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—— methyl (2S)-2-[[(4aR,7R,7aS)-6-(4-amino-2-oxopyrimidin-1-yl)-7-azido-7-methyl-2-oxo-4,4a,6,7a-tetrahydrofuro[3,2-d][1,3,2]dioxaphosphinin-2-yl]amino]propanoate —— C14H20N7O7P
methyl (2S)-2-[[(4aR,7R,7aS)-6-(4-amino-2-oxopyrimidin-1-yl)-7-azido-7-methyl-2-oxo-4,4a,6,7a-tetrahydrofuro[3,2-d][1,3,2]dioxaphosphinin-2-yl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-(3,4-dichlorophenoxy)phosphoryl]amino]propanoate —— C19H19Cl2N6O9P
methyl (2S)-2-[[[(2R,3S)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-(3,4-dichlorophenoxy)phosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(2-chlorophenoxy)phosphoryl]amino]propanoate —— C20H24ClN6O9P
methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(2-chlorophenoxy)phosphoryl]amino]propanoate
—— methyl (2R)-2-[3-chloro-5-[(2S)-1-methoxy-1-oxopropan-2-yl]oxy-4-methyl-2-oxochromen-7-yl]oxypropanoate —— C18H19ClO8
methyl (2R)-2-[3-chloro-5-[(2S)-1-methoxy-1-oxopropan-2-yl]oxy-4-methyl-2-oxochromen-7-yl]oxypropanoate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-4-amino-5-(2-amino-6-ethoxypurin-9-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate —— C22H32N7O11P
methyl (2S)-2-[[[(2R,3S,4R,5R)-4-amino-5-(2-amino-6-ethoxypurin-9-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate
—— Methyl 5-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxylate 1620412-21-6 C10H11F3N2O2
Methyl 5-(trifluoromethyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridine-3-carboxylate
—— methyl 2-[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-[[(2S)-1-methoxy-1-oxopropan-2-yl]amino]phosphoryl]oxybenzoate —— C22H27N6O11P
methyl 2-[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-[[(2S)-1-methoxy-1-oxopropan-2-yl]amino]phosphoryl]oxybenzoate
—— methyl (2S)-2-[[[(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate —— C20H25FN7O8P
methyl (2S)-2-[[[(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate —— C19H20FN6O9P
methyl (2S)-2-[[[(2R,3S)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate
—— Methyl 2,3-dihydro-4-hydroxy-7-benzofurancarboxylate 1620412-65-8 C10H10O4
Methyl 2,3-dihydro-4-hydroxy-7-benzofurancarboxylate
—— methyl N-[(2S)-1-[(2S)-4-fluoro-2-[5-[4-[2-[(5R)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-3,3-dimethyl-1,3-azasilolidin-5-yl]-3H-benzo[e]benzimidazol-7-yl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1334312-51-4 C43H53FN8O6Si
methyl N-[(2S)-1-[(2S)-4-fluoro-2-[5-[4-[2-[(5R)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-3,3-dimethyl-1,3-azasilolidin-5-yl]-3H-benzo[e]benzimidazol-7-yl]phenyl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(5-methyl-2-propan-2-ylphenoxy)phosphoryl]amino]propanoate —— C24H33N6O9P
methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(5-methyl-2-propan-2-ylphenoxy)phosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R,5S)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate 1403574-35-5 C26H29N8O7P
methyl (2S)-2-[[[(2R,3S,4R,5S)-5-(4-aminopyrrolo[2,1-f][1,2,4]triazin-7-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate —— C24H27N6O9P
methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate —— C20H25N6O9P
methyl (2S)-2-[[[(2R,3S,4R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate —— C23H24N7O8P
methyl (2S)-2-[[[(2R,3S)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-2,3-dihydrofuran-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-methoxyphosphoryl]amino]propanoate —— C15H24N7O8P
methyl (2S)-2-[[[(2R,3S,4R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-methoxyphosphoryl]amino]propanoate
—— methyl (2S)-2-[3-chloro-5-[(2S)-1-methoxy-1-oxopropan-2-yl]oxy-4-methyl-2-oxochromen-7-yl]oxypropanoate —— C18H19ClO8
methyl (2S)-2-[3-chloro-5-[(2S)-1-methoxy-1-oxopropan-2-yl]oxy-4-methyl-2-oxochromen-7-yl]oxypropanoate
