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—— 6-{cis-3-[(7-chloroquinolin-4-yl)amino]cyclobutyl}-2-(methoxymethyl)pyrimidin-4(3H)-one —— C19H19ClN4O2
6-{cis-3-[(7-chloroquinolin-4-yl)amino]cyclobutyl}-2-(methoxymethyl)pyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-N~4~-{[1-(dimethylamino)cyclopentyl]methyl}pyrimidine-2,4-diamine —— C16H28N6
6-(3-aminocyclobutyl)-N~4~-{[1-(dimethylamino)cyclopentyl]methyl}pyrimidine-2,4-diamine
—— 6-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}-4-oxo-1,4-dihydropyridine-3-carboxamide —— C17H24N2O4
6-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}-4-oxo-1,4-dihydropyridine-3-carboxamide
—— 6-(trans-3-aminocyclobutyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine —— C16H24N6O
6-(trans-3-aminocyclobutyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-[(2-Hydroxyphenyl)methylamino]-2-phenylbenzo[de]isoquinoline-1,3-dione —— C25H18N2O3
6-[(2-Hydroxyphenyl)methylamino]-2-phenylbenzo[de]isoquinoline-1,3-dione
—— 6-[(4-Ethoxyphenyl)sulfamoyl]-N-[2-(4-methylphenyl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide —— C27H27N3O5S
6-[(4-Ethoxyphenyl)sulfamoyl]-N-[2-(4-methylphenyl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
—— 6-[3-[(2-chloro-4-nitrobenzoyl)amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide —— C28H24ClN5O4S
6-[3-[(2-chloro-4-nitrobenzoyl)amino]phenyl]-8-methyl-N-phenyl-2,3,4,6-tetrahydropyrimido[2,1-b][1,3]thiazine-7-carboxamide
—— 6a,9a-dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-8-(4-fluorophenyl)-6-(6-hydroxy-4H-chromen-3-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C36H25Cl3F4N4O6
6a,9a-dichloro-2-[[3-chloro-6-(trifluoromethyl)pyridin-2-yl]-methylamino]-8-(4-fluorophenyl)-6-(6-hydroxy-4H-chromen-3-yl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-{[5-(cis-3-aminocyclobutyl)-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-3,5,6,7-tetrahydro-4H-pyrrolo[3,4-d]pyrimidin-4-one —— C17H25N7O2
6-{[5-(cis-3-aminocyclobutyl)-4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-methyl-3,5,6,7-tetrahydro-4H-pyrrolo[3,4-d]pyrimidin-4-one
—— 6,8-dibromo-3-(diethylaminomethyl)-7-methyl-3-[(4-methylphenyl)methyl]-2H-chromen-4-one —— C23H27Br2NO2
6,8-dibromo-3-(diethylaminomethyl)-7-methyl-3-[(4-methylphenyl)methyl]-2H-chromen-4-one
—— 6-(trans-3-{[1-(2-thienylcarbonyl)piperidin-4-yl]amino}cyclobutyl)pyrimidin-4(3H)-one —— C18H22N4O2S
6-(trans-3-{[1-(2-thienylcarbonyl)piperidin-4-yl]amino}cyclobutyl)pyrimidin-4(3H)-one
—— 6-(Morpholin-4-yl)-5-nitro-2-(piperidin-1-yl)pyrimidin-4-amine —— C13H20N6O3
6-(Morpholin-4-yl)-5-nitro-2-(piperidin-1-yl)pyrimidin-4-amine
—— 6-[6-(5-bromo-2-hydroxyphenyl)-8-(3-chlorophenyl)-1,3,7,9-tetraoxo-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid —— C38H34BrClN2O7
6-[6-(5-bromo-2-hydroxyphenyl)-8-(3-chlorophenyl)-1,3,7,9-tetraoxo-6a-phenyl-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindol-2-yl]hexanoic acid
—— 6-(1-(3-Chloro-5-(trifluoromethyl)-2-pyridinyl)-1H-pyrazol-5-yl)-4-methyl-2-(3-(trifluoromethyl)phenyl)-1,2,4-triazine-3,5(2H,4H)-dione —— C20H11ClF6N6O2
6-(1-(3-Chloro-5-(trifluoromethyl)-2-pyridinyl)-1H-pyrazol-5-yl)-4-methyl-2-(3-(trifluoromethyl)phenyl)-1,2,4-triazine-3,5(2H,4H)-dione
—— 6-methyl-4-oxo-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]-4H-pyran-2-carboxamide —— C17H21N5O3
6-methyl-4-oxo-N-[2-(4-pyrimidin-2-ylpiperazin-1-yl)ethyl]-4H-pyran-2-carboxamide
—— 6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(2-phenylethyl)pyrimidin-4-amine —— C20H26N4
6-(trans-3-aminocyclobutyl)-2-cyclopropyl-N-methyl-N-(2-phenylethyl)pyrimidin-4-amine
—— 6-(trans-3-aminocyclobutyl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]pyrimidin-4-amine —— C19H25N5
