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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S-{1S-[2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidine-1-carbonyl]-2-methyl-propylcarbamoyl}-ethyl)-carbamic acid tert-butyl ester 874774-44-4 C28H40N4O5
(1S-{1S-[2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidine-1-carbonyl]-2-methyl-propylcarbamoyl}-ethyl)-carbamic acid tert-butyl ester
—— (S)-N4-[3-chloro-4-(thiazol-2-ylmethoxy)-phenyl]-N6-(4-methyl-4,5-dihydro-oxazol-2-yl)-quinazoline-4,6-diamine 845272-22-2 C22H19ClN6O2S
(S)-N4-[3-chloro-4-(thiazol-2-ylmethoxy)-phenyl]-N6-(4-methyl-4,5-dihydro-oxazol-2-yl)-quinazoline-4,6-diamine
—— (3S,9S)-3-amino-18,23-dioxa-5-azapentacyclo[22.2.2.05,9.011,19.012,17]octacosa-1(27),11(19),12,14,16,24(28),25-heptaen-4-one 874774-27-3 C25H28N2O3
(3S,9S)-3-amino-18,23-dioxa-5-azapentacyclo[22.2.2.05,9.011,19.012,17]octacosa-1(27),11(19),12,14,16,24(28),25-heptaen-4-one
—— 4-(4-chloro-phenyl)-4-{[3-(2,4-dimethoxy-benzyl)-4-oxo-3,4-dihydro-quinazolin-7-ylamino]-methyl}-piperidine-1-carboxylic acid tert-butyl ester 887129-10-4 C34H39ClN4O5
4-(4-chloro-phenyl)-4-{[3-(2,4-dimethoxy-benzyl)-4-oxo-3,4-dihydro-quinazolin-7-ylamino]-methyl}-piperidine-1-carboxylic acid tert-butyl ester
—— 6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-3-pyrrolidin-2-ylmethyl-1H-indole 874774-60-4 C20H29FN2O3
6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-3-pyrrolidin-2-ylmethyl-1H-indole
—— (3-Bromo-4-fluorophenyl)-(1,4,5,6-tetrahydropyrimidin-2-yl)-[4-(trifluoromethoxy)phenyl]methanol 871942-14-2 C18H15BrF4N2O2
(3-Bromo-4-fluorophenyl)-(1,4,5,6-tetrahydropyrimidin-2-yl)-[4-(trifluoromethoxy)phenyl]methanol
—— trans-2S-amino-1-{2S-[3-(2-ethyl-phenoxy)-propenyl]-4S-phenoxy-pyrrolidin-1-yl}-3-methyl-butan-1-one 874773-28-1 C26H34N2O3
trans-2S-amino-1-{2S-[3-(2-ethyl-phenoxy)-propenyl]-4S-phenoxy-pyrrolidin-1-yl}-3-methyl-butan-1-one
—— tert-butyl N-[8-[3-(2-fluoropyridin-3-yl)phenyl]-8-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-imidazo[1,5-a]pyrimidin-6-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 871942-45-9 C34H35F4N5O5
tert-butyl N-[8-[3-(2-fluoropyridin-3-yl)phenyl]-8-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-imidazo[1,5-a]pyrimidin-6-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— 2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester 874773-78-1 C18H22BrNO3
2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester
—— benzyl 4-(4-bromobenzenesulfonyl)piperidine-1-carboxylate 867331-39-3 C19H20BrNO4S
benzyl 4-(4-bromobenzenesulfonyl)piperidine-1-carboxylate
—— 7-(2,6-Dimethylphenyl)-N-[2-(4-methyl-1-piperazinyl)ethyl]-1,2,4-benzotriazin-3-amine 867333-44-6 C22H28N6
7-(2,6-Dimethylphenyl)-N-[2-(4-methyl-1-piperazinyl)ethyl]-1,2,4-benzotriazin-3-amine
