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—— (R)-2-[3,5-dichloro-4'-(4-trifluoromethyl-piperidine-1-carbonyl)-biphenyl-4-ylmethyl]-5-(1-trifluoromethanesulfonyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-pyrrolidin-2-one 955406-72-1 C32H30Cl2F6N4O4S
(R)-2-[3,5-dichloro-4'-(4-trifluoromethyl-piperidine-1-carbonyl)-biphenyl-4-ylmethyl]-5-(1-trifluoromethanesulfonyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-pyrrolidin-2-one
—— 8-chloromethyl-7-(5-fluoro-2-methoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one 949891-73-0 C18H18ClFN2O2
8-chloromethyl-7-(5-fluoro-2-methoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— phenylmethyl 3-(4-bromo-6-methyl-1H-indazol-1-yl)benzoate 955946-37-9 C22H17BrN2O2
phenylmethyl 3-(4-bromo-6-methyl-1H-indazol-1-yl)benzoate
—— (3R)-3-(3,5-Dichloro-4'-trifluoromethyl-biphenyl-4-ylmethyl)-1-(4,5,6,7-tetrahydro-1H-indazol-4-yl)-pyrrolidin-2-one 955407-77-9 C25H22Cl2F3N3O
(3R)-3-(3,5-Dichloro-4'-trifluoromethyl-biphenyl-4-ylmethyl)-1-(4,5,6,7-tetrahydro-1H-indazol-4-yl)-pyrrolidin-2-one
—— methyl 2-(6-chloro-2,3-dihydro-1H-indol-3-yl)acetate 929005-86-7 C11H12ClNO2
methyl 2-(6-chloro-2,3-dihydro-1H-indol-3-yl)acetate
—— ([1,1'-Biphenyl]-2,2'-diyl)bis[(piperazin-1-yl)methanone] 904958-94-7 C22H26N4O2
([1,1'-Biphenyl]-2,2'-diyl)bis[(piperazin-1-yl)methanone]
—— (R)-[1-(3-fluoro-4-methanesulfonylamino-5-vinylphenyl)ethyl] carbamic acid tert-butyl ester 911124-29-3 C16H23FN2O4S
(R)-[1-(3-fluoro-4-methanesulfonylamino-5-vinylphenyl)ethyl] carbamic acid tert-butyl ester
—— 7-(5-Chloro-2-methoxyphenyl)-8-hydroxymethyl-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one 949892-03-9 C19H21ClN2O3
7-(5-Chloro-2-methoxyphenyl)-8-hydroxymethyl-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— 8-Benzoyloxymethyl-7-(2-methoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one 949888-52-2 C25H24N2O4
8-Benzoyloxymethyl-7-(2-methoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— tert-butyl 3-ethynyl-5-fluoro-4-(methylsulfonamido)benzylcarbamate 911124-11-3 C15H19FN2O4S
tert-butyl 3-ethynyl-5-fluoro-4-(methylsulfonamido)benzylcarbamate
—— (+/-)-ethyl (4-nitro-2-oxo-2,3-dihydro-1H-indol-3-yl)acetate 939036-69-8 C12H12N2O5
(+/-)-ethyl (4-nitro-2-oxo-2,3-dihydro-1H-indol-3-yl)acetate
—— (1R)-2-[{[(1-methylethyl)amino]carbonyl}(4-{[(2-nitrophenyl)sulfonyl]amino}butyl)amino]-1-[(methyloxy)methyl]ethyl phenylcarbamate 929281-16-3 C25H35N5O8S
(1R)-2-[{[(1-methylethyl)amino]carbonyl}(4-{[(2-nitrophenyl)sulfonyl]amino}butyl)amino]-1-[(methyloxy)methyl]ethyl phenylcarbamate
—— 3-[5-(isopropoxycarbonyl)-2-thienyl]propanoic acid 924301-26-8 C11H14O4S
3-[5-(isopropoxycarbonyl)-2-thienyl]propanoic acid
—— 4-oxo-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester 955406-76-5 C12H16N2O3
4-oxo-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester
—— 3-(3,5-dichloro-4'-carboxyl-biphenyl-4-ylmethyl)-1-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-pyrrolidin-2-one 955407-12-2 C25H23Cl2N3O3
3-(3,5-dichloro-4'-carboxyl-biphenyl-4-ylmethyl)-1-(4,5,6,7-tetrahydro-2H-indazol-5-yl)-pyrrolidin-2-one
—— —— 951217-70-2 C64H76N20O4
—— 8-chloromethyl-7-(2-methoxy-4-methoxymethoxyphenyl)-3,3-di methyl-3,4-dihydro-1H-quinoxalin-2-one 949891-74-1 C20H23ClN2O4
8-chloromethyl-7-(2-methoxy-4-methoxymethoxyphenyl)-3,3-di methyl-3,4-dihydro-1H-quinoxalin-2-one
—— methyl 6-[(1S,4S)-2,5-diazabicyclo[2.2.1]hept-2-yl]nicotinate 936706-52-4 C12H15N3O2
