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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-((2-bromo-4-(1-tert-butoxy-1-oxopropan-2-yl)phenylamino)methyl)benzoic acid 950741-87-4 C21H24BrNO4
2-((2-bromo-4-(1-tert-butoxy-1-oxopropan-2-yl)phenylamino)methyl)benzoic acid
—— 2-(isopropylamino)thiazolo[4,5-c]pyridine-6-carbaldehyde 924287-79-6 C10H11N3OS
2-(isopropylamino)thiazolo[4,5-c]pyridine-6-carbaldehyde
—— (R)-3-acetyl-5-((1-phenylethyl)carbamoyl)benzoic acid 924650-34-0 C18H17NO4
(R)-3-acetyl-5-((1-phenylethyl)carbamoyl)benzoic acid
—— N-butyryl-N-[(2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl)methyl]-L-valine 934736-49-9 C24H27N3O5
N-butyryl-N-[(2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl)methyl]-L-valine
—— tert-butyl N-[(2R,3S)-3-[[3-acetyl-5-[[(1R)-1-phenylethyl]carbamoyl]benzoyl]amino]-4-(3,5-difluorophenyl)-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate 924650-35-1 C41H45F2N3O7
tert-butyl N-[(2R,3S)-3-[[3-acetyl-5-[[(1R)-1-phenylethyl]carbamoyl]benzoyl]amino]-4-(3,5-difluorophenyl)-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate
—— N-valeryl-N-[(2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl)methyl]-L-valine 934736-50-2 C25H29N3O5
N-valeryl-N-[(2'-(4,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl)biphenyl-4-yl)methyl]-L-valine
—— tert-butyl 3-methoxybenzyl((2R,3S)-3-(3-acetyl-5-(N-methylmethan-2-ylsulfonamido)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate 924650-20-4 C34H41F2N3O8S
tert-butyl 3-methoxybenzyl((2R,3S)-3-(3-acetyl-5-(N-methylmethan-2-ylsulfonamido)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate
—— tert-butyl {6-[3-(tert-butyldimethylsilanyloxy)-2-hydroxypropyl]-5-chloropyrazolo[1,5-a]pyrimidin-7-yl}(4-ethoxyphenyl)carbamate 910214-23-2 C28H41ClN4O5Si
tert-butyl {6-[3-(tert-butyldimethylsilanyloxy)-2-hydroxypropyl]-5-chloropyrazolo[1,5-a]pyrimidin-7-yl}(4-ethoxyphenyl)carbamate
—— 5-Chloro-4-(hexylamino)-2-phenylpyridazin-3(2H)-one 923027-35-4 C16H20ClN3O
5-Chloro-4-(hexylamino)-2-phenylpyridazin-3(2H)-one
—— [(2R,3S)-3-{3-Acetyl-5-[1-(4-fluoro-phenyl)-ethylcarbamoyl]-benzoylamino}-4-(3,5-difluoro-phenyl)-2-hydroxy-butyl]-(3-methoxy-benzyl)-carbamic acid tert-butyl ester 924650-40-8 C41H44F3N3O7
[(2R,3S)-3-{3-Acetyl-5-[1-(4-fluoro-phenyl)-ethylcarbamoyl]-benzoylamino}-4-(3,5-difluoro-phenyl)-2-hydroxy-butyl]-(3-methoxy-benzyl)-carbamic acid tert-butyl ester
—— ethyl (2E)-4-(1-azabicyclo[3.2.1]oct-5-yl)-4-oxobut-2-enoate 926910-87-4 C13H19NO3
ethyl (2E)-4-(1-azabicyclo[3.2.1]oct-5-yl)-4-oxobut-2-enoate
—— tert-butyl [5-chloro-6-(3-oxopropyl)pyrazolo[1,5-a]pyrimidin-7-yl]-(4-ethoxyphenyl)carbamate 910214-21-0 C22H25ClN4O4