—— 3-Benzyl-3-azabicyclo[3.2.1]octan-6-ol 833458-91-6 C14H19NO
3-Benzyl-3-azabicyclo[3.2.1]octan-6-ol
—— 2S-amino-1-(2S-benzofuran-3-ylmethyl-pyrrolidin-1-yl)-3-methyl-butan-1-one 874773-56-5 C18H24N2O2
2S-amino-1-(2S-benzofuran-3-ylmethyl-pyrrolidin-1-yl)-3-methyl-butan-1-one
—— 4-[5-amino-7-(2,6-dimethyl-phenyl)-benzo[1,2,4]triazin-3-ylamino]-N-(2-pyrrolidin-1-yl-ethyl)-benzenesulfonamide 867331-01-9 C27H31N7O2S
4-[5-amino-7-(2,6-dimethyl-phenyl)-benzo[1,2,4]triazin-3-ylamino]-N-(2-pyrrolidin-1-yl-ethyl)-benzenesulfonamide
—— 3-cyclopentyl-3-hydroxy-2-oxo-propionic acid ethyl ester 811467-30-8 C10H16O4
3-cyclopentyl-3-hydroxy-2-oxo-propionic acid ethyl ester
—— tert-butyl N-[(3S,9S)-4-oxo-18,23-dioxa-5-azapentacyclo[22.2.2.05,9.011,19.012,17]octacosa-1(27),11(19),12,14,16,24(28),25-heptaen-3-yl]carbamate 874774-25-1 C30H36N2O5
tert-butyl N-[(3S,9S)-4-oxo-18,23-dioxa-5-azapentacyclo[22.2.2.05,9.011,19.012,17]octacosa-1(27),11(19),12,14,16,24(28),25-heptaen-3-yl]carbamate
—— 1-{4-[3-(2,2-dimethylpyrrolidin-1-yl)propoxy]phenyl}-cyclohexanecarbonitrile 868849-27-8 C22H32N2O
1-{4-[3-(2,2-dimethylpyrrolidin-1-yl)propoxy]phenyl}-cyclohexanecarbonitrile
—— (6aR,8R,9aR)-8-(4-chloro-5-fluoropyrrolo[2,3-d]pyrimidin-7-yl)-2,2,4,4-tetra(propan-2-yl)-6a,9a-dihydro-6H-furo[3,2-f][1,3,5,2,4]trioxadisilocin-9-one 892389-19-4 C23H35ClFN3O5Si2
(6aR,8R,9aR)-8-(4-chloro-5-fluoropyrrolo[2,3-d]pyrimidin-7-yl)-2,2,4,4-tetra(propan-2-yl)-6a,9a-dihydro-6H-furo[3,2-f][1,3,5,2,4]trioxadisilocin-9-one
—— {1S-[1S-(2S-benzofuran-3-ylmethyl-pyrrolidine-1-carbonyl)-2-methyl-propylcarbamoyl]-ethyl}-carbamic acid tert-butyl ester 874773-58-7 C26H37N3O5
{1S-[1S-(2S-benzofuran-3-ylmethyl-pyrrolidine-1-carbonyl)-2-methyl-propylcarbamoyl]-ethyl}-carbamic acid tert-butyl ester
—— 8-[3-(2-fluoro-1-oxy-pyridin-3-yl)-phenyl]-8-(4-trifluoromethoxyphenyl)-2,3,4,8-tetrahydro-imidazo[1,5-a]pyrimidin-6-ylamine 871942-47-1 C24H19F4N5O2
8-[3-(2-fluoro-1-oxy-pyridin-3-yl)-phenyl]-8-(4-trifluoromethoxyphenyl)-2,3,4,8-tetrahydro-imidazo[1,5-a]pyrimidin-6-ylamine
—— 5-(5-methyl-7-(2,6-dimethylphenyl)benzo[e][1,2,4]triazin-3-ylamino)-1-(3-(pyrrolidin-1-yl)propyl)pyridin-2(1H)-one 867331-84-8 C28H32N6O
5-(5-methyl-7-(2,6-dimethylphenyl)benzo[e][1,2,4]triazin-3-ylamino)-1-(3-(pyrrolidin-1-yl)propyl)pyridin-2(1H)-one
—— 2-[(4-Bromo-benzyl)-isopropyl-amino]-ethanol 867333-39-9 C12H18BrNO
2-[(4-Bromo-benzyl)-isopropyl-amino]-ethanol
—— trans-2S-[3-(2-ethyl-phenoxy)-propenyl]-4S-phenoxy-pyrrolidine 874773-24-7 C21H25NO2
trans-2S-[3-(2-ethyl-phenoxy)-propenyl]-4S-phenoxy-pyrrolidine
—— 9-benzyl-3-(4-fluoro-phenyl)-3,4,9-triaza-tricyclo[5.3.1.0<SP>2,6</SP>]undeca-2(6),4-diene 833458-99-4 C21H20FN3
