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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-bromo-4-((S)-2,2,2-trifluoro-1-methyl-ethoxy)-pyridine-2-carboxylic acid [2-methanesulfonyl-1-methyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide 1613238-97-3 C16H18BrF3N4O5S
5-bromo-4-((S)-2,2,2-trifluoro-1-methyl-ethoxy)-pyridine-2-carboxylic acid [2-methanesulfonyl-1-methyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide
—— 5,6-Dimethyl-pyrazin-2,3-dicarbonsaeure-monomethylester 92658-95-2 C9H10N2O4
5,6-Dimethyl-pyrazin-2,3-dicarbonsaeure-monomethylester
—— 7-(2-methyl-1H-benzimidazol-6-yl)-4-({2-[3-(trifluoromethyl)phenyl]piperidin-1-yl}carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1257299-22-1 C30H29F3N4O2
7-(2-methyl-1H-benzimidazol-6-yl)-4-({2-[3-(trifluoromethyl)phenyl]piperidin-1-yl}carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 7-{(E)-2-[2-(cyclopropylmethoxy)-3-methoxyphenyl]vinyl}-6-iodo-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one 1192871-96-7 C21H21IN2O3S
7-{(E)-2-[2-(cyclopropylmethoxy)-3-methoxyphenyl]vinyl}-6-iodo-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (4-(5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-5,6-dihydropyridin-1(2H)-yl)(2,6-difluorophenyl)methanone 1225061-49-3 C24H18F2N6O2
(4-(5-amino-6-(5-phenyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-5,6-dihydropyridin-1(2H)-yl)(2,6-difluorophenyl)methanone
—— 2-(3-cyano-1-cyclobutyl-5-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-(propan-2-yl)pyrimidine-5-sulfonamide 1247933-81-8 C21H24N6O2S
2-(3-cyano-1-cyclobutyl-5-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-(propan-2-yl)pyrimidine-5-sulfonamide
—— 6-(3-cyano-1-cyclopentyl-5-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide 1247934-84-4 C23H24F3N5O2S
6-(3-cyano-1-cyclopentyl-5-ethyl-1H-pyrrolo[2,3-b]pyridin-2-yl)-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide
—— 2-[3-cyano-1-cyclobutyl-6-(difluoromethyl)-1H-indol-2-yl]-N-(1,3-difluoropropan-2-yl)pyrimidine-5-sulfonamide 1248577-01-6 C21H19F4N5O2S
2-[3-cyano-1-cyclobutyl-6-(difluoromethyl)-1H-indol-2-yl]-N-(1,3-difluoropropan-2-yl)pyrimidine-5-sulfonamide
—— 5-(4-cyanophenoxy)-1-indanol 906673-47-0 C16H13NO2
5-(4-cyanophenoxy)-1-indanol
—— 3-methyl-1-[(2-methylcyclopropyl)methyl]-5-phenyl-1,3-dihydro-2H-benzimidazol-2-one 1359758-75-0 C19H20N2O
3-methyl-1-[(2-methylcyclopropyl)methyl]-5-phenyl-1,3-dihydro-2H-benzimidazol-2-one
—— 8-[2-(3-chloro-4-trifluoromethylphenyl)ethyl]-3-ethyl-5,6-dihydro-8H-imidazo[1,5-a]pyrazine-7-carboxylic acid tert-butyl ester 1036400-14-2 C22H27ClF3N3O2
8-[2-(3-chloro-4-trifluoromethylphenyl)ethyl]-3-ethyl-5,6-dihydro-8H-imidazo[1,5-a]pyrazine-7-carboxylic acid tert-butyl ester
