(S)-2-{2-[9-(Benzylamino-methyl)-6,10-dioxo-1,4,7,8,9,10-hexahydro-6H-pyridazino[1,2-a][1,2]diazepin-1-yl]-acetylamino}-4-methyl-pentanoic acid ((R)-1-carboxy-2-phenyl-ethylcarbamoyl)-methyl ester 在
antibody 2E11.2E7 作用下,
以
various solvent(s) 为溶剂,
反应 168.0h,
生成
(R)-2-(2-Hydroxy-acetylamino)-3-phenyl-propionic acid 、 (S)-2-{2-[9-(Benzylamino-methyl)-6,10-dioxo-1,4,7,8,9,10-hexahydro-6H-pyridazino[1,2-a][1,2]diazepin-1-yl]-acetylamino}-4-methyl-pentanoic acid