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—— 2-{4-[({4-[(5-{2-[(2,3-difluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)methyl]piperidin-1-yl}ethyl dihydrogen phosphate 722543-19-3 C27H30F2N7O6P
2-{4-[({4-[(5-{2-[(2,3-difluorophenyl)amino]-2-oxoethyl}-1H-pyrazol-3-yl)amino]quinazolin-7-yl}oxy)methyl]piperidin-1-yl}ethyl dihydrogen phosphate
—— N-[3-[[5-bromo-4-[[3-[[[1-(trifluoromethyl)cyclobutyl]carbonyl]amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide 702676-87-7 C24H29BrF3N7O2
N-[3-[[5-bromo-4-[[3-[[[1-(trifluoromethyl)cyclobutyl]carbonyl]amino]propyl]amino]-2-pyrimidinyl]amino]phenyl]-1-pyrrolidinecarboxamide
—— 1-benzyl-5-[(2R)-2-({(2R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethylphenyl) ethyl}amino)propyl]-N-(2-methoxybenzyl)-1H-indole-2-carboxamide 757963-61-4 C36H39N3O5
1-benzyl-5-[(2R)-2-({(2R)-2-hydroxy-2-(4-hydroxy-3-hydroxymethylphenyl) ethyl}amino)propyl]-N-(2-methoxybenzyl)-1H-indole-2-carboxamide
—— (2R,2'S,5'S)-2-amino-N-[5-(4-ethoxy-benzyl)-3,6-dioxo-1-(4-phenoxy-benzyl)-piperazin-2-ylmethyl]-3-(1H-imidazol-4-yl)-propionamide 702690-17-3 C33H36N6O5
(2R,2'S,5'S)-2-amino-N-[5-(4-ethoxy-benzyl)-3,6-dioxo-1-(4-phenoxy-benzyl)-piperazin-2-ylmethyl]-3-(1H-imidazol-4-yl)-propionamide
—— (15S)-11-[[(3S,4S)-1-[(2,4-dichlorophenyl)methyl]-4-thiophen-3-ylpyrrolidin-3-yl]methyl]-3,14-dioxa-11-azadispiro[5.1.58.26]pentadecane-15-carboxylic acid 723287-94-3 C29H36Cl2N2O4S
(15S)-11-[[(3S,4S)-1-[(2,4-dichlorophenyl)methyl]-4-thiophen-3-ylpyrrolidin-3-yl]methyl]-3,14-dioxa-11-azadispiro[5.1.58.26]pentadecane-15-carboxylic acid
—— 5,5-bis(4-fluorophenyl)-2-methyl-3-{[1-(2-phenylethyl)-3-azetidinyl]methyl}-3,5-dihydro-4H-imidazol-4-one trifluoroacetate 721949-61-7 C2HF3O2*C28H27F2N3O
5,5-bis(4-fluorophenyl)-2-methyl-3-{[1-(2-phenylethyl)-3-azetidinyl]methyl}-3,5-dihydro-4H-imidazol-4-one trifluoroacetate
—— 2-[5-(5-chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-5-(thiazolidine-3-carbonyl)-2H-pyrazole-3-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide 713143-24-9 C24H29ClN6O3S2
2-[5-(5-chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-5-(thiazolidine-3-carbonyl)-2H-pyrazole-3-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
—— 2-[5-(5-chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-5-methanesulfonylaminocarbonyl-2H-pyrazole-3-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide 713142-87-1 C22H27ClN6O5S2
