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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-chloro-9-methyl-6,7,8,9-tetrahydro-5-oxa-2,3,9-triazabenzocycloheptene 1417632-92-8 C8H10ClN3O
4-chloro-9-methyl-6,7,8,9-tetrahydro-5-oxa-2,3,9-triazabenzocycloheptene
—— (4R,5R)-5-(2,4-difluorophenyl)-4-( 6-((3-fluorophenyl)ethynyl)pyridin-2-yl)oxazolidin-2-one 1375752-25-2 C22H13F3N2O2
(4R,5R)-5-(2,4-difluorophenyl)-4-( 6-((3-fluorophenyl)ethynyl)pyridin-2-yl)oxazolidin-2-one
—— 2-(4-chloro-2-(trifluoromethyl)phenyl)-2-methylpropanenitrile 1095544-17-4 C11H9ClF3N
2-(4-chloro-2-(trifluoromethyl)phenyl)-2-methylpropanenitrile
—— 1-bromo-3-(phenethylsulfonyl)benzene 1215077-96-5 C14H13BrO2S
1-bromo-3-(phenethylsulfonyl)benzene
—— [(R)-2-hydroxy-1-(6-methoxy-[1,5]naphthyridin-4-yl)-ethyl]-carbamic acid tert-butyl ester 1220978-34-6 C16H21N3O4
[(R)-2-hydroxy-1-(6-methoxy-[1,5]naphthyridin-4-yl)-ethyl]-carbamic acid tert-butyl ester
—— 2,2-Dimethyl-6-(trifluoromethyl)morpholine 1478030-16-8 C7H12F3NO
2,2-Dimethyl-6-(trifluoromethyl)morpholine
—— 6-(3-methylpyrazol-1-yl)-N-[(4-methylsulfonylphenyl)methyl]pyridine-2-carboxamide 1038409-13-0 C18H18N4O3S
6-(3-methylpyrazol-1-yl)-N-[(4-methylsulfonylphenyl)methyl]pyridine-2-carboxamide
—— 4-hydroxy-5,6-dimethoxy-3-(2-methyl-5-phenylpentanoyl)-1H-pyridin-2-one 1231946-08-9 C19H23NO5
4-hydroxy-5,6-dimethoxy-3-(2-methyl-5-phenylpentanoyl)-1H-pyridin-2-one
—— 4-[[[(2S)-2-cyano-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)propyl]-methylamino]methyl]benzonitrile 1056888-14-2 C24H24N4O
4-[[[(2S)-2-cyano-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)propyl]-methylamino]methyl]benzonitrile
—— ((1S*,5R*)-3-azabicyclo[3.3.0]octane-7-yl)(2,6-dimethylmorpholin-1-yl)methanone 1069113-09-2 C14H24N2O2
((1S*,5R*)-3-azabicyclo[3.3.0]octane-7-yl)(2,6-dimethylmorpholin-1-yl)methanone
—— [4-[4-[4-Bis[(2-methylquinolin-8-yl)oxy]alumanyloxyphenyl]-2,3,5,6-tetradeuteriophenyl]phenoxy]-bis[(2-methylquinolin-8-yl)oxy]alumane 1130088-24-2 C58H44Al2N4O6
[4-[4-[4-Bis[(2-methylquinolin-8-yl)oxy]alumanyloxyphenyl]-2,3,5,6-tetradeuteriophenyl]phenoxy]-bis[(2-methylquinolin-8-yl)oxy]alumane
—— 5-{6-[(2-imidazol-1-yl-ethylamino)-methyl]-pyrimidin-4-yloxy}-indole-1-carboxylic acid (3-trifluoromethyl-phenyl)-amide 1229448-67-2 C26H22F3N7O2
5-{6-[(2-imidazol-1-yl-ethylamino)-methyl]-pyrimidin-4-yloxy}-indole-1-carboxylic acid (3-trifluoromethyl-phenyl)-amide
—— 2-Cyclopropyl-2-(3-ethyl-2-methoxyquinolin-7-yl)-3-phenylpropanenitrile 1056892-60-4 C24H24N2O
2-Cyclopropyl-2-(3-ethyl-2-methoxyquinolin-7-yl)-3-phenylpropanenitrile
—— N-benzyl-3-azabicyclo[3.3.1]nonane-7-carboxamide 1068582-94-4 C16H22N2O
N-benzyl-3-azabicyclo[3.3.1]nonane-7-carboxamide
—— 6-(2-methylpropanoylamino)-N-[[1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]methyl]pyridine-2-carboxamide 1038409-45-8 C21H20F3N5O2
6-(2-methylpropanoylamino)-N-[[1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]methyl]pyridine-2-carboxamide
—— 5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid [1-methyl-5-(2,2,2-trifluoro-1-methoxy-1-methyl-ethyl)-1H-pyrazol-3-yl]-amide 1229452-81-6 C23H22F3N7O3
5-(6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-4-yloxy)-indole-1-carboxylic acid [1-methyl-5-(2,2,2-trifluoro-1-methoxy-1-methyl-ethyl)-1H-pyrazol-3-yl]-amide
—— 3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile 1056889-84-9 C23H22N2O3
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methylpropanenitrile
