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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[2-(4-tert-butoxycarbonylaminofurazan-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-7-yloxy]piperidine-1-carboxylic acid tert-butyl ester 842144-00-7 C25H35N7O6
4-[2-(4-tert-butoxycarbonylaminofurazan-3-yl)-1-ethyl-1H-imidazo[4,5-c]pyridin-7-yloxy]piperidine-1-carboxylic acid tert-butyl ester
—— ethyl 2-(4-amino-1,2,5-oxadiazol-3-yl)-1-(1-methylethyl)-4-phenyl-1H-imidazo[4,5-c]pyridine-7-carboxylate 842145-08-8 C20H20N6O3
ethyl 2-(4-amino-1,2,5-oxadiazol-3-yl)-1-(1-methylethyl)-4-phenyl-1H-imidazo[4,5-c]pyridine-7-carboxylate
—— [5-methyl-2-(3-methylbenzyl)-1,3-oxazol-4-yl]methanol 867314-58-7 C13H15NO2
[5-methyl-2-(3-methylbenzyl)-1,3-oxazol-4-yl]methanol
—— 4-(chloromethyl)-5-methyl-2-(3-methylbenzyl)-1,3-oxazole 867314-72-5 C13H14ClNO
4-(chloromethyl)-5-methyl-2-(3-methylbenzyl)-1,3-oxazole
—— 2-[(4-{[(2-ethoxy-2-oxoethyl)(2-methoxyethyl)amino]methyl}phenyl)thio]-2-methyl-propionic acid tert-butylester 867314-30-5 C22H35NO5S
2-[(4-{[(2-ethoxy-2-oxoethyl)(2-methoxyethyl)amino]methyl}phenyl)thio]-2-methyl-propionic acid tert-butylester
—— 1-[2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-2S-amino-3-methyl-butan-1-one 874774-42-2 C20H27N3O2
1-[2S-(1-acetyl-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-2S-amino-3-methyl-butan-1-one
—— 2-(4-amino-1,2,5-oxadiazol-3-yl)-1-(1-methylethyl)-4-phenyl-1H-imidazo[4,5-c]pyridine-7-carboxylic acid 842145-09-9 C18H16N6O3
2-(4-amino-1,2,5-oxadiazol-3-yl)-1-(1-methylethyl)-4-phenyl-1H-imidazo[4,5-c]pyridine-7-carboxylic acid
—— 3-(2-chlorophenyl)-6-methylsulfanyl-1H-pyrazolo[3,4-d]-pyrimidine 864543-60-2 C12H9ClN4S
3-(2-chlorophenyl)-6-methylsulfanyl-1H-pyrazolo[3,4-d]-pyrimidine
—— N-(4-[(2-tert.-butoxy-1,1-dimethyl-2-oxoethyl)thio]benzyl)-N-(2-methoxyethyl)glycine 867314-31-6 C20H31NO5S
N-(4-[(2-tert.-butoxy-1,1-dimethyl-2-oxoethyl)thio]benzyl)-N-(2-methoxyethyl)glycine
—— [2-(3-chloro-phenoxy)-thiazol-5-yl]-methanol 867315-09-1 C10H8ClNO2S
[2-(3-chloro-phenoxy)-thiazol-5-yl]-methanol
—— 9-(2-methoxy-ethyl)-9H-carbazol-4-ol 890017-28-4 C15H15NO2
9-(2-methoxy-ethyl)-9H-carbazol-4-ol
—— tert-butyl 3-fluoro-4-(2-oxo-2-phenylethoxy)cyclohexylcarbamate 847417-29-2 C19H26FNO4
tert-butyl 3-fluoro-4-(2-oxo-2-phenylethoxy)cyclohexylcarbamate
—— 3-{3-[1-(5-benzyloxycarbonylamino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid 874774-07-9 C34H43N3O8