tert-butyl [5-chloro-6-(3-oxopropyl)pyrazolo[1,5-a]pyrimidin-7-yl]-(4-ethoxyphenyl)carbamate
—— 13-Amino-5-cyclohexyl-12-nitro-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one 902745-62-4 C15H15N5O3S
13-Amino-5-cyclohexyl-12-nitro-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
—— tert-butyl (S)-3-[7-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6-(2-methanesulfonyloxyethyl)pyrazolo[1,5-a]pyrimidin-5-ylamino]piperidine-1-carboxylate 910214-15-2 C33H48N6O9S
tert-butyl (S)-3-[7-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6-(2-methanesulfonyloxyethyl)pyrazolo[1,5-a]pyrimidin-5-ylamino]piperidine-1-carboxylate
—— 2-(5,7-dichloropyrazolo[1,5-a]pyrimidin-6-yl)ethanol 910214-11-8 C8H7Cl2N3O
2-(5,7-dichloropyrazolo[1,5-a]pyrimidin-6-yl)ethanol
—— 6-[2-(tert-butyldimethylsilanyloxy)ethyl]-5,7-dichloropyrazolo[1,5-a]pyrimidine 910214-12-9 C14H21Cl2N3OSi
6-[2-(tert-butyldimethylsilanyloxy)ethyl]-5,7-dichloropyrazolo[1,5-a]pyrimidine
—— tert-butyl (S)-3-{7-[tert-butoxycarbonyl-(4-ethoxyphenyl)amino]-6-[3-(tert-butyldimethylsilanyloxy)-2-hydroxypropyl]pyrazolo[1,5-a]pyrimidin-5-ylamino}piperidine-1-carboxylate 910214-29-8 C38H60N6O7Si
tert-butyl (S)-3-{7-[tert-butoxycarbonyl-(4-ethoxyphenyl)amino]-6-[3-(tert-butyldimethylsilanyloxy)-2-hydroxypropyl]pyrazolo[1,5-a]pyrimidin-5-ylamino}piperidine-1-carboxylate
—— 5-(2-Bromo-1,3-benzothiazol-6-yl)-4-phenyl-1,3-oxazole 924287-05-8 C16H9BrN2OS
5-(2-Bromo-1,3-benzothiazol-6-yl)-4-phenyl-1,3-oxazole
—— 2-(isopropylamino)thiazolo[4,5-b]pyridine-6-carbaldehyde 924287-75-2 C10H11N3OS
2-(isopropylamino)thiazolo[4,5-b]pyridine-6-carbaldehyde
—— 13-cyclohexyl-N-[(morpholin-4-yl)sulfonyl]-6-carboxy-7H-indolo[2,1-a][2]benzazepine-10-carboxamide 929629-08-3 C29H31N3O6S
13-cyclohexyl-N-[(morpholin-4-yl)sulfonyl]-6-carboxy-7H-indolo[2,1-a][2]benzazepine-10-carboxamide
—— [(2R,3S)-3-[3-acetyl-5-(1,1-dioxo-1λ6-[1,2]thiazinan-2-yl)-benzoylamino]-4-(3,5-difluoro-phenyl)-2-hydroxy-butyl]-(3-methoxy-benzyl)-carbamic acid tert-butyl ester 924650-15-7 C36H43F2N3O8S
[(2R,3S)-3-[3-acetyl-5-(1,1-dioxo-1λ6-[1,2]thiazinan-2-yl)-benzoylamino]-4-(3,5-difluoro-phenyl)-2-hydroxy-butyl]-(3-methoxy-benzyl)-carbamic acid tert-butyl ester
—— tert-butyl (S)-3-(8-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6,7-dihydro-1,4,5,8a-tetraaza-s-indacen-5-yl)piperidine-1-carboxylate 910214-34-5 C32H44N6O6
tert-butyl (S)-3-(8-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6,7-dihydro-1,4,5,8a-tetraaza-s-indacen-5-yl)piperidine-1-carboxylate
—— 1-(6-chloropyridazin-3-yl)-1-(2,6-difluorophenyl)but-3-yn-2-one 940891-91-8 C14H7ClF2N2O
1-(6-chloropyridazin-3-yl)-1-(2,6-difluorophenyl)but-3-yn-2-one