6-(trans-3-aminocyclobutyl)-N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]pyrimidin-4-amine
—— 6-chloro-2'-(4-methoxyphenyl)-7-methyl-3a',6',7',8',8a',8b'-hexahydro-1'H-spiro[indole-3,4'-pyrrolo[3,4-a]pyrrolizine]-1',2,3'(1H,2'H)-trione —— C24H22ClN3O4
6-chloro-2'-(4-methoxyphenyl)-7-methyl-3a',6',7',8',8a',8b'-hexahydro-1'H-spiro[indole-3,4'-pyrrolo[3,4-a]pyrrolizine]-1',2,3'(1H,2'H)-trione
—— 6-hydroxy-5-[(3-hydroxy-4-methoxyphenyl)-(6-hydroxy-1-methyl-4-oxo-2-propylsulfanylpyrimidin-5-yl)methyl]-1-methyl-2-propylsulfanylpyrimidin-4-one —— C24H30N4O6S2
6-hydroxy-5-[(3-hydroxy-4-methoxyphenyl)-(6-hydroxy-1-methyl-4-oxo-2-propylsulfanylpyrimidin-5-yl)methyl]-1-methyl-2-propylsulfanylpyrimidin-4-one
—— 6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpyrimidin-4-amine —— C19H28N6
6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylpyrimidin-4-amine
—— 6-(3-ethoxy-4-hydroxyphenyl)-8-(4-methylanilino)-6a-phenyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C40H37N3O6S
6-(3-ethoxy-4-hydroxyphenyl)-8-(4-methylanilino)-6a-phenyl-2-(thiophen-2-ylmethyl)-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(trans-3-aminocyclobutyl)-N-(1-isobutyrylpiperidin-4-yl)-2-(methoxymethyl)pyrimidin-4-amine —— C19H31N5O2
6-(trans-3-aminocyclobutyl)-N-(1-isobutyrylpiperidin-4-yl)-2-(methoxymethyl)pyrimidin-4-amine
—— 6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(4-hydroxy-2-methoxyphenyl)-2-[2-(4-hydroxyphenyl)ethyl]-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C41H33Cl2F3N4O7
6a-(4-chlorophenyl)-8-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]amino]-6-(4-hydroxy-2-methoxyphenyl)-2-[2-(4-hydroxyphenyl)ethyl]-4,6,9a,10,10a,10b-hexahydro-3aH-isoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(cis-3-aminocyclobutyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]-2-methylpyrimidin-4-amine —— C19H23N5O
6-(cis-3-aminocyclobutyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]-2-methylpyrimidin-4-amine
—— 6-N-(3,5-dichlorophenyl)-2-N-(2,3-dimethylcyclohexyl)-3-(2-morpholin-4-ylethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-2,6-dicarboxamide —— C30H38Cl2N4O5
6-N-(3,5-dichlorophenyl)-2-N-(2,3-dimethylcyclohexyl)-3-(2-morpholin-4-ylethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-2,6-dicarboxamide
—— 6-[[3-Chloro-4-[2-(4-methoxyphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C26H20ClN5O4S
6-[[3-Chloro-4-[2-(4-methoxyphenoxy)ethoxy]phenyl]methylidene]-5-imino-2-pyridin-3-yl-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}carbonyl)pyridin-2-amine —— C17H23N5O
6-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}carbonyl)pyridin-2-amine
—— 6-amino-N-[4-(1-ethyl-4,5-diphenylimidazol-2-yl)sulfanylbutyl]hexanamide —— C27H36N4OS
6-amino-N-[4-(1-ethyl-4,5-diphenylimidazol-2-yl)sulfanylbutyl]hexanamide
—— 6-(4-Methylphenyl)-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1,4-dihydropyridazin-3-one —— C19H25N3O2
6-(4-Methylphenyl)-2-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]-1,4-dihydropyridazin-3-one
—— 6-{1-[(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}-2-methylpyrimidin-4-ol —— C16H20ClN5O2
6-{1-[(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}-2-methylpyrimidin-4-ol
—— 6-[[1-(2,5-Dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one —— C20H19N5O3S
6-[[1-(2,5-Dimethoxyphenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-5-imino-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-one
—— 6a,9a-Dichloro-8-(4-fluorophenyl)-6-[4-(2-hydroxyethoxy)phenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone —— C34H26Cl2FN3O8
6a,9a-Dichloro-8-(4-fluorophenyl)-6-[4-(2-hydroxyethoxy)phenyl]-2-(3-nitrophenyl)-3a,4,6,10,10a,10b-hexahydroisoindolo[5,6-e]isoindole-1,3,7,9-tetrone