3-{3-[1-(5-benzyloxycarbonylamino-2-tert-butoxycarbonylamino-pentanoyl)-pyrrolidin-2-ylmethyl]-benzofuran-2-yl}-propionic acid
—— 4-methyl-3,5,10-triaza-tricyclo[6.3.1.0<SP>2,7</SP>]dodeca-2(7),3,5-triene 833458-98-3 C10H13N3
4-methyl-3,5,10-triaza-tricyclo[6.3.1.0<SP>2,7</SP>]dodeca-2(7),3,5-triene
—— 4,8-Dichloro-2-trifluoromethylbenzo[4,5]furo[3,2-d]pyrimidine 887281-53-0 C11H3Cl2F3N2O
4,8-Dichloro-2-trifluoromethylbenzo[4,5]furo[3,2-d]pyrimidine
—— 1-(6-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-(2,3-difluoro-phenyl)-ethanone 849068-51-5 C15H9ClF2N2O
1-(6-chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)-2-(2,3-difluoro-phenyl)-ethanone
—— [1S-(2S-benzofuran-3-ylmethyl-pyrrolidine-1-carbonyl)-2-methyl-propyl]-carbamic acid tert-butyl ester 874773-54-3 C23H32N2O4
[1S-(2S-benzofuran-3-ylmethyl-pyrrolidine-1-carbonyl)-2-methyl-propyl]-carbamic acid tert-butyl ester
—— tert-butyl-2-methyl-2-{[4-({[6-(3-methylphenyl)pyrimidin-4-yl]amino}methyl)-phenyl]thio}-2-methylpropanoate 881687-31-6 C26H31N3O2S
tert-butyl-2-methyl-2-{[4-({[6-(3-methylphenyl)pyrimidin-4-yl]amino}methyl)-phenyl]thio}-2-methylpropanoate
—— [2-(3-chloro-phenylamino)-4-cyclopropyl-pyrimidin-5-yl]-methanol 863774-14-5 C14H14ClN3O
[2-(3-chloro-phenylamino)-4-cyclopropyl-pyrimidin-5-yl]-methanol
—— (2-{[4-azido-2-fluorocyclohexyl]oxy}-1-phenylethoxy)(tert-butyl)dimethylsilane 847417-21-4 C20H32FN3O2Si
(2-{[4-azido-2-fluorocyclohexyl]oxy}-1-phenylethoxy)(tert-butyl)dimethylsilane
—— tert-butyl-2-({4-[((2-methoxyethyl){6-[4-methylphenyl]pyrimidin-4-yl}amino)methyl]-phenyl}thio)-2-methylpropanoate 881687-28-1 C29H37N3O3S
tert-butyl-2-({4-[((2-methoxyethyl){6-[4-methylphenyl]pyrimidin-4-yl}amino)methyl]-phenyl}thio)-2-methylpropanoate
—— (1S,4S)-4-[(tert-butoxycarbonyl)amino]-1-(2-methoxyethyl)cyclopent-2-ene-1-carboxylic acid 872592-84-2 C14H23NO5
(1S,4S)-4-[(tert-butoxycarbonyl)amino]-1-(2-methoxyethyl)cyclopent-2-ene-1-carboxylic acid
—— tert-Butyl 2-methyl-2-({4-[(prop-2-yn-1-ylamino)methyl]phenyl}thio)propanoate 881687-43-0 C18H25NO2S
tert-Butyl 2-methyl-2-({4-[(prop-2-yn-1-ylamino)methyl]phenyl}thio)propanoate
—— 1-[4-(2,3-dihydro-benzo[1,4]dioxin-6-ylsulfonylmethyl)-phenyl]-ethanone 890847-40-2 C17H16O5S
1-[4-(2,3-dihydro-benzo[1,4]dioxin-6-ylsulfonylmethyl)-phenyl]-ethanone
—— tert-butyl-2-{[4-({(6-chloropyrimidm-4-yl)[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-phenyl]thio}-2-methylpropanoate 881687-58-7 C24H29ClN4O2S2
tert-butyl-2-{[4-({(6-chloropyrimidm-4-yl)[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-phenyl]thio}-2-methylpropanoate
