| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 3-[(2R)-1-(cyclopropylmethyl)pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C14H23N5 |
| —— | 1-[3-[(2S)-1-(cyclopropylmethyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C16H25N5O |
| —— | 4-(4-fluorophenyl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]butan-1-one | —— | C21H28FN5O |
| —— | 3-[(2R)-1-(4-fluoro-3-methylphenyl)sulfonylpyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22FN5O2S |
| —— | 4-(azepan-1-yl)-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]butan-1-one | —— | C20H34N6O |
| —— | 2-(2-methylindol-1-yl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C22H28N6O |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-cyclopentylpropan-1-one | —— | C20H31N5O2 |
| —— | [4-(ethoxymethyl)phenyl]-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H27N5O2 |
| —— | 3-[(2R)-1-[(3-cyclopentyloxyphenyl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | 1-[3-[(2S)-1-(2-methylpropyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C16H27N5O |
| —— | 1-[3-[(2S)-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O2 |
| —— | 1-[3-[(2R)-1-(3-methoxybenzoyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H25N5O3 |
| —— | 3-[(2S)-1-(cyclopropylmethyl)pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C14H23N5 |
| —— | 2-[(4-methoxyphenyl)methyl-methylamino]-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C21H30N6O2 |
| —— | (5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C19H28N6O2 |
| —— | [1-(2-fluorophenyl)cyclopentyl]-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C22H28FN5O |
| —— | 2-(2-fluorophenoxy)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H24FN5O2 |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C21H30N6O2 |
| —— | 3-[(2R)-1-[(3-methylphenyl)methylsulfonyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O2S |
| —— | 3-[(2R)-1-(4-fluoro-3-methylphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | (2-methyl-1,3-benzothiazol-6-yl)-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H24N6OS |
| —— | 3-(3-chlorophenyl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C19H24ClN5O |
| —— | 1-[3-[(2S)-1-[(2-methylphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O |
| —— | 3-(2-methylphenoxy)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H27N5O2 |
| —— | 3-(3-chlorophenyl)-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C19H24ClN5O |
| —— | 1-[3-[(2R)-1-(benzenesulfonyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H23N5O3S |
| —— | 3-(4-methoxyphenyl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H27N5O2 |
| —— | (3-methyl-1-benzofuran-2-yl)-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H23N5O2 |
| —— | 1-[3-[(2S)-1-[(2-chlorophenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24ClN5O |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C21H30N6O2 |
| —— | 3-[(2R)-1-[(4-cyclopentyloxyphenyl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | 1-[3-[(2R)-1-(cyclopropylmethyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C16H25N5O |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-cyclopentylethanone | —— | C19H29N5O2 |
| —— | 1-[3-[(2S)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C21H29N5O2 |
| —— | [3-(4-fluorophenyl)-1,2-oxazol-5-yl]-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H21FN6O2 |
| —— | 3-(3-chlorophenyl)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H26ClN5O |
| —— | 1-[3-[(2R)-1-[(2-methoxy-4-methylphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C21H29N5O2 |
| —— | 3-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |
| —— | 2-(2-methylindol-1-yl)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C22H28N6O |
| —— | (2-methyl-1,3-benzothiazol-6-yl)-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C20H24N6OS |
| —— | 4-(azepan-1-yl)-1-[(2R)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]butan-1-one | —— | C20H34N6O |
| —— | 1-[3-[(2R)-1-benzylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H25N5O |
| —— | 3-[(2R)-1-[(2,2-dimethyl-3H-1-benzofuran-5-yl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C21H29N5O |
| —— | (5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C19H28N6O2 |
| —— | 3-(2-methylphenoxy)-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C20H27N5O2 |
| —— | 1-[3-[(2R)-1-[(2-methylphenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27N5O |
| —— | 1-[3-[(2S)-1-benzylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H25N5O |
| —— | 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-cyclopentylethanone | —— | C19H29N5O2 |
| —— | 3-[(2S)-1-[(4-cyclopentyloxyphenyl)methyl]pyrrolidin-2-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | [4-(ethoxymethyl)phenyl]-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]methanone | —— | C21H29N5O2 |