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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(E)-2-(4-chloro-6-pyrrolidin-1-ylpyrimidin-2-yl)ethenyl]-6-fluoro-2-methylquinoxaline 1214254-44-0 C19H17ClFN5
3-[(E)-2-(4-chloro-6-pyrrolidin-1-ylpyrimidin-2-yl)ethenyl]-6-fluoro-2-methylquinoxaline
—— 4-bromo-N1-(tetrahydro2H-pyran-4-yl)benzene-1,2-diamine 1153229-26-5 C11H15BrN2O
4-bromo-N1-(tetrahydro2H-pyran-4-yl)benzene-1,2-diamine
—— 5-(3,4-dichlorophenyl)-3-(4-tetrahydropyranyl)imino-2-(2-methoxy-3-pyridyl)amino-3,5-dihydrophenazine 1353733-65-9 C29H25Cl2N5O2
5-(3,4-dichlorophenyl)-3-(4-tetrahydropyranyl)imino-2-(2-methoxy-3-pyridyl)amino-3,5-dihydrophenazine
—— 4-(naphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1-(tetrahydrofuran-3-yl)-1H-1,2,4-triazol-5(4H)-one 1268247-65-9 C26H27N5O3
4-(naphthalen-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1-(tetrahydrofuran-3-yl)-1H-1,2,4-triazol-5(4H)-one
—— 2-[(1S)-1'-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-5-chloro-6-methylspiro[1,2-dihydroindene-3,4'-piperidine]-1-yl]-2-methyl-N-(oxan-4-yl)propanamide 1243675-48-0 C38H50ClF2N3O3
2-[(1S)-1'-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-5-chloro-6-methylspiro[1,2-dihydroindene-3,4'-piperidine]-1-yl]-2-methyl-N-(oxan-4-yl)propanamide
—— 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-[1-(tetrahydro-pyran-4-yl)-1H-imidazol-4-yl]-1H-pyrazole 1191899-46-3 C24H21Cl3N4O
5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-3-[1-(tetrahydro-pyran-4-yl)-1H-imidazol-4-yl]-1H-pyrazole
—— 2-(3-azadicyclo[3.1.0]hexan-3-yl)-4-(3-chloro-4-methoxybenzyloxy)-N-(4-fluorobenzyl)pyrimidine-5-carboxamide 1418759-16-6 C25H24ClFN4O3
2-(3-azadicyclo[3.1.0]hexan-3-yl)-4-(3-chloro-4-methoxybenzyloxy)-N-(4-fluorobenzyl)pyrimidine-5-carboxamide
—— 4-(6-((tetrahydro-2H-pyran-4-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one 1453852-20-4 C14H16N4O2
4-(6-((tetrahydro-2H-pyran-4-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one
—— 4-(naphthalen-2-yl)-1-(pyridin-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one 1268247-66-0 C27H24N6O2
4-(naphthalen-2-yl)-1-(pyridin-2-yl)-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-1H-1,2,4-triazol-5(4H)-one
—— 2-(3-azadicyclo[3.1.0]hexan-3-yl)-4-(3-chloro-4-methoxybenzyloxy)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide 1418759-14-4 C24H24ClN5O3
2-(3-azadicyclo[3.1.0]hexan-3-yl)-4-(3-chloro-4-methoxybenzyloxy)-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
—— 4-methyl-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid 1159251-32-7 C17H15N3O4
4-methyl-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid
—— 1-{3-[2-(tetrahydropyran-4-ylamino)pyridin-4-yl][2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid ethylamide 1071133-33-9 C26H32N6O2
1-{3-[2-(tetrahydropyran-4-ylamino)pyridin-4-yl][2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid ethylamide
—— 4-[3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl]-N-(1(R)-phenylethyl)pyridin-2-amine 1177418-29-9 C25H24FN3O
4-[3-(4-fluorophenyl)-5-isopropylisoxazol-4-yl]-N-(1(R)-phenylethyl)pyridin-2-amine
—— Ethyl 2-methyl-2-[2-methyl-4-[2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]propanoate 1030367-91-9 C34H33F3O3S
Ethyl 2-methyl-2-[2-methyl-4-[2-phenyl-1-[4-[4-(trifluoromethyl)phenyl]phenyl]ethyl]sulfanylphenoxy]propanoate
—— 6-chloro-N-(oxan-4-yl)pyridine-3-carboxamide 1101793-11-6 C11H13ClN2O2
6-chloro-N-(oxan-4-yl)pyridine-3-carboxamide
—— dimethyl 4-(6-azidohexyl)-3,5-dioxoheptanedioate 1609644-10-1 C15H23N3O6