—— 4-tert-butyl-2-(3-chloro-phenylamino)-pyrimidine-5-carboxylic acid ethyl ester 863323-34-6 C17H20ClN3O2
4-tert-butyl-2-(3-chloro-phenylamino)-pyrimidine-5-carboxylic acid ethyl ester
—— intermediate 42 840537-55-5 C13H10ClN5O
intermediate 42
—— (6aR,8R,9S,9aR)-8-(4-chloro-5-fluoropyrrolo[2,3-d]pyrimidin-7-yl)-9-methyl-2,2,4,4-tetra(propan-2-yl)-6,6a,8,9a-tetrahydrofuro[3,2-f][1,3,5,2,4]trioxadisilocin-9-ol 892389-21-8 C24H39ClFN3O5Si2
(6aR,8R,9S,9aR)-8-(4-chloro-5-fluoropyrrolo[2,3-d]pyrimidin-7-yl)-9-methyl-2,2,4,4-tetra(propan-2-yl)-6,6a,8,9a-tetrahydrofuro[3,2-f][1,3,5,2,4]trioxadisilocin-9-ol
—— 2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine 874773-79-2 C13H14BrNO
2S-(2-bromo-benzofuran-3-ylmethyl)-pyrrolidine
—— benzyl-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-cyclohex-3-enyl]-carbamic acid tert-butyl ester 849069-11-0 C24H36BNO4
benzyl-[4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-cyclohex-3-enyl]-carbamic acid tert-butyl ester
—— [1-(6-chloro-4-isopropyl-pyridin-3-yl)-ethyl]-cyclobutylmethyl-amine 863894-39-7 C15H23ClN2
[1-(6-chloro-4-isopropyl-pyridin-3-yl)-ethyl]-cyclobutylmethyl-amine
—— tert-butyl-2-({4-[((2-furylmethyl){6-[3-chlorophenyl]pyrimidin-4-yl}amino)methyl]-phenyl}thio)-2-methylpropanoate 881687-30-5 C30H32ClN3O3S
tert-butyl-2-({4-[((2-furylmethyl){6-[3-chlorophenyl]pyrimidin-4-yl}amino)methyl]-phenyl}thio)-2-methylpropanoate
—— tert-butyl-2-{[4-({(2-methoxyethyl)[6-(4-methylphenoxy)pyrimidin-4-yl]amino}methyl)phenyl]-thio}-2-methylpropanoate 881687-66-7 C29H37N3O4S
tert-butyl-2-{[4-({(2-methoxyethyl)[6-(4-methylphenoxy)pyrimidin-4-yl]amino}methyl)phenyl]-thio}-2-methylpropanoate
—— tert-butyl-2-methyl-2-{[4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]thio}-propanoate 881687-57-6 C20H28N2O2S2
tert-butyl-2-methyl-2-{[4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenyl]thio}-propanoate
—— tert-butyl-2-{[4-({[6-(cyclohexyloxy)pyrimidin-4-yl][(3,5-dimethylisoxazol-4-yl)methyl]amino}-methyl)phenyl]thio}-2-methylpropanoate 881687-56-5 C31H42N4O4S
tert-butyl-2-{[4-({[6-(cyclohexyloxy)pyrimidin-4-yl][(3,5-dimethylisoxazol-4-yl)methyl]amino}-methyl)phenyl]thio}-2-methylpropanoate
—— 2-amino-2-cyclohexyl-1-[2-(6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-ethanone 874774-64-8 C28H42FN3O4
2-amino-2-cyclohexyl-1-[2-(6-fluoro-1-{2-[2-(2-methoxy-ethoxy)-ethoxy]-ethyl}-1H-indol-3-ylmethyl)-pyrrolidin-1-yl]-ethanone
—— 5-(Trifluoromethyl)-1',2',3',6'-tetrahydro-3,4'-bipyridine 872673-21-7 C11H11F3N2
