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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-({[(1-{[6-({4-[(cyclopropylsulfonyl)amino]phenyl}oxy)-2-methyl-3-pyridinyl]methyl}-4-piperidinyl)(3-fluorophenyl)amino]carbonyl}amino)-2,4-difluorobenzamide 1150100-15-4 C35H35F3N6O5S
5-({[(1-{[6-({4-[(cyclopropylsulfonyl)amino]phenyl}oxy)-2-methyl-3-pyridinyl]methyl}-4-piperidinyl)(3-fluorophenyl)amino]carbonyl}amino)-2,4-difluorobenzamide
—— 2-[3,5-Bis(4-fluorophenyl)-1,2,4-triazol-1-yl]-1-[4-(1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethanone 1443254-49-6 C23H20F2N6O2
2-[3,5-Bis(4-fluorophenyl)-1,2,4-triazol-1-yl]-1-[4-(1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethanone
—— 1-[(4R)-2,2-bis(fluoromethyl)-7-(trifluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea 1444800-62-7 C21H18F5N3O4
1-[(4R)-2,2-bis(fluoromethyl)-7-(trifluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
—— 1-Methyl-4-phenyl-benzofuro[3,2-d]pyrimidin-2-one 1251585-62-2 C17H12N2O2
1-Methyl-4-phenyl-benzofuro[3,2-d]pyrimidin-2-one
—— meso-4,4'-((ethane-1,2-diylbis(4,1-phenylene))bis(methylene))bis(1-(hydroxymethyl)-5,7-dimethyl-2,3-dithia-5,7-diazabicyclo[2.2.2]octane-6,8-dione) 1427176-96-2 C30H34N4O6S4
meso-4,4'-((ethane-1,2-diylbis(4,1-phenylene))bis(methylene))bis(1-(hydroxymethyl)-5,7-dimethyl-2,3-dithia-5,7-diazabicyclo[2.2.2]octane-6,8-dione)
—— 4-((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-3a-((2-(4-(methylsulfonyl)piperazin-1-yl)ethylamino)methyl)-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysen-9-yl)benzoic acid 1392113-04-0 C44H67N3O4S
4-((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-3a-((2-(4-(methylsulfonyl)piperazin-1-yl)ethylamino)methyl)-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysen-9-yl)benzoic acid
—— 8-methyl-3-{3-[(S)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-1H-quinazoline-2,4-dione 1422209-08-2 C23H22N4O5S
8-methyl-3-{3-[(S)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propyl}-1H-quinazoline-2,4-dione
—— 1-[(4R)-7-chloro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-[(2R)-7-fluoro-2-hydroxy-2,3-dihydro-1H-inden-4-yl]urea 1443654-07-6 C21H20ClF3N2O3
1-[(4R)-7-chloro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-[(2R)-7-fluoro-2-hydroxy-2,3-dihydro-1H-inden-4-yl]urea
—— (3S,3aR,4S,5aS,7R,8S,9bR)-8-hydroxy-3-methoxy-3,4,7-trimethyl-2-oxo-4,5,6,7,8,9b-hexahydro-3aH-benzo[g][1]benzofuran-5a-carbonitrile 1429194-85-3 C17H23NO4
(3S,3aR,4S,5aS,7R,8S,9bR)-8-hydroxy-3-methoxy-3,4,7-trimethyl-2-oxo-4,5,6,7,8,9b-hexahydro-3aH-benzo[g][1]benzofuran-5a-carbonitrile
—— N-[3-(1-amino-3-methyl-4H-2,7-naphthyridin-3-yl)-4-fluorophenyl]-3,5-difluoropyridine-2-carboxamide 1373686-74-8 C21H16F3N5O
N-[3-(1-amino-3-methyl-4H-2,7-naphthyridin-3-yl)-4-fluorophenyl]-3,5-difluoropyridine-2-carboxamide
—— 2-(3,4-Difluorophenyl)-N-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]acetamide 1227094-22-5 C18H19F2N3O
2-(3,4-Difluorophenyl)-N-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]acetamide
