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—— ethyl 5-(4-bromophenyl)-2-[(2-hydroxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H21BrN2O4S
ethyl 5-(4-bromophenyl)-2-[(2-hydroxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[(2-hydroxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H20N2O4S2
ethyl 2-[(2-hydroxynaphthalen-1-yl)methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[(5-bromo-2-hydroxyphenyl)methylidene]-5-(4-bromophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H18Br2N2O4S
ethyl 2-[(5-bromo-2-hydroxyphenyl)methylidene]-5-(4-bromophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 2-[2-(4-hexoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H31N3O6S
Ethyl 2-[2-(4-hexoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 2-[2-[3-ethoxy-4-(3-methylbutoxy)phenyl]-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H33N3O7S
Ethyl 2-[2-[3-ethoxy-4-(3-methylbutoxy)phenyl]-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 2-[2-(3-ethoxy-4-pentoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H33N3O7S
Ethyl 2-[2-(3-ethoxy-4-pentoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[3-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)carbamoyl]phenoxy]acetate —— C19H17ClN2O6
ethyl 2-[3-[(6-chloro-3-oxo-4H-1,4-benzoxazin-7-yl)carbamoyl]phenoxy]acetate
—— Ethyl 4-[(15,18,18-trimethyl-7,9-dioxa-3,13-diazapentacyclo[13.2.1.02,14.04,12.06,10]octadeca-2,4,6(10),11,13-pentaene-1-carbonyl)amino]benzoate —— C27H27N3O5
Ethyl 4-[(15,18,18-trimethyl-7,9-dioxa-3,13-diazapentacyclo[13.2.1.02,14.04,12.06,10]octadeca-2,4,6(10),11,13-pentaene-1-carbonyl)amino]benzoate
—— ethyl 2-[3-[[2-(prop-2-enylcarbamoyl)phenyl]carbamoyl]phenoxy]acetate —— C21H22N2O5
ethyl 2-[3-[[2-(prop-2-enylcarbamoyl)phenyl]carbamoyl]phenoxy]acetate
—— Ethyl 2-[2-(3-ethoxy-4-phenylmethoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H29N3O7S
Ethyl 2-[2-(3-ethoxy-4-phenylmethoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— Ethyl 2-[2-(4-butoxy-3-ethoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H31N3O7S
Ethyl 2-[2-(4-butoxy-3-ethoxyphenyl)-3-[hydroxy(pyridin-4-yl)methylidene]-4,5-dioxopyrrolidin-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl N-[4-[[2-[methyl-[(2R)-2-pyrazol-1-ylpropanoyl]amino]acetyl]amino]phenyl]carbamate —— C18H23N5O4
ethyl N-[4-[[2-[methyl-[(2R)-2-pyrazol-1-ylpropanoyl]amino]acetyl]amino]phenyl]carbamate
—— ethyl 2-[3-[[2-(piperidine-1-carbonyl)phenyl]carbamoyl]phenoxy]acetate —— C23H26N2O5
ethyl 2-[3-[[2-(piperidine-1-carbonyl)phenyl]carbamoyl]phenoxy]acetate
—— Ethyl 2-[(5-bromo-6-chloropyridin-3-yl)sulfonylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C16H16BrClN2O4S2
Ethyl 2-[(5-bromo-6-chloropyridin-3-yl)sulfonylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl N-[4-[[(2S)-3-methyl-2-(5-phenyltetrazol-2-yl)butanoyl]amino]phenyl]carbamate —— C21H24N6O3
ethyl N-[4-[[(2S)-3-methyl-2-(5-phenyltetrazol-2-yl)butanoyl]amino]phenyl]carbamate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(3-methoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H24N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(3-methoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-phenylmethoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C34H28N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-phenylmethoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C33H34N2O9S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-[3-methoxy-4-(3-methylbutoxy)phenyl]-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— (E)-N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C16H16N4O5S
(E)-N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— ethyl 2-[2-(3-bromo-4-hydroxy-5-methoxyphenyl)-4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H23BrN2O9S
ethyl 2-[2-(3-bromo-4-hydroxy-5-methoxyphenyl)-4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-[6-(3-methoxyphenyl)sulfonyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C27H31N5O5S
ethyl 1-[6-(3-methoxyphenyl)sulfonyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(4-methoxycarbonylphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C29H24N2O9S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(4-methoxycarbonylphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(3-methoxy-4-phenylmethoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C35H30N2O9S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(3-methoxy-4-phenylmethoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl N-[4-[[2-[methyl-[(2S)-2-pyrazol-1-ylpropanoyl]amino]acetyl]amino]phenyl]carbamate —— C18H23N5O4