—— 6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-methyl-N-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]pyrimidin-4-amine —— C19H23N7O2
6-(3-aminocyclobutyl)-2-(methoxymethyl)-N-methyl-N-[(3-pyridin-4-yl-1,2,4-oxadiazol-5-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(2-pyrrolidin-1-ylethyl)pyrimidine-2,4-diamine —— C15H26N6
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(2-pyrrolidin-1-ylethyl)pyrimidine-2,4-diamine
—— 6-N-(4-bromophenyl)-2-N-cyclohexyl-3-[3-(3-methylpiperidin-1-yl)propyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-2,6-dicarboxamide —— C31H41BrN4O4
6-N-(4-bromophenyl)-2-N-cyclohexyl-3-[3-(3-methylpiperidin-1-yl)propyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-2,6-dicarboxamide
—— 6-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}-2-oxo-1,2-dihydroquinoline-4-carboxamide —— C21H26N2O4
6-methyl-N-{trans-3-[(3-methylbut-2-en-1-yl)oxy]tetrahydro-2H-pyran-4-yl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
—— 6-oxo-N-[(3R,4R)-4-piperidin-1-yloxolan-3-yl]-1H-pyridine-2-carboxamide —— C15H21N3O3
6-oxo-N-[(3R,4R)-4-piperidin-1-yloxolan-3-yl]-1H-pyridine-2-carboxamide
—— 6-{2-[2-(3-Methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethoxy}[1,2,4]triazolo[4,3-b]pyridazine —— C15H17N7O3
6-{2-[2-(3-Methyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]-2-oxoethoxy}[1,2,4]triazolo[4,3-b]pyridazine
—— 6-(cis-3-aminocyclobutyl)-N-[2-(4,5-dimethyl-3-thienyl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine —— C18H26N4OS
6-(cis-3-aminocyclobutyl)-N-[2-(4,5-dimethyl-3-thienyl)ethyl]-2-(methoxymethyl)pyrimidin-4-amine
—— 6-(3,5-dimethylpiperidin-1-yl)-N~2~-(4-methylbenzyl)-5-nitropyrimidine-2,4-diamine —— C19H26N6O2
6-(3,5-dimethylpiperidin-1-yl)-N~2~-(4-methylbenzyl)-5-nitropyrimidine-2,4-diamine
—— 6-(3-Aminocyclobutyl)-N-[(3S)-1-benzylpyrrolidin-3-YL]pyrimidin-4-amine —— C19H25N5
6-(3-Aminocyclobutyl)-N-[(3S)-1-benzylpyrrolidin-3-YL]pyrimidin-4-amine
—— 6-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide —— C14H18N4O2S
6-oxo-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
—— 6-(4-Methylphenyl)-2-(2-morpholin-4-yl-2-oxoethyl)-1,4-dihydropyridazin-3-one —— C17H21N3O3
6-(4-Methylphenyl)-2-(2-morpholin-4-yl-2-oxoethyl)-1,4-dihydropyridazin-3-one
—— 6-{[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-1,3-dimethylpyrimidine-2,4(1H,3H)-dione —— C16H21N5O5
6-{[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-1,3-dimethylpyrimidine-2,4(1H,3H)-dione
—— 6-(3-aminocyclobutyl)-N~4~-{2-[(dimethylamino)methyl]benzyl}pyrimidine-2,4-diamine —— C18H26N6
6-(3-aminocyclobutyl)-N~4~-{2-[(dimethylamino)methyl]benzyl}pyrimidine-2,4-diamine
—— 6-{[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-2-methyl-4,5-dihydropyridazin-3(2H)-one —— C15H21N5O4
6-{[2-(1,2-dihydroxyethyl)-7,8-dihydro-4H-pyrazolo[1,5-a][1,4]diazepin-5(6H)-yl]carbonyl}-2-methyl-4,5-dihydropyridazin-3(2H)-one
—— 6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(3-pyridin-2-ylisoxazol-5-yl)methyl]pyrimidin-4-amine —— C19H22N6O2
6-(trans-3-aminocyclobutyl)-2-(methoxymethyl)-N-[(3-pyridin-2-ylisoxazol-5-yl)methyl]pyrimidin-4-amine
—— 6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(2-morpholin-4-ylethyl)pyrimidine-2,4-diamine —— C15H26N6O
6-(3-aminocyclobutyl)-N~4~-methyl-N~4~-(2-morpholin-4-ylethyl)pyrimidine-2,4-diamine
—— 6-{cis-3-[(5-chloropyridin-2-yl)amino]cyclobutyl}-2-cyclopropylpyrimidin-4(3H)-one —— C16H17ClN4O
6-{cis-3-[(5-chloropyridin-2-yl)amino]cyclobutyl}-2-cyclopropylpyrimidin-4(3H)-one
—— 6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidin-4-amine —— C21H26N6
6-(3-aminocyclobutyl)-2-cyclopropyl-N-[2-(1-methyl-1H-benzimidazol-2-yl)ethyl]pyrimidin-4-amine