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中文名称 英文名称 CAS号 化学式 结构式图片
—— Oscillapeptilide 97-A 264909-19-5 C53H75N9O13
Oscillapeptilide 97-A
—— (2R)-N-cyclopropyl-N-{[1-(3-methoxypropyl)-4-methylindol-3-yl]methyl}morpholine-2-carboxamide 1093080-24-0 C22H31N3O3
(2R)-N-cyclopropyl-N-{[1-(3-methoxypropyl)-4-methylindol-3-yl]methyl}morpholine-2-carboxamide
—— 9-hydroxy-N,N-dimethyl-9-(trifluoromethyl)fluorene-4-carboxamide 1220961-12-5 C17H14F3NO2
9-hydroxy-N,N-dimethyl-9-(trifluoromethyl)fluorene-4-carboxamide
—— 6-(3-Fluoro-4-methylphenyl)-2-(3-methylbutyl)-4-(trifluoromethyl)nicotinic acid 1130343-99-5 C19H19F4NO2
6-(3-Fluoro-4-methylphenyl)-2-(3-methylbutyl)-4-(trifluoromethyl)nicotinic acid
—— 8-[[3-chloro-5-[[(2R)-oxolan-2-yl]methylsulfanyl]pyridin-4-yl]methoxy]-2-methyl-4-(2-methylpyrazol-3-yl)quinoline 1064670-44-5 C25H25ClN4O2S
8-[[3-chloro-5-[[(2R)-oxolan-2-yl]methylsulfanyl]pyridin-4-yl]methoxy]-2-methyl-4-(2-methylpyrazol-3-yl)quinoline
—— Ethyl 4-[3-[3-(4-acetyloxybutoxy)phenyl]-4-cyanopyrrol-1-yl]benzoate 1072199-06-4 C26H26N2O5
Ethyl 4-[3-[3-(4-acetyloxybutoxy)phenyl]-4-cyanopyrrol-1-yl]benzoate
—— —— 1448423-45-7 C20H16N2O4
—— —— 1451261-34-9 C11H23NO2S
—— —— 1613389-55-1 C15H17NO3
—— 3-(2-chloro-5,6,7,8-tetrahydroquinolin-8-yl)-5-fluoro-2-oxo-N-1,3-thiazol-2-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide 1432514-14-1 C19H14ClFN4O4S2
3-(2-chloro-5,6,7,8-tetrahydroquinolin-8-yl)-5-fluoro-2-oxo-N-1,3-thiazol-2-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide
—— 1-[6-(5-fluoro-2-((6-(3,4-dichlorophenoxy)pyridin-3-yl)methyloxy)-phenyl)pyridin-2-yl]-5-trifluoromethyl-pyrazole-4-carboxylic acid 1160429-52-6 C28H16Cl2F4N4O4
1-[6-(5-fluoro-2-((6-(3,4-dichlorophenoxy)pyridin-3-yl)methyloxy)-phenyl)pyridin-2-yl]-5-trifluoromethyl-pyrazole-4-carboxylic acid
—— 4-[(3-aminopyridin-4-yl)methyl]piperazin-2-one 1334713-27-7 C10H14N4O
4-[(3-aminopyridin-4-yl)methyl]piperazin-2-one
—— (8Z)-3(R)-(4-fluorophenyl)-5,6-dihydro-8-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]methylene]-3,6(R)-dimethyl-3H,8H-[1,2,4]oxadiazolo[3,4-c][1,4]oxazine 1080671-18-6 C25H25FN4O3
(8Z)-3(R)-(4-fluorophenyl)-5,6-dihydro-8-[[3-methoxy-4-(4-methyl-1H-imidazol-1-yl)phenyl]methylene]-3,6(R)-dimethyl-3H,8H-[1,2,4]oxadiazolo[3,4-c][1,4]oxazine
—— 3-[2-(2-{2-[((1R,2S)-1-tert-butoxycarbonylamino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylamino}-ethoxy)-ethoxy]-propionic acid methyl ester 1051392-11-0 C25H37N3O9S
3-[2-(2-{2-[((1R,2S)-1-tert-butoxycarbonylamino-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylamino}-ethoxy)-ethoxy]-propionic acid methyl ester
—— N-benzyl-N-methyl-6,7-dihydro-3H-pyrazolo[4',3':5,6]pyrido[4,3-f]quinazolin-9-amine 1234372-21-4 C20H18N6
N-benzyl-N-methyl-6,7-dihydro-3H-pyrazolo[4',3':5,6]pyrido[4,3-f]quinazolin-9-amine
—— methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[2-[(2S)-1-[(2S,3R)-3-methoxy-2-(methoxycarbonylamino)butanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1242088-49-8 C40H48N8O7