—— 5-(3-chloro-2-fluoro-phenyl)-4-(4-chloro-2-methyl-phenyl)-2-(4-chloro-phenyl)-3-isopropyl-4,5-dihydro-2H-pyrrolo[3,4-c]pyrazol-6-one 1441748-70-4 C27H21Cl3FN3O
5-(3-chloro-2-fluoro-phenyl)-4-(4-chloro-2-methyl-phenyl)-2-(4-chloro-phenyl)-3-isopropyl-4,5-dihydro-2H-pyrrolo[3,4-c]pyrazol-6-one
—— [3-chloro-2-fluoro-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-phenyl]-morpholin-4-yl-methanone 1441202-63-6 C17H16ClF4N5O2
[3-chloro-2-fluoro-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-phenyl]-morpholin-4-yl-methanone
—— 3-(5-(3-acetylphenyl)nicotinoyl)-1-methylpyrrolidin-2-one 1434288-90-0 C19H18N2O3
3-(5-(3-acetylphenyl)nicotinoyl)-1-methylpyrrolidin-2-one
—— 2-chloro-5-((N-methylpivalamido)methyl)-N-(4-oxo-3-(4-(trifluoromethyl)phenyl)-3,4-dihydrophthalazin-6-yl)benzamide 1436500-55-8 C29H26ClF3N4O3
2-chloro-5-((N-methylpivalamido)methyl)-N-(4-oxo-3-(4-(trifluoromethyl)phenyl)-3,4-dihydrophthalazin-6-yl)benzamide
—— 4-(5-chloro-4-(methylamino)pyrimidin-2-ylamino)-3-methoxybenzonitrile 1441720-81-5 C13H12ClN5O
4-(5-chloro-4-(methylamino)pyrimidin-2-ylamino)-3-methoxybenzonitrile
—— 6-methoxy-4-((R)-pyrrolidin-3-yloxy)-quinazoline 1163127-76-1 C13H15N3O2
6-methoxy-4-((R)-pyrrolidin-3-yloxy)-quinazoline
—— 1-(2-fluoro-4-(trifluoromethyl)phenyl)cyclobutanecarbonitrile 1314650-24-2 C12H9F4N
1-(2-fluoro-4-(trifluoromethyl)phenyl)cyclobutanecarbonitrile
—— 2-(3-methyl-2-oxo-1-propyl-2,3-dihydro-1H-benzimidazol-5-yl)benzonitrile 1359760-29-4 C18H17N3O
2-(3-methyl-2-oxo-1-propyl-2,3-dihydro-1H-benzimidazol-5-yl)benzonitrile
—— 5-bromo-2-(dibenzylphosphono)oxy-N-{3,5-bis[(1,1-dimethyl)ethyl]phenyl}benzamide 634914-28-6 C35H39BrNO5P
5-bromo-2-(dibenzylphosphono)oxy-N-{3,5-bis[(1,1-dimethyl)ethyl]phenyl}benzamide
—— (R)-2-(1-amino-1-oxobutan-2-ylamino)-4-(isoquinolin-7-ylamino)pyrimidin-5-carboxamide 1439906-28-1 C18H19N7O2
(R)-2-(1-amino-1-oxobutan-2-ylamino)-4-(isoquinolin-7-ylamino)pyrimidin-5-carboxamide
—— (E)-4-(2-(bis(4-fluorobenzyl)amino)phenyl)but-3-en-2-one 1417628-18-2 C24H21F2NO
(E)-4-(2-(bis(4-fluorobenzyl)amino)phenyl)but-3-en-2-one
—— (3S,6R,7S)-methyl 6-bromo-6-methyl-4-((4-nitrophenyl)sulfonyl)-7-phenyl-1,4-oxazepane-3-carboxylate 1421070-75-8 C20H21BrN2O7S
(3S,6R,7S)-methyl 6-bromo-6-methyl-4-((4-nitrophenyl)sulfonyl)-7-phenyl-1,4-oxazepane-3-carboxylate
—— 2-[4-(4-Fluorophenyl)-2-phenylimidazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone 1443145-17-2 C26H24FN5O
2-[4-(4-Fluorophenyl)-2-phenylimidazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone
—— 6-chloro-4-(2-chloro-benzyl)-2-dimethylamino-quinoline-3-carboxylic acid 1433901-76-8 C19H16Cl2N2O2