dimethyl 4-(6-azidohexyl)-3,5-dioxoheptanedioate
—— (1E,3E,5E,7E)-1,2,3,4,5,6,7,8-octa(3-methoxyphenyl)-1,3,5,7-octatetraene 1326244-52-3 C64H58O8
(1E,3E,5E,7E)-1,2,3,4,5,6,7,8-octa(3-methoxyphenyl)-1,3,5,7-octatetraene
—— N1-(tetrahydro-2H-pyran-4-yl)benzene-1,2-diamine 1154930-46-7 C11H16N2O
N1-(tetrahydro-2H-pyran-4-yl)benzene-1,2-diamine
—— 3-hydroxy-8,9,10-trimethoxy-benzo[<i>c</i>]chromen-6-one 107100-41-4 C16H14O6
3-hydroxy-8,9,10-trimethoxy-benzo[<i>c</i>]chromen-6-one
—— 1-(3-fluorophenyl)-7-methyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-6(7H)-one 1186491-26-8 C18H19FN4O2
1-(3-fluorophenyl)-7-methyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-6(7H)-one
—— 4-(2-chloro-4-pyrimidinyl)-N-(tetrahydro-2H-pyran-4-yl)-1,3,5-triazin-2-amine 1150111-28-6 C12H13ClN6O
4-(2-chloro-4-pyrimidinyl)-N-(tetrahydro-2H-pyran-4-yl)-1,3,5-triazin-2-amine
—— 1-{3-[2-(tetrahydropyran-4-ylamino)pyridin-4-yl][2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid amide 1071131-85-5 C24H28N6O2
1-{3-[2-(tetrahydropyran-4-ylamino)pyridin-4-yl][2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid amide
—— 6-{[3-(4-Fluoro-phenyl)-5-methyl-isoxazol-4-ylmethyl]-amino}-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide 1159251-82-7 C21H22FN5O3
6-{[3-(4-Fluoro-phenyl)-5-methyl-isoxazol-4-ylmethyl]-amino}-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide
—— 4-methyl-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide 1159251-33-8 C22H24N4O4
4-methyl-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide
—— N-((R)-cyano-methyl-methyl)-3-[5-(4-{[(tetrahydropyran-4-yl)-(2,2,2-trifluoroacetyl)amino]methyl}phenyl)isoxazol-3-yl]benzamide 1333335-02-6 C27H25F3N4O4
N-((R)-cyano-methyl-methyl)-3-[5-(4-{[(tetrahydropyran-4-yl)-(2,2,2-trifluoroacetyl)amino]methyl}phenyl)isoxazol-3-yl]benzamide
—— 4-chloro-1-(3-fluorophenyl)-7-methyl-1H-pyrazolo[3,4-b]pyridin-6(7H)-one 1148051-72-2 C13H9ClFN3O
4-chloro-1-(3-fluorophenyl)-7-methyl-1H-pyrazolo[3,4-b]pyridin-6(7H)-one
—— 1-[5-(2-oxo-2-phenylethyl)-furan-2-yl]hex-5-en-2-one 1195869-37-4 C18H18O3
1-[5-(2-oxo-2-phenylethyl)-furan-2-yl]hex-5-en-2-one
—— (S)-N-(1-cyanoethyl)-3-(5-(4-((2,2,2-trifluoro-N-(tetrahydro-2H-pyran-4-yl)acetamido)methyl)phenyl)isoxazol-3-yl)benzamide 1333341-24-4 C27H25F3N4O4
(S)-N-(1-cyanoethyl)-3-(5-(4-((2,2,2-trifluoro-N-(tetrahydro-2H-pyran-4-yl)acetamido)methyl)phenyl)isoxazol-3-yl)benzamide
—— N-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-pyran-4-ylamino)-7,8-dihydro-pyrido[2,3-d]pyrimidin-6-yl]-benzamide 1026662-97-4 C24H27N5O3
N-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-pyran-4-ylamino)-7,8-dihydro-pyrido[2,3-d]pyrimidin-6-yl]-benzamide
—— 1-(6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)piperidin-4-amine 1565849-97-9 C24H31N5O2
1-(6-ethyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)piperidin-4-amine
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-90-1 C25H29F3N6O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-N-(tetrahydro-pyran-4-yl)-benzamide
—— [<sup>14</sup>C]3-(3-chloro-4-methoxybenzyl)-5-ethyl-2-((tetrahydro-2H-pyran-4-yl)amino)-7,8-dihydro-3H-imidazo[2,1-b]purin-4(5H)-one 1542204-84-1 C22H27ClN6O3
[<sup>14</sup>C]3-(3-chloro-4-methoxybenzyl)-5-ethyl-2-((tetrahydro-2H-pyran-4-yl)amino)-7,8-dihydro-3H-imidazo[2,1-b]purin-4(5H)-one
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methyl-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-58-1 C26H32F2N6O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methyl-N-(tetrahydro-pyran-4-yl)-benzamide
