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—— 3-{2-methoxy-4-[4-methyl-3-oxy-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-phenyl}-4H-[1,2,4]oxadiazol-5-one 933772-91-9 C21H16F3N3O5S
3-{2-methoxy-4-[4-methyl-3-oxy-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— N-[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]-7-(5-piperidin-1-ylpent-2-ynoyl)-5,6,7,8-tetrahydropyrido[4',3':4,5]-thieno[2,3-d]pyrimidin-4-amine 951034-55-2 C31H31ClN6O2S
N-[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]-7-(5-piperidin-1-ylpent-2-ynoyl)-5,6,7,8-tetrahydropyrido[4',3':4,5]-thieno[2,3-d]pyrimidin-4-amine
—— 4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazole-5-carboxylic acid 933772-47-5 C14H9F6NO4
4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazole-5-carboxylic acid
—— 2-pentyl-2H-pyrazolo[3,4-d]pyrimidine-4,6-diol 959432-66-7 C10H14N4O2
2-pentyl-2H-pyrazolo[3,4-d]pyrimidine-4,6-diol
—— 3-(3-fluoro-4-hydroxy-5-methoxy-phenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one 910814-29-8 C21H23FO3S
3-(3-fluoro-4-hydroxy-5-methoxy-phenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one
—— 4-(2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)thiazol-2-amine 956393-37-6 C13H12ClN5OS2
4-(2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)thiazol-2-amine
—— 3,5-diamino-6-chloropyrazine-2-carbothioamide 952751-46-1 C5H6ClN5S
3,5-diamino-6-chloropyrazine-2-carbothioamide
—— 5-(pyridin-3-yl)benzofuran-2-ylboronic acid 939050-30-3 C13H10BNO3
5-(pyridin-3-yl)benzofuran-2-ylboronic acid
—— ethyl 3-ureidofuran-2-carboxylate 956034-05-2 C8H10N2O4
ethyl 3-ureidofuran-2-carboxylate
—— 6-(4-trifluoromethyl-benzylamino)-pyridine-3-carbaldehyde 923562-77-0 C14H11F3N2O
6-(4-trifluoromethyl-benzylamino)-pyridine-3-carbaldehyde
—— N-{4-[(1R)-1-aminoethyl]-2,6-difluorophenyl}methanesulfonamide 957103-01-4 C9H12F2N2O2S
N-{4-[(1R)-1-aminoethyl]-2,6-difluorophenyl}methanesulfonamide
—— {4-[(4-benzyloxycarbonylamino)phenoxy]pyridin-2-yl}carbamic acid tert-butyl ester 928038-15-7 C24H25N3O5
{4-[(4-benzyloxycarbonylamino)phenoxy]pyridin-2-yl}carbamic acid tert-butyl ester
—— 4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-N-hydroxy-2-methoxy-benzamidine 933772-84-0 C29H28F3N3O4S
4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-N-hydroxy-2-methoxy-benzamidine
—— 3-{4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-phenyl}-4H-[1,2,4]oxadiazol-5-one 933773-18-3 C29H23F4N3O4S
3-{4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— N-[3-(2-chloro-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl)phenyl]propane-2-sulfonamide 956388-20-8 C19H21ClN4O3S2
N-[3-(2-chloro-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl)phenyl]propane-2-sulfonamide
—— 3-{4-[4-azidomethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-phenyl}-4H-[1,2,4]oxadiazol-5-one 933773-10-5 C20H12F4N6O3S
3-{4-[4-azidomethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— 4-[4-(benzyloxycarbonylamino)phenoxy]pyridine-2-carboxylic acid 928038-14-6 C20H16N2O5
4-[4-(benzyloxycarbonylamino)phenoxy]pyridine-2-carboxylic acid
—— 2-(1,3-oxazol-2-yl)-3,4'-bipyridin-5,6-diamine 933998-70-0 C13H11N5O
2-(1,3-oxazol-2-yl)-3,4'-bipyridin-5,6-diamine