9-benzyl-3-(4-fluoro-phenyl)-3,4,9-triaza-tricyclo[5.3.1.0<SP>2,6</SP>]undeca-2(6),4-diene
—— 1-(3-bromophenyl)-1-(imidazol-2-yl)-1-[4-(trifluoromethoxy)phenyl]methanol 871942-06-2 C17H12BrF3N2O2
1-(3-bromophenyl)-1-(imidazol-2-yl)-1-[4-(trifluoromethoxy)phenyl]methanol
—— 3-{3-[1-(2-tert-butoxycarbonylamino-3-methyl-butyryl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester 874773-97-4 C28H40N2O6
3-{3-[1-(2-tert-butoxycarbonylamino-3-methyl-butyryl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester
—— 2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester 874774-37-5 C20H26N2O3
2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester
—— {1S-[2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine-1-carbonyl]-2-methyl-propyl}-carbamic acid tert-butyl ester 874773-80-5 C23H31BrN2O4
{1S-[2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine-1-carbonyl]-2-methyl-propyl}-carbamic acid tert-butyl ester
—— 2S-Benzofuran-3-ylmethyl-pyrrolidine-1-carboxylic acid tert-butyl ester 874773-51-0 C18H23NO3
2S-Benzofuran-3-ylmethyl-pyrrolidine-1-carboxylic acid tert-butyl ester
—— 3-{3-[1-(5-amino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid 874774-09-1 C26H37N3O6
3-{3-[1-(5-amino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid
—— {1S-[2-methyl-1S-(4S-phenoxy-2S-phenoxymethyl-pyrrolidine-1-carbonyl)-propylcarbamoyl]-ethyl}-carbamic acid tert-butyl ester 874773-16-7 C30H41N3O6
{1S-[2-methyl-1S-(4S-phenoxy-2S-phenoxymethyl-pyrrolidine-1-carbonyl)-propylcarbamoyl]-ethyl}-carbamic acid tert-butyl ester
—— 3-{3-[1-(5-benzyloxycarbonylamino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester 874774-05-7 C36H47N3O8
3-{3-[1-(5-benzyloxycarbonylamino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester
—— 1-(3-pyrrolidin-2S-ylmethyl-indol-1-yl)-ethanone 874774-39-7 C15H18N2O
1-(3-pyrrolidin-2S-ylmethyl-indol-1-yl)-ethanone
—— (1S-{2-methyl-1S-[2S-(2-pyridin-4-yl-benzofuran-3-ylmethyl)-pyrrolidine-1-carbonyl]-propylcarbamoyl}-ethyl)-carbamic acid tert-butyl ester 874773-85-0 C31H40N4O5
(1S-{2-methyl-1S-[2S-(2-pyridin-4-yl-benzofuran-3-ylmethyl)-pyrrolidine-1-carbonyl]-propylcarbamoyl}-ethyl)-carbamic acid tert-butyl ester
—— [1S-(1S-{2R-[3-(2-ethyl-phenoxy)-propyl]-4S-phenoxy-pyrrolidine-1-carbonyl}-2-methyl-propylcarbamoyl)-ethyl]-carbamic acid tert-butyl ester 874773-44-1 C34H49N3O6
[1S-(1S-{2R-[3-(2-ethyl-phenoxy)-propyl]-4S-phenoxy-pyrrolidine-1-carbonyl}-2-methyl-propylcarbamoyl)-ethyl]-carbamic acid tert-butyl ester
—— 6-(4-fluorophenyl)-3-[2-(2,4,6-trifluorophenyl)-acetylamino]-pyrazine-2-carboxylic acid methyl ester 872088-75-0 C20H13F4N3O3
6-(4-fluorophenyl)-3-[2-(2,4,6-trifluorophenyl)-acetylamino]-pyrazine-2-carboxylic acid methyl ester
—— 6-chloro-2-cyclopropyl-nicotinic acid methyl ester 862695-74-7 C10H10ClNO2
