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—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(5-methyl-2-thienyl)methyl]pyrimidin-4-amine —— C17H22N4S
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-[(5-methyl-2-thienyl)methyl]pyrimidin-4-amine
—— 6-amino-N-[1-(3-methylpyridin-2-yl)propyl]nicotinamide —— C15H18N4O
6-amino-N-[1-(3-methylpyridin-2-yl)propyl]nicotinamide
—— 6-{cis-3-[(3,5-dichloropyridin-2-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one —— C17H19Cl2N5O
6-{cis-3-[(3,5-dichloropyridin-2-yl)amino]cyclobutyl}-2-pyrrolidin-1-ylpyrimidin-4(3H)-one
—— 6-[2-[hydroxy(1-methyl-1H-pyrazol-5-yl)methyl]-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]nicotinonitrile —— C18H19N7O
6-[2-[hydroxy(1-methyl-1H-pyrazol-5-yl)methyl]-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]nicotinonitrile
—— 6-Bromo-8-methyl-2-[4-(8-methyl-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl)phenyl]quinoline-4-carboxylic acid —— C27H21BrN2O4
6-Bromo-8-methyl-2-[4-(8-methyl-3,5-dioxo-4-azatricyclo[5.2.1.02,6]dec-8-en-4-yl)phenyl]quinoline-4-carboxylic acid
—— 6-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]carbonyl}pyridin-2(1H)-one —— C19H21N3O2
6-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]carbonyl}pyridin-2(1H)-one
—— 6-bromo-3-cyclohexyl-3,4-dihydro-2H-1,3-benzoxazin-3-ium —— C14H19BrNO+
6-bromo-3-cyclohexyl-3,4-dihydro-2H-1,3-benzoxazin-3-ium
—— 6-Amino-8-thiophen-2-yl-4-thia-2-azoniatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-5-carboxamide —— C15H14N3OS2+
6-Amino-8-thiophen-2-yl-4-thia-2-azoniatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-5-carboxamide
—— 6-butyl-2-methyl-3-(pyrrolidin-1-ium-1-ylmethyl)-1H-quinolin-4-one —— C19H27N2O+
6-butyl-2-methyl-3-(pyrrolidin-1-ium-1-ylmethyl)-1H-quinolin-4-one
—— 6-acetamido-N-[[3-[4-[4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide —— C42H49N3O6S
6-acetamido-N-[[3-[4-[4-[(4-acetamidophenyl)sulfanylmethyl]-6-[4-(hydroxymethyl)phenyl]-5-methyl-1,3-dioxan-2-yl]phenyl]phenyl]methyl]hexanamide
—— 6-(3-aminocyclobutyl)-N~4~-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidine-2,4-diamine —— C18H23N7
6-(3-aminocyclobutyl)-N~4~-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidine-2,4-diamine
—— 6-[4-[(3,4-difluorophenyl)carbamoylamino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C29H27F2N5O3S
6-[4-[(3,4-difluorophenyl)carbamoylamino]phenyl]-N-(4-methoxyphenyl)-8-methyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6-(cis-3-aminocyclobutyl)-N-[(5-chloro-1H-benzimidazol-2-yl)methyl]-N-methylpyrimidin-4-amine —— C17H19ClN6
6-(cis-3-aminocyclobutyl)-N-[(5-chloro-1H-benzimidazol-2-yl)methyl]-N-methylpyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine —— C20H27N5O
6-(trans-3-aminocyclobutyl)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-{[4-(Pyridin-3-ylmethoxy)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridine —— C19H20N4O2
6-{[4-(Pyridin-3-ylmethoxy)piperidin-1-yl]carbonyl}imidazo[1,2-a]pyridine
—— 6-Methyl 3-[2-(propan-2-yloxy)ethyl] 4-(4-hydroxyphenyl)-2,7-dimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3,6-dicarboxylate —— C25H31NO7
6-Methyl 3-[2-(propan-2-yloxy)ethyl] 4-(4-hydroxyphenyl)-2,7-dimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3,6-dicarboxylate
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-[4-(2-hydroxyethoxy)phenyl]-2-(4-morpholin-4-ylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C44H38Cl2F3N5O7
