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—— 6-acetamido-N-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H56N4O5
6-acetamido-N-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-6-[[2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]methyl}pyrimidine-2,4(1H,3H)-dione —— C13H17N5O3
6-{[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]methyl}pyrimidine-2,4(1H,3H)-dione
—— 6-(3-Aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(4-methyl-1H-imidazol-2-YL)methyl]pyrimidin-4-amine —— C17H24N6
6-(3-Aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[(4-methyl-1H-imidazol-2-YL)methyl]pyrimidin-4-amine
—— 6-Chloro-2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]imidazo[1,2-a]pyridine —— C19H17Cl2N5OS
6-Chloro-2-[[5-(4-chlorophenyl)-4-(2-methoxyethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]imidazo[1,2-a]pyridine
—— 6-(cis-3-aminocyclobutyl)-N-(2-pyridin-3-ylethyl)-2-pyrrolidin-1-ylpyrimidin-4-amine —— C19H26N6
6-(cis-3-aminocyclobutyl)-N-(2-pyridin-3-ylethyl)-2-pyrrolidin-1-ylpyrimidin-4-amine
—— 6-Pyrrolidin-1-ylhex-4-yn-3-ol —— C10H17NO
6-Pyrrolidin-1-ylhex-4-yn-3-ol
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine —— C18H22N8O
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine
—— 6-acetamido-N-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C40H46N2O6S
6-acetamido-N-[[2-[4-[4-[4-(hydroxymethyl)phenyl]-6-[(2-methoxyphenyl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-[[(3-Carboxyphenyl)hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid —— C17H16N2O6
6-[[(3-Carboxyphenyl)hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid
—— 6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-3,4-dihydroquinolin-2(1H)-one —— C16H18N4O4S
6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-3,4-dihydroquinolin-2(1H)-one
—— 6-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-9-methyl-2,3,4,9-tetrahydro-1H-carbazol-1-one —— C21H26N2O3
6-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-9-methyl-2,3,4,9-tetrahydro-1H-carbazol-1-one
—— 6-{[4-(2-Thienylmethyl)-1,4-diazepan-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C18H21N5O2S
6-{[4-(2-Thienylmethyl)-1,4-diazepan-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— (6E)-6-[(2-ethoxyanilino)methylidene]-3-methyl-[1,3]thiazolo[2,3-b][1,3]thiazol-4-ium-5-one —— C15H15N2O2S2+
(6E)-6-[(2-ethoxyanilino)methylidene]-3-methyl-[1,3]thiazolo[2,3-b][1,3]thiazol-4-ium-5-one
—— 6,7-Diethoxy-3-[4-oxo-4-(1-pyrrolidinyl)butyl]-2,4(1H,3H)-quinazolinedione —— C20H27N3O5
6,7-Diethoxy-3-[4-oxo-4-(1-pyrrolidinyl)butyl]-2,4(1H,3H)-quinazolinedione
—— 6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[(5-methylpyrazin-2-YL)methyl]pyrimidin-4-amine —— C17H22N6
6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[(5-methylpyrazin-2-YL)methyl]pyrimidin-4-amine
—— 6-(trans-3-{[1-(2-furylmethyl)piperidin-4-yl]amino}cyclobutyl)pyrimidin-4(3H)-one —— C18H24N4O2
6-(trans-3-{[1-(2-furylmethyl)piperidin-4-yl]amino}cyclobutyl)pyrimidin-4(3H)-one
—— 6-{trans-3-[(3-fluoropyridin-4-yl)amino]cyclobutyl}-2-methylpyrimidin-4(3H)-one —— C14H15FN4O
6-{trans-3-[(3-fluoropyridin-4-yl)amino]cyclobutyl}-2-methylpyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-[2-(3-chlorophenyl)ethyl]pyrimidine-2,4-diamine —— C16H20ClN5
6-(3-aminocyclobutyl)-N~4~-[2-(3-chlorophenyl)ethyl]pyrimidine-2,4-diamine