—— {5-[[5-(2-morpholin-4-yl)-ethoxy]-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl]-pyridin-2-yl}-(4-trifluoromethyl-benzyl)-amine 923562-21-4 C27H28F3N5O2
{5-[[5-(2-morpholin-4-yl)-ethoxy]-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl]-pyridin-2-yl}-(4-trifluoromethyl-benzyl)-amine
—— 3-(4-dimethylamino-2-methoxyphenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one 910813-79-5 C23H29NO2S
3-(4-dimethylamino-2-methoxyphenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one
—— 5-chloromethyl-4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazole 933772-49-7 C14H10ClF6NO2
5-chloromethyl-4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazole
—— 3-amino-1-pentyl-1H-pyrazole-4-caroboxylic acid amide 959432-64-5 C9H16N4O
3-amino-1-pentyl-1H-pyrazole-4-caroboxylic acid amide
—— diethyl-[2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-ethyl]-amine 918523-69-0 C13H19N3O
diethyl-[2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)-ethyl]-amine
—— 4,6-dichloro-2-pentyl-2H-pyrazolo[3,4-d]pyrimidine 959432-67-8 C10H12Cl2N4
4,6-dichloro-2-pentyl-2H-pyrazolo[3,4-d]pyrimidine
—— 4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-benzonitrile 933773-16-1 C28H22F4N2O2S
4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-fluoro-benzonitrile
—— 2-(2-Chloro-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl)ethanol 956388-24-2 C12H14ClN3O2S
2-(2-Chloro-4-morpholin-4-ylthieno[3,2-d]pyrimidin-6-yl)ethanol
—— (2E)-3-{1-[(4-bromophenyl)sulfonyl]-1H-indol-2-yl}acrylic acid 948581-74-6 C17H12BrNO4S
(2E)-3-{1-[(4-bromophenyl)sulfonyl]-1H-indol-2-yl}acrylic acid
—— 5-[[2-[(18S,25S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-methylamino]-5-oxopentanoic acid 960061-84-1 C53H53N13O10S6
5-[[2-[(18S,25S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-methylamino]-5-oxopentanoic acid
—— 3-{4-[4-hydroxymethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-methoxy-phenyl}-4H-[1,2,4]oxadiazol-5-one 933772-94-2 C21H16F3N3O5S
3-{4-[4-hydroxymethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-methoxy-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— 4-[4-hydroxymethyl-2-(4-methoxy-phenyl)-oxazol-5-ylmethoxy]-2-methyl-benzonitrile 933773-03-6 C20H18N2O4
4-[4-hydroxymethyl-2-(4-methoxy-phenyl)-oxazol-5-ylmethoxy]-2-methyl-benzonitrile
—— (5-{hydroxy-[5-(2-morpholin-4-yl-ethoxy)-1H-pyrrolo[2,3-b]pyridin-3-yl]-methyl}-pyridin-2-yl)-(4-trifluoromethyl-benzyl)-carbamic acid tert-butyl ester 923562-78-1 C32H36F3N5O5
(5-{hydroxy-[5-(2-morpholin-4-yl-ethoxy)-1H-pyrrolo[2,3-b]pyridin-3-yl]-methyl}-pyridin-2-yl)-(4-trifluoromethyl-benzyl)-carbamic acid tert-butyl ester
—— N,N-Dimethyl-5-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]pyridin-2-amine 918517-14-3 C15H16N4
N,N-Dimethyl-5-[(1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]pyridin-2-amine
—— (2S)-5-amino-6-(2-aminoethyl)-1,3-dihydrohydrospiro[indeno-2,3'-pyrrolo[2,3-b]pyridin]-2'(1H')-one 938460-92-5 C17H18N4O
(2S)-5-amino-6-(2-aminoethyl)-1,3-dihydrohydrospiro[indeno-2,3'-pyrrolo[2,3-b]pyridin]-2'(1H')-one
—— 3-{4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-methoxy-phenyl}-4H-[1,2,4]oxadiazol-5-one 933772-85-1 C30H26F3N3O5S
3-{4-[4-(3-benzyloxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-2-methoxy-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— N-(4-(hydroxy(7-(methyloxy)-4-quinolinyl)methyl)phenyl)-5-methyl-3-oxo-2-phenyl-1-propyl-2,3-dihydro-1H-pyrazole-4-carboxamide 913377-88-5 C31H30N4O4