—— 6-(3-fluorophenyl)hexan-1-ol 1005407-94-2 C12H17FO
6-(3-fluorophenyl)hexan-1-ol
—— 3-fluoro-4-(1-methylisoquinolin-4-yloxy)benzonitrile 1087351-46-9 C17H11FN2O
3-fluoro-4-(1-methylisoquinolin-4-yloxy)benzonitrile
—— 2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-[4-(trifluoromethyl)phenyl]propanenitrile 1056889-67-8 C22H19F3N2O
2-(3-ethyl-2-oxo-1H-quinolin-7-yl)-2-methyl-3-[4-(trifluoromethyl)phenyl]propanenitrile
—— N-(3-bromo-5-methylphenyl)-6-chloro-4-pyrimidinamine 1316066-22-4 C11H9BrClN3
N-(3-bromo-5-methylphenyl)-6-chloro-4-pyrimidinamine
—— 2-[(4-Hexanoyloxyphenyl)methyl-[4-[[2-[4-methoxy-2-(trifluoromethyl)phenyl]acetyl]amino]benzoyl]amino]acetic acid 1415672-61-5 C32H33F3N2O7
2-[(4-Hexanoyloxyphenyl)methyl-[4-[[2-[4-methoxy-2-(trifluoromethyl)phenyl]acetyl]amino]benzoyl]amino]acetic acid
—— (5R,7aS,11aS)-5-butyloctahydro-1H-pyrrolo[2,1-j]quinolin-7(7aH)-one 1431968-39-6 C16H27NO
(5R,7aS,11aS)-5-butyloctahydro-1H-pyrrolo[2,1-j]quinolin-7(7aH)-one
—— N-(4-Chloro-phenyl)-N-(2-diethylamino-ethyl)-propionamide 132465-49-7 C15H23ClN2O
N-(4-Chloro-phenyl)-N-(2-diethylamino-ethyl)-propionamide
—— N-(3,3-Dichloro-2-methyl-allyl)-N-p-tolyl-benzenesulfonamide 109503-72-2 C17H17Cl2NO2S
N-(3,3-Dichloro-2-methyl-allyl)-N-p-tolyl-benzenesulfonamide
—— O<sup>3</sup>-Propionyl-oestron-17-mandelsaeurehydrazon 124463-62-3 C29H34N2O4
O<sup>3</sup>-Propionyl-oestron-17-mandelsaeurehydrazon
—— (S)-N2-(3-(difluoromethoxy)-4-(tetrahydrofuran-3-yloxy)phenyl)-5-fluoro-N4-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidine-2,4-diamine 1239595-79-9 C24H32F3N5O3
(S)-N2-(3-(difluoromethoxy)-4-(tetrahydrofuran-3-yloxy)phenyl)-5-fluoro-N4-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidine-2,4-diamine
—— N2-(3,5-difluoro-4-(1-(methylsulfonyl)azepan-4-yloxy)phenyl)-5-fluoro-N4-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidine-2,4-diamine 1239595-61-9 C26H37F3N6O3S
N2-(3,5-difluoro-4-(1-(methylsulfonyl)azepan-4-yloxy)phenyl)-5-fluoro-N4-(2,2,6,6-tetramethylpiperidin-4-yl)pyrimidine-2,4-diamine
—— (1S,5S)-3-(pentanoyl)-3,6-diazabicyclo[3.2.1]octane 1215170-32-3 C11H20N2O
(1S,5S)-3-(pentanoyl)-3,6-diazabicyclo[3.2.1]octane
—— (1S,5S)-3-(spiro[2.3]hexan-1-ylcarbonyl)-3,6-diazabicyclo[3.2.1]octane 1215170-31-2 C13H20N2O
(1S,5S)-3-(spiro[2.3]hexan-1-ylcarbonyl)-3,6-diazabicyclo[3.2.1]octane
—— 1,1-diphenyl-1,2,3,4-tetrhydroisoquinoline 1085538-60-8 C21H19N
1,1-diphenyl-1,2,3,4-tetrhydroisoquinoline
—— 1-[(5-{2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl}pyrimidin-2-yl)carbonyl]azetidin-3-ol 1233525-60-4 C27H33N9O2
1-[(5-{2-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-3-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl}pyrimidin-2-yl)carbonyl]azetidin-3-ol
—— 2-bromo-5-({(3R,6R)-6-methyl-1-[2-(2H-1,2,3-triazol-2-yl)benzoyl]piperidin-3-yl}methoxy)pyridine 1088992-26-0 C21H22BrN5O2
2-bromo-5-({(3R,6R)-6-methyl-1-[2-(2H-1,2,3-triazol-2-yl)benzoyl]piperidin-3-yl}methoxy)pyridine
—— 4-{4-[8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxalin-2-yl]-5-methyl-pyrazol-1-yl}-piperidine-1-carboxylic acid tert-butyl ester 1092500-18-9 C33H38F2N6O3
4-{4-[8-(3,5-difluoro-4-morpholin-4-ylmethyl-phenyl)-quinoxalin-2-yl]-5-methyl-pyrazol-1-yl}-piperidine-1-carboxylic acid tert-butyl ester
—— N-[4-cyclopentyl-2-[3-(dimethylamino)prop-1-ynyl]-5-methoxyphenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide 1233530-42-1 C27H30F3N3O4