2-[5-(5-chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-5-methanesulfonylaminocarbonyl-2H-pyrazole-3-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
—— 2-({6-methoxy-5-[2-(4-methyl-piperazin-1-yl)-ethylamino]-pyridin-3-ylmethyl}-amino)-N-(3-trifluoromethyl-phenyl)-benzamide 709045-10-3 C28H33F3N6O2
2-({6-methoxy-5-[2-(4-methyl-piperazin-1-yl)-ethylamino]-pyridin-3-ylmethyl}-amino)-N-(3-trifluoromethyl-phenyl)-benzamide
—— 3-(2-(((4-(benzothiophen-2-yl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)-4-(3,5-dimethylphenoxy)phenyl)propanoic acid 740852-41-9 C31H31NO5S
3-(2-(((4-(benzothiophen-2-yl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)-4-(3,5-dimethylphenoxy)phenyl)propanoic acid
—— 3-(4-(2-chloro-5-fluorophenoxymethyl)-2-(((4-(3-methylphenyl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid 740850-65-1 C29H29ClFNO5
3-(4-(2-chloro-5-fluorophenoxymethyl)-2-(((4-(3-methylphenyl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid
—— (3-{4-[3-phenethyl-1-(3-phenylpropyl)ureido]phenylsulphanyl}phenyl)acetic acid 735273-63-9 C32H32N2O3S
(3-{4-[3-phenethyl-1-(3-phenylpropyl)ureido]phenylsulphanyl}phenyl)acetic acid
—— (4S)-2-[[6-[(3-bromo-2-thienyl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(2-methylpropyl)-2,4-dioxo-thieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-methyl-4-isoxazolidinol 733809-39-7 C21H24BrN3O5S2
(4S)-2-[[6-[(3-bromo-2-thienyl)methyl]-1,2,3,4-tetrahydro-3-methyl-1-(2-methylpropyl)-2,4-dioxo-thieno[2,3-d]pyrimidin-5-yl]carbonyl]-4-methyl-4-isoxazolidinol
—— 3-(4-(3,5-dimethylphenoxy)-2-(((4-(naphthalen-2-yl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid 740852-13-5 C33H33NO5
3-(4-(3,5-dimethylphenoxy)-2-(((4-(naphthalen-2-yl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid
—— (S,S)-6-(4-Amino-butyl)-3-naphthalen-2-ylmethyl-1-(4-o-tolyloxy-benzyl)-piperazine-2,5-dione 702689-39-2 C33H35N3O3
(S,S)-6-(4-Amino-butyl)-3-naphthalen-2-ylmethyl-1-(4-o-tolyloxy-benzyl)-piperazine-2,5-dione
—— (+/-)-N-[4-(1-butyryl-3,3-dimethyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-benzamide 723305-32-6 C29H35N3O4S
(+/-)-N-[4-(1-butyryl-3,3-dimethyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-2-methyl-benzamide
—— 3-amino-6-[4-[[(1ethyl-3-piperidinyl)amino]sulfonyl]phenyl]-N-3-pyridinyl-2-pyrazinecarboxamide hydrochloride 714237-27-1 C23H27N7O3S*ClH
3-amino-6-[4-[[(1ethyl-3-piperidinyl)amino]sulfonyl]phenyl]-N-3-pyridinyl-2-pyrazinecarboxamide hydrochloride
—— 3-amino-6-[4-[[(1-ethyl-3-piperidinyl)amino]sulfonyl]phenyl]-N-3-pyridinyl-2-pyrazinecarboxamide 714237-39-5 C23H27N7O3S
