| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 3-[(2S)-1-[(4-chlorophenyl)methylsulfonyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22ClN5O2S |
| —— | (3-methyl-1-benzofuran-2-yl)-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H23N5O2 |
| —— | 1-[3-[(2R)-1-[(1-methylindol-3-yl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H28N6O |
| —— | 3-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |
| —— | 1-[3-[(2S)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O |
| —— | 1-[3-[(2R)-1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O |
| —— | (2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C21H29N5O2 |
| —— | 1-[3-[(2S)-1-[(3-methylphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O |
| —— | [1-(2-fluorophenyl)cyclopentyl]-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C22H28FN5O |
| —— | 2-(1H-indol-3-yl)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H26N6O |
| —— | 3-[(2R)-1-(4-methoxy-3-methylphenyl)sulfonylpyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |
| —— | 3-[(2S)-1-[(4-methoxy-2,3,6-trimethylphenyl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C21H31N5O |
| —— | 2-[(4-methoxyphenyl)methyl-methylamino]-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H30N6O2 |
| —— | 2-(2-methoxy-4-methylphenoxy)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H29N5O3 |
| —— | 1-[3-[(2R)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | 3-(3-chlorophenyl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H26ClN5O |
| —— | 3-[(2S)-1-(4-fluoro-3-methylphenyl)sulfonylpyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22FN5O2S |
| —— | [4-(ethoxymethyl)phenyl]-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C21H29N5O2 |
| —— | 1-[3-[(2S)-1-(2-phenylethyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O |
| —— | 1-[3-[(2S)-1-(benzenesulfonyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H23N5O3S |
| —— | 3-[(2R)-1-(2-methoxyphenyl)sulfonylpyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H23N5O3S |
| —— | 4-(4-fluorophenyl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]butan-1-one | —— | C20H26FN5O |
| —— | 2-(2-methoxy-4-methylphenoxy)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H29N5O3 |
| —— | [3-(4-fluorophenyl)-1,2-oxazol-5-yl]-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H21FN6O2 |
| —— | 2-(2,6-dimethylphenoxy)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H29N5O2 |
| —— | 2-(1H-indol-3-yl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H26N6O |
| —— | 3-[(2S)-1-[(6-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C20H27N5O3 |
| —— | 2,3-dihydro-1,4-benzodioxin-6-yl-[3-[(3S)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H27N5O3 |
| —— | 2-(4-ethoxyphenyl)-1-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | 3-(2-methoxyphenyl)-1-[3-[(3S)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | 1-[4-(7-Acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-2-cyclopentylethanone | —— | C20H31N5O2 |
| —— | 2-(3-fluorophenyl)-2-methyl-1-[4-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]propan-1-one | —— | C21H28FN5O |
| —— | 3-[(3S)-1-(2-phenylethyl)piperidin-3-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C19H27N5 |
| —— | (3-methyl-1-benzofuran-2-yl)-[3-[(3S)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C22H27N5O2 |
| —— | 3-[1-[[(2S)-2-methyl-2,3-dihydro-1-benzofuran-5-yl]methyl]piperidin-4-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C21H29N5O |
| —— | 1-[(3R)-3-[7-[(2-methoxy-4-methylphenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]piperidin-1-yl]ethanone | —— | C22H31N5O2 |
| —— | 1-[4-(7-Acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-2-(3-methylphenyl)ethanone | —— | C22H29N5O2 |
| —— | 3-[(3S)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]piperidin-3-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | 3-(1-cyclopentylsulfonylpiperidin-4-yl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C16H27N5O2S |
| —— | 2-cyclohexyl-1-[3-[(3S)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H33N5O |
| —— | 3-methyl-1-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one | —— | C17H29N5O |
| —— | 1-[4-(7-Acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-2-(4-fluorophenyl)ethanone | —— | C21H26FN5O2 |
| —— | 1-[3-[(3S)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenoxyethanone | —— | C20H27N5O2 |
| —— | 2-(3,4-Dimethylphenyl)-1-[4-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]ethanone | —— | C22H31N5O |
| —— | 3-(2-methoxyphenyl)-1-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | 1-[4-(7-Acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-2-(3-fluorophenyl)ethanone | —— | C21H26FN5O2 |
| —— | 2-cyclopentyl-1-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H31N5O |
| —— | (2-Methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)-[4-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]methanone | —— | C22H31N5O2 |
| —— | 2,2-dimethyl-1-[3-[(3R)-1-methylpiperidin-3-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C17H29N5O |
| —— | (2S)-1-[4-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-2-phenylpropan-1-one | —— | C22H29N5O2 |