| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C14H23N5O |
| —— | 2,3-dihydro-1,4-benzodioxin-6-yl-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C19H23N5O3 |
| —— | [3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C22H31N5O2 |
| —— | [3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(4-methyl-1,3-thiazol-5-yl)methanone | —— | C17H24N6OS |
| —— | (3-methoxyphenyl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C19H25N5O2 |
| —— | 1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenoxyethanone | —— | C19H25N5O2 |
| —— | 1-[3-[(2R)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-cyclopentylpropan-1-one | —— | C20H31N5O2 |
| —— | 4-(4-fluorophenyl)-1-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one | —— | C22H30FN5O |
| —— | (2,4-dimethyl-1,3-oxazol-5-yl)-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H26N6O2 |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenoxyethanone | —— | C20H25N5O3 |
| —— | 1-[(2S)-2-[7-[(4-fluorophenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone | —— | C19H24FN5O |
| —— | 1-[3-[(2S)-1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C17H29N5O |
| —— | 3-[(2S)-1-(4-fluoro-2-methylphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | 2-cyclohexyl-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H31N5O |
| —— | 2-(3-methoxyphenyl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C20H27N5O2 |
| —— | 7-(2-fluoro-5-methylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22FN5O2S |
| —— | 3-(2-methoxyphenyl)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C21H29N5O2 |
| —— | 1-[2-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-oxoethyl]azepan-2-one | —— | C20H32N6O2 |
| —— | 1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C14H23N5O |
| —— | 7-(2-fluoro-5-methylphenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | (5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C19H28N6O2 |
| —— | 2-methyl-2-(4-methylphenyl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C21H29N5O |
| —— | 7-(4-methoxyphenyl)sulfonyl-3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |
| —— | 7-(2-chlorophenyl)sulfonyl-3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22ClN5O2S |
| —— | 2-(2,6-dimethylphenoxy)-1-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | 2-(2,4-difluorophenoxy)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H23F2N5O2 |
| —— | 7-[(4-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | N-benzyl-N-propan-2-yl-2-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]acetamide | —— | C22H32N6O |
| —— | 2-cyclopentyl-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H29N5O |
| —— | 2-(3-methoxyphenyl)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | 2-(3-methoxyphenyl)-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | [3-(2-fluorophenyl)-1,2-oxazol-5-yl]-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H21FN6O2 |
| —— | 2-(4-fluorophenoxy)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O2 |
| —— | [3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)methanone | —— | C20H30N6O2 |
| —— | 2-(2,6-dimethylphenoxy)-1-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | [3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-phenylmethanone | —— | C18H23N5O |
| —— | 4-(4-fluorophenyl)-1-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]butan-1-one | —— | C22H30FN5O |
| —— | (5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H26N6O2 |
| —— | 1-[3-[(2S)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H31N5O |
| —— | 2,3-dihydro-1,4-benzodioxin-6-yl-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H25N5O3 |
| —— | 7-(2-fluoro-5-methylphenyl)sulfonyl-3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-(4-fluorophenyl)ethanone | —— | C20H24FN5O2 |
| —— | 2-(2,4-difluorophenoxy)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H23F2N5O2 |
| —— | 2-(4-fluorophenyl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C18H22FN5O |
| —— | 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenoxyethanone | —— | C20H25N5O3 |
| —— | 7-(2-fluoro-5-methylphenyl)sulfonyl-3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22FN5O2S |
| —— | 1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenoxyethanone | —— | C19H25N5O2 |
| —— | (2,4-dimethyl-1,3-thiazol-5-yl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C17H24N6OS |
| —— | 2-[(2-fluorophenyl)methyl-methylamino]-1-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27FN6O |
| —— | 7-(2-methoxy-5-methylphenyl)sulfonyl-3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |