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—— 6-(trans-3-aminocyclobutyl)-N-[3-(1,3-benzothiazol-2-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine —— C20H25N5OS
6-(trans-3-aminocyclobutyl)-N-[3-(1,3-benzothiazol-2-yl)propyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(2,3-Dibromo-4-hydroxy-5-methoxyphenyl)-2,8-bis[2-(4-hydroxyphenyl)ethyl]-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C37H34Br2N2O8
6-(2,3-Dibromo-4-hydroxy-5-methoxyphenyl)-2,8-bis[2-(4-hydroxyphenyl)ethyl]-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3,4-Dimethoxyphenyl)-5-methylsulfanyl-3-phenyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C20H17N3O3S3
6-(3,4-Dimethoxyphenyl)-5-methylsulfanyl-3-phenyl-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-N-[3-(1H-indazol-1-yl)propyl]pyrimidin-4-amine —— C18H22N6
6-(cis-3-aminocyclobutyl)-N-[3-(1H-indazol-1-yl)propyl]pyrimidin-4-amine
—— 6-ethyl 3-methyl 2-(4-(N,N-bis(2-methoxyethyl)sulfamoyl)benzamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate —— C25H33N3O9S2
6-ethyl 3-methyl 2-(4-(N,N-bis(2-methoxyethyl)sulfamoyl)benzamido)-4,5-dihydrothieno[2,3-c]pyridine-3,6(7H)-dicarboxylate
—— 6-(3-aminocyclobutyl)-N~4~-[(5-methylpyrazin-2-yl)methyl]pyrimidine-2,4-diamine —— C14H19N7
6-(3-aminocyclobutyl)-N~4~-[(5-methylpyrazin-2-yl)methyl]pyrimidine-2,4-diamine
—— 6a,9a-Dichloro-6-(3-ethoxy-2-hydroxyphenyl)-8-(4-fluorophenyl)-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C34H26Cl2FN3O8
6a,9a-Dichloro-6-(3-ethoxy-2-hydroxyphenyl)-8-(4-fluorophenyl)-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(cis-3-aminocyclobutyl)-N-methyl-N-(1-naphthylmethyl)pyrimidin-4-amine —— C20H22N4
6-(cis-3-aminocyclobutyl)-N-methyl-N-(1-naphthylmethyl)pyrimidin-4-amine
—— 6-amino-N-[(1S,5S,6R,7S)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]heptan-6-yl]pyridine-3-carboxamide —— C14H19N3O3
6-amino-N-[(1S,5S,6R,7S)-7-(methoxymethyl)-2-oxabicyclo[3.2.0]heptan-6-yl]pyridine-3-carboxamide
—— 6-Methoxy-2-(2-morpholin-4-ylbenzoyl)-1,2,3,4-tetrahydroisoquinoline —— C21H24N2O3
6-Methoxy-2-(2-morpholin-4-ylbenzoyl)-1,2,3,4-tetrahydroisoquinoline
—— 6-Amino-4-(4-phenylmethoxyphenyl)-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C21H15F3N4O2
6-Amino-4-(4-phenylmethoxyphenyl)-3-(trifluoromethyl)-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-Amino-N-[2-(2-oxopiperidin-1-YL)ethyl]pyridine-2-carboxamide —— C13H18N4O2
6-Amino-N-[2-(2-oxopiperidin-1-YL)ethyl]pyridine-2-carboxamide
—— 6-Amino-4-[1-[2-(4-tert-butylphenoxy)ethyl]indol-3-yl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile —— C28H29N5O2
6-Amino-4-[1-[2-(4-tert-butylphenoxy)ethyl]indol-3-yl]-3-methyl-2,4-dihydropyrano[2,3-c]pyrazole-5-carbonitrile
—— 6-(4-methoxyphenyl)-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxo-1H-pyridine-3-carboxamide —— C19H20N2O4
6-(4-methoxyphenyl)-N-[(1S,5R,6S)-2-oxabicyclo[3.2.0]heptan-6-yl]-2-oxo-1H-pyridine-3-carboxamide
—— 6-Amino-3-(3-hydroxyphenyl)-4-phenyl-4,7-dihydro-[1,2]oxazolo[5,4-b]pyridine-5-carbonitrile —— C19H14N4O2
6-Amino-3-(3-hydroxyphenyl)-4-phenyl-4,7-dihydro-[1,2]oxazolo[5,4-b]pyridine-5-carbonitrile
—— 6-(3-aminocyclobutyl)-N~4~-(4-phenylbutyl)pyrimidine-2,4-diamine —— C18H25N5
6-(3-aminocyclobutyl)-N~4~-(4-phenylbutyl)pyrimidine-2,4-diamine
—— 6-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]carbonyl}pyridin-2(1H)-one —— C15H18N4O3