—— (2S)-2-tert-butoxy-2-[4-(4-chlorophenyl)-6-(5,6-dihydro-4H-cyclopenta[d]thiazol-2-ylcarbamoyl)-2,5-dimethyl-3-pyridyl]acetic acid 1256251-62-3 C26H28ClN3O4S
(2S)-2-tert-butoxy-2-[4-(4-chlorophenyl)-6-(5,6-dihydro-4H-cyclopenta[d]thiazol-2-ylcarbamoyl)-2,5-dimethyl-3-pyridyl]acetic acid
—— 2-fluoro-5-methoxy-N-methyl-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide 1441200-16-3 C21H26F4N6O2
2-fluoro-5-methoxy-N-methyl-4-(4-methylamino-5-(trifluoromethyl)pyrimidin-2-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide
—— N-(3-{2-[2-(2-hydroxyethoxy)ethoxy]-3,5-dimethoxyphenylamino}quinoxalin-2-yl)-4-methoxybenzenesulfonamide 1373670-45-1 C27H30N4O8S
N-(3-{2-[2-(2-hydroxyethoxy)ethoxy]-3,5-dimethoxyphenylamino}quinoxalin-2-yl)-4-methoxybenzenesulfonamide
—— Propan-2-yl 24-oxo-5-(2,2,2-trifluoroethoxy)-14-oxa-2,4,6,8,17,23,32-heptazatetracyclo[23.2.2.210,13.13,7]dotriaconta-1(27),3,5,7(32),10(31),11,13(30),25,28-nonaene-17-carboxylate 1373163-43-9 C30H36F3N7O5
Propan-2-yl 24-oxo-5-(2,2,2-trifluoroethoxy)-14-oxa-2,4,6,8,17,23,32-heptazatetracyclo[23.2.2.210,13.13,7]dotriaconta-1(27),3,5,7(32),10(31),11,13(30),25,28-nonaene-17-carboxylate
—— (2R)-1-((2S)-2-((dimethylamino)methyl)pyrrolidin-1-yl)-2-methylamino-3-phenylpropan-1-one 254905-73-2 C17H27N3O
(2R)-1-((2S)-2-((dimethylamino)methyl)pyrrolidin-1-yl)-2-methylamino-3-phenylpropan-1-one
—— (S)-3-[(2S,3R)-2-Hydroxy-5-methyl-3-(2,4,6-trimethyl-benzenesulfonylamino)-hexylamino]-N-isopropyl-succinamic acid tert-butyl ester 433922-95-3 C27H47N3O6S
(S)-3-[(2S,3R)-2-Hydroxy-5-methyl-3-(2,4,6-trimethyl-benzenesulfonylamino)-hexylamino]-N-isopropyl-succinamic acid tert-butyl ester
—— 4-[4-[[4-(4-fluorophenyl)-2-methylsulfinyl-1H-imidazole-5-carbonyl]amino]phenoxy]-N-methylpyridine-2-carboxamide 1422175-84-5 C24H20FN5O4S
4-[4-[[4-(4-fluorophenyl)-2-methylsulfinyl-1H-imidazole-5-carbonyl]amino]phenoxy]-N-methylpyridine-2-carboxamide
—— 2-([1,4]dioxan-2-ylmethoxy)-9-(3-hydroxy-5-methyl-hex-1-ynyl)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one 1445847-07-3 C24H28N2O5
2-([1,4]dioxan-2-ylmethoxy)-9-(3-hydroxy-5-methyl-hex-1-ynyl)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one
—— 2-O-benzyl-4,6-O-benzylidene-1-allyl-1,3-dideoxy-α-D-glucopyranose 1403351-24-5 C23H26O4
2-O-benzyl-4,6-O-benzylidene-1-allyl-1,3-dideoxy-α-D-glucopyranose
—— (S)-ethyl 2-((diphenoxyphosphoryl)oxy)-7-((R)-5-oxo-2,5-dihydrofuran-2-yl)cyclohept-1-enecarboxylate 1425314-19-7 C26H27O8P
(S)-ethyl 2-((diphenoxyphosphoryl)oxy)-7-((R)-5-oxo-2,5-dihydrofuran-2-yl)cyclohept-1-enecarboxylate
—— 3-[4-(4-cyano-phenyl)-[1,2,3]triazol-1-ylmethyl]-N-[6-(cyclopropyl-methyl-amino)-4,5,6,7-tetrahydro-benzothiazol-2-yl]-benzamide 1373515-96-8 C28H27N7OS
3-[4-(4-cyano-phenyl)-[1,2,3]triazol-1-ylmethyl]-N-[6-(cyclopropyl-methyl-amino)-4,5,6,7-tetrahydro-benzothiazol-2-yl]-benzamide
—— 1-[(5-Bromo-2-{2-ethylbutyloxy}phenyl)methyl]-5-methyl-1H-pyrazole-4-carboxylic acid 1444367-32-1 C18H23BrN2O3