methyl N-[(2S)-1-[(2S)-2-[5-[4-[2-[2-[(2S)-1-[(2S,3R)-3-methoxy-2-(methoxycarbonylamino)butanoyl]pyrrolidin-2-yl]-3H-benzimidazol-5-yl]ethynyl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 7-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-N-[(1S,2R)-2-methoxy-2,3-dihydro-1H-inden-1-yl]-3,4-dihydroisoquinoline-2(1H)-carboxamide 1246207-81-7 C29H35N7O2
7-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-N-[(1S,2R)-2-methoxy-2,3-dihydro-1H-inden-1-yl]-3,4-dihydroisoquinoline-2(1H)-carboxamide
—— (3-Hydroxyazetidin-1-yl)-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]methanone 1220961-57-8 C18H14F3NO3
(3-Hydroxyazetidin-1-yl)-[9-hydroxy-9-(trifluoromethyl)fluoren-2-yl]methanone
—— 6-(3,4-difluorophenyl)-N-(4-(2-(4-(2-methoxyethyl)piperazin-1-yl)ethyl)phenyl)-5,6-dihydrobenzo[h]quinazolin-2-amine 1234350-49-2 C33H35F2N5O
6-(3,4-difluorophenyl)-N-(4-(2-(4-(2-methoxyethyl)piperazin-1-yl)ethyl)phenyl)-5,6-dihydrobenzo[h]quinazolin-2-amine
—— 1-(3,4-dimethyl-3<i>H</i>-thiazol-2-ylidene)-2,3-dimethyl-isothiourea 75398-92-4 C8H13N3S2
1-(3,4-dimethyl-3<i>H</i>-thiazol-2-ylidene)-2,3-dimethyl-isothiourea
—— N-(3,4-dichlorophenyl)-N-{1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}propionamide hydrochloride 1161704-89-7 C23H28Cl2N2O2*ClH
N-(3,4-dichlorophenyl)-N-{1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}propionamide hydrochloride
—— 3-phenylsulphonylmethylcyclopropane-trans-1,2-dicarboxylate 115373-58-5 C14H16O6S
3-phenylsulphonylmethylcyclopropane-trans-1,2-dicarboxylate
—— tert-butyl 4-(3-(1-((1-benzylpiperidin-4-yl)(methyl)carbamoyl)-1H-imidazol-4-yl)benzoyl)piperazine-1-carboxylate 1356960-63-8 C33H42N6O4
tert-butyl 4-(3-(1-((1-benzylpiperidin-4-yl)(methyl)carbamoyl)-1H-imidazol-4-yl)benzoyl)piperazine-1-carboxylate
—— (E)-2-(phenyl(phenylselanyl)methylene)tetrahydroselenophene 1414875-00-5 C17H16Se2
(E)-2-(phenyl(phenylselanyl)methylene)tetrahydroselenophene
—— 2-(difluoromethyl)-5-(methylsulfonyl)pyridine 1574401-82-3 C7H7F2NO2S
2-(difluoromethyl)-5-(methylsulfonyl)pyridine
—— 1-(2,5-difluorobenzyl)-7-methoxy-3-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydronaphthalene 1245637-15-3 C26H26F2O2
1-(2,5-difluorobenzyl)-7-methoxy-3-(4-methoxy-phenyl)-2-methyl-1,2,3,4-tetrahydronaphthalene
—— 7-(2-chlorophenyl)-6,7-dihydro-3H-benzo[f]pyrazolo[3,4-c]isoquinoline 1234371-51-7 C20H14ClN3
7-(2-chlorophenyl)-6,7-dihydro-3H-benzo[f]pyrazolo[3,4-c]isoquinoline
—— (R)-2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenethyl methanesulfonate 1234352-30-7 C27H23F2N3O3S
(R)-2-fluoro-5-(6-(2-fluorophenyl)-5,6-dihydrobenzo[h]quinazolin-2-ylamino)phenethyl methanesulfonate
—— 1-acetyl-4-(4-(4-chlorophenyl)-5-(4-methoxyphenyl)oxazol-2-yl)piperidine 951744-38-0 C23H23ClN2O3
1-acetyl-4-(4-(4-chlorophenyl)-5-(4-methoxyphenyl)oxazol-2-yl)piperidine
—— methyl 2,6-di-tert-butylisonicotinate 69209-41-2 C15H23NO2
methyl 2,6-di-tert-butylisonicotinate
—— (S)-2-(8-(5-(hydroxymethyl)thiazol-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid 1080639-65-1 C21H20N2O6S2
(S)-2-(8-(5-(hydroxymethyl)thiazol-2-yl)dibenzo[b,d]furan-3-sulfonamido)-3-methylbutanoic acid
—— —— 1356687-03-0 C13H18O6
—— N-{[4-(3-methoxypropoxy)-2-naphthyl]methyl}cyclopropanamine 1093083-13-6 C18H23NO2
N-{[4-(3-methoxypropoxy)-2-naphthyl]methyl}cyclopropanamine