N-(4-(hydroxy(7-(methyloxy)-4-quinolinyl)methyl)phenyl)-5-methyl-3-oxo-2-phenyl-1-propyl-2,3-dihydro-1H-pyrazole-4-carboxamide
—— 3-nitro-6-(1,3-oxazol-2-yl)pyridin-2-amine 933998-72-2 C8H6N4O3
3-nitro-6-(1,3-oxazol-2-yl)pyridin-2-amine
—— (5-formyl-pyridin-2-yl)-(4-trifluoromethyl-benzyl)-carbamic acid tert-butyl ester 923562-50-9 C19H19F3N2O3
(5-formyl-pyridin-2-yl)-(4-trifluoromethyl-benzyl)-carbamic acid tert-butyl ester
—— tert-butyl 3-(6-(5-cyclopentylbenzofuran-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate 939050-87-0 C29H35NO3
tert-butyl 3-(6-(5-cyclopentylbenzofuran-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate
—— 3-{2-fluoro-4-[4-(3-hydroxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-phenyl}-4H-[1,2,4]oxadiazol-5-one 933773-19-4 C22H17F4N3O4S
3-{2-fluoro-4-[4-(3-hydroxy-propyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-phenyl}-4H-[1,2,4]oxadiazol-5-one
—— 3-(4-dimethylamino-phenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one 910813-77-3 C22H27NOS
3-(4-dimethylamino-phenyl)-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one
—— tert-butyl N-[2-[(18S,25S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-N-methylcarbamate 960061-85-2 C53H55N13O9S6
tert-butyl N-[2-[(18S,25S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-N-methylcarbamate
—— 3-[4-(2,3-dihydroxy-propyl)-3,5-dimethyl-phenyl]-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one 910811-41-5 C25H32O3S
3-[4-(2,3-dihydroxy-propyl)-3,5-dimethyl-phenyl]-1-((1aS,5aR)-1,1,2-trimethyl-1,1a,5,5a-tetrahydro-3-thia-cyclopropa[a]pentalen-4-yl)-propan-1-one
—— [4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazol-5-yl]-methanol 933772-48-6 C14H11F6NO3
[4-(2,2,2-trifluoro-ethoxymethyl)-2-(4-trifluoromethyl-phenyl)-oxazol-5-yl]-methanol
—— 2-methyl-4-[4-(tetrahydro-pyran-2-yloxymethyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-benzonitrile 933772-97-5 C25H23F3N2O3S
2-methyl-4-[4-(tetrahydro-pyran-2-yloxymethyl)-2-(4-trifluoromethyl-phenyl)-thiazol-5-ylmethoxy]-benzonitrile
—— [4-morpholin-4-ylmethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-yl]-methanol 933772-27-1 C16H17F3N2O2S
[4-morpholin-4-ylmethyl-2-(4-trifluoromethyl-phenyl)-thiazol-5-yl]-methanol
—— 1-allyl-3-amino-1H-pyrazole-4-carboxylic acid amide 959430-10-5 C7H10N4O
1-allyl-3-amino-1H-pyrazole-4-carboxylic acid amide
—— 4-bromomethyl-2-(4-trifluoromethyl-phenyl)-oxazole-5-carboxylic acid ethyl ester 933772-45-3 C14H11BrF3NO3
4-bromomethyl-2-(4-trifluoromethyl-phenyl)-oxazole-5-carboxylic acid ethyl ester
—— tert-butyl 3-(6-(trifluoromethylsulfonyloxy)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate 939050-85-8 C17H22F3NO5S
tert-butyl 3-(6-(trifluoromethylsulfonyloxy)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate
—— [4-difluoromethyl-2-(4-methoxy-phenyl)-thiazol-5-yl]-methanol 933772-63-5 C12H11F2NO2S
[4-difluoromethyl-2-(4-methoxy-phenyl)-thiazol-5-yl]-methanol
—— tert-butyl 3-(6-(5-benzylbenzofuran-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate 939050-67-6 C31H33NO3
tert-butyl 3-(6-(5-benzylbenzofuran-2-yl)-3,4-dihydroisoquinolin-2(1H)-yl)propanoate