—— methyl (Z)-5-aminopent-3-enoate —— C6H11NO2
methyl (Z)-5-aminopent-3-enoate
—— methyl 3-[(4-bromobenzoyl)amino]-1H-1,2,4-triazole-5-carboxylate —— C11H9BrN4O3
methyl 3-[(4-bromobenzoyl)amino]-1H-1,2,4-triazole-5-carboxylate
—— methyl N-[1-[(2S)-2-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C36H36ClN5O4S
methyl N-[1-[(2S)-2-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-ethoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-tert-butyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate —— C25H36N9O11P
methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-ethoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-tert-butyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate —— C20H24FN6O9P
methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(4-fluorophenoxy)phosphoryl]amino]propanoate
—— methyl N-[1-(2,2-dimethyloxan-4-yl)-2-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate —— C56H68FN9O9S
methyl N-[1-(2,2-dimethyloxan-4-yl)-2-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-10-[2-[(2S)-pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1620559-78-5 C45H51FN8O5S
methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-10-[2-[(2S)-pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-ethoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate —— C22H30N9O11P
methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-ethoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-[(5-methyl-2-oxo-1,3-dioxol-4-yl)methoxy]phosphoryl]amino]propanoate
—— methyl N-[1-[(2R,6S)-2,6-dimethyloxan-4-yl]-2-[(2R)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2-methylbutyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate —— C56H68FN9O8S
methyl N-[1-[(2R,6S)-2,6-dimethyloxan-4-yl]-2-[(2R)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2-methylbutyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(5-methyl-2-propan-2-ylphenoxy)phosphoryl]amino]propanoate —— C24H33N6O9P
methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-(5-methyl-2-propan-2-ylphenoxy)phosphoryl]amino]propanoate
—— methyl N-[(1S,2S)-1-[(2S)-2-[1-[[1-[(3S,7aS,11aS,12bR)-6-[(3aS)-5,6,7,7a-tetrahydro-3aH-thieno[3,2-b]pyran-2-yl]-10-[(2R)-1-amino-6-[[(1R,2S)-2-(2,2-dimethyloxan-4-yl)-1-hydroxy-2-[[hydroxy(methoxy)methyl]amino]ethyl]amino]-3-ethyl-3-methylhexan-2-yl]-1-fluoro-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-3-yl]-2-aminoethyl]amino]ethenyl]pyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate —— C57H97FN8O9S
methyl N-[(1S,2S)-1-[(2S)-2-[1-[[1-[(3S,7aS,11aS,12bR)-6-[(3aS)-5,6,7,7a-tetrahydro-3aH-thieno[3,2-b]pyran-2-yl]-10-[(2R)-1-amino-6-[[(1R,2S)-2-(2,2-dimethyloxan-4-yl)-1-hydroxy-2-[[hydroxy(methoxy)methyl]amino]ethyl]amino]-3-ethyl-3-methylhexan-2-yl]-1-fluoro-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-3-yl]-2-aminoethyl]amino]ethenyl]pyrrolidin-1-yl]-1-hydroxy-3-methylbutan-2-yl]carbamate
—— methoxy-[[(2S)-3-methyl-1-(methylamino)butan-2-yl]amino]methanol —— C8H20N2O2
methoxy-[[(2S)-3-methyl-1-(methylamino)butan-2-yl]amino]methanol
—— methyl N-[1-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2,2,2-trifluoroethyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate —— C53H59F4N9O8S
methyl N-[1-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-[5-(2,2,2-trifluoroethyl)thiophen-2-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-methoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate —— C26H30N9O8P
methyl (2S)-2-[[[(2R,3S,4R,5R)-5-(2-amino-6-methoxypurin-9-yl)-4-azido-3-hydroxy-4-methyloxolan-2-yl]methoxy-naphthalen-1-yloxyphosphoryl]amino]propanoate
—— methyl N-[(2S)-1-[(2S)-2-[5-[6-[5-(difluoromethyl)thiophen-2-yl]-1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxymethylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C48H54F3N9O6S