N-[4-cyclopentyl-2-[3-(dimethylamino)prop-1-ynyl]-5-methoxyphenyl]-6-(trifluoromethoxy)-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
—— 2-benzyl-3-cyclopropyl-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)propanenitrile 1056887-64-9 C24H24N2O
2-benzyl-3-cyclopropyl-2-(3-ethyl-2-oxo-1H-quinolin-7-yl)propanenitrile
—— 3-(3-iodophenyl)-2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)propanenitrile 1056890-49-3 C20H17IN2O
3-(3-iodophenyl)-2-methyl-2-(3-methyl-2-oxo-1H-quinolin-7-yl)propanenitrile
—— N-(4-(3-bromophenylamino)quinazolin-6-yl)-2-(1-(2-methoxyethyl)piperidin-4-ylidene)acetamide 1005195-24-3 C24H26BrN5O2
N-(4-(3-bromophenylamino)quinazolin-6-yl)-2-(1-(2-methoxyethyl)piperidin-4-ylidene)acetamide
—— 2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (2-dimethylamino-4,5-dimethoxy-phenyl)-amide 1232687-78-3 C22H24FN3O4
2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (2-dimethylamino-4,5-dimethoxy-phenyl)-amide
—— 2-{2-[((2R,5R)-5-{[(5-fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl)carbonyl]phenyl}pyrimidine 1088992-04-4 C23H23FN4O2
2-{2-[((2R,5R)-5-{[(5-fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl)carbonyl]phenyl}pyrimidine
—— N-(2-(diethylamino)ethyl)-2-methyl-7-[5-(piperidin-1-ylsulfonyl)-1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide 1032266-65-1 C29H39N5O4S
N-(2-(diethylamino)ethyl)-2-methyl-7-[5-(piperidin-1-ylsulfonyl)-1,2-dihydro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
—— 3-cyclopropyl-5-phenoxycarbonylamino-pyrazole-1-carboxylic acid tert-butyl ester 1229454-51-6 C18H21N3O4
3-cyclopropyl-5-phenoxycarbonylamino-pyrazole-1-carboxylic acid tert-butyl ester
—— (1R2R,1S2S)-3-(2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenyl 2-(1-((ethoxycarbonylamino)methyl)cyclohexyl)acetate 1345016-67-2 C27H42N2O5
(1R2R,1S2S)-3-(2-((dimethylamino)methyl)-1-hydroxycyclohexyl)phenyl 2-(1-((ethoxycarbonylamino)methyl)cyclohexyl)acetate
—— N-(6-fluoro-3-methylimidazo[1,2-a]pyridin-2-yl)-N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]methanesulfonamide 1381784-33-3 C17H14F5N3O2S
N-(6-fluoro-3-methylimidazo[1,2-a]pyridin-2-yl)-N-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]methanesulfonamide
—— N-cyclopropyl-3-fluoro-5-(1-(4-fluoro-2-methylphenyl)-1H-benzotriazol-5-yl)-4-methylbenzamide 1135352-04-3 C24H20F2N4O
N-cyclopropyl-3-fluoro-5-(1-(4-fluoro-2-methylphenyl)-1H-benzotriazol-5-yl)-4-methylbenzamide
—— 3-oxo-3-(7-oxo-1,5-cycloheptadien-1-yl)propionic acid ethyl ester 1092980-12-5 C12H14O4
3-oxo-3-(7-oxo-1,5-cycloheptadien-1-yl)propionic acid ethyl ester
—— 4'-[(2-cyclohexyl-ethylamino)methyl]-2'-methylbiphenyl-3-carboxylic acid amide 1131794-97-2 C23H30N2O
4'-[(2-cyclohexyl-ethylamino)methyl]-2'-methylbiphenyl-3-carboxylic acid amide
—— N-cycloheptyl-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-10-carboxamide 1029686-50-7 C17H21N3O2S
N-cycloheptyl-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-triene-10-carboxamide
—— 3-(2,6-dichloro-4-{5-[8-chloro-6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,2,4-oxadiazol-3-yl}phenyl)propanoic acid 1228371-42-3 C19H10Cl3F3N4O3
3-(2,6-dichloro-4-{5-[8-chloro-6-(trifluoromethyl)imidazo[1,2-a]pyridin-2-yl]-1,2,4-oxadiazol-3-yl}phenyl)propanoic acid
—— (S)-2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (4,5-difluoro-2-methyl-phenyl)-amide 1232688-18-4 C19H15F3N2O2
(S)-2-(4-fluoro-phenyl)-4-oxo-3,4-dihydro-2H-pyridine-1-carboxylic acid (4,5-difluoro-2-methyl-phenyl)-amide