1-[(5-Bromo-2-{2-ethylbutyloxy}phenyl)methyl]-5-methyl-1H-pyrazole-4-carboxylic acid
—— N-((6-methyl-2-phenylquinolin-4-yl)methyl)-N-(p-tolyl)acetamide 1402150-87-1 C26H24N2O
N-((6-methyl-2-phenylquinolin-4-yl)methyl)-N-(p-tolyl)acetamide
—— 2-(3-((R)-1-((S)-1-(4-chlorobenzylsulfonyl)piperidine-2-carbonyloxy)-3-(3,4-dimethoxyphenyl)propyl)phenoxy)acetic acid 1373829-93-6 C32H36ClNO9S
2-(3-((R)-1-((S)-1-(4-chlorobenzylsulfonyl)piperidine-2-carbonyloxy)-3-(3,4-dimethoxyphenyl)propyl)phenoxy)acetic acid
—— (rac)-4-(4,5-difluoro-2-methoxyphenyl)-N-{3-[(S-methylsulfonimidoyl)methyl]phenyl}-1,3,5-triazin-2-amine 1414944-07-2 C18H17F2N5O2S
(rac)-4-(4,5-difluoro-2-methoxyphenyl)-N-{3-[(S-methylsulfonimidoyl)methyl]phenyl}-1,3,5-triazin-2-amine
—— ethyl {[(3-{[4-(2,3-dihydro-1-benzofuran-7-yl)-1,3,5-triazin-2-yl]amino}phenyl)methyl](methyl)oxo-λ<sup>6</sup>-sulfanylidene}carbamate 1415248-63-3 C22H23N5O4S
ethyl {[(3-{[4-(2,3-dihydro-1-benzofuran-7-yl)-1,3,5-triazin-2-yl]amino}phenyl)methyl](methyl)oxo-λ<sup>6</sup>-sulfanylidene}carbamate
—— 1-((2-methyl-1H-indol-4-yl)methyl)-9-(4-methylpyrimidin-2-yl)-1,9-diazaspiro[5.5]undecan-2-one 1373766-01-8 C24H29N5O
1-((2-methyl-1H-indol-4-yl)methyl)-9-(4-methylpyrimidin-2-yl)-1,9-diazaspiro[5.5]undecan-2-one
—— Methyl 4-cyclohexyl-2-ethoxyfuro[2,3-c]quinoline-1-carboxylate 1374336-87-4 C21H23NO4
Methyl 4-cyclohexyl-2-ethoxyfuro[2,3-c]quinoline-1-carboxylate
—— 1-[2-cyclopentyl-3-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)piperidin-1-yl]-2-(3,5-dichloroanilino)ethanone 1374240-44-4 C24H28Cl2N6O
1-[2-cyclopentyl-3-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)piperidin-1-yl]-2-(3,5-dichloroanilino)ethanone
—— 2,2-dimethyl-3-[1-[5-(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)pyridin-2-yl]piperidin-4-yl]oxypropanoic acid 1445205-79-7 C21H25N5O3S
2,2-dimethyl-3-[1-[5-(5-thiophen-2-yl-1H-1,2,4-triazol-3-yl)pyridin-2-yl]piperidin-4-yl]oxypropanoic acid
—— 9-tert-butoxymethyl-2-([1,4]dioxan-2-ylmethoxy)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one 1445846-94-5 C22H28N2O5
9-tert-butoxymethyl-2-([1,4]dioxan-2-ylmethoxy)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one
—— 1-[(4R)-7,8-dichloro-2,2-diethyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-5-yl)urea 1444792-67-9 C23H26Cl2N4O3
1-[(4R)-7,8-dichloro-2,2-diethyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-5-yl)urea
—— [3,3-Dimethyl-4-(1-phenyl-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-[3-(2-methylpropoxy)phenyl]methanone 1443757-06-9 C26H31N5O3
[3,3-Dimethyl-4-(1-phenyl-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-[3-(2-methylpropoxy)phenyl]methanone
—— [(1S,3S,4R,6R,8S,9R,10R,12R)-6-cyano-3,12-dimethoxy-4,8,10-trimethyl-2-oxo-11-oxatricyclo[7.2.1.01,6]dodecan-10-yl]methyl acetate 1429194-94-4 C20H29NO6
[(1S,3S,4R,6R,8S,9R,10R,12R)-6-cyano-3,12-dimethoxy-4,8,10-trimethyl-2-oxo-11-oxatricyclo[7.2.1.01,6]dodecan-10-yl]methyl acetate
—— [(1R)-1-{[4-(2-methoxyphenyl)-4-oxobutanoyl]amino}-2-(3-thienyl)ethyl]boronic acid 1444009-59-9 C17H20BNO5S
