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—— (6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-(propylamino)-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C38H48BClN4O4
(6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-(propylamino)-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-4-oxo-8-(3-phenylpropyl)-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C39H45BClF3N4O4
(6S,8R)-1-chloro-4-oxo-8-(3-phenylpropyl)-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-3-amino-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C35H42BClN4O4
(6S,8R)-3-amino-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-3-[(3-methoxyphenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C43H50BClN4O5
(6S,8R)-1-chloro-3-[(3-methoxyphenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-4-oxo-8-[(4-phenylphenyl)methyl]-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C43H45BClF3N4O4
(6S,8R)-1-chloro-4-oxo-8-[(4-phenylphenyl)methyl]-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C43H47BClF3N4O4
(6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-3-[(3-nitrophenyl)methylamino]-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C42H47BClN5O6
(6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-3-[(3-nitrophenyl)methylamino]-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-3-[(3,4-dihydroxyphenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C42H48BClN4O6
(6S,8R)-1-chloro-3-[(3,4-dihydroxyphenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-3-(benzylamino)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C42H48BClN4O4
(6S,8R)-3-(benzylamino)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-8-(3-naphthalen-2-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]propyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C42H47BClF3N4O4
(6S,8R)-1-chloro-8-(3-naphthalen-2-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]propyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-3-(butylamino)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C39H50BClN4O4
(6S,8R)-3-(butylamino)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[2-({2-[(methylamino)carbonyl]phenyl}amino)-2-oxoethyl]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C40H48BF3N6O6
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[2-({2-[(methylamino)carbonyl]phenyl}amino)-2-oxoethyl]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S)-1-chloro-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C30H35BClF3N4O4
(6S)-1-chloro-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(4-fluorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C37H43BF4N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(4-fluorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[({[3-(methylthio)phenyl]amino}carbonyl)amino]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H46BF3N6O5S
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[({[3-(methylthio)phenyl]amino}carbonyl)amino]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-1-chloro-3-(methylamino)-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C36H44BClN4O4
(6S,8R)-1-chloro-3-(methylamino)-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-3-[(3-fluorophenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C42H47BClFN4O4
(6S,8R)-1-chloro-3-[(3-fluorophenyl)methylamino]-8-(3-naphthalen-1-ylpropyl)-4-oxo-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-4-oxo-8-({[(4-phenoxyphenyl)amino]carbonyl}amino)-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C43H48BF3N6O6
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-4-oxo-8-({[(4-phenoxyphenyl)amino]carbonyl}amino)-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(2-chlorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C37H43BClF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(2-chlorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-(pyridin-2-ylmethylamino)-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C41H47BClN5O4
(6S,8R)-1-chloro-8-(3-naphthalen-1-ylpropyl)-4-oxo-3-(pyridin-2-ylmethylamino)-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-chloro-8-(3-naphthalen-2-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide —— C43H47BClF3N4O4
(6S,8R)-1-chloro-8-(3-naphthalen-2-ylpropyl)-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(2R)-2,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]but-3-enyl]-7,8-dihydro-6H-pyrrolo[1,2-a]pyrazine-6-carboxamide
—— (6S,8R)-1-Chloro-3-cyclohexylamino-8-(3-naphthalen-1-yl-propyl)-4-oxo-4,6,7,8-tetrahydro-pyrrolo[1,2-a]pyrazine-6-carboxylic acid, [(R)-1-((R)-2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0%2,6&]dec-4-yl)-but-3-enyl]-amide —— C41H52BClN4O4
(6S,8R)-1-Chloro-3-cyclohexylamino-8-(3-naphthalen-1-yl-propyl)-4-oxo-4,6,7,8-tetrahydro-pyrrolo[1,2-a]pyrazine-6-carboxylic acid, [(R)-1-((R)-2,9,9-trimethyl-3,5-dioxa-4-bora-tricyclo[6.1.1.0%2,6&]dec-4-yl)-but-3-enyl]-amide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[2-(1-naphthylamino)-2-oxoethyl]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C42H47BF3N5O5
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[2-(1-naphthylamino)-2-oxoethyl]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{[(1,1'-biphenyl-2-ylamino)carbonyl]amino}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C43H48BF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{[(1,1'-biphenyl-2-ylamino)carbonyl]amino}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— 6-(2-Phenylsulfanylethyl)pteridine-2,4-diamine —— C14H14N6S
6-(2-Phenylsulfanylethyl)pteridine-2,4-diamine