methyl 6-[(1S,4S)-2,5-diazabicyclo[2.2.1]hept-2-yl]nicotinate
—— (1R)-2-[{[(1-methylethyl)amino]carbonyl}(4-{[(2-nitrophenyl)sulfonyl]amino}butyl)amino]-1-[(methyloxy)methyl]ethyl phenylcarbamate 929281-28-7 C26H37N5O8S
(1R)-2-[{[(1-methylethyl)amino]carbonyl}(4-{[(2-nitrophenyl)sulfonyl]amino}butyl)amino]-1-[(methyloxy)methyl]ethyl phenylcarbamate
—— 2-[[(cyclohexylamino)carbonyl](4-{[(2,4-dichlorophenyl)sulfonyl]amino}butyl)amino]ethyl phenylcarbamate 929281-32-3 C26H34Cl2N4O5S
2-[[(cyclohexylamino)carbonyl](4-{[(2,4-dichlorophenyl)sulfonyl]amino}butyl)amino]ethyl phenylcarbamate
—— 2-(oxan-2-yloxy)ethyl 4-(4-cyanophenyl)-3-[8-[8-[4-(4-cyanophenyl)-6-methyl-5-[2-(oxan-2-yloxy)ethoxycarbonyl]-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidin-3-yl]octyl-ethylamino]octyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate 904958-57-2 C72H87F6N7O10
2-(oxan-2-yloxy)ethyl 4-(4-cyanophenyl)-3-[8-[8-[4-(4-cyanophenyl)-6-methyl-5-[2-(oxan-2-yloxy)ethoxycarbonyl]-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidin-3-yl]octyl-ethylamino]octyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate
—— [1-(4-ethenesulfonylamino-3-vinylphenyl)ethyl]carbamic acid tert-butyl ester 911124-89-5 C17H24N2O4S
[1-(4-ethenesulfonylamino-3-vinylphenyl)ethyl]carbamic acid tert-butyl ester
—— 7-(2-Methoxy-4-methoxymethoxyphenyl)-8-(5-methylthiophen-2-ylcarbonyloxymethyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one 949888-71-5 C26H28N2O6S
7-(2-Methoxy-4-methoxymethoxyphenyl)-8-(5-methylthiophen-2-ylcarbonyloxymethyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— 5-Bromo-4-[tert-butyl(dimethyl)silyl]oxy-3-methoxy-2-methylbenzaldehyde 905450-25-1 C15H23BrO3Si
5-Bromo-4-[tert-butyl(dimethyl)silyl]oxy-3-methoxy-2-methylbenzaldehyde
—— ethyl (4R)-4-(4-cyanophenyl)-6-methyl-2-oxo-3-(3-oxopropyl)-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate 904959-00-8 C25H22F3N3O4
ethyl (4R)-4-(4-cyanophenyl)-6-methyl-2-oxo-3-(3-oxopropyl)-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate
—— ethyl (4R)-4-(4-cyanophenyl)-3-[3-(1,3-dioxoisoindol-2-yl)propyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate 904958-62-9 C33H27F3N4O5
ethyl (4R)-4-(4-cyanophenyl)-3-[3-(1,3-dioxoisoindol-2-yl)propyl]-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate
—— (R)-4-[3-(2,6-dichloro-4-hydroxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester 955406-87-8 C23H27Cl2N3O4
(R)-4-[3-(2,6-dichloro-4-hydroxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester
—— 3-(benzyloxy)-N-methoxy-5-[(1S)-2-methoxy-1-methylethoxy]-N-methylbenzamide 929614-69-7 C20H25NO5
3-(benzyloxy)-N-methoxy-5-[(1S)-2-methoxy-1-methylethoxy]-N-methylbenzamide
—— tert-butyl [1-(4-ethyl-5-oxo-2,5-dihydro-1H-pyrazol-3-yl)-ethyl]-carbamate 957129-22-5 C12H21N3O3
tert-butyl [1-(4-ethyl-5-oxo-2,5-dihydro-1H-pyrazol-3-yl)-ethyl]-carbamate
—— 4-hydroxy-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester 955406-77-6 C12H18N2O3
4-hydroxy-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester
—— (2S)-2,6-dimethyl-6-triethylsilanyloxyheptanal 928257-65-2 C15H32O2Si
(2S)-2,6-dimethyl-6-triethylsilanyloxyheptanal
—— 8-hydroxymethyl-7-(2-methoxy-4-methoxymethoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one 949891-70-7 C20H24N2O5
8-hydroxymethyl-7-(2-methoxy-4-methoxymethoxyphenyl)-3,3-dimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— (R)-4-[3-(2,6-dichloro-4-hydroxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester 955406-86-7 C23H27Cl2N3O4