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-[4-(2-hydroxyethoxy)phenyl]-2-(4-morpholin-4-ylphenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-aminocyclobutyl)-N~4~-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine —— C15H23N7
6-(3-aminocyclobutyl)-N~4~-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyrimidine-2,4-diamine
—— 6-(3-bromo-4-hydroxy-5-methoxyphenyl)-6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide —— C34H25BrCl2F3N5O7
6-(3-bromo-4-hydroxy-5-methoxyphenyl)-6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-1,3,7,9-tetraoxo-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-2-carboxamide
—— 6-(2-chloro-4-hydroxyphenyl)-6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-(4-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C38H25Cl3F3N5O7
6-(2-chloro-4-hydroxyphenyl)-6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-(4-nitrophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(cis-3-aminocyclobutyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-4-amine —— C15H23N7O
6-(cis-3-aminocyclobutyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-4-amine
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(3-ethoxy-2-hydroxyphenyl)-2-(4-iodophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H30Cl2F3IN4O6
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(3-ethoxy-2-hydroxyphenyl)-2-(4-iodophenyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-Aminocyclobutyl)-N-[(5-isopropyl-1,2,4-oxadiazol-3-YL)methyl]pyrimidin-4-amine —— C14H20N6O
6-(3-Aminocyclobutyl)-N-[(5-isopropyl-1,2,4-oxadiazol-3-YL)methyl]pyrimidin-4-amine
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C49H36Cl2F6N4O8
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-2-[4-[2-(2,5-dimethoxyphenyl)ethenyl]phenyl]-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-aminocyclobutyl)-N-{2-[(trifluoromethyl)thio]ethyl}pyrimidin-4-amine —— C11H15F3N4S
6-(3-aminocyclobutyl)-N-{2-[(trifluoromethyl)thio]ethyl}pyrimidin-4-amine
—— 6a,9a-Dichloro-6-[5-(hydroxymethyl)furan-2-yl]-8-(2,3,4,5,6-pentafluorophenyl)-2-(thiophen-2-ylmethyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H19Cl2F5N2O6S
6a,9a-Dichloro-6-[5-(hydroxymethyl)furan-2-yl]-8-(2,3,4,5,6-pentafluorophenyl)-2-(thiophen-2-ylmethyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-methyl-2-[(1-methyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)thio]pyrimidin-4(3H)-one —— C17H23N5O3S
6-methyl-2-[(1-methyl-2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)thio]pyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-{3-[(5-methylpyridin-2-yl)amino]propyl}pyrimidine-2,4-diamine —— C17H25N7
6-(3-aminocyclobutyl)-N~4~-{3-[(5-methylpyridin-2-yl)amino]propyl}pyrimidine-2,4-diamine
—— 6-(trans-3-aminocyclobutyl)-N-[3-(2-furyl)propyl]pyrimidin-4-amine —— C15H20N4O
6-(trans-3-aminocyclobutyl)-N-[3-(2-furyl)propyl]pyrimidin-4-amine
—— 6-{[(2-Methoxyethyl)(2-thienylmethyl)amino]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid —— C16H18N4O3S
6-{[(2-Methoxyethyl)(2-thienylmethyl)amino]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
—— 6-[[1-(2-Ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one —— C22H22N4OS
6-[[1-(2-Ethylphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-7-one
—— 6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-pyridin-2-ylpropyl)pyrimidin-4-amine —— C18H25N5O
6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-(3-pyridin-2-ylpropyl)pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine —— C13H19N7
6-(3-aminocyclobutyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