3-amino-6-[4-[[(1-ethyl-3-piperidinyl)amino]sulfonyl]phenyl]-N-3-pyridinyl-2-pyrazinecarboxamide
—— (S,S)-6-(4-Amino-butyl)-1-(4-phenoxy-benzyl)-3-(5,6,7,8-tetrahydro-naphthalen-2-ylmethyl)-piperazine-2,5-dione 702689-38-1 C32H37N3O3
(S,S)-6-(4-Amino-butyl)-1-(4-phenoxy-benzyl)-3-(5,6,7,8-tetrahydro-naphthalen-2-ylmethyl)-piperazine-2,5-dione
—— {3-[3-(1,3-diphenethylureido)phenylsulphanyl]phenyl}acetic acid 735273-88-8 C31H30N2O3S
{3-[3-(1,3-diphenethylureido)phenylsulphanyl]phenyl}acetic acid
—— 3-(4-(3,5-dimethylphenylamino)-2-(((4-(2-(2-fluorophenyl)ethyl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid 740852-45-3 C31H35FN2O4
3-(4-(3,5-dimethylphenylamino)-2-(((4-(2-(2-fluorophenyl)ethyl)tetrahydro-2H-pyran-4-yl)amino)carbonyl)phenyl)propanoic acid
—— 1-[2-[4-[3-chloro-5-(1-pyrrolidinylcarbonyl)-2-pyridinyl]-1-piperazinyl]-4-pyrimidinyl]-3-piperidinecarboxamide 749908-46-1 C24H31ClN8O2
1-[2-[4-[3-chloro-5-(1-pyrrolidinylcarbonyl)-2-pyridinyl]-1-piperazinyl]-4-pyrimidinyl]-3-piperidinecarboxamide
—— 3-{2-methyl-4-[2-(4-trifluoromethylphenyl)benzothiazol-5-ylmethylsulfanyl]phenyl}propionic acid 729591-48-4 C25H20F3NO2S2
3-{2-methyl-4-[2-(4-trifluoromethylphenyl)benzothiazol-5-ylmethylsulfanyl]phenyl}propionic acid
—— 4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalene-1-carboxylic acid m-tolylamide 723307-54-8 C27H31N3O4S
4-(1-butyryl-piperidin-4-ylsulfamoyl)-naphthalene-1-carboxylic acid m-tolylamide
—— (S)-N-[3-[3-FLUORO-4-[N-1-[4-{2-FURYL-(5-nitro) methyl} piperazinylcarbonyl] PHENYL]-2-OXO-5-OXAZOLIDINYL] METHYL]-ACETAMIDE 741294-18-8 C22H24FN5O7
(S)-N-[3-[3-FLUORO-4-[N-1-[4-{2-FURYL-(5-nitro) methyl} piperazinylcarbonyl] PHENYL]-2-OXO-5-OXAZOLIDINYL] METHYL]-ACETAMIDE
—— {3-[4-(3-benzyl-1-heptylureido)phenylsulphanyl]phenyl}acetic acid 735273-96-8 C29H34N2O3S
{3-[4-(3-benzyl-1-heptylureido)phenylsulphanyl]phenyl}acetic acid
—— 3-(7-Acetylamino-1-oxo-1,3-dihydro-isoindol-2-yl)-3-(4-difluoromethoxy-3-ethoxy-phenyl)-N,N-dimethyl-propionamide 725256-92-8 C24H27F2N3O5
3-(7-Acetylamino-1-oxo-1,3-dihydro-isoindol-2-yl)-3-(4-difluoromethoxy-3-ethoxy-phenyl)-N,N-dimethyl-propionamide
—— (E)-5-(8-fluoro-11H-10-oxa-1-aza-dibenzo[a,d]cyclohepten-5-ylidenemethyl)-1-(2-morpholin-4-ylethyl)-1,3-dihydrobenzoimidazol-2-one 710345-86-1 C27H25FN4O3
(E)-5-(8-fluoro-11H-10-oxa-1-aza-dibenzo[a,d]cyclohepten-5-ylidenemethyl)-1-(2-morpholin-4-ylethyl)-1,3-dihydrobenzoimidazol-2-one