—— N-cyclopropyl-3-(2-methanesulfonyl-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-6-yl)-4-methyl-benzamide 1026663-24-0 C20H20N4O4S
N-cyclopropyl-3-(2-methanesulfonyl-8-methyl-7-oxo-7,8-dihydro-pyrido[2,3-d]pyrimidin-6-yl)-4-methyl-benzamide
—— 3-(7-(2-hydroxyethyl)-8-oxo-9-(tetrahydro-2H-pyran-4-yl)-8,9-dihydro-7H-purin-2-yl)pyrazolo[1,5-a]pyridin-5-carbonitrile 1299418-91-9 C20H19N7O3
3-(7-(2-hydroxyethyl)-8-oxo-9-(tetrahydro-2H-pyran-4-yl)-8,9-dihydro-7H-purin-2-yl)pyrazolo[1,5-a]pyridin-5-carbonitrile
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-66-1 C27H34F2N6O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-N-(tetrahydro-pyran-4-yl)-benzamide
—— 4-chloro-5-(3-fluoro-4-(trifluoromethyl)phenyl)isoxazole-3-carboxylic acid 1110771-93-1 C11H4ClF4NO3
4-chloro-5-(3-fluoro-4-(trifluoromethyl)phenyl)isoxazole-3-carboxylic acid
—— 6-[3-(4-fluoro-phenyl)-5-methyl-isoxazol-4-ylmethoxy]-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide 1159251-53-2 C21H21FN4O4
6-[3-(4-fluoro-phenyl)-5-methyl-isoxazol-4-ylmethoxy]-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide
—— tert-butyl 4-((5-(hydroxymethyl)-2-(methylthio)pyrimidin-4-yl)amino)piperidine-1-carboxylate 1222315-78-7 C16H26N4O3S
tert-butyl 4-((5-(hydroxymethyl)-2-(methylthio)pyrimidin-4-yl)amino)piperidine-1-carboxylate
—— 2-[(4-methyl-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carbonyl)amino]-N-(oxan-4-yl)-1,3-thiazole-4-carboxamide 1014694-97-3 C22H23N5O4S
2-[(4-methyl-1-oxo-3,4-dihydro-2H-pyrazino[1,2-a]indole-7-carbonyl)amino]-N-(oxan-4-yl)-1,3-thiazole-4-carboxamide
—— 6-(5-methyl-3-pyridin-2-yl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid ethyl ester 1159251-91-8 C17H16N4O4
6-(5-methyl-3-pyridin-2-yl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid ethyl ester
—— 4-chloro-N-(tetrahydro-2H-pyran-4-yl)benzenesulfonamide 1429647-66-4 C11H14ClNO3S
4-chloro-N-(tetrahydro-2H-pyran-4-yl)benzenesulfonamide
—— N-methyl-2-propylsulfanyl-N-tetrahydropyran-4-ylpyridine-3-carboxamide 1383624-87-0 C15H22N2O2S
N-methyl-2-propylsulfanyl-N-tetrahydropyran-4-ylpyridine-3-carboxamide
—— 6-(5-Methyl-3-pyridin-4-yl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide 1159251-64-5 C20H21N5O4
6-(5-Methyl-3-pyridin-4-yl-isoxazol-4-ylmethoxy)-pyridazine-3-carboxylic acid (tetrahydro-pyran-4-yl)-amide
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-pyran-4-yl)-3-trifluoromethyl-benzamide 1201692-74-1 C26H29F5N6O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-pyran-4-yl)-3-trifluoromethyl-benzamide
—— [7-(2,6-Difluorophenyl)-2-(tetrahydro-pyran-4-ylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-(4-fluorophenyl)-methanone 1001128-48-8 C24H19F3N4O2
[7-(2,6-Difluorophenyl)-2-(tetrahydro-pyran-4-ylamino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]-(4-fluorophenyl)-methanone
—— N-(3-chlorophenyl)-4-[2-[(tetrahydro-2H-pyran-4-yl)amino]-4-pyrimidinyl]-1,3,5-triazin-2-amine 1150110-19-2 C18H18ClN7O
N-(3-chlorophenyl)-4-[2-[(tetrahydro-2H-pyran-4-yl)amino]-4-pyrimidinyl]-1,3,5-triazin-2-amine
—— 2-(trimethylsilyl)-1,3-benzodithiole 175167-20-1 C10H14S2Si
2-(trimethylsilyl)-1,3-benzodithiole
—— 7,8-[<sup>2</sup>H<sub>4</sub>]-2-chloro-3-(3-chloro-4-methoxybenzyl)-5-ethyl-7,8-dihydro-3H-imidazo[2,1-b]purin-4(5H)-one 1542204-52-3 C17H17Cl2N5O2
7,8-[<sup>2</sup>H<sub>4</sub>]-2-chloro-3-(3-chloro-4-methoxybenzyl)-5-ethyl-7,8-dihydro-3H-imidazo[2,1-b]purin-4(5H)-one
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-82-1 C27H34F2N6O4
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethoxy-N-(tetrahydro-pyran-4-yl)-benzamide