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-({[(2-methylphenyl)amino]carbonyl}amino)-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H46BF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-({[(2-methylphenyl)amino]carbonyl}amino)-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(3-fluorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C37H43BF4N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(3-fluorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-{[(1-naphthylamino)carbonyl]amino}-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C41H46BF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-{[(1-naphthylamino)carbonyl]amino}-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-[2-({2-[(dimethylamino)carbonyl]phenyl}amino)-2-oxoethyl]-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C41H50BF3N6O6
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-[2-({2-[(dimethylamino)carbonyl]phenyl}amino)-2-oxoethyl]-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-(2-{[2-(aminocarbonyl)phenyl]amino}-2-oxoethyl)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C39H46BF3N6O6
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-(2-{[2-(aminocarbonyl)phenyl]amino}-2-oxoethyl)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-4-oxo-8-({[(2-phenoxyphenyl)amino]carbonyl}amino)-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C43H48BF3N6O6
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-4-oxo-8-({[(2-phenoxyphenyl)amino]carbonyl}amino)-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-(2-{[3-(methylthio)phenyl]amino}-2-oxoethyl)-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C39H47BF3N5O5S
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-(2-{[3-(methylthio)phenyl]amino}-2-oxoethyl)-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-[2-(1-isoquinolinylamino)-2-oxoethyl]-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C41H46BF3N6O5
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-[2-(1-isoquinolinylamino)-2-oxoethyl]-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-(2-anilino-2-oxoethyl)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H45BF3N5O5
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-(2-anilino-2-oxoethyl)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(2-ethoxyphenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C39H48BF3N6O6
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(2-ethoxyphenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{[(benzylamino)carbonyl]amino}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H46BF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{[(benzylamino)carbonyl]amino}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8S)-8-methyl-8-[2-(2-nitroanilino)-2-oxoethyl]-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(6S)-6,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]propyl]-6,7-dihydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H44BF3N6O7
(6S,8S)-8-methyl-8-[2-(2-nitroanilino)-2-oxoethyl]-4-oxo-3-[[3-(trifluoromethyl)phenyl]methylamino]-N-[(1R)-1-[(6S)-6,9,9-trimethyl-3,5-dioxa-4-boratricyclo[6.1.1.02,6]decan-4-yl]propyl]-6,7-dihydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[({[4-(methylthio)phenyl]amino}carbonyl)amino]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C38H46BF3N6O5S
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-methyl-8-[({[4-(methylthio)phenyl]amino}carbonyl)amino]-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— 6-[1-(2,6-Difluoro-phenyl)-ethyl]-2-methylamino-3H-pyrimidin-4-one —— C13H13F2N3O
6-[1-(2,6-Difluoro-phenyl)-ethyl]-2-methylamino-3H-pyrimidin-4-one
—— (6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{2-[(2-methoxyphenyl)amino]-2-oxoethyl}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C39H47BF3N5O6
(6S,8S)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-{2-[(2-methoxyphenyl)amino]-2-oxoethyl}-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— (6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(4-chlorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide —— C37H43BClF3N6O5
(6S,8R)-N-{(1R)-1-[(7aS)-5,5,7a-Trimethylhexahydro-4,6-methano-1,3,2-benzodioxaborol-2-yl]propyl}-8-({[(4-chlorophenyl)amino]carbonyl}amino)-8-methyl-4-oxo-3-{[3-(trifluoromethyl)benzyl]amino}-4,6,7,8-tetrahydropyrrolo[1,2-a]pyrimidine-6-carboxamide
—— 6-[1-(2,6-Difluoro-phenyl)-ethyl]-5-methyl-2-methylamino-3H-pyrimidin-4-one —— C14H15F2N3O
6-[1-(2,6-Difluoro-phenyl)-ethyl]-5-methyl-2-methylamino-3H-pyrimidin-4-one
—— 6-[3-(2,4-Diamino-pyrimidin-5-ylmethyl)-4-methoxy-phenyl]-hexanoic acid —— C18H24N4O3
6-[3-(2,4-Diamino-pyrimidin-5-ylmethyl)-4-methoxy-phenyl]-hexanoic acid
—— 6-[1-(2,6-Difluoro-phenyl)-ethyl]-2-isopropylamino-3H-pyrimidin-4-one —— C15H17F2N3O
6-[1-(2,6-Difluoro-phenyl)-ethyl]-2-isopropylamino-3H-pyrimidin-4-one
—— 6-(2,6-Difluoro-benzyl)-2-methylamino-3H-pyrimidin-4-one —— C12H11F2N3O
6-(2,6-Difluoro-benzyl)-2-methylamino-3H-pyrimidin-4-one
—— 6-(2,6-Difluorophenylmethyl)-3,4-dihydro-2-N,N-dimethylaminopyrimidin-4-(3H)-one —— C13H13F2N3O
6-(2,6-Difluorophenylmethyl)-3,4-dihydro-2-N,N-dimethylaminopyrimidin-4-(3H)-one
—— 6-(2,6-Difluoro-benzyl)-5-methyl-2-methylamino-3H-pyrimidin-4-one —— C13H13F2N3O
6-(2,6-Difluoro-benzyl)-5-methyl-2-methylamino-3H-pyrimidin-4-one
—— 6-(Dodecylamino)-3,7-dihydroimidazo[4,5-e][1,3]diazepine-4,8-dione —— C18H29N5O2
6-(Dodecylamino)-3,7-dihydroimidazo[4,5-e][1,3]diazepine-4,8-dione
—— 6-Chloro-4-(1,3-dioxolan-2-ylmethoxy)-3-propyl-2(1H)-quinolinone 345912-92-7 C16H18ClNO4
6-Chloro-4-(1,3-dioxolan-2-ylmethoxy)-3-propyl-2(1H)-quinolinone
—— 6-amino-3-[2-(phosphanylmethoxy)ethoxymethyl]-7H-imidazo[4,5-e][1,3]diazepine-4,8-dione —— C10H14N5O4P
6-amino-3-[2-(phosphanylmethoxy)ethoxymethyl]-7H-imidazo[4,5-e][1,3]diazepine-4,8-dione