methyl N-[(2S)-1-[(2S)-2-[5-[6-[5-(difluoromethyl)thiophen-2-yl]-1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxymethylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-10-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C44H53BFN5O7S
methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(2-methoxy-2-methylpropyl)thiophen-2-yl]-10-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(1R,2S)-1-[[5-[(3S,7aS,11aS,12bR)-6-[(2R)-2-cyclopropyl-2,3-dihydrothiophen-5-yl]-3-[2-[(2S)-1-[2-[(2R,6S)-2,6-dimethyloxan-4-yl]-1-hydroxy-2-(methoxycarbonylamino)ethyl]pyrrolidin-2-yl]-4,5-dihydro-1H-imidazol-5-yl]-1-fluoro-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-10-yl]-4-ethyl-4-methyl-6-(methylideneamino)hexyl]amino]-1-hydroxy-3-methylbutan-2-yl]carbamate —— C57H91FN8O8S
methyl N-[(1R,2S)-1-[[5-[(3S,7aS,11aS,12bR)-6-[(2R)-2-cyclopropyl-2,3-dihydrothiophen-5-yl]-3-[2-[(2S)-1-[2-[(2R,6S)-2,6-dimethyloxan-4-yl]-1-hydroxy-2-(methoxycarbonylamino)ethyl]pyrrolidin-2-yl]-4,5-dihydro-1H-imidazol-5-yl]-1-fluoro-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-10-yl]-4-ethyl-4-methyl-6-(methylideneamino)hexyl]amino]-1-hydroxy-3-methylbutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[10-[(2Z)-2-[(1R,5R)-2-azabicyclo[3.1.0]hexan-3-ylidene]imidazol-4-yl]-6-(5-cyclopropylthiophen-2-yl)-12-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C44H43FN8O4S
methyl N-[(2S)-1-[(2S)-2-[5-[10-[(2Z)-2-[(1R,5R)-2-azabicyclo[3.1.0]hexan-3-ylidene]imidazol-4-yl]-6-(5-cyclopropylthiophen-2-yl)-12-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[1-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-(5-prop-1-en-2-ylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C50H56FN9O7S
methyl N-[1-[(2S)-2-[5-[1-fluoro-3-[2-[(2S)-1-[2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-(5-prop-1-en-2-ylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(1S)-2-[(1R,3S,5R)-3-[5-[6-(5-cyclopropylthiophen-2-yl)-1-fluoro-3-[2-[1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-1-(oxan-4-yl)-2-oxoethyl]carbamate —— C53H58FN9O8S
methyl N-[(1S)-2-[(1R,3S,5R)-3-[5-[6-(5-cyclopropylthiophen-2-yl)-1-fluoro-3-[2-[1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-1-(oxan-4-yl)-2-oxoethyl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[3-[2-[(2S)-1-ethylpyrrolidin-2-yl]-1H-imidazol-5-yl]-1-fluoro-6-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C46H51FN8O4S
methyl N-[(2S)-1-[(2S)-2-[5-[3-[2-[(2S)-1-ethylpyrrolidin-2-yl]-1H-imidazol-5-yl]-1-fluoro-6-(4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(1R)-1-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-[(3S,5S)-5-[5-[1-fluoro-3-[2-[(2R)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-(5-propan-2-ylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]-2,3-dimethylpyrrolidin-1-yl]-2-oxoethyl]carbamate —— C56H68FN9O8S
methyl N-[(1R)-1-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-[(3S,5S)-5-[5-[1-fluoro-3-[2-[(2R)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6-(5-propan-2-ylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]-2,3-dimethylpyrrolidin-1-yl]-2-oxoethyl]carbamate
—— methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate —— C20H25N6O9P
methyl (2S)-2-[[[(2R,3S,4R,5R)-4-azido-5-(2,4-dioxopyrimidin-1-yl)-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
—— methyl N-[(1R,2S)-1-[[(E)-8-[(3R,8S,10aR)-10-fluoro-5-[2-(1-methoxy-2-methylpropan-2-yl)-2,3-dihydrothiophen-5-yl]-8-[(5S)-2-[(2S)-1-methylpyrrolidin-2-yl]-4,5-dihydro-1H-imidazol-5-yl]-2,3,5,6a,7,8,10a,10b-octahydro-1H-pyrrolo[1,2-c][1,3]benzoxazin-3-yl]-4,6-diethyl-4-methyl-5-(methylaminomethyl)oct-6-enyl]amino]-1-hydroxy-3-methylbutan-2-yl]carbamate —— C50H86FN7O5S
