| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | (3S)-3-[2-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-oxoethyl]-2,3-dihydroisoindol-1-one | —— | C22H24N4O4S |
| —— | 1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-(2-ethylimidazol-1-yl)propan-1-one | —— | C20H27N5O3S |
| —— | (1R,4S)-4-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1,7,7-trimethylbicyclo[2.2.1]heptan-2-one | —— | C23H31N3O4S |
| —— | 1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-(6-methylpyridin-2-yl)propan-1-one | —— | C21H26N4O3S |
| —— | 1-[4-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-4-oxobutyl]pyrrolidin-2-one | —— | C20H28N4O4S |
| —— | (2S)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methylpropan-1-one | —— | C21H29N5O3S |
| —— | (2R)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methylpropan-1-one | —— | C21H29N5O3S |
| —— | 2-(4-chloro-3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]ethanone | —— | C19H24ClN5O3S |
| —— | 2-(1,3-benzodioxol-5-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]ethanone | —— | C21H23N3O5S |
| —— | 3-(benzotriazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one | —— | C21H24N6O3S |
| —— | (3S)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one | —— | C21H29N5O3S |
| —— | [5-(diethylaminomethyl)furan-3-yl]-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone | —— | C22H30N4O4S |
| —— | (3R)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-(furan-2-yl)-4-methylpentan-1-one | —— | C22H29N3O4S |
| —— | (3R)-3-[2-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-oxoethyl]-5,5-dimethyloxolan-2-one | —— | C20H27N3O5S |
| —— | (3R)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one | —— | C21H29N5O3S |
| —— | 4-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one | —— | C21H29N5O3S |
| —— | (4R)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one | —— | C20H28N4O5S |
| —— | 4-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]butan-1-one | —— | C21H29N5O3S |
| —— | (3R)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C19H25N5O3S |
| —— | (2S)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methylpropan-1-one | —— | C21H29N5O3S |
| —— | [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[5-ethyl-4-(methoxymethyl)furan-2-yl]methanone | —— | C21H27N3O5S |
| —— | (2S)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methyl-3-(3-methylpyrazol-1-yl)propan-1-one | —— | C20H27N5O3S |
| —— | [2-(dimethylamino)pyrimidin-5-yl]-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone | —— | C19H24N6O3S |
| —— | [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-pyrazolo[1,5-a]pyrimidin-2-ylmethanone | —— | C19H20N6O3S |
| —— | [2-(dimethylamino)pyrimidin-5-yl]-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]methanone | —— | C19H24N6O3S |
| —— | [4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[(5S)-5-methyl-4,5,6,7-tetrahydro-1H-indazol-3-yl]methanone | —— | C21H27N5O3S |
| —— | (3R)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C19H25N5O3S |
| —— | 1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-(4-ethylpiperazin-1-yl)propan-1-one | —— | C21H33N5O3S |
| —— | [4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[(5S)-5-methyl-4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl]methanone | —— | C21H26N4O4S |
| —— | (2R)-3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methylpropan-1-one | —— | C21H29N5O3S |
| —— | [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-(5-propyl-1,2-oxazol-3-yl)methanone | —— | C19H24N4O4S |
| —— | (3S)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-imidazol-1-ylbutan-1-one | —— | C19H25N5O3S |
| —— | [4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-[(5S)-5-methyl-4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl]methanone | —— | C21H26N4O4S |
| —— | (2S)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methyl-3-morpholin-4-ylpropan-1-one | —— | C20H30N4O4S |
| —— | 1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-indazol-1-ylpropan-1-one | —— | C22H25N5O3S |
| —— | 3-(3,5-dimethylpyrazol-1-yl)-1-[4-[(3R)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]propan-1-one | —— | C20H27N5O3S |
| —— | 1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-pyridin-2-ylethanone | —— | C19H22N4O3S |
| —— | 1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-3-(6-methylpyridin-2-yl)propan-1-one | —— | C21H26N4O3S |
| —— | (2R)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1lambda6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]-2-methyl-3-morpholin-4-ylpropan-1-one | —— | C20H30N4O4S |
| —— | 2-(1,3-dihydroisoindol-2-yl)-1-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidin-1-yl]ethanone | —— | C22H26N4O3S |
| —— | (4S)-4-[4-[(3S)-1,1-dioxo-3,4-dihydro-2H-1λ6,2,4-benzothiadiazin-3-yl]piperidine-1-carbonyl]-1-(2-methoxyethyl)pyrrolidin-2-one | —— | C20H28N4O5S |
| —— | Isoquinolin-1-yl-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone | —— | C22H22N4O4S |
| —— | (6-Methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-pyridin-4-ylmethanone | —— | C18H20N4O4S |
| —— | 2-(1,3-Benzodioxol-5-yl)-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone | —— | C21H23N3O6S |
| —— | 2H-chromen-3-yl-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone | —— | C22H23N3O5S |
| —— | Furan-2-yl-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)methanone | —— | C17H19N3O5S |
| —— | 2-(1H-indol-3-yl)-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone | —— | C22H24N4O4S |
| —— | 2-[(1S,3R)-3-acetyl-2,2-dimethylcyclobutyl]-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone | —— | C22H31N3O5S |
| —— | 1-(6-Methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)-3-phenylpropan-1-one | —— | C21H25N3O4S |
| —— | 2-[(1R,3R)-3-acetyl-2,2-dimethylcyclobutyl]-1-(6-methoxy-1,1-dioxospiro[2,4-dihydro-1lambda6,2,4-benzothiadiazine-3,4'-piperidine]-1'-yl)ethanone | —— | C22H31N3O5S |