—— 2-Cyclohexyl-9-(trifluoromethyl)fluoren-9-ol 1220962-47-9 C20H19F3O
2-Cyclohexyl-9-(trifluoromethyl)fluoren-9-ol
—— tert-butyl 3-hexylcyclobut-2-enecarboxylate 1422357-14-9 C15H26O2
tert-butyl 3-hexylcyclobut-2-enecarboxylate
—— Dimethyl 5-[(4-ethynylphenyl)carbamoylamino]benzene-1,3-dicarboxylate 1137673-93-8 C19H16N2O5
Dimethyl 5-[(4-ethynylphenyl)carbamoylamino]benzene-1,3-dicarboxylate
—— (3R,4R)-3-(2,4-dichlorophenyl)-1-oxo-2-[(3R)-2-oxopiperidin-3-yl]-N-phenylmethoxy-3,4-dihydroisoquinoline-4-carboxamide 1091588-96-3 C28H25Cl2N3O4
(3R,4R)-3-(2,4-dichlorophenyl)-1-oxo-2-[(3R)-2-oxopiperidin-3-yl]-N-phenylmethoxy-3,4-dihydroisoquinoline-4-carboxamide
—— 4-(3-Benzoyl-4-cyanopyrrol-1-yl)benzoic acid 1072200-88-4 C19H12N2O3
4-(3-Benzoyl-4-cyanopyrrol-1-yl)benzoic acid
—— 4-methylphenyl 3-(4-fluorophenylthio)-2-methyl-N-(4-methylphenyl)-2-propenimidothioate 1158848-18-0 C24H22FNS2
4-methylphenyl 3-(4-fluorophenylthio)-2-methyl-N-(4-methylphenyl)-2-propenimidothioate
—— N'-[5-bromo-2-methyl-6-[[3-(2-phenylethyl)phenyl]methoxy]pyridin-3-yl]-N-ethyl-N-methylmethanimidamide 1404444-66-1 C25H28BrN3O
N'-[5-bromo-2-methyl-6-[[3-(2-phenylethyl)phenyl]methoxy]pyridin-3-yl]-N-ethyl-N-methylmethanimidamide
—— 6-Methoxy-2-[(3-methylphenoxy)methyl]-4(3H)-pyrimidinone 67386-41-8 C13H14N2O3
6-Methoxy-2-[(3-methylphenoxy)methyl]-4(3H)-pyrimidinone
—— N-(adamantan-1-ylmethyl)-2-{[4-(2-methoxyethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine-5-carboxamide 1031829-87-4 C27H37N5O3
N-(adamantan-1-ylmethyl)-2-{[4-(2-methoxyethyl)piperazin-1-yl]carbonyl}imidazo[1,2-a]pyridine-5-carboxamide
—— 2-bromo-1-[(3S,5R,8R,9R,10S,13S,14S,17S)-3-(fluoromethyl)-3-hydroxy-13-methyl-2,4,5,6,7,8,9,10,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]ethanone 1430063-72-1 C21H32BrFO2
2-bromo-1-[(3S,5R,8R,9R,10S,13S,14S,17S)-3-(fluoromethyl)-3-hydroxy-13-methyl-2,4,5,6,7,8,9,10,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]ethanone
—— (1R,2S,4R,5S,8S,12R)-7-(3,4-dichlorophenyl)-2-hydroxy-4-methyl-9,13-dioxa-7-azatetracyclo[6.3.1.1(1,4).0(5,12)]tridecan-6-one 1095183-31-5 C17H17Cl2NO4
(1R,2S,4R,5S,8S,12R)-7-(3,4-dichlorophenyl)-2-hydroxy-4-methyl-9,13-dioxa-7-azatetracyclo[6.3.1.1(1,4).0(5,12)]tridecan-6-one
—— 3-(5-Methoxy-benzotriazol-2-yl)-propan-1-ol 362613-83-0 C10H13N3O2
3-(5-Methoxy-benzotriazol-2-yl)-propan-1-ol
—— US10280167, Example 32 1434586-42-1 C15H12N6O2
US10280167, Example 32
—— 1-(3,5-bis(trifluoromethyl)phenyl)-5-(3-chlorophenyl)-1H-pyrazole-3-carboxylic acid methylester 1610952-61-8 C19H11ClF6N2O2
1-(3,5-bis(trifluoromethyl)phenyl)-5-(3-chlorophenyl)-1H-pyrazole-3-carboxylic acid methylester
—— N-methylcarbamate-N-phenyl-O-THP-hydroxylamine 1093102-68-1 C13H17NO4
N-methylcarbamate-N-phenyl-O-THP-hydroxylamine
—— 1-Chloro-1-phenylstanninane 82744-03-4 C11H15ClSn
1-Chloro-1-phenylstanninane
—— (7R)-7-benzyl-8-[5-fluoro-2-(trifluoromethoxy)phenyl]sulfonyl-2,5,8,11,13-pentazatricyclo[8.4.0.02,6]tetradeca-1(14),3,5,10,12-pentaene 1433992-47-2 C23H17F4N5O3S
(7R)-7-benzyl-8-[5-fluoro-2-(trifluoromethoxy)phenyl]sulfonyl-2,5,8,11,13-pentazatricyclo[8.4.0.02,6]tetradeca-1(14),3,5,10,12-pentaene