—— 6-[5-(3,5-Dichlorophenyl)-2,4-dimethylfuran-3-yl]-3-phenyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole —— C21H14Cl2N4OS
6-[5-(3,5-Dichlorophenyl)-2,4-dimethylfuran-3-yl]-3-phenyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
—— (6,6-Difluoro-2,16-dimethyl-15-pentacyclo[9.7.0.02,8.05,7.012,16]octadec-8-enyl) acetate —— C22H30F2O2
(6,6-Difluoro-2,16-dimethyl-15-pentacyclo[9.7.0.02,8.05,7.012,16]octadec-8-enyl) acetate
—— 6-acetamido-N-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C38H46N4O5S
6-acetamido-N-[[3-[4-[4-[4-(hydroxymethyl)phenyl]-5-methyl-6-[(1-methylimidazol-2-yl)sulfanylmethyl]-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-chloro-2-(2-methylphenyl)-N-(2,4,4-trimethylpentan-2-yl)imidazo[1,2-a]pyridin-3-amine —— C22H28ClN3
6-chloro-2-(2-methylphenyl)-N-(2,4,4-trimethylpentan-2-yl)imidazo[1,2-a]pyridin-3-amine
—— 6-(3-Aminocyclobutyl)-N-(2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl)pyrimidin-4-amine —— C17H26N6
6-(3-Aminocyclobutyl)-N-(2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl)pyrimidin-4-amine
—— 6-chloro-2-methyl-N-{cis-3-[6-(methylamino)pyrimidin-4-yl]cyclobutyl}imidazo[1,2-a]pyridine-3-carboxamide —— C18H19ClN6O
6-chloro-2-methyl-N-{cis-3-[6-(methylamino)pyrimidin-4-yl]cyclobutyl}imidazo[1,2-a]pyridine-3-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine —— C14H21N7
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-2,4-diamine
—— 6-{[2-(Pyrrolidin-1-ylmethyl)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridine —— C18H24N4O
6-{[2-(Pyrrolidin-1-ylmethyl)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridine
—— 6-(3-aminocyclobutyl)-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,2-dimethylpyrimidin-4-amine —— C16H25N7O
6-(3-aminocyclobutyl)-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,2-dimethylpyrimidin-4-amine
—— 6-(1-{[(3-Methoxyphenyl)thio]acetyl}piperidin-3-yl)-2-methylpyrimidin-4-ol —— C19H23N3O3S
6-(1-{[(3-Methoxyphenyl)thio]acetyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
—— 6-{3-[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]-3-oxopropyl}-4,5-dihydropyridazin-3(2H)-one —— C15H21N5O3
6-{3-[2-(hydroxymethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]-3-oxopropyl}-4,5-dihydropyridazin-3(2H)-one
—— 6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)pyrimidin-4-amine —— C16H24N4O2S
6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-(imidazo[1,2-a]pyrazin-3-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine —— C17H21N7O
6-(3-aminocyclobutyl)-N-(imidazo[1,2-a]pyrazin-3-ylmethyl)-2-(methoxymethyl)pyrimidin-4-amine
—— 6-amino-N-[2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethyl]nicotinamide —— C16H15N5OS
6-amino-N-[2-(2-pyridin-3-yl-1,3-thiazol-4-yl)ethyl]nicotinamide
—— 6-(cis-3-aminocyclobutyl)-N~4~-(2-imidazo[1,2-a]pyrimidin-2-ylethyl)pyrimidine-2,4-diamine —— C16H20N8
6-(cis-3-aminocyclobutyl)-N~4~-(2-imidazo[1,2-a]pyrimidin-2-ylethyl)pyrimidine-2,4-diamine
—— 6-Methyl-3-[3-[3-[3-(6-methyl-2,4-dioxopyran-3-yl)-3-oxoprop-1-enyl]phenyl]prop-2-enoyl]pyran-2,4-dione —— C24H18O8
6-Methyl-3-[3-[3-[3-(6-methyl-2,4-dioxopyran-3-yl)-3-oxoprop-1-enyl]phenyl]prop-2-enoyl]pyran-2,4-dione
—— 6-(cis-3-aminocyclobutyl)-N-methyl-N-[3-(methylthio)benzyl]pyrimidin-4-amine —— C17H22N4S
6-(cis-3-aminocyclobutyl)-N-methyl-N-[3-(methylthio)benzyl]pyrimidin-4-amine