6-chloro-2-cyclopropyl-nicotinic acid methyl ester
—— tert-butyl N-[(3S,9S)-8,14-dioxo-18-oxa-7,13-diazatetracyclo[15.7.0.03,7.019,24]tetracosa-1(17),19,21,23-tetraen-9-yl]carbamate 874774-11-5 C26H35N3O5
tert-butyl N-[(3S,9S)-8,14-dioxo-18-oxa-7,13-diazatetracyclo[15.7.0.03,7.019,24]tetracosa-1(17),19,21,23-tetraen-9-yl]carbamate
—— 3-{3-[1-(2-amino-3-methyl-butyryl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester 874773-99-6 C23H32N2O4
3-{3-[1-(2-amino-3-methyl-butyryl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid ethyl ester
—— 2-(6-fluoro-1H-indol-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester 874774-56-8 C18H23FN2O2
2-(6-fluoro-1H-indol-3-ylmethyl)-pyrrolidine-1-carboxylic acid tert-butyl ester
—— {1-cyclohexyl-2-[2-(6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-2-oxo-ethyl}-carbamic acid tert-butyl ester 874774-62-6 C33H50FN3O6
{1-cyclohexyl-2-[2-(6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-2-oxo-ethyl}-carbamic acid tert-butyl ester
—— 3-(3-{1-[2-(2-tert-butoxycarbonylamino-propionylamino)-3-methyl-butyryl]-pyrrolidin-2-ylmethyl}-benzofuran-2-yl)-propionic acid ethyl ester 874774-01-3 C31H45N3O7
3-(3-{1-[2-(2-tert-butoxycarbonylamino-propionylamino)-3-methyl-butyryl]-pyrrolidin-2-ylmethyl}-benzofuran-2-yl)-propionic acid ethyl ester
—— 5-methanesulfonyl-2-methyl-4-oxo-3,4-dihydro-thieno[3,4-]pyrimidine-7-carboxylic acid ethyl ester 873190-01-3 C11H12N2O5S2
5-methanesulfonyl-2-methyl-4-oxo-3,4-dihydro-thieno[3,4-]pyrimidine-7-carboxylic acid ethyl ester
—— 1-hydroxymethyl-3-methanesulfonyl-6,6-dimethyl-6,7-dihydro-5H-benzo[c]thiophen-4-one 873190-12-6 C12H16O4S2
1-hydroxymethyl-3-methanesulfonyl-6,6-dimethyl-6,7-dihydro-5H-benzo[c]thiophen-4-one
—— 2-[3-[2-Fluoro-6-(trifluoromethoxy)phenyl]phenyl]-2-oxoacetic acid 866632-59-9 C15H8F4O4
2-[3-[2-Fluoro-6-(trifluoromethoxy)phenyl]phenyl]-2-oxoacetic acid
—— N-(2a(2),4a(2)-Difluoro[1,1a(2)-biphenyl]-4-yl)-4-morpholinepentanamide 874450-45-0 C21H24F2N2O2
N-(2a(2),4a(2)-Difluoro[1,1a(2)-biphenyl]-4-yl)-4-morpholinepentanamide
—— Methyl 6-(3-bromophenyl)-4-methyl-5-oxopyrazine-2-carboxylate 866631-17-6 C13H11BrN2O3
Methyl 6-(3-bromophenyl)-4-methyl-5-oxopyrazine-2-carboxylate
—— 2-[4-(hydroxymethyl)phenyl]-3-phenyl-1,6-naphthyridin-5(6H)-one 893423-86-4 C21H16N2O2
2-[4-(hydroxymethyl)phenyl]-3-phenyl-1,6-naphthyridin-5(6H)-one
—— 1-[3-[2-Fluoro-6-(trifluoromethoxy)phenyl]phenyl]ethanone 866632-58-8 C15H10F4O2
1-[3-[2-Fluoro-6-(trifluoromethoxy)phenyl]phenyl]ethanone
—— Tert-butyl 2-[bis[(2-methylpropan-2-yl)oxycarbonyl]amino]-4-(5-ethoxycarbonylthiophen-2-yl)imidazole-1-carboxylate 866524-05-2 C25H35N3O8S
Tert-butyl 2-[bis[(2-methylpropan-2-yl)oxycarbonyl]amino]-4-(5-ethoxycarbonylthiophen-2-yl)imidazole-1-carboxylate