6-{[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]carbonyl}pyridin-2(1H)-one
—— 6-benzyl-2,5-dimethyl-N-[3-(morpholin-4-yl)propyl]-3-phenylpyrazolo[1,5-a]pyrimidin-7-amine —— C28H33N5O
6-benzyl-2,5-dimethyl-N-[3-(morpholin-4-yl)propyl]-3-phenylpyrazolo[1,5-a]pyrimidin-7-amine
—— 6-imino-N-(2-methylpropyl)-2-oxo-7-(1-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C24H25N5O2
6-imino-N-(2-methylpropyl)-2-oxo-7-(1-phenylethyl)-1,7,9-triazatricyclo[8.4.0.03,8]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 6-(2-methoxyphenyl)-5-(methylsulfanyl)-3-(2-phenylethyl)-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-d]pyrimidin-7-one —— C21H19N3O2S3
6-(2-methoxyphenyl)-5-(methylsulfanyl)-3-(2-phenylethyl)-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-d]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-N~4~-[3-(1H-pyrazol-1-yl)benzyl]pyrimidine-2,4-diamine —— C18H21N7
6-(3-aminocyclobutyl)-N~4~-[3-(1H-pyrazol-1-yl)benzyl]pyrimidine-2,4-diamine
—— 6-[[1-(4-Chloro-2-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C22H22ClN5OS
6-[[1-(4-Chloro-2-methylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-propyl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-amino-N-[1-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)piperidin-4-yl]nicotinamide —— C16H24N4O3S
6-amino-N-[1-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)piperidin-4-yl]nicotinamide
—— 6-(trans-3-aminocyclobutyl)-N~4~-[3-(4-methyl-1,3-thiazol-5-yl)propyl]pyrimidine-2,4-diamine —— C15H22N6S
6-(trans-3-aminocyclobutyl)-N~4~-[3-(4-methyl-1,3-thiazol-5-yl)propyl]pyrimidine-2,4-diamine
—— (6Z)-6-(4-hydroxybenzylidene)-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C19H14N4O2S
(6Z)-6-(4-hydroxybenzylidene)-5-imino-2-(4-methylphenyl)-5,6-dihydro-7H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(3-isobutyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylpyrimidin-4-amine —— C19H28N6O
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(3-isobutyl-1,2,4-oxadiazol-5-yl)methyl]-N-methylpyrimidin-4-amine
—— 6-[(4-phenoxyphenyl)amino]-7H-benzo[e]perimidin-7-one —— C27H17N3O2
6-[(4-phenoxyphenyl)amino]-7H-benzo[e]perimidin-7-one
—— 6-(trans-3-aminocyclobutyl)-N~4~-(3-pyridin-3-ylpropyl)pyrimidine-2,4-diamine —— C16H22N6
6-(trans-3-aminocyclobutyl)-N~4~-(3-pyridin-3-ylpropyl)pyrimidine-2,4-diamine
—— 6-(3-aminocyclobutyl)-N~4~-[(1-benzyl-1H-imidazol-2-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine —— C20H25N7
6-(3-aminocyclobutyl)-N~4~-[(1-benzyl-1H-imidazol-2-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine
—— 6-[6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-yl]-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4(3H)-one —— C17H22N6O2
6-[6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)pyrimidin-4-yl]-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4(3H)-one
—— [6-[[(1R,5R,6S,7R)-7-(dimethylamino)-2-oxabicyclo[3.2.0]heptan-6-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone —— C17H25N5O2
[6-[[(1R,5R,6S,7R)-7-(dimethylamino)-2-oxabicyclo[3.2.0]heptan-6-yl]amino]pyrazin-2-yl]-pyrrolidin-1-ylmethanone
—— 6-Chloro-9-(2,4-dichlorophenyl)-3,4-dimethyl-8,10-dihydropyrano[2,3-f][1,3]benzoxazin-2-one —— C19H14Cl3NO3
6-Chloro-9-(2,4-dichlorophenyl)-3,4-dimethyl-8,10-dihydropyrano[2,3-f][1,3]benzoxazin-2-one
—— 6,8-Dibromo-3-(4-methylphenyl)sulfanyl-3-(morpholin-4-ylmethyl)-2,4-dihydrochromen-4-ol —— C21H23Br2NO3S