(R)-4-[3-(2,6-dichloro-4-hydroxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester
—— (1S,4R,6S,7Z,18R)-N-cyclopropylsulfonyl-18-hydroxy-14-[(4-methoxyphenyl)methyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide 923946-75-2 C28H38N4O7S
(1S,4R,6S,7Z,18R)-N-cyclopropylsulfonyl-18-hydroxy-14-[(4-methoxyphenyl)methyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— 1-[4-(3-chloropropoxy)phenyl]-2-methyl-1H-indole 934840-33-2 C18H18ClNO
1-[4-(3-chloropropoxy)phenyl]-2-methyl-1H-indole
—— (1S,4R,6S,7Z,18R)-18-[tert-butyl(dimethyl)silyl]oxy-14-[(4-methoxyphenyl)methyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid 923946-73-0 C31H47N3O6Si
(1S,4R,6S,7Z,18R)-18-[tert-butyl(dimethyl)silyl]oxy-14-[(4-methoxyphenyl)methyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— 5-(2,5-bis(trimethylsilanylethynyl)-phenoxy)-pyrimidine-2,4-diamine 927872-70-6 C20H26N4OSi2
5-(2,5-bis(trimethylsilanylethynyl)-phenoxy)-pyrimidine-2,4-diamine
—— 4,5,6,7-tetrahydro-2H-indazol-4-ol 955406-79-8 C7H10N2O
4,5,6,7-tetrahydro-2H-indazol-4-ol
—— 1-(1,5-dimethyl-1H-imidazol-2-yl)-2-phenylethanamine 955028-24-7 C13H17N3
1-(1,5-dimethyl-1H-imidazol-2-yl)-2-phenylethanamine
—— 2-[2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidin-7-amine 942590-16-1 C18H20BClN4O2
2-[2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidin-7-amine
—— 2-[1-(4-benzyloxyphenyl)-1H-indol-2-yl]ethanol 934840-39-8 C23H21NO2
2-[1-(4-benzyloxyphenyl)-1H-indol-2-yl]ethanol
—— 5-methyl-2-oxazol-2-yl-phenylamine 923947-66-4 C10H10N2O
5-methyl-2-oxazol-2-yl-phenylamine
—— (R)-4-[3-(2,6-dichloro-4-trifluoromethanesulfonyloxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester 955406-88-9 C24H26Cl2F3N3O6S
(R)-4-[3-(2,6-dichloro-4-trifluoromethanesulfonyloxy-benzyl)-2-oxo-pyrrolidin-1-yl]-4,5,6,7-tetrahydro-indazole-1-carboxylic acid tert-butyl ester
—— 4-hydroxy-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester 955406-78-7 C12H18N2O3
4-hydroxy-4,5,6,7-tetrahydro-indazole-2-carboxylic acid tert-butyl ester
—— 7-(5-Chloro-2-methoxyphenyl)-8-chloromethyl-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one 949892-05-1 C19H20Cl2N2O2
7-(5-Chloro-2-methoxyphenyl)-8-chloromethyl-1,3,3-trimethyl-3,4-dihydro-1H-quinoxalin-2-one
—— Ethyl 3-(4-cyanophenyl)-2-(2-methyl-1,3-dioxolan-2-yl)-3-(prop-2-enoxycarbonylamino)propanoate 904959-13-3 C20H24N2O6
Ethyl 3-(4-cyanophenyl)-2-(2-methyl-1,3-dioxolan-2-yl)-3-(prop-2-enoxycarbonylamino)propanoate
—— Methyl (3-{[(3-[(4-{[6-amino-8-methoxy-2-(2-methoxyethoxy)-9H-purin-9-yl]methyl}benzyl)(methyl)amino]propyl}(tert-butoxycarbonyl)amino]methyl}phenyl)acetate 930785-45-8 C36H49N7O7
Methyl (3-{[(3-[(4-{[6-amino-8-methoxy-2-(2-methoxyethoxy)-9H-purin-9-yl]methyl}benzyl)(methyl)amino]propyl}(tert-butoxycarbonyl)amino]methyl}phenyl)acetate
—— ethyl (4R)-3-(3-aminopropyl)-4-(4-cyanophenyl)-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate 904958-63-0 C25H25F3N4O3
ethyl (4R)-3-(3-aminopropyl)-4-(4-cyanophenyl)-6-methyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-4H-pyrimidine-5-carboxylate
—— 2-(4-tert-Butyl-phenyl)-4-piperazin-1-yl-benzooxazole 915135-24-9 C21H25N3O
2-(4-tert-Butyl-phenyl)-4-piperazin-1-yl-benzooxazole
—— [5-Bromo-4-[tert-butyl(dimethyl)silyl]oxy-3-methoxy-2-methylphenyl] 4-methylbenzenesulfonate 905450-28-4 C21H29BrO5SSi
[5-Bromo-4-[tert-butyl(dimethyl)silyl]oxy-3-methoxy-2-methylphenyl] 4-methylbenzenesulfonate