—— 4-(2-Methylsulfanyl-4,5-diphenylimidazol-1-yl)phenol 902780-91-0 C22H18N2OS
4-(2-Methylsulfanyl-4,5-diphenylimidazol-1-yl)phenol
—— tert-butyl (S)-3-[7-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-5-ylamino]piperidine-1-carboxylate 910214-14-1 C32H46N6O7
tert-butyl (S)-3-[7-{tert-butoxycarbonyl-[4-(2-methoxyethoxy)phenyl]amino}-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-5-ylamino]piperidine-1-carboxylate
—— 3-bromo-5-(thien-3-yl)benzonitrile 914484-77-8 C11H6BrNS
3-bromo-5-(thien-3-yl)benzonitrile
—— tert-butyl [5-chloro-6-(2,3-dihydroxypropyl)pyrazolo[1,5-a]pyrimidin-7-yl](4-ethoxyphenyl)carbamate 910214-22-1 C22H27ClN4O5
tert-butyl [5-chloro-6-(2,3-dihydroxypropyl)pyrazolo[1,5-a]pyrimidin-7-yl](4-ethoxyphenyl)carbamate
—— tert-butyl [5-chloro-6-(2-oxoethyl)pyrazolo[1,5-a]pyrimidin-7-yl](4-ethoxyphenyl)carbamate 910214-19-6 C21H23ClN4O4
tert-butyl [5-chloro-6-(2-oxoethyl)pyrazolo[1,5-a]pyrimidin-7-yl](4-ethoxyphenyl)carbamate
—— 3-acetyl-5-((1-(4-fluorophenyl)ethyl)carbamoyl)benzoic acid 924650-39-5 C18H16FNO4
3-acetyl-5-((1-(4-fluorophenyl)ethyl)carbamoyl)benzoic acid
—— tert-butyl 3-methoxybenzyl((2R,3S)-3-(3-acetyl-5-(N-phenylmethan-10-ylsulfonamido)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate 924650-29-3 C39H43F2N3O8S
tert-butyl 3-methoxybenzyl((2R,3S)-3-(3-acetyl-5-(N-phenylmethan-10-ylsulfonamido)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate
—— 3-(4-Phenoxyphenyl)sulfonylpropane-1,2-diol 915156-52-4 C15H16O5S
3-(4-Phenoxyphenyl)sulfonylpropane-1,2-diol
—— {(2R,3S)-4-(3,5-difluoro-phenyl)-3-[3-(1,1-dioxo-1λ6-[1,2]thiazinan-2-yl)-5-(1-hydroxy-ethyl)-benzoylamino]-2-hydroxy-butyl}-(3-methoxy-benzyl)-carbamic acid tert-butyl ester 924650-16-8 C36H45F2N3O8S
{(2R,3S)-4-(3,5-difluoro-phenyl)-3-[3-(1,1-dioxo-1λ6-[1,2]thiazinan-2-yl)-5-(1-hydroxy-ethyl)-benzoylamino]-2-hydroxy-butyl}-(3-methoxy-benzyl)-carbamic acid tert-butyl ester
—— 2-(isopropylamino)benzo[d]thiazole-6-carbaldehyde 924288-01-7 C11H12N2OS
2-(isopropylamino)benzo[d]thiazole-6-carbaldehyde
—— ethyl 4-(1-azabicyclo[3.2.1]oct-5-yl)-4-oxobutanoate 926910-88-5 C13H21NO3
ethyl 4-(1-azabicyclo[3.2.1]oct-5-yl)-4-oxobutanoate
—— 3-acetyl-5-(dipropylcarbamoyl)benzoic acid 924650-02-2 C16H21NO4
3-acetyl-5-(dipropylcarbamoyl)benzoic acid
—— (2-Bromo-4-fluorobenzo[d]thiazol-6-yl)methanol 924287-66-1 C8H5BrFNOS
(2-Bromo-4-fluorobenzo[d]thiazol-6-yl)methanol
—— tert-butyl N-[(2R,3S)-4-(3,5-difluorophenyl)-2-hydroxy-3-[[3-[(E)-N-hydroxy-C-methylcarbonimidoyl]-5-[methyl(propyl)carbamoyl]benzoyl]amino]butyl]-N-[(3-methoxyphenyl)methyl]carbamate 924650-08-8 C37H46F2N4O7