5-(Trifluoromethyl)-1',2',3',6'-tetrahydro-3,4'-bipyridine
—— 5-bromo-1H-pyrrolo[2,3-b]pyridine-3-carbothioic acid (2,3-difluoro-phenyl)-amide 849068-63-9 C14H8BrF2N3S
5-bromo-1H-pyrrolo[2,3-b]pyridine-3-carbothioic acid (2,3-difluoro-phenyl)-amide
—— (2S)-Pyrrolidine-1,2-dicarbaldehyde 88218-11-5 C6H9NO2
(2S)-Pyrrolidine-1,2-dicarbaldehyde
—— 3-(4-(trifluoromethyl)piperidin-1-yl)propan-1-amine 869493-49-2 C9H17F3N2
3-(4-(trifluoromethyl)piperidin-1-yl)propan-1-amine
—— 2-biphenyl-4-yl-benzooxazole-7-carboxylic acid 884849-21-2 C20H13NO3
2-biphenyl-4-yl-benzooxazole-7-carboxylic acid
—— (R)-benzyl 1-(imidazo[1,5-a]pyridin-3-yl)-2-(7-methyl-1H-indazol-5-yl)ethylcarbamate 890044-61-8 C25H23N5O2
(R)-benzyl 1-(imidazo[1,5-a]pyridin-3-yl)-2-(7-methyl-1H-indazol-5-yl)ethylcarbamate
—— 4,11-diazatricyclo[7,3,1,0<sup>2,7</sup>]trideca-2,4,6-triene 833459-31-7 C11H14N2
4,11-diazatricyclo[7,3,1,0<sup>2,7</sup>]trideca-2,4,6-triene
—— tert-butyl 3-[7-(hydroxymethyl)-5-phenyl-1H-indol-3-yl]pyrrolidine-1-carboxylate 860625-01-0 C24H28N2O3
tert-butyl 3-[7-(hydroxymethyl)-5-phenyl-1H-indol-3-yl]pyrrolidine-1-carboxylate
—— 2-(tert-butyl-dimethyl-silanyloxy)-9-[4'-(2'-chloro-ethoxy)-phenyl]-11,14-spiro[4,5]-5,6,7,8-tetrahydro-9H-benzo[c]chromene 874281-35-3 C29H37ClO3S2Si
2-(tert-butyl-dimethyl-silanyloxy)-9-[4'-(2'-chloro-ethoxy)-phenyl]-11,14-spiro[4,5]-5,6,7,8-tetrahydro-9H-benzo[c]chromene
—— (2-chlorophenyl)-(2,6-dichloropyridin-3-yl)methanone 864543-73-7 C12H6Cl3NO
(2-chlorophenyl)-(2,6-dichloropyridin-3-yl)methanone
—— 6-bromo-2,2-diethyl-8-isopropyl-4,4-dimethyl chroman 856251-45-1 C18H27BrO
6-bromo-2,2-diethyl-8-isopropyl-4,4-dimethyl chroman
—— 3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-4-methylbenzoyl chloride 882739-69-7 C19H12Cl2F2N2O3
3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-4-methylbenzoyl chloride
—— tert-butyl N-[8-[3-(2-fluoro-1-oxidopyridin-1-ium-3-yl)phenyl]-8-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-imidazo[1,5-a]pyrimidin-6-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 871942-46-0 C34H35F4N5O6
tert-butyl N-[8-[3-(2-fluoro-1-oxidopyridin-1-ium-3-yl)phenyl]-8-[4-(trifluoromethoxy)phenyl]-3,4-dihydro-2H-imidazo[1,5-a]pyrimidin-6-yl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate
—— 4-{2-[2-(3,4-dimethoxy-phenyl)-5,7-dimethoxy-4-oxo-4H-chromen-3-yloxy]-ethoxy}-benzoic acid 851133-90-9 C28H26O10
4-{2-[2-(3,4-dimethoxy-phenyl)-5,7-dimethoxy-4-oxo-4H-chromen-3-yloxy]-ethoxy}-benzoic acid