ethyl N-[4-[[2-[methyl-[(2S)-2-pyrazol-1-ylpropanoyl]amino]acetyl]amino]phenyl]carbamate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-prop-2-enoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H26N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-prop-2-enoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[2-(2-fluorophenyl)-4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H21FN2O7S
ethyl 2-[2-(2-fluorophenyl)-4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-propoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H28N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(4-propoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C24H32N4O4S
ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-methyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(3-pentoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H32N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(3-pentoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-(6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C23H29N5O2
ethyl 1-(6-prop-2-enyl-2-pyridin-3-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— Ethyl 1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C20H25N5O2
Ethyl 1-(2-pyridin-3-yl-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-[3-(3-methylbutoxy)phenyl]-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C32H32N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-[3-(3-methylbutoxy)phenyl]-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(3-propoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C30H28N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2-(3-propoxyphenyl)-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[4-hydroxy-2-(3-hydroxyphenyl)-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C27H22N2O8S
ethyl 2-[4-hydroxy-2-(3-hydroxyphenyl)-3-(7-methoxy-1-benzofuran-2-carbonyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 2-[3-[[2-(2-amino-2-oxoethyl)phenyl]carbamoyl]phenoxy]acetate —— C19H20N2O5
ethyl 2-[3-[[2-(2-amino-2-oxoethyl)phenyl]carbamoyl]phenoxy]acetate
—— ethyl 1-[6-(ethylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C23H30N6O3
ethyl 1-[6-(ethylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 1-(2-phenyl-6-prop-2-enyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C24H30N4O2
ethyl 1-(2-phenyl-6-prop-2-enyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— ethyl 1-[6-[(3-cyanophenyl)carbamoyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H29N7O3
ethyl 1-[6-[(3-cyanophenyl)carbamoyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 2-[3-[(5-acetamido-2-fluorophenyl)carbamoyl]phenoxy]acetate —— C19H19FN2O5
ethyl 2-[3-[(5-acetamido-2-fluorophenyl)carbamoyl]phenoxy]acetate
—— Ethane ethyl 1-{6-[2-(benzenesulfonyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl}piperidine-4-carboxylate —— C28H33N5O4S
Ethane ethyl 1-{6-[2-(benzenesulfonyl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl}piperidine-4-carboxylate
—— ethyl 1-[2-pyridin-2-yl-6-(thiophene-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C25H27N5O3S
ethyl 1-[2-pyridin-2-yl-6-(thiophene-2-carbonyl)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— (E)-N-[4-(2,2-dimethylpropanoyl)-2,3-dihydro-1,4-benzoxazin-6-yl]-3-thiophen-2-ylprop-2-enamide —— C20H22N2O3S
(E)-N-[4-(2,2-dimethylpropanoyl)-2,3-dihydro-1,4-benzoxazin-6-yl]-3-thiophen-2-ylprop-2-enamide
—— ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O4S
ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-4-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 2-[3-[[2-(2-amino-2-oxoethyl)sulfanylphenyl]carbamoyl]phenoxy]acetate —— C19H20N2O5S
ethyl 2-[3-[[2-(2-amino-2-oxoethyl)sulfanylphenyl]carbamoyl]phenoxy]acetate
—— ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(4-methoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate —— C28H24N2O8S
ethyl 2-[4-hydroxy-3-(7-methoxy-1-benzofuran-2-carbonyl)-2-(4-methoxyphenyl)-5-oxo-2H-pyrrol-1-yl]-4-methyl-1,3-thiazole-5-carboxylate
—— ethyl 1-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C23H29N5O2
ethyl 1-(6-prop-2-enyl-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate
—— ethyl 1-[6-[(3-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O3
ethyl 1-[6-[(3-methoxyphenyl)methyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C28H33N5O4S
ethyl 1-[6-[2-(benzenesulfonyl)ethyl]-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 1-[6-(benzenesulfonylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate —— C27H30N6O5S
ethyl 1-[6-(benzenesulfonylcarbamoyl)-2-pyridin-2-yl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]piperidine-4-carboxylate
—— ethyl 1-(2-pyridin-2-yl-6-thiophen-2-ylsulfonyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate —— C24H27N5O4S2
ethyl 1-(2-pyridin-2-yl-6-thiophen-2-ylsulfonyl-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl)piperidine-4-carboxylate