—— 6-bromo-N-(2,6-dimethylphenyl)-2-(pyridin-2-yl)imidazo[1,2-a]pyridin-3-amine —— C20H17BrN4
6-bromo-N-(2,6-dimethylphenyl)-2-(pyridin-2-yl)imidazo[1,2-a]pyridin-3-amine
—— 6-chloro-N-[rac-(1S,5R,6R)-2-oxabicyclo[3.2.0]hept-6-yl]-2H-chromene-3-carboxamide —— C16H16ClNO3
6-chloro-N-[rac-(1S,5R,6R)-2-oxabicyclo[3.2.0]hept-6-yl]-2H-chromene-3-carboxamide
—— 6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]carbonyl}-1,4-dihydroquinoxaline-2,3-dione —— C18H19N5O3
6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]carbonyl}-1,4-dihydroquinoxaline-2,3-dione
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(1-piperidin-1-ylcyclohexyl)methyl]pyrimidine-2,4-diamine —— C21H36N6
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-[(1-piperidin-1-ylcyclohexyl)methyl]pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(3-methoxyphenyl)ethyl]pyrimidine-2,4-diamine —— C17H23N5O
6-(3-aminocyclobutyl)-N~4~-[2-(3-methoxyphenyl)ethyl]pyrimidine-2,4-diamine
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-hydroxy-6-(2-hydroxy-4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C33H25Cl2F3N4O7
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-hydroxy-6-(2-hydroxy-4-methoxyphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6a,9a-Dichloro-6-[2-(2-hydroxyethoxy)phenyl]-8-methyl-2-phenyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H26Cl2N2O6
6a,9a-Dichloro-6-[2-(2-hydroxyethoxy)phenyl]-8-methyl-2-phenyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6a,9a-Dichloro-2-cyclohexyl-6-(4-hydroxynaphthalen-1-yl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C31H30Cl2N2O5
6a,9a-Dichloro-2-cyclohexyl-6-(4-hydroxynaphthalen-1-yl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-ethyl-4-{[2-[hydroxy(1-methyl-1H-pyrazol-5-yl)methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]carbonyl}pyridin-2(1H)-one —— C19H22N6O3
6-ethyl-4-{[2-[hydroxy(1-methyl-1H-pyrazol-5-yl)methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]carbonyl}pyridin-2(1H)-one
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[3-(trifluoromethyl)benzyl]pyrimidin-4-amine —— C20H23F3N4
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-[3-(trifluoromethyl)benzyl]pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N~4~-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]pyrimidine-2,4-diamine —— C16H20N8
6-(trans-3-aminocyclobutyl)-N~4~-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]pyrimidine-2,4-diamine
—— 6-{[(2R*,6S*)-2,6-dimethylmorpholin-4-yl]methyl}-1-methyl-1H-indole —— C16H22N2O
6-{[(2R*,6S*)-2,6-dimethylmorpholin-4-yl]methyl}-1-methyl-1H-indole
—— 6-(cis-3-aminocyclobutyl)-N-[2-(2-isopropyl-1,3-thiazol-4-yl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine —— C18H27N5OS
6-(cis-3-aminocyclobutyl)-N-[2-(2-isopropyl-1,3-thiazol-4-yl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-[(trans-3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}cyclobutyl)amino]-N,N-dimethylpyrazine-2-carboxamide —— C17H26N8O
6-[(trans-3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}cyclobutyl)amino]-N,N-dimethylpyrazine-2-carboxamide
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[3-(1H-imidazol-1-yl)propyl]pyrimidin-4-amine —— C17H24N6
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[3-(1H-imidazol-1-yl)propyl]pyrimidin-4-amine