—— 5-{3-[2-(3-ethoxy-4-methoxy-phenyl)-ethyl]-ureido}-3-(pyridin-3-ylmethoxy)-isothiazole-4-carboxylic acid amide 727359-44-6 C22H25N5O5S
5-{3-[2-(3-ethoxy-4-methoxy-phenyl)-ethyl]-ureido}-3-(pyridin-3-ylmethoxy)-isothiazole-4-carboxylic acid amide
—— [2-(1-(4'-isopropylbenzenesulfonyl)-5-bromo-1H-indol-3-yloxy)ethyl]dimethylamine 700838-31-9 C21H25BrN2O3S
[2-(1-(4'-isopropylbenzenesulfonyl)-5-bromo-1H-indol-3-yloxy)ethyl]dimethylamine
—— 4-(3,4-Dichloro-benzyl)-8-fluoro-6-(4-oxo-2-thioxo-thiazolidin-5-ylidenemethyl)-4H-benzo[1,4]oxazin-3-one 711026-03-8 C19H11Cl2FN2O3S2
4-(3,4-Dichloro-benzyl)-8-fluoro-6-(4-oxo-2-thioxo-thiazolidin-5-ylidenemethyl)-4H-benzo[1,4]oxazin-3-one
—— ethyl 6-oxo-5-{2-[(phenylsulfonyl)methyl](1,3-thiazol-4-yl)}-2-(trifluoromethyl)-1,6-dihydro-3-pyridinecarboxylate 727382-51-6 C19H15F3N2O5S2
ethyl 6-oxo-5-{2-[(phenylsulfonyl)methyl](1,3-thiazol-4-yl)}-2-(trifluoromethyl)-1,6-dihydro-3-pyridinecarboxylate
—— 1-cyclohexylmethyl-5-[2-(4-methoxyphenyl)thiazol-4-yl]-2-methyl-1H-pyrrole-3-carboxylic acid cyclobutylamide 726179-79-9 C27H33N3O2S
1-cyclohexylmethyl-5-[2-(4-methoxyphenyl)thiazol-4-yl]-2-methyl-1H-pyrrole-3-carboxylic acid cyclobutylamide
—— 5-[3-(3-dibutylamino-propyl)-ureidomethyl]thiophene-2-carboxylic acid (2-amino-phenyl)amide 709664-61-9 C24H37N5O2S
5-[3-(3-dibutylamino-propyl)-ureidomethyl]thiophene-2-carboxylic acid (2-amino-phenyl)amide
—— {3-[4-(3-butyl-1-heptylureido)phenylsulphanyl]phenyl}acetic acid 735274-20-1 C26H36N2O3S
{3-[4-(3-butyl-1-heptylureido)phenylsulphanyl]phenyl}acetic acid
—— 9-[2-(2-methoxyphenyl)-2-oxoethyl]-8-phenyl-2-(4-pyridinyl)-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one 760975-03-9 C27H24N4O3
9-[2-(2-methoxyphenyl)-2-oxoethyl]-8-phenyl-2-(4-pyridinyl)-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one
—— {3-[2-({[(1Z)-1-biphenyl-4-yl-2-(dimethylamino)ethylidene]amino}oxy)ethoxy]-2-methylphenyl}acetic acid 760986-85-4 C27H30N2O4
{3-[2-({[(1Z)-1-biphenyl-4-yl-2-(dimethylamino)ethylidene]amino}oxy)ethoxy]-2-methylphenyl}acetic acid
—— 1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-3-(5-fluoro-2-methyl-phenyl)-urea 717899-25-7 C24H23FN6O2
1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-3-(5-fluoro-2-methyl-phenyl)-urea
—— {3-[4-(3-benzyl-1-butylureido)phenylsulphanyl]phenyl}acetic acid 735273-98-0 C26H28N2O3S
{3-[4-(3-benzyl-1-butylureido)phenylsulphanyl]phenyl}acetic acid
—— 4-(4-phenethyl-piperazin-1-yl)-9-thiazol-2-yl-5,6,7,8-tetrahydro-1,3,4b-triaza-fluorene 731824-38-7 C25H28N6S
