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噻吩并嘧啶酮衍生物

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[cyclohexyl(methyl)amino]-5-methyl-N-[(1R)-1-phenylethyl]thieno[2,3-d]pyrimidine-6-carboxamide —— C23H28N4OS
4-[cyclohexyl(methyl)amino]-5-methyl-N-[(1R)-1-phenylethyl]thieno[2,3-d]pyrimidine-6-carboxamide
—— N-[(2R)-butan-2-yl]-2-[3-(4-ethylphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide —— C24H29N3O3S
N-[(2R)-butan-2-yl]-2-[3-(4-ethylphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide
—— 6-[1-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide —— C24H30N4O4S
6-[1-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-phenylhexanamide
—— N-[(4-methylphenyl)methyl]-6-[1-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]hexanamide —— C28H36N4O4S
N-[(4-methylphenyl)methyl]-6-[1-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]hexanamide
—— 11-(4-chlorophenyl)-9-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6)-diene-10,12-dione —— C23H24ClN3O3S
11-(4-chlorophenyl)-9-[2-[(2R)-2-methylpiperidin-1-yl]-2-oxoethyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6)-diene-10,12-dione
—— N-[(2S)-butan-2-yl]-2-[3-(4-ethylphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide —— C24H29N3O3S
N-[(2S)-butan-2-yl]-2-[3-(4-ethylphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide
—— N-[(2R)-butan-2-yl]-2-[3-(4-ethoxyphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide —— C24H29N3O4S
N-[(2R)-butan-2-yl]-2-[3-(4-ethoxyphenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide
—— N-[(2S)-butan-2-yl]-2-[3-(4-chlorophenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide —— C22H24ClN3O3S
N-[(2S)-butan-2-yl]-2-[3-(4-chlorophenyl)-2,4-dioxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-1-yl]acetamide
—— 6-[1-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-fluorophenyl)methyl]hexanamide —— C28H35FN4O4S
6-[1-[2-[(2R)-2-ethylpiperidin-1-yl]-2-oxoethyl]-2,4-dioxothieno[3,2-d]pyrimidin-3-yl]-N-[(4-fluorophenyl)methyl]hexanamide
—— (2R)-2-(4-oxo-6-propylthieno[2,3-d]pyrimidin-3-yl)-N-[(E)-1-thiophen-2-ylpropylideneamino]propanamide —— C19H22N4O2S2
(2R)-2-(4-oxo-6-propylthieno[2,3-d]pyrimidin-3-yl)-N-[(E)-1-thiophen-2-ylpropylideneamino]propanamide
—— (2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2,4-dimethylphenyl)propanamide —— C21H24N4OS2
(2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2,4-dimethylphenyl)propanamide
—— (2S)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(3-fluorophenyl)propanamide —— C19H19FN4OS2
(2S)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(3-fluorophenyl)propanamide
—— (2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2-phenylethyl)propanamide —— C21H24N4OS2
(2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(2-phenylethyl)propanamide
—— 2-[[3-(4-chlorophenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide —— C27H25ClN4O5S2
2-[[3-(4-chlorophenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide
—— 2-[[11-(4-chlorophenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide —— C26H23ClN4O5S2
2-[[11-(4-chlorophenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide
—— N-benzyl-3-[(7R)-7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl]propanamide —— C21H23N3O2S
N-benzyl-3-[(7R)-7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl]propanamide
—— ethyl (3S)-1-[2-(4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-3-yl)acetyl]piperidine-3-carboxylate —— C20H25N3O4S
ethyl (3S)-1-[2-(4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-3-yl)acetyl]piperidine-3-carboxylate
—— N-[(Z)-(2-chlorophenyl)methylideneamino]-2-[(4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]acetamide —— C25H21ClN4O2S2
N-[(Z)-(2-chlorophenyl)methylideneamino]-2-[(4-oxo-3-phenyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]acetamide
—— 2-[(Z)-[[2-[[3-(4-methylphenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]hydrazinylidene]methyl]benzoic acid —— C27H24N4O4S2
2-[(Z)-[[2-[[3-(4-methylphenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]hydrazinylidene]methyl]benzoic acid
—— N'-[(Z)-(4-chloro-3-nitrophenyl)methylidene]-2-{[3-(4-methylphenyl)-4-oxo-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl]sulfanyl}acetohydrazide —— C26H22ClN5O4S2
N'-[(Z)-(4-chloro-3-nitrophenyl)methylidene]-2-{[3-(4-methylphenyl)-4-oxo-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl]sulfanyl}acetohydrazide
—— (E)-N'-(1-(4-bromophenyl)ethylidene)-2-((4-oxo-3-(p-tolyl)-3,4,5,6,7,8-hexahydrobenzo[4,5]thieno[2,3-d]pyrimidin-2-yl)thio)acetohydrazide —— C27H25BrN4O2S2
(E)-N'-(1-(4-bromophenyl)ethylidene)-2-((4-oxo-3-(p-tolyl)-3,4,5,6,7,8-hexahydrobenzo[4,5]thieno[2,3-d]pyrimidin-2-yl)thio)acetohydrazide
—— N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C20H28N4O2S
N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— 4-methyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C21H30N4O2S
4-methyl-N-[2-[(2R)-2-methylpiperidin-1-yl]ethyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— 4-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C22H32N4O2S
4-methyl-N-[3-[(2S)-2-methylpiperidin-1-yl]propyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— 4-methyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C21H30N4O2S
4-methyl-N-[2-[(2S)-2-methylpiperidin-1-yl]ethyl]-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide —— C21H30N4O2S