[(1R)-1-{[4-(2-methoxyphenyl)-4-oxobutanoyl]amino}-2-(3-thienyl)ethyl]boronic acid
—— [2,6-dichloro-4-(2-methoxypyrimidin-5-yl)phenyl](1H-pyrrolo[2,3-c]pyridin-3-yl)methanone 1415123-00-0 C19H12Cl2N4O2
[2,6-dichloro-4-(2-methoxypyrimidin-5-yl)phenyl](1H-pyrrolo[2,3-c]pyridin-3-yl)methanone
—— (2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid 1443788-31-5 C32H35N3O4
(2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-tert-butylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]propanoic acid
—— 3,4-dihydroxy-1-(4-methoxyphenyl)-N,N-dimethyl-5-(piperidine-1-carbonyl)-1H-pyrrole-2-carboxamide 1443052-95-6 C20H25N3O5
3,4-dihydroxy-1-(4-methoxyphenyl)-N,N-dimethyl-5-(piperidine-1-carbonyl)-1H-pyrrole-2-carboxamide
—— 2-(2,6-dichlorophenyl)-N-(pyrimidin-4-yl)thiazolo[5,4-c]pyridin-4-amine 1365989-64-5 C16H9Cl2N5S
2-(2,6-dichlorophenyl)-N-(pyrimidin-4-yl)thiazolo[5,4-c]pyridin-4-amine
—— {4-[2-((S)-2-amino-4,5-dihydro-oxazol-4-yl)-ethyl]-phenyl}-(4-methoxy-pyrimidin-2-yl)-amine 1374037-87-2 C16H19N5O2
{4-[2-((S)-2-amino-4,5-dihydro-oxazol-4-yl)-ethyl]-phenyl}-(4-methoxy-pyrimidin-2-yl)-amine
—— N-[3-(1-amino-3-methyl-4H-2,6-naphthyridin-3-yl)-4-fluorophenyl]-5-chloropyridine-2-carboxamide 1373686-92-0 C21H17ClFN5O
N-[3-(1-amino-3-methyl-4H-2,6-naphthyridin-3-yl)-4-fluorophenyl]-5-chloropyridine-2-carboxamide
—— N-[(3-aminoisoindol-1-ylidene)amino]isoquinoline-3-carboxamide 1356546-43-4 C18H13N5O
N-[(3-aminoisoindol-1-ylidene)amino]isoquinoline-3-carboxamide
—— 2-[4-(4-Fluoro-3-methylphenyl)-1-(4-fluorophenyl)imidazol-2-yl]-1-[4-(1,3,5-triazin-2-yl)piperazin-1-yl]ethanone 1443769-70-7 C25H23F2N7O
2-[4-(4-Fluoro-3-methylphenyl)-1-(4-fluorophenyl)imidazol-2-yl]-1-[4-(1,3,5-triazin-2-yl)piperazin-1-yl]ethanone
—— [(1,1-dimethylethyl)oxy][2-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1-oxo-1,2-dihydro-3-isoquinolinyl]acetic acid 1392118-59-0 C20H23N3O4
[(1,1-dimethylethyl)oxy][2-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1-oxo-1,2-dihydro-3-isoquinolinyl]acetic acid
—— 2',3',5'-tri-O-benzoyl-5-iodocytidine 1109220-17-8 C30H24IN3O8
2',3',5'-tri-O-benzoyl-5-iodocytidine
—— (2R,3R,5R,6R)-5,6-bis(iodomethyl)-2,3-dimethoxy-2,3-dimethyl-1,4-dioxane 1203603-60-4 C10H18I2O4
(2R,3R,5R,6R)-5,6-bis(iodomethyl)-2,3-dimethoxy-2,3-dimethyl-1,4-dioxane
—— N-[1-({5-bromo-2-[(phenylmethyl)oxy]phenyl}methyl)-1H-pyrazol-4-yl]-2,6-difluorobenzamide 1373394-76-3 C24H18BrF2N3O2
N-[1-({5-bromo-2-[(phenylmethyl)oxy]phenyl}methyl)-1H-pyrazol-4-yl]-2,6-difluorobenzamide
—— 2-[(2,6-dichlorophenyl)amino]-7,7-dimethyl-N-[2-(morpholin-4-yl)ethyl]-7,8-dihydro-1H-furo[3,2-e]benzimidazole-5-carboxamide 1374296-65-7 C24H27Cl2N5O3
2-[(2,6-dichlorophenyl)amino]-7,7-dimethyl-N-[2-(morpholin-4-yl)ethyl]-7,8-dihydro-1H-furo[3,2-e]benzimidazole-5-carboxamide
—— 2-Cyclohexylimino-3-cyclohexyl-4,5-diphenyl-Δ<sup>4</sup>-oxazolin 6652-41-1 C27H32N2O
2-Cyclohexylimino-3-cyclohexyl-4,5-diphenyl-Δ<sup>4</sup>-oxazolin