methyl N-[(1R,2S)-1-[[(E)-8-[(3R,8S,10aR)-10-fluoro-5-[2-(1-methoxy-2-methylpropan-2-yl)-2,3-dihydrothiophen-5-yl]-8-[(5S)-2-[(2S)-1-methylpyrrolidin-2-yl]-4,5-dihydro-1H-imidazol-5-yl]-2,3,5,6a,7,8,10a,10b-octahydro-1H-pyrrolo[1,2-c][1,3]benzoxazin-3-yl]-4,6-diethyl-4-methyl-5-(methylaminomethyl)oct-6-enyl]amino]-1-hydroxy-3-methylbutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[5-[6-(5-cyclobutylthiophen-2-yl)-10-[2-[(2S)-1-[2-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-(methoxycarbonylamino)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-1-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C55H64FN9O8S
methyl N-[(2S)-1-[(2S)-2-[5-[6-(5-cyclobutylthiophen-2-yl)-10-[2-[(2S)-1-[2-[(2S,6R)-2,6-dimethyloxan-4-yl]-2-(methoxycarbonylamino)acetyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-1-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— Methyl 3-amino-3-(oxan-4-ylsulfanyl)propanoate —— C9H17NO3S
Methyl 3-amino-3-(oxan-4-ylsulfanyl)propanoate
—— methyl N-[(2S)-1-[[(1S)-1-[5-[6-(5-cyclopropylthiophen-2-yl)-10-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-3-methylbutyl]-methylamino]-3-methyl-1-oxobutan-2-yl]carbamate —— C44H54BN5O6S
methyl N-[(2S)-1-[[(1S)-1-[5-[6-(5-cyclopropylthiophen-2-yl)-10-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-3-methylbutyl]-methylamino]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(1R)-1-[(2R,6S)-2,6-dimethyloxan-4-yl]-2-[(2S)-2-[5-[6-(5-ethylthiophen-2-yl)-1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate —— C53H62FN9O8S
methyl N-[(1R)-1-[(2R,6S)-2,6-dimethyloxan-4-yl]-2-[(2S)-2-[5-[6-(5-ethylthiophen-2-yl)-1-fluoro-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-2-oxoethyl]carbamate
—— methyl N-[1-[(2S)-2-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-1-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-2-methylpyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C37H37ClFN5O4S
methyl N-[1-[(2S)-2-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-1-fluoro-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-2-methylpyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(1R,3S)-3-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C37H36ClN5O4S
methyl N-[(2S)-1-[(1R,3S)-3-[5-[10-chloro-6-(5-cyclopropylthiophen-2-yl)-6H-indolo[1,2-c][1,3]benzoxazin-3-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— methyl N-[(2S)-1-[(2S)-2-[(4S)-4-[(3S,7aS,11aR,12bR)-6-(2-cyclopropyl-2,3-dihydrothiophen-5-yl)-1,12-difluoro-10-[2-[1-[(2R)-1-[(2S)-2-[[hydroxy(methoxy)methyl]amino]-3-methylbutanoyl]-2-methylpyrrolidin-2-yl]ethyl]-4,5-dihydro-1H-imidazol-5-yl]-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-3-yl]imidazolidin-2-yl]pyrrolidin-1-yl]-3-methylbutan-2-yl]-N-methylcarbamate —— C54H85F2N9O6S
methyl N-[(2S)-1-[(2S)-2-[(4S)-4-[(3S,7aS,11aR,12bR)-6-(2-cyclopropyl-2,3-dihydrothiophen-5-yl)-1,12-difluoro-10-[2-[1-[(2R)-1-[(2S)-2-[[hydroxy(methoxy)methyl]amino]-3-methylbutanoyl]-2-methylpyrrolidin-2-yl]ethyl]-4,5-dihydro-1H-imidazol-5-yl]-4,4a,6,7a,8,11,11a,12,12a,12b-decahydro-3H-indolo[1,2-c][1,3]benzoxazin-3-yl]imidazolidin-2-yl]pyrrolidin-1-yl]-3-methylbutan-2-yl]-N-methylcarbamate
—— methyl N-[(2S)-1-[(2S,4R)-2-[1-[[(Z,3E)-2-amino-3-[[1-(4,5-dimethylthiophen-2-yl)-4-ethenyl-7-ethyl-3-[(E)-2-[2-[(2S,4R)-4-fluoro-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]prop-1-enyl]-1H-pyrrolo[1,2-c][1,3]oxazin-6-yl]methylidene]pent-1-enyl]amino]ethenyl]-4-fluoropyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate —— C53H71F2N9O7S
methyl N-[(2S)-1-[(2S,4R)-2-[1-[[(Z,3E)-2-amino-3-[[1-(4,5-dimethylthiophen-2-yl)-4-ethenyl-7-ethyl-3-[(E)-2-[2-[(2S,4R)-4-fluoro-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]prop-1-enyl]-1H-pyrrolo[1,2-c][1,3]oxazin-6-yl]methylidene]pent-1-enyl]amino]ethenyl]-4-fluoropyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate