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三唑并二氮卓类

中文名称 英文名称 CAS号 化学式
—— (2-phenylmethoxyphenyl)-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methanone —— C23H26N4O2
—— (1-phenylcyclopentyl)-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methanone —— C21H28N4O
—— 1-(2,3-dihydroindol-1-yl)-4-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)butane-1,4-dione —— C21H27N5O2
—— 2-(4-propan-2-yloxyphenyl)-1-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)ethanone —— C20H28N4O2
—— 2-methyl-N-[4-[2-oxo-2-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)ethyl]phenyl]propanamide —— C21H29N5O2
—— 2-(1,3-benzodioxol-5-yl)-1-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)ethanone —— C18H22N4O3
—— N-[4-[2-oxo-2-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)ethyl]phenyl]cyclohexanecarboxamide —— C24H33N5O2
—— 3-(4-cyclopentyloxyphenyl)-1-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)propan-1-one —— C23H32N4O2
—— [1-(4-methoxyphenyl)cyclopentyl]-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)methanone —— C22H30N4O2
—— (3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)-[4-(thiophen-2-ylmethoxy)phenyl]methanone —— C21H24N4O2S
—— 2-(4-phenylmethoxyphenyl)-1-(3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)ethanone —— C24H28N4O2
—— (3-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)-[1-[2-[(2R)-piperidin-2-yl]ethyl]triazol-4-yl]methanone —— C17H26N8O
—— (3-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)-[1-[2-[(2S)-piperidin-2-yl]ethyl]triazol-4-yl]methanone —— C17H26N8O
—— 4-[3-[(2R)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]-1-(3-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)butan-1-one —— C21H29N7O2
—— 4-[3-[(2S)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]-1-(3-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)butan-1-one —— C21H29N7O2
—— (3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)-[(4S)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]methanone —— C16H23N7O
—— (3-propan-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl)-[(4R)-4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridin-4-yl]methanone —— C16H23N7O
—— (3S)-3-[[3-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl]piperidin-3-ol —— C18H26N6O
—— (3R)-3-[[3-(pyridin-3-ylmethyl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl]piperidin-3-ol —— C18H26N6O
—— 2-(4-methoxyphenyl)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C20H27N5O2
—— 3-(4-fluorophenyl)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one —— C20H26FN5O
—— 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-(4-fluorophenoxy)ethanone —— C20H24FN5O3
—— 1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-phenylpropan-1-one —— C20H27N5O
—— 1-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-(4-chlorophenyl)ethanone —— C20H24ClN5O2
—— 3-(4-fluorophenyl)-1-[3-[(2S)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one —— C20H26FN5O
—— 1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-3-phenylpropan-1-one —— C20H27N5O
—— 1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-phenylpropan-1-one —— C20H27N5O
—— 1-[(2S)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-3-phenylpropan-1-one —— C20H27N5O
—— 1-[3-[(2S)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C18H22FN5O3S
—— 1-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]-2-(4-chlorophenyl)ethanone —— C20H24ClN5O2
—— 1-[3-[(2R)-1-(4-fluorophenyl)sulfonylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C18H22FN5O3S
—— 7-[(2-methoxy-4-methylphenyl)methyl]-3-[(2R)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C20H29N5O
—— 1-[(2R)-2-[7-[(3-methylphenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone —— C20H27N5O
—— 7-(2-phenylethyl)-3-[(2R)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H27N5
—— 1-[3-[(2R)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C14H21N5O2
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2S)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C23H33N5O
—— 2-[(2R)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-1-piperidin-1-ylethanone —— C20H32N6O2
—— 2-(1H-indol-3-yl)-1-[3-[(2R)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C21H26N6O
—— 1-[(2S)-2-[7-[(2-methoxy-4-methylphenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone —— C21H29N5O2
—— 1-[(2S)-2-(7-pyrimidin-2-yl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone —— C16H21N7O
—— 7-[(3-cyclopentyloxyphenyl)methyl]-3-[(2R)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C23H33N5O
—— 3-(4-methoxyphenyl)-1-[3-[(2R)-1-methylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]propan-1-one —— C21H29N5O2
—— 7-(2-phenylethyl)-3-[(2S)-piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C19H27N5
—— 1-[(2R)-2-[7-[(2-chlorophenyl)methyl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]pyrrolidin-1-yl]ethanone —— C19H24ClN5O
—— 1-[3-[(2S)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C14H21N5O2
—— 2-[(2S)-2-(7-acetyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)piperidin-1-yl]-1-piperidin-1-ylethanone —— C20H32N6O2
—— 1-[3-[(2S)-1-acetylpyrrolidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-2-cyclohexylethanone —— C20H31N5O2
—— 1-[(2R)-2-(7-methyl-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)pyrrolidin-1-yl]ethanone —— C13H21N5O
—— 1-[3-[(2S)-1-(cyclopropylmethyl)piperidin-2-yl]-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethanone —— C17H27N5O
—— 3-[(2R)-piperidin-2-yl]-7-(quinolin-4-ylmethyl)-5,6,8,9-tetrahydro-[1,2,4]triazolo[4,3-d][1,4]diazepine —— C21H26N6