4-(4-phenethyl-piperazin-1-yl)-9-thiazol-2-yl-5,6,7,8-tetrahydro-1,3,4b-triaza-fluorene
—— 1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-3-(2,5-difluoro-phenyl)-urea 717899-30-4 C23H20F2N6O2
1-[3-(4-amino-7-isopropyl-7H-pyrrolo[2,3-d]pyrimidine-5-carbonyl)-phenyl]-3-(2,5-difluoro-phenyl)-urea
—— 2-[5-(4-pyrrolidinylcarbonylphenyl)-3,6-dihydro-2H-pyridin-1-yl]-3-methyl-6-pyrimidin-4-yl-3H-pyrimidin-4-one 712343-99-2 C25H26N6O2
2-[5-(4-pyrrolidinylcarbonylphenyl)-3,6-dihydro-2H-pyridin-1-yl]-3-methyl-6-pyrimidin-4-yl-3H-pyrimidin-4-one
—— (E)-N-methyl-N-(2-methyl-benzofuran-3-ylmethyl)-3-(4-methyl-2-oxo-2,3,4,5-tetrahydro-1H-pyrido[2,3-e][1,4]diazepin-7-yl)acrylamide hydrochloride 709651-53-6 C23H24N4O3*ClH
(E)-N-methyl-N-(2-methyl-benzofuran-3-ylmethyl)-3-(4-methyl-2-oxo-2,3,4,5-tetrahydro-1H-pyrido[2,3-e][1,4]diazepin-7-yl)acrylamide hydrochloride
—— 2-[(aminocarbonyl)amino]-5-[2-{[1-benzylpyrrolidin-3-yl]oxy}phenyl]thiophene-3-carboxamide 727741-87-9 C23H24N4O3S
2-[(aminocarbonyl)amino]-5-[2-{[1-benzylpyrrolidin-3-yl]oxy}phenyl]thiophene-3-carboxamide
—— N-[3-[(1Z)-1-(8-methoxy-6H-benzo[c][1]benzoxepin-11-ylidene)propyl]phenyl]methanesulfonamide 710347-67-4 C25H25NO4S
N-[3-[(1Z)-1-(8-methoxy-6H-benzo[c][1]benzoxepin-11-ylidene)propyl]phenyl]methanesulfonamide
—— 1-[(3S)-5-[4-(4-fluorophenyl)phenoxy]-3-methylpentyl]-3-pyridin-4-ylimidazolidin-2-one 708208-52-0 C26H28FN3O2
1-[(3S)-5-[4-(4-fluorophenyl)phenoxy]-3-methylpentyl]-3-pyridin-4-ylimidazolidin-2-one
—— 1-(2,5-dimethyl-2H-pyrazol-3-yl)-3-[2-(3-isopropyl-[1,2,4]triazolo[4,3-a]pyridin-6-ylsulfanyl)-benzyl]-urea 745827-37-6 C22H25N7OS
1-(2,5-dimethyl-2H-pyrazol-3-yl)-3-[2-(3-isopropyl-[1,2,4]triazolo[4,3-a]pyridin-6-ylsulfanyl)-benzyl]-urea
—— (E)-(6-{2-[methyl-(1-methyl-1H-indol-2-ylmethyl)carbamoyl]vinyl}-2-oxo-1,4-dihydro-2H-pyrido[2,3-d]pyrimidin-3-yl)acetic acid 709652-36-8 C23H23N5O4
(E)-(6-{2-[methyl-(1-methyl-1H-indol-2-ylmethyl)carbamoyl]vinyl}-2-oxo-1,4-dihydro-2H-pyrido[2,3-d]pyrimidin-3-yl)acetic acid
—— 1-[5-(4-chloro-phenyl)-1-(2-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-2-morpholin-4-yl-ethanone 709033-17-0 C22H21Cl2N3O2
1-[5-(4-chloro-phenyl)-1-(2-chloro-phenyl)-4-methyl-1H-pyrazol-3-yl]-2-morpholin-4-yl-ethanone
—— N-(2,4-dichlorophenyl)-7-[3-trifluoromethyl-2-pyridinyl][1,2,4]triazolo[4,3-b]pyridazin-3-amine 749258-22-8 C17H9Cl2F3N6
N-(2,4-dichlorophenyl)-7-[3-trifluoromethyl-2-pyridinyl][1,2,4]triazolo[4,3-b]pyridazin-3-amine