6-chloro-4-(2-chloro-benzyl)-2-dimethylamino-quinoline-3-carboxylic acid
—— N-(2-diisopropylamino-ethyl)-2-methoxy-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide 617244-48-1 C29H36N4O4
N-(2-diisopropylamino-ethyl)-2-methoxy-4-[3-(4-phenoxy-phenyl)-ureido]-benzamide
—— 4-(2-aminoethoxy)-N-[(2-fluoro-5-phenyl)phenyl]-3-methoxybenzenethanamide 729557-42-0 C23H23FN2O3
4-(2-aminoethoxy)-N-[(2-fluoro-5-phenyl)phenyl]-3-methoxybenzenethanamide
—— (2R)-2-{[4-(5-{1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)phenoxy]propyl}-1,2,4-oxadiazol-3-yl)-2-fluorobenzoyl]amino}propyl N-(tert-butoxycarbonyl)glycinate 1263483-73-3 C33H37FN6O8
(2R)-2-{[4-(5-{1-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)phenoxy]propyl}-1,2,4-oxadiazol-3-yl)-2-fluorobenzoyl]amino}propyl N-(tert-butoxycarbonyl)glycinate
—— 5-chloro-2-{[(3R)-3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1H-indole 917356-66-2 C14H18ClN3O2S
5-chloro-2-{[(3R)-3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1H-indole
—— litophynol A diacetate 162244-61-3 C28H42O7
litophynol A diacetate
—— 1-[[2-(3,5-difluorophenyl)-5-(trifluoromethyl)-2H-pyrazol-3-yl]methyl]-3-[3-fluoro-4-(hydroxymethyl)phenyl]urea 1402582-65-3 C19H14F6N4O2
1-[[2-(3,5-difluorophenyl)-5-(trifluoromethyl)-2H-pyrazol-3-yl]methyl]-3-[3-fluoro-4-(hydroxymethyl)phenyl]urea
—— 4-methyl-2,3,4,5-tetrahydro-1H-1-benzazepine 1251853-40-3 C11H15N
4-methyl-2,3,4,5-tetrahydro-1H-1-benzazepine
—— 2H-Pyrazolo[3,4-c]pyridine, 3-(fluoromethyl)-4,5,6,7-tetrahydro-2-methyl- 1782805-92-8 C8H12FN3
2H-Pyrazolo[3,4-c]pyridine, 3-(fluoromethyl)-4,5,6,7-tetrahydro-2-methyl-
—— (2S,4R)-N-((S)-1-(butylamino)-1,2-dioxopentan-3-yl)-1-(1-(5-chloro-3-fluoropyridin-2-yl)cyclopropanecarbonyl)-4-(2-chlorophenylsulfonyl)pyrrolidine-2-carboxamide 1439404-18-8 C29H33Cl2FN4O6S
(2S,4R)-N-((S)-1-(butylamino)-1,2-dioxopentan-3-yl)-1-(1-(5-chloro-3-fluoropyridin-2-yl)cyclopropanecarbonyl)-4-(2-chlorophenylsulfonyl)pyrrolidine-2-carboxamide
—— kravanhin B 1422517-73-4 C20H28O3
kravanhin B
—— 2-[[5-cyano-2-(4-fluorophenyl)-1H-pyrrolo-[2,3-b]pyridin-4-yl]amino]-N-methylbenzamide 1420885-81-9 C22H16FN5O
2-[[5-cyano-2-(4-fluorophenyl)-1H-pyrrolo-[2,3-b]pyridin-4-yl]amino]-N-methylbenzamide
—— 2-[2-(2,6-dichloro-phenyl)-2H-pyrazolo[4,3-c]pyridin-4-ylamino]-isonicotinamide 1378038-09-5 C18H12Cl2N6O
2-[2-(2,6-dichloro-phenyl)-2H-pyrazolo[4,3-c]pyridin-4-ylamino]-isonicotinamide
—— {6-[7-bromo-2-(2,6-dichlorophenyl)-2H-pyrazolo[4,3-c]pyridin-4-ylamino]-pyrimidin-4-yl}-carbamic acid tert-butyl ester 1378040-04-0 C21H18BrCl2N7O2
{6-[7-bromo-2-(2,6-dichlorophenyl)-2H-pyrazolo[4,3-c]pyridin-4-ylamino]-pyrimidin-4-yl}-carbamic acid tert-butyl ester
