| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 1-[3-[1-(Cyclohexanecarbonyl)piperidin-4-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H31N5O2 |
| —— | 1-[4-(7-Acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-3-phenylpropan-1-one | —— | C22H29N5O2 |
| —— | 2-(4-Methoxyphenyl)-1-[3-(1-methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C21H29N5O2 |
| —— | (3-Ethyl-1,2-oxazol-5-yl)-[3-(1-methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H26N6O2 |
| —— | N-cyclohexyl-N-methyl-2-(3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)acetamide | —— | C20H34N6O |
| —— | [3-(1-Methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C22H31N5O2 |
| —— | 1-[3-(1-Acetylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(2-fluorophenyl)ethanone | —— | C21H26FN5O2 |
| —— | 7-(4-Fluoro-3-methylphenyl)sulfonyl-3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | 7-[(2-Cyclopentyloxyphenyl)methyl]-3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C23H33N5O |
| —— | 1-[3-(1-methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-[(2R)-oxan-2-yl]ethanone | —— | C19H31N5O2 |
| —— | 1-[3-[1-(2,2-Dimethylpropyl)piperidin-4-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H31N5O |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-(4-fluorophenyl)propan-1-one | —— | C21H26FN5O2 |
| —— | 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-(4-fluorophenyl)propan-1-one | —— | C21H26FN5O2 |
| —— | 1-[3-[1-(Quinolin-6-ylmethyl)piperidin-4-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C23H28N6O |
| —— | 1-[3-[(2R)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H25N5O4S |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-phenylpropan-1-one | —— | C21H27N5O2 |
| —— | 1-[(2S)-2-[7-(4-methoxyphenyl)sulfonyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone | —— | C19H25N5O4S |
| —— | 1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenylethanone | —— | C19H25N5O |
| —— | 1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenylethanone | —— | C19H25N5O |
| —— | 1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenylethanone | —— | C19H25N5O |
| —— | 1-[3-[(2S)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-phenylpropan-1-one | —— | C21H27N5O2 |
| —— | 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-phenylpropan-1-one | —— | C21H27N5O2 |
| —— | 1-[(2R)-2-[7-[(4-fluorophenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone | —— | C19H24FN5O |
| —— | 1-[3-[(2S)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O |
| —— | 2-(2,3-dimethylphenoxy)-2-methyl-1-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | [(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-phenylmethanone | —— | C18H23N5O |
| —— | 2,3-dihydro-1,4-benzodioxin-6-yl-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H25N5O3 |
| —— | N-benzyl-N-propan-2-yl-2-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]acetamide | —— | C22H32N6O |
| —— | (2-methyl-1,3-benzothiazol-6-yl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H24N6OS |
| —— | 7-(4-methoxyphenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H25N5O3S |
| —— | 2-methyl-1-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C16H27N5O |
| —— | (2,4-dimethyl-1,3-thiazol-5-yl)-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H26N6OS |
| —— | 2-(2-fluorophenoxy)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O2 |
| —— | 2-[(2-fluorophenyl)methyl-methylamino]-1-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H27FN6O |
| —— | 1-[3-[(2R)-1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C17H29N5O |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H30N6O2 |
| —— | 3-[(2R)-1-(4-fluoro-2-methylphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | N-cyclohexyl-N-methyl-2-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]acetamide | —— | C19H32N6O |
| —— | 2-(1H-indol-3-yl)-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C21H26N6O |
| —— | 2-(4-fluorophenyl)-1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H24FN5O |
| —— | 1-(4-methylpiperidin-1-yl)-2-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H30N6O |
| —— | [3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C21H29N5O2 |
| —— | 2-(2,4-difluorophenoxy)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H23F2N5O2 |
| —— | [3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(2-methyl-4,5,6,7-tetrahydro-1-benzofuran-3-yl)methanone | —— | C21H29N5O2 |
| —— | 1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenoxyethanone | —— | C19H25N5O2 |
| —— | 2-methyl-2-(4-methylphenyl)-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]propan-1-one | —— | C21H29N5O |
| —— | (3-methyl-1-benzofuran-2-yl)-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C22H27N5O2 |
| —— | 2-(4-fluorophenyl)-1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C19H24FN5O |
| —— | (3-methyl-1-benzofuran-2-yl)-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C22H27N5O2 |
| —— | 7-(4-fluoro-2-methylphenyl)sulfonyl-3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |