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三唑并二氮卓类

中文名称 英文名称 CAS号 化学式
—— 2-{7-[(3,5-Dimethyl-1,2-oxazol-4-YL)sulfonyl]-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-2-YL}acetonitrile —— C13H16N6O4S
—— 7-[2-(2-Fluorophenyl)acetyl]-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C15H17FN4O2
—— 7-[(5-Chlorothiophen-2-YL)sulfonyl]-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C11H13ClN4O3S2
—— 2-(Cyclopropylmethyl)-7-(pyridine-3-sulfonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C15H19N5O3S
—— 2-(Cyclopropylmethyl)-7-(2,3-dihydro-1H-indene-5-sulfonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C19H24N4O3S
—— 3-{[2-(2-Methoxyethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-7-YL]methyl}benzonitrile —— C17H21N5O2
—— 2-[7-(2,3-Dihydro-1,4-benzodioxine-6-sulfonyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-2-YL]acetonitrile —— C16H17N5O5S
—— 7-(Butane-1-sulfonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C10H18N4O3S
—— 7-(2,4-Dimethoxybenzoyl)-2-(2-methoxyethyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C18H24N4O5
—— 7-(5-Chloro-2-fluorobenzoyl)-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H14ClFN4O2
—— 2-(Cyclopropylmethyl)-7-[2-(4-methylphenyl)acetyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C19H24N4O2
—— 7-[2-(4-Chloro-2-methylphenoxy)acetyl]-2-(2-methoxyethyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C18H23ClN4O4
—— 7-(2-Chloro-4-fluorobenzoyl)-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H14ClFN4O2
—— 7-[2-(4-Chloro-2-methylphenoxy)acetyl]-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C16H19ClN4O3
—— 2-Methyl-7-(3-methylthiophene-2-carbonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C13H16N4O2S
—— 7-(2,6-Dimethoxypyridine-3-carbonyl)-2-(2-methoxyethyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C17H23N5O5
—— 7-{5-[(3,5-Dimethyl-1,2-oxazol-4-YL)methyl]furan-2-carbonyl}-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C18H21N5O4
—— 2-(Cyclopropylmethyl)-7-[(1-ethyl-1H-pyrazol-4-YL)sulfonyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C15H22N6O3S
—— 3-{2-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-7-YL]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one —— C19H21N5O4
—— 7-[3-(2-Methoxyphenyl)propanoyl]-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C17H22N4O3
—— 4-({3-Oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-7-YL}sulfonyl)benzonitrile —— C13H13N5O3S
—— 7-(5-Bromopyridine-3-carbonyl)-2-(2-methoxyethyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C15H18BrN5O3
—— 7-(5-Fluoro-2-methoxybenzenesulfonyl)-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H17FN4O4S
—— 7-[(3-fluoro-4-pyridyl)methyl]-2-methyl-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-one —— C13H16FN5O
—— 7-[(3,5-Dimethyl-1,2-oxazol-4-YL)sulfonyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C11H15N5O4S
—— 2-Methyl-7-(5,6,7,8-tetrahydronaphthalene-2-sulfonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C17H22N4O3S
—— 7-[3-(3-methoxy-5-isoxazolyl)propanoyl]-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-one —— C13H17N5O4
—— 7-(4-Chloro-2-methylbenzenesulfonyl)-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H17ClN4O3S
—— 2-Benzyl-7-[2-(benzyloxy)acetyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C22H24N4O3
—— 7-[(1-Ethyl-1H-pyrazol-4-YL)sulfonyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C11H16N6O3S
—— 7-[2-(4-Methanesulfonylphenyl)acetyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C15H18N4O4S
—— 7-[3-(3-Methoxyphenyl)propanoyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C16H20N4O3
—— 3-({3-Oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-7-YL}sulfonyl)benzonitrile —— C13H13N5O3S
—— 7-[2-(2-Methoxyphenyl)acetyl]-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C16H20N4O3
—— 7-(5-Bromofuran-2-carbonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C11H11BrN4O3
—— N-(2-furylmethyl)-3-oxo-2,3,5,6,8,9-hexahydro-7H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide —— C12H15N5O3
—— 7-[(5-Chlorothiophen-2-YL)sulfonyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C10H11ClN4O3S2
—— 7-[2-(4-Chlorophenyl)acetyl]-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H15ClN4O2
—— N-(2-Methoxyethyl)-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepine-7-carboxamide —— C11H19N5O3
—— 2-methyl-7-[2-(3-thienyl)acetyl]-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-one —— C13H16N4O2S
—— 7-(2,3-Dihydro-1,4-benzodioxine-6-sulfonyl)-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepin-3-one —— C14H16N4O5S
—— 3-Cyclopropyl-N-(4-methoxyphenyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepine-7-carboxamide —— C17H21N5O2
—— 3-Cyclopropyl-N-(3-methylphenyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepine-7-carboxamide —— C17H21N5O
—— 3-Cyclopropyl-N-[(4-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepine-7-carboxamide —— C18H23N5O
—— 3-Cyclopropyl-N-(3-fluorophenyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-D][1,4]diazepine-7-carboxamide —— C16H18FN5O
—— 3-cyclopropyl-N-(2-fluorophenyl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide —— C16H18FN5O
—— 3-benzyl-7-[(3-ethyl-4,5-dihydroisoxazol-5-yl)methyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H25N5O
—— 5-[(3-benzyl-5,6,8,9-tetrahydro-7H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methyl]-N,N-dimethylpyridin-2-amine —— C21H26N6
—— 3-benzyl-7-[(3-isopropyl-1,2,4-oxadiazol-5-yl)methyl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H24N6O
—— 3-benzyl-7-(2-morpholin-4-yl-2-oxoethyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H25N5O2