| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | [3-(1-Methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(5-propyl-1,2-oxazol-3-yl)methanone | —— | C19H28N6O2 |
| —— | 3-[(3R)-1-(2-phenylethyl)piperidin-3-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C19H27N5 |
| —— | 2-(4-Methoxy-3-methylphenyl)-1-[3-(1-methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H31N5O2 |
| —— | [4-(methoxymethyl)phenyl]-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H29N5O2 |
| —— | 3-(2-Methylphenoxy)-1-[3-(1-methylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | 2-methyl-2-(4-methylphenyl)-1-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C23H33N5O |
| —— | (5-cyclopropyl-1,2-oxazol-3-yl)-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H24N6O2 |
| —— | 1-[3-(1-Cycloheptylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C20H33N5O |
| —— | 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-cyclohexylethanone | —— | C20H31N5O2 |
| —— | 1-[(2R)-2-[7-(4-methoxyphenyl)sulfonyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone | —— | C19H25N5O4S |
| —— | [3-(2-fluorophenyl)-1,2-oxazol-5-yl]-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H21FN6O2 |
| —— | 1-[3-(1-Acetylpiperidin-4-yl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-(4-fluorophenyl)ethanone | —— | C21H26FN5O2 |
| —— | 7-(2-Fluoro-5-methylphenyl)sulfonyl-3-piperidin-4-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | 1-[3-[(2S)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-cyclopentylpropan-1-one | —— | C20H31N5O2 |
| —— | 1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenylethanone | —— | C19H25N5O |
| —— | 1-[3-[(2R)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-phenylpropan-1-one | —— | C21H27N5O2 |
| —— | 3-[(2R)-1-(2-chlorophenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22ClN5O2S |
| —— | 2-(4-fluorophenoxy)-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O2 |
| —— | 2-cyclopentyl-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C18H29N5O |
| —— | 3-(2-methylphenoxy)-1-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | (5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H26N6O2 |
| —— | 1-[3-[(2S)-1-(4-methoxyphenyl)sulfonylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H25N5O4S |
| —— | [3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-phenylmethanone | —— | C18H23N5O |
| —— | 2-(4-fluorophenyl)-1-[(2S)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone | —— | C18H22FN5O |
| —— | 1-[3-[(2R)-1-(cyclohexylmethyl)pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H31N5O |
| —— | 7-(4-fluoro-2-methylphenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | 2-(2,4-difluorophenoxy)-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H23F2N5O2 |
| —— | 1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-phenoxyethanone | —— | C19H25N5O2 |
| —— | [3-[2-(dimethylamino)ethoxy]phenyl]-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H30N6O2 |
| —— | 3-(2-methylphenoxy)-1-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one | —— | C22H31N5O2 |
| —— | (3-cyclohexyl-1,2-oxazol-5-yl)-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H30N6O2 |
| —— | [3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-(5-methyl-3-propan-2-yl-1,2-oxazol-4-yl)methanone | —— | C20H30N6O2 |
| —— | 3-[(2S)-1-(2-fluoro-5-methylphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |
| —— | N,N-dimethyl-3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-sulfonamide | —— | C14H26N6O2S |
| —— | (5-cyclopropyl-1,2-oxazol-3-yl)-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C18H24N6O2 |
| —— | 1-[3-[(2R)-1-[(2-fluorophenyl)methyl]pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C19H24FN5O |
| —— | 2-(1H-indol-3-yl)-1-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone | —— | C22H28N6O |
| —— | N-cyclohexyl-N-methyl-2-[3-[(2R)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]acetamide | —— | C19H32N6O |
| —— | 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C22H31N5O |
| —— | N,N-dimethyl-3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-sulfonamide | —— | C14H26N6O2S |
| —— | 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-cyclohexylethanone | —— | C20H31N5O2 |
| —— | 1-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-phenoxyethanone | —— | C20H27N5O2 |
| —— | 1-[2-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-oxoethyl]azepan-2-one | —— | C20H32N6O2 |
| —— | [3-[2-(dimethylamino)ethoxy]phenyl]-[3-[(2S)-pyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H30N6O2 |
| —— | 7-(2-chlorophenyl)sulfonyl-3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C17H22ClN5O2S |
| —— | (3-methoxyphenyl)-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C19H25N5O2 |
| —— | [4-(methoxymethyl)phenyl]-[3-[(2S)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C21H29N5O2 |
| —— | isoquinolin-1-yl-[3-[(2R)-1-methylpiperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C22H26N6O |
| —— | [4-(methoxymethyl)phenyl]-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methanone | —— | C20H27N5O2 |
| —— | 3-[(2R)-1-(2-fluoro-5-methylphenyl)sulfonylpyrrolidin-2-yl]-7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine | —— | C18H24FN5O2S |