—— 6a,9a-Dichloro-2-(4-ethenylphenyl)-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C30H26Cl2N2O5
6a,9a-Dichloro-2-(4-ethenylphenyl)-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-({2-[(3-Ethoxyphenyl)carbonyl]hydrazinyl}carbonyl)-3,4-dimethylcyclohex-3-ene-1-carboxylic acid —— C19H24N2O5
6-({2-[(3-Ethoxyphenyl)carbonyl]hydrazinyl}carbonyl)-3,4-dimethylcyclohex-3-ene-1-carboxylic acid
—— 6-(2-Fluorophenyl)-3-(2-methylphenyl)-5-(methylsulfanyl)-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-D]pyrimidin-7-one —— C19H14FN3OS3
6-(2-Fluorophenyl)-3-(2-methylphenyl)-5-(methylsulfanyl)-2-sulfanylidene-2H,3H,6H,7H-[1,3]thiazolo[4,5-D]pyrimidin-7-one
—— 6a,9a-Dichloro-2-(3-chloro-4-methylphenyl)-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C29H25Cl3N2O5
6a,9a-Dichloro-2-(3-chloro-4-methylphenyl)-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-aminocyclobutyl)-N~4~-[3-(methylthio)benzyl]pyrimidine-2,4-diamine —— C16H21N5S
6-(3-aminocyclobutyl)-N~4~-[3-(methylthio)benzyl]pyrimidine-2,4-diamine
—— 6-(6-bromo-4-oxo-2-thioxo-1,2-dihydroquinazolin-3(4H)-yl)-N-butylhexanamide —— C18H24BrN3O2S
6-(6-bromo-4-oxo-2-thioxo-1,2-dihydroquinazolin-3(4H)-yl)-N-butylhexanamide
—— 6-(3-aminocyclobutyl)-N~4~-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidine-2,4-diamine —— C18H25N7
6-(3-aminocyclobutyl)-N~4~-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidine-2,4-diamine
—— 6a,9a-Dichloro-2-cyclohexyl-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C28H30Cl2N2O5
6a,9a-Dichloro-2-cyclohexyl-6-(4-hydroxy-3-methylphenyl)-8-methyl-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-aminocyclobutyl)-N~4~-[(1-ethylcyclobutyl)methyl]pyrimidine-2,4-diamine —— C15H25N5
6-(3-aminocyclobutyl)-N~4~-[(1-ethylcyclobutyl)methyl]pyrimidine-2,4-diamine
—— 6-amino-N-[rac-(1R,5S,6R,7R)-7-benzyl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide —— C19H21N3O2
6-amino-N-[rac-(1R,5S,6R,7R)-7-benzyl-2-oxabicyclo[3.2.0]hept-6-yl]nicotinamide
—— 6-{1-[3-(1H-benzimidazol-2-yl)propanoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol —— C20H23N5O2
6-{1-[3-(1H-benzimidazol-2-yl)propanoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
—— 6-(3-aminocyclobutyl)-N~4~-[(2-isopropyl-4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-2,4-diamine —— C16H24N6S
6-(3-aminocyclobutyl)-N~4~-[(2-isopropyl-4-methyl-1,3-thiazol-5-yl)methyl]pyrimidine-2,4-diamine
—— 6-methoxy-N~4~-{cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}pyrimidine-2,4-diamine —— C16H21N9O
6-methoxy-N~4~-{cis-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]cyclobutyl}pyrimidine-2,4-diamine
—— 6-[8-(5-Carboxypentyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-1,3,7,9-tetraoxo-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C33H37F3N2O10
6-[8-(5-Carboxypentyl)-6-[2-hydroxy-5-(trifluoromethoxy)phenyl]-1,3,7,9-tetraoxo-3a,4,6,6a,9a,10,10a,10b-octahydroisoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— 6-methoxy-2-[3-(5-methyl-1H-tetrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline —— C15H19N5O2
6-methoxy-2-[3-(5-methyl-1H-tetrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline
—— 6-(3-Aminocyclobutyl)-N-(cyclopentylmethyl)-N-methylpyrimidin-4-amine —— C15H24N4
6-(3-Aminocyclobutyl)-N-(cyclopentylmethyl)-N-methylpyrimidin-4-amine
—— 6-Chloro-1-[3-(dimethylamino)propyl]-4-methyl-3,4-dihydroquinolin-2-one —— C15H21ClN2O
6-Chloro-1-[3-(dimethylamino)propyl]-4-methyl-3,4-dihydroquinolin-2-one