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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R,3R,4R,5R)-2-(4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-3-fluoro-4-hydroxy-5-(hydroxymethyl)-3-methyloxolane-2-carbonitrile 1273029-46-1 C12H13FN6O3
(2R,3R,4R,5R)-2-(4-aminoimidazo[2,1-f][1,2,4]triazin-7-yl)-3-fluoro-4-hydroxy-5-(hydroxymethyl)-3-methyloxolane-2-carbonitrile
—— trans-{4-[4-(4-fluorophenyl)-2-methylsulfanyl-1H-imidazol-5-yl]pyridin-2-yl}-(4-methylcyclohexyl)amine 1041850-68-3 C22H25FN4S
trans-{4-[4-(4-fluorophenyl)-2-methylsulfanyl-1H-imidazol-5-yl]pyridin-2-yl}-(4-methylcyclohexyl)amine
—— tert-butyl 3-(1-(7-(hydroxydimethylsilyl)-1-naphthoyl)piperidin-4-yl)benzylcarbamate 1431289-28-9 C30H38N2O4Si
tert-butyl 3-(1-(7-(hydroxydimethylsilyl)-1-naphthoyl)piperidin-4-yl)benzylcarbamate
—— 1'-(benzyl)-spiro[isobenzofuran-1(3H),4'-piperidin]-3-thione 1254981-82-2 C19H19NOS
1'-(benzyl)-spiro[isobenzofuran-1(3H),4'-piperidin]-3-thione
—— (S)-2-(benzyloxy)but-3-yn-1-ol 1429480-80-7 C11H12O2
(S)-2-(benzyloxy)but-3-yn-1-ol
—— 3-(2-fluoro-5-(5-(3,4,5-trichlorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)benzylamino)-3-oxopropanoic acid 1338473-79-2 C20H13Cl3F4N2O4
3-(2-fluoro-5-(5-(3,4,5-trichlorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)benzylamino)-3-oxopropanoic acid
—— (E)-5-(methylthio)-8-phenyl-7-styryl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene 1264117-41-0 C22H20OS
(E)-5-(methylthio)-8-phenyl-7-styryl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene
—