6,8-Dibromo-3-(4-methylphenyl)sulfanyl-3-(morpholin-4-ylmethyl)-2,4-dihydrochromen-4-ol
—— 6-isobutyl-2-oxo-N-[2-(tetrahydro-1H-pyrrolo[1,2-a]pyrrol-7a(5H)-yl)ethyl]-1,2-dihydropyrimidine-4-carboxamide —— C18H28N4O2
6-isobutyl-2-oxo-N-[2-(tetrahydro-1H-pyrrolo[1,2-a]pyrrol-7a(5H)-yl)ethyl]-1,2-dihydropyrimidine-4-carboxamide
—— 6-(cis-3-aminocyclobutyl)-N~4~-[3-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)propyl]pyrimidine-2,4-diamine —— C15H24N8
6-(cis-3-aminocyclobutyl)-N~4~-[3-(3,5-dimethyl-1H-1,2,4-triazol-1-yl)propyl]pyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-N~4~-[2-(2-fluorophenoxy)ethyl]pyrimidine-2,4-diamine —— C16H20FN5O
6-(cis-3-aminocyclobutyl)-N~4~-[2-(2-fluorophenoxy)ethyl]pyrimidine-2,4-diamine
—— 6-(trans-3-aminocyclobutyl)-N-[(5-isopropylisoxazol-3-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine —— C17H25N5O2
6-(trans-3-aminocyclobutyl)-N-[(5-isopropylisoxazol-3-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylpyrimidin-4-amine —— C17H26N6
6-(3-aminocyclobutyl)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methylpyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1H-1,2,4-triazol-1-yl)benzyl]pyrimidine-2,4-diamine —— C17H20N8
6-(3-aminocyclobutyl)-N~4~-[2-(1H-1,2,4-triazol-1-yl)benzyl]pyrimidine-2,4-diamine
—— 6-benzyl-N-methyl-2-[[4-(2-methylpiperidin-1-yl)sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide —— C29H34N4O4S2
6-benzyl-N-methyl-2-[[4-(2-methylpiperidin-1-yl)sulfonylbenzoyl]amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide
—— 6-(3-aminocyclobutyl)-N~4~-{3-[(dimethylamino)methyl]benzyl}-N~4~-methylpyrimidine-2,4-diamine —— C19H28N6
6-(3-aminocyclobutyl)-N~4~-{3-[(dimethylamino)methyl]benzyl}-N~4~-methylpyrimidine-2,4-diamine
—— 6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(2-methoxyphenyl)ethyl]pyrimidin-4-amine —— C20H26N4O
6-(3-Aminocyclobutyl)-2-cyclopropyl-N-[2-(2-methoxyphenyl)ethyl]pyrimidin-4-amine
—— 6-chloro-2-(3-chloro-4-methoxyphenyl)-7-methyl-1H-indole-3-carbaldehyde —— C17H13Cl2NO2
6-chloro-2-(3-chloro-4-methoxyphenyl)-7-methyl-1H-indole-3-carbaldehyde
—— 6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-4-methylquinolin-2-ol —— C17H18N4O4S
6-{[2-(hydroxymethyl)-6,7-dihydropyrazolo[1,5-a]pyrazin-5(4H)-yl]sulfonyl}-4-methylquinolin-2-ol
—— 6-(3-aminocyclobutyl)-N~4~-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine —— C16H23N7O
6-(3-aminocyclobutyl)-N~4~-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N~4~-methylpyrimidine-2,4-diamine
—— 6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(5-methyl-1H-benzimidazol-2-yl)methyl]pyrimidin-4-amine —— C19H24N6O
6-(cis-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(5-methyl-1H-benzimidazol-2-yl)methyl]pyrimidin-4-amine
—— 6-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}carbonyl)imidazo[1,2-a]pyridine —— C18H21N5O
6-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}carbonyl)imidazo[1,2-a]pyridine
—— 6-[[1-(4-Ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C27H30N6O2S
6-[[1-(4-Ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-2-(2-oxo-2-piperidin-1-ylethyl)-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]pyrimidin-4-amine —— C18H26N6
6-(cis-3-aminocyclobutyl)-2-cyclopropyl-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]pyrimidin-4-amine
—— 6-methyl-4-oxo-N-[2-(2-oxopiperidin-1-yl)ethyl]-4H-pyran-2-carboxamide —— C14H18N2O4
6-methyl-4-oxo-N-[2-(2-oxopiperidin-1-yl)ethyl]-4H-pyran-2-carboxamide