tert-butyl N-[(2R,3S)-4-(3,5-difluorophenyl)-2-hydroxy-3-[[3-[(E)-N-hydroxy-C-methylcarbonimidoyl]-5-[methyl(propyl)carbamoyl]benzoyl]amino]butyl]-N-[(3-methoxyphenyl)methyl]carbamate
—— N-(2,2-Dimethylpropyl)-3,3-dimethyl-1-butanamine 951160-87-5 C11H25N
N-(2,2-Dimethylpropyl)-3,3-dimethyl-1-butanamine
—— DPEphos 923039-20-7 C36H28P2S
DPEphos
—— tert-butyl 3-methoxybenzyl(2R,3S)-3-(3-(benzamido)-5-(1-(hydroxyethyl)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate 924650-09-9 C37H47F2N3O7
tert-butyl 3-methoxybenzyl(2R,3S)-3-(3-(benzamido)-5-(1-(hydroxyethyl)benzamido)-4-(3,5-difluorophenyl)-2-hydroxybutyl)carbamate
—— tert-butyl 4-[2-(6-methoxy-3-oxo-1H-isoindol-2-yl)acetyl]piperidine-1-carboxylate 916450-86-7 C21H28N2O5
tert-butyl 4-[2-(6-methoxy-3-oxo-1H-isoindol-2-yl)acetyl]piperidine-1-carboxylate
—— 3-acetyl-5-(N-phenylmethan-10-ylsulfonamido)benzoic acid 924650-26-0 C16H15NO5S
3-acetyl-5-(N-phenylmethan-10-ylsulfonamido)benzoic acid
—— tert-butyl N-[(2R,3S)-3-[[3-acetyl-5-(dipropylcarbamoyl)benzoyl]amino]-4-(3,5-difluorophenyl)-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate 924650-03-3 C39H49F2N3O7
tert-butyl N-[(2R,3S)-3-[[3-acetyl-5-(dipropylcarbamoyl)benzoyl]amino]-4-(3,5-difluorophenyl)-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate
—— ethyl 4-(4-hydroxy-6-oxo-1H-pyrimidin-5-yl)butanoate 905085-69-0 C10H14N2O4
ethyl 4-(4-hydroxy-6-oxo-1H-pyrimidin-5-yl)butanoate
—— N-methyl-1-(1,3-thiazol-2-yl)propan-2-amine 92932-27-9 C7H12N2S
N-methyl-1-(1,3-thiazol-2-yl)propan-2-amine
—— tert-butyl N-[(2R,3S)-4-(3,5-difluorophenyl)-3-[[3-(dipropylcarbamoyl)-5-[(E)-N-hydroxy-C-methylcarbonimidoyl]benzoyl]amino]-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate 924650-05-5 C39H50F2N4O7
tert-butyl N-[(2R,3S)-4-(3,5-difluorophenyl)-3-[[3-(dipropylcarbamoyl)-5-[(E)-N-hydroxy-C-methylcarbonimidoyl]benzoyl]amino]-2-hydroxybutyl]-N-[(3-methoxyphenyl)methyl]carbamate
—— 6-(1-azabicyclo[3.2.1]oct-5-yl)-4,5-dihydropyridazin-3-ol 926910-89-6 C11H17N3O
6-(1-azabicyclo[3.2.1]oct-5-yl)-4,5-dihydropyridazin-3-ol
—— 4-(4-bromo-3-methoxyphenyl)-1H-pyrazine-2,3-dione 942910-26-1 C11H9BrN2O3
4-(4-bromo-3-methoxyphenyl)-1H-pyrazine-2,3-dione
—— tert-butyl 3-methoxybenzyl((2R,3S)-4-(3,5-difluorophenyl)-2-hydroxy-3-(3-(1-hydroxyethyl)-5-(N-methylmethan-2-ylsulfonamido)benzamido)butyl)carbamate 924650-21-5 C34H43F2N3O8S
tert-butyl 3-methoxybenzyl((2R,3S)-4-(3,5-difluorophenyl)-2-hydroxy-3-(3-(1-hydroxyethyl)-5-(N-methylmethan-2-ylsulfonamido)benzamido)butyl)carbamate
—— Methyl 2-[4-[[ethyl-[(3-methylbenzotriazol-5-yl)methyl]amino]methyl]piperidin-1-yl]pyrimidine-5-carboxylate 944556-18-7 C22H29N7O2
Methyl 2-[4-[[ethyl-[(3-methylbenzotriazol-5-yl)methyl]amino]methyl]piperidin-1-yl]pyrimidine-5-carboxylate