—— 4-{[4-bromo-3-(tetrahydropyran-2-yloxy)benzyl][1,2,4]triazol-4-ylamino}benzonitrile 870779-66-1 C21H20BrN5O2
4-{[4-bromo-3-(tetrahydropyran-2-yloxy)benzyl][1,2,4]triazol-4-ylamino}benzonitrile
—— (Diethyldithiocarbamato)bis(triethylphosphin)palladium(II)-iodid 73887-87-3 C17H40NP2PdS2*I
(Diethyldithiocarbamato)bis(triethylphosphin)palladium(II)-iodid
—— 3-[4-[(1S,3S)-3-[[(1R)-1-(4-fluoro-3-methoxy-phenyl)ethyl]amino]cyclopentyl]-2-(trifluoromethyl)phenyl]propanoic acid 1256944-73-6 C24H27F4NO3
3-[4-[(1S,3S)-3-[[(1R)-1-(4-fluoro-3-methoxy-phenyl)ethyl]amino]cyclopentyl]-2-(trifluoromethyl)phenyl]propanoic acid
—— N-cyclopropyl-4-{7,8-difluoro-4-[(4-hydroxybutyl)amino]imidazo[1,2-a]quinoxalin-1-yl}benzamide 1254194-53-0 C24H23F2N5O2
N-cyclopropyl-4-{7,8-difluoro-4-[(4-hydroxybutyl)amino]imidazo[1,2-a]quinoxalin-1-yl}benzamide
—— (R)-(+)-5-(1-Aminoaethyl)-3-isoxazolol-zwitterion 69489-06-1 C5H8N2O2
(R)-(+)-5-(1-Aminoaethyl)-3-isoxazolol-zwitterion
—— (S)-3-((3R,4S)-6-iodo-3-vinylchroman-4-ylamino)-4-isopropyl-2-oxazolidinone 1187455-25-9 C17H21IN2O3
(S)-3-((3R,4S)-6-iodo-3-vinylchroman-4-ylamino)-4-isopropyl-2-oxazolidinone
—— N-(4-(4-methyl-1-piperazinyl)phenyl)-spiro[chromeno[3,4-d]pyrimidine-5,4'-piperidine]-3-amine 1190961-37-5 C26H30N6O
N-(4-(4-methyl-1-piperazinyl)phenyl)-spiro[chromeno[3,4-d]pyrimidine-5,4'-piperidine]-3-amine
—— 5-amino-2-tert-butyl-4-(6-methylpyridin-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide 1190976-74-9 C17H19N5OS
5-amino-2-tert-butyl-4-(6-methylpyridin-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
—— 4-((R)-2-[(4-phenyl-6-p-tolyl-pyridine-2-carbonyl)-amino]-3-phosphono-propionyl)-piperazine-1-carboxylic acid butyl ester 1191263-54-3 C31H37N4O7P
4-((R)-2-[(4-phenyl-6-p-tolyl-pyridine-2-carbonyl)-amino]-3-phosphono-propionyl)-piperazine-1-carboxylic acid butyl ester
—— 2-[1-(4-Fluorophenyl)-4-(3-methoxyphenyl)imidazol-2-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone 1443769-83-2 C27H26FN5O2
2-[1-(4-Fluorophenyl)-4-(3-methoxyphenyl)imidazol-2-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone
—— (4R)-4-[(3R,5R,8R,9S,10S,12S,13R,14S,17R)-3,12-dihydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]-N-[2-(prop-2-enoylamino)ethyl]pentanamide 1423138-41-3 C29H48N2O4
(4R)-4-[(3R,5R,8R,9S,10S,12S,13R,14S,17R)-3,12-dihydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]-N-[2-(prop-2-enoylamino)ethyl]pentanamide
—— cyclopropylmethyl (2S)-2-[[(4-fluorophenoxy)-[[(2R,4R)-4-(5-methyl-2,4-dioxo-pyrimidin-1-yl)-1,3-dioxolan-2-yl]methoxy]phosphoryl]amino]propanoate 1142818-11-8 C22H27FN3O9P
cyclopropylmethyl (2S)-2-[[(4-fluorophenoxy)-[[(2R,4R)-4-(5-methyl-2,4-dioxo-pyrimidin-1-yl)-1,3-dioxolan-2-yl]methoxy]phosphoryl]amino]propanoate