N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]-4-methyl-2-oxo-6-thia-1,8-diazatricyclo[7.3.0.03,7]dodeca-3(7),4,8-triene-5-carboxamide
—— (3R)-1-(9-fluoro-[1]benzothiolo[3,2-d]pyrimidin-4-yl)-N-(4-methylcyclohexyl)piperidine-3-carboxamide —— C23H27FN4OS
(3R)-1-(9-fluoro-[1]benzothiolo[3,2-d]pyrimidin-4-yl)-N-(4-methylcyclohexyl)piperidine-3-carboxamide
—— N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-2,3,5-trimethyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide —— C18H25N3O2S
N-[(1S,2S,3S)-2,3-dimethylcyclohexyl]-2,3,5-trimethyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide
—— 1-(5-chloropyridin-2-yl)-3-[(12R)-4,12-dimethyl-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-5-yl]urea —— C19H20ClN5O2S
1-(5-chloropyridin-2-yl)-3-[(12R)-4,12-dimethyl-2-oxo-6-thia-1,8-diazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-5-yl]urea
—— (12R)-5-hexylsulfanyl-12-propan-2-yl-4-prop-2-enyl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one —— C21H30N2O2S2
(12R)-5-hexylsulfanyl-12-propan-2-yl-4-prop-2-enyl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
—— 5-(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)-N-[(1R,2R)-2-methylcyclohexyl]pentanamide —— C18H25N3O3S
5-(2,4-dioxo-1H-thieno[3,2-d]pyrimidin-3-yl)-N-[(1R,2R)-2-methylcyclohexyl]pentanamide
—— N-butyl-3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide —— C21H30N4O3S
N-butyl-3-[2-[(3R,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide
—— N-butyl-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide —— C21H30N4O3S
N-butyl-3-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethyl]-5-methyl-4-oxothieno[2,3-d]pyrimidine-6-carboxamide
—— (12R)-12-ethyl-5-(2-methoxyethylsulfanyl)-12-methyl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine —— C15H21N3O2S2
(12R)-12-ethyl-5-(2-methoxyethylsulfanyl)-12-methyl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
—— methyl (2S)-2-[(12R)-3-oxo-4-phenyl-12-propan-2-yl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-5-yl]propanoate —— C22H24N2O4S
methyl (2S)-2-[(12R)-3-oxo-4-phenyl-12-propan-2-yl-11-oxa-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-5-yl]propanoate
—— (6S)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one —— C21H25N3O2S2
(6S)-6-methyl-2-(2-oxo-2-pyrrolidin-1-ylethyl)sulfanyl-3-(2-phenylethyl)-6,7-dihydrothieno[3,2-d]pyrimidin-4-one
—— (2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(3-cyanophenyl)propanamide —— C20H19N5OS2
(2R)-2-[(4-amino-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl)sulfanyl]-N-(3-cyanophenyl)propanamide
—— (2R)-2-(5,6-dimethyl-4-oxo-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanyl-N-phenylpropanamide —— C20H21N3O2S2
(2R)-2-(5,6-dimethyl-4-oxo-3-prop-2-enylthieno[2,3-d]pyrimidin-2-yl)sulfanyl-N-phenylpropanamide
—— ethyl (6R)-6-methyl-2-[[2-[6-methyl-4-oxo-3-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-2-yl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H28N4O4S3
ethyl (6R)-6-methyl-2-[[2-[6-methyl-4-oxo-3-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidin-2-yl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetohydrazide —— C28H28N4O6S2
N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]-2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]acetohydrazide
—— 2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)propyl]acetohydrazide —— C28H28N4O4S2
2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)propyl]acetohydrazide
—— 2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide —— C26H24N4O4S2
2-[[11-(4-ethoxyphenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[(4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide
—— (6R)-N-[(Z)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C24H30N4S
(6R)-N-[(Z)-(4-ethylphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 2-[[11-(4-chlorophenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)propyl]acetohydrazide —— C26H23ClN4O3S2
2-[[11-(4-chlorophenyl)-12-oxo-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(8),2(6),9-trien-10-yl]sulfanyl]-N'-[1-(4-oxocyclohexa-2,5-dien-1-ylidene)propyl]acetohydrazide
—— 2-[[3-(4-bromophenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide —— C27H25BrN4O5S2
2-[[3-(4-bromophenyl)-4-oxo-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-2-yl]sulfanyl]-N'-[(3,5-dimethoxy-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]acetohydrazide
—— 4-(dimethylamino)benzaldehyde [3-(4-methylphenyl)-4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl]hydrazone —— C25H25N5OS
4-(dimethylamino)benzaldehyde [3-(4-methylphenyl)-4-oxo-3,5,6,7-tetrahydro-4H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl]hydrazone
—— (6R)-N-[(Z)-(4-methoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C23H28N4OS
(6R)-N-[(Z)-(4-methoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— 6-[[2-[(6S)-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one —— C22H26N4OS
6-[[2-[(6S)-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-yl]hydrazinyl]methylidene]cyclohexa-2,4-dien-1-one
—— (6R)-N-[(Z)-(2-methoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C23H28N4OS
(6R)-N-[(Z)-(2-methoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine
—— (6S)-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine —— C24H30N4OS
(6S)-N-[(Z)-(4-ethoxyphenyl)methylideneamino]-6-(2-methylbutan-2-yl)-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-amine