1(2H)-yl]propyl}phenoxy)propanoate
—— 2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one 1079353-14-2 C19H20ClF3N4O
2-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-5-(1-ethylpropyl)-3,7-dimethylpyrrolo[2,1-f][1,2,4]triazin-4(3H)-one
—— 4-(6-amino-3-azabicyclo[3.1.0]hexan-3-yl)-6-fluoro-N-methyl-2-pyrimidin-5-yloxy-9H-pyrimido[4,5-b]indol-8-amine 1400803-14-6 C20H19FN8O
4-(6-amino-3-azabicyclo[3.1.0]hexan-3-yl)-6-fluoro-N-methyl-2-pyrimidin-5-yloxy-9H-pyrimido[4,5-b]indol-8-amine
—— N-[(2R)-2,3-dihydroxypropyl]-3-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)benzamide 1020169-39-4 C32H36F4N4O5
N-[(2R)-2,3-dihydroxypropyl]-3-(4-{[4-[5-fluoro-2-(methyloxy)phenyl]-2-hydroxy-4-methyl-2-(trifluoromethyl)pentyl]amino}-6-methyl-1H-indazol-1-yl)benzamide
—— 5-acetyl-4,7-dimethoxy-6-benzofuranyl 2,3,4-tri-O-acetyl-5-thio-β-D-xylopyranoside 1001434-05-4 C23H26O11S
5-acetyl-4,7-dimethoxy-6-benzofuranyl 2,3,4-tri-O-acetyl-5-thio-β-D-xylopyranoside
—— 6-Bromobenzo[f][1,3]benzodioxole 1235379-17-5 C11H7BrO2
6-Bromobenzo[f][1,3]benzodioxole
—— (R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(3,4-difluoro-phenyl)-ethyl]-2-isopropylamino-3-phenyl-propionamide 1194094-05-7 C27H31F2N5O2
(R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(3,4-difluoro-phenyl)-ethyl]-2-isopropylamino-3-phenyl-propionamide
—— 2-[4-(2,3-difluoro-phenyl)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-morpholin-4-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one 1082988-44-0 C30H30F2N4O3
2-[4-(2,3-difluoro-phenyl)-2-oxo-1,2-dihydro-indol-3-ylidenemethyl]-3-methyl-5-(2-morpholin-4-yl-ethyl)-5,6,7,8-tetrahydro-1H-pyrrolo[3,2-c]azepin-4-one
—— 2-(2-chloro-4-methoxyphenyl)-3,7-dimethyl-4-oxo-3,4-dihydropyrrolo[2,1-f][1,2,4]triazin-5-carboxylic acid 1079360-15-8 C16H14ClN3O4
2-(2-chloro-4-methoxyphenyl)-3,7-dimethyl-4-oxo-3,4-dihydropyrrolo[2,1-f][1,2,4]triazin-5-carboxylic acid
—— 5,6-dichloro-2-(3-fluoropyridin-4-yl)-1-methyl-1H-benzimidazole 1356481-23-6 C13H8Cl2FN3
5,6-dichloro-2-(3-fluoropyridin-4-yl)-1-methyl-1H-benzimidazole
—— 2-(3-fluoropyridin-4-yl)-1-cyclopropyl-1H-benzimidazole-6-carbonitrile 1356480-21-1 C16H11FN4
2-(3-fluoropyridin-4-yl)-1-cyclopropyl-1H-benzimidazole-6-carbonitrile
—— 1-cyclopropyl-2-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl]-5-(trifluoromethyl)-1H-benzimidazole 1356480-67-5 C20H16F3N5
1-cyclopropyl-2-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-3-yl]-5-(trifluoromethyl)-1H-benzimidazole
—— methyl 2-(7-(methylamino)-2-(trifluoromethoxy)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetate 1403368-15-9 C17H19F3N2O3
methyl 2-(7-(methylamino)-2-(trifluoromethoxy)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetate
—— 4-{4-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-3-(phenylethynyl)-2-thienyl}morpholine 1203508-89-7 C23H27N3O2S
4-{4-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-3-(phenylethynyl)-2-thienyl}morpholine
—— N'-(5-bromo-2-cyano-4-pyrimidinyl)-N'-cyclohexyl-3-{[4-(4-morpholinyl)-1-piperidinyl]methyl}benzohydrazide trifluoroacetate 1024588-04-2 C2HF3O2*C28H36BrN7O2
N'-(5-bromo-2-cyano-4-pyrimidinyl)-N'-cyclohexyl-3-{[4-(4-morpholinyl)-1-piperidinyl]methyl}benzohydrazide trifluoroacetate
—— 4-[2-(3-{4-[2-(2,4-dichlorophenoxy)phenylsulfamoyl]benzoylamino}propionylamino)ethyl]piperidine-1-carboxylic acid tert-butyl ester 1021363-65-4 C34H40Cl2N4O7S
4-[2-(3-{4-[2-(2,4-dichlorophenoxy)phenylsulfamoyl]benzoylamino}propionylamino)ethyl]piperidine-1-carboxylic acid tert-butyl ester
—— 4-[2-(2-chloro-4-fluorophenoxy)phenylsulfamoyl]-N-(2-piperidin-1-ylethyl)benzamide 1021362-50-4 C26H27ClFN3O4S
4-[2-(2-chloro-4-fluorophenoxy)phenylsulfamoyl]-N-(2-piperidin-1-ylethyl)benzamide