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噻二嗪

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(2,3-Dihydro-1,4-benzoxazin-4-yl)-2-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone —— C21H24N4O4S
1-(2,3-Dihydro-1,4-benzoxazin-4-yl)-2-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone
—— 1-(1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-3,3-dimethylbutan-2-one —— C17H25N3O3S
1-(1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-3,3-dimethylbutan-2-one
—— 2-(4-Fluorophenyl)-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone —— C20H22FN3O4S
2-(4-Fluorophenyl)-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone
—— (1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-(1,3-thiazol-4-yl)methanone —— C15H16N4O3S2
(1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-(1,3-thiazol-4-yl)methanone
—— Cycloheptyl-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone —— C19H27N3O3S
Cycloheptyl-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone
—— (5,7-Dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone —— C20H22N6O3S
(5,7-Dimethylpyrazolo[1,5-a]pyrimidin-2-yl)-(1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone
—— 1-(1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-2-(2-methylbenzimidazol-1-yl)ethanone —— C21H23N5O3S
1-(1,1-Dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-2-(2-methylbenzimidazol-1-yl)ethanone
—— (3S)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide —— C18H22N4O2S
(3S)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide
—— (5-cyclopropyl-2-methylfuran-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C21H25N3O4S
(5-cyclopropyl-2-methylfuran-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— 3-(3-chloro-1,2-oxazol-5-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one —— C18H21ClN4O4S
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one
—— [4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone —— C19H22N4O3S
[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[2-methyl-5-(2-methylpropyl)furan-3-yl]methanone —— C22H29N3O4S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[2-methyl-5-(2-methylpropyl)furan-3-yl]methanone
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[1-(2-fluorophenyl)cyclopropyl]methanone —— C22H24FN3O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[1-(2-fluorophenyl)cyclopropyl]methanone
—— [4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone —— C19H20N6O3S
[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone
—— (3R)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide —— C18H22N4O2S
(3R)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide
—— (5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C21H24N6O3S
(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone —— C19H20N6O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-pyrazolo[1,5-a]pyrimidin-3-ylmethanone
—— [4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(5-propylfuran-2-yl)methanone —— C20H25N3O4S
[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(5-propylfuran-2-yl)methanone
—— (3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one —— C20H28N6O3S
(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one
—— 3-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one —— C20H26N4O4S
3-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one
—— (3R)-3-[1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H25N3O5S
(3R)-3-[1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(1-ethyl-3,5-dimethylpyrazol-4-yl)methanone —— C20H27N5O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(1-ethyl-3,5-dimethylpyrazol-4-yl)methanone
—— (4S)-4-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one —— C20H28N4O4S
(4S)-4-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one
—— (3R)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H29N3O3S
(3R)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(3-methyl-1-propylpyrazol-4-yl)methanone —— C20H27N5O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(3-methyl-1-propylpyrazol-4-yl)methanone
—— (5-cyclopropyl-2-methylfuran-3-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C21H25N3O4S
(5-cyclopropyl-2-methylfuran-3-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (3S)-3-[1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C22H24FN5O2S
(3S)-3-[1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(5-methyl-1-propylpyrazol-4-yl)methanone —— C20H27N5O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(5-methyl-1-propylpyrazol-4-yl)methanone
—— (3R)-3-[1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C22H24FN5O2S
(3R)-3-[1-[[1-(4-fluorophenyl)pyrazol-4-yl]methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— (3S)-3-[1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H25N3O5S
(3S)-3-[1-[(6-methoxy-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— (3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one —— C20H28N6O3S
(3S)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one
—— (3R)-3-[1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C22H25FN4O2S
(3R)-3-[1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— (5-tert-butyl-2-methylpyrazol-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C21H29N5O3S
(5-tert-butyl-2-methylpyrazol-3-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (3,5-dimethyl-1-benzofuran-2-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C23H25N3O4S
(3,5-dimethyl-1-benzofuran-2-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (1,3-dimethylpyrazol-4-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C18H23N5O3S
(1,3-dimethylpyrazol-4-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— 3-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one —— C21H21N5O4S
3-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one
—— (3R)-3-[1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide —— C23H27N3O4S
(3R)-3-[1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazine 1,1-dioxide
—— (3S)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H29N3O3S
(3S)-3-[1-[(3R)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— (1,3-dimethylpyrazol-4-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C18H23N5O3S
(1,3-dimethylpyrazol-4-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (3S)-3-[1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C22H25FN4O2S
(3S)-3-[1-[(5-fluoro-1-methylindol-3-yl)methyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— (4S)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one —— C20H28N4O4S
(4S)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one
—— [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone —— C19H22N4O3S
[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(6-methylpyridin-3-yl)methanone
—— (5-tert-butyl-3-methylfuran-2-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C22H29N3O4S
(5-tert-butyl-3-methylfuran-2-yl)-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (3,5-dimethyl-1-benzofuran-2-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C23H25N3O4S
(3,5-dimethyl-1-benzofuran-2-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (4R)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one —— C20H28N4O4S
(4R)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-propan-2-ylpyrrolidin-2-one
—— (3,5-dimethyl-1-propylpyrazol-4-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone —— C21H29N5O3S
(3,5-dimethyl-1-propylpyrazol-4-yl)-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone
—— (3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one —— C20H28N6O3S
(3R)-3-(3,5-dimethyl-1,2,4-triazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one
—— (3S)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H29N3O3S
(3S)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide
—— 3-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one —— C21H21N5O4S
3-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]pyrido[1,2-a]pyrimidin-4-one
—— (3R)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide —— C21H29N3O3S
(3R)-3-[1-[(3S)-3-(5-methylfuran-2-yl)butyl]piperidin-4-yl]-3,4-dihydro-2H-1λ6,2,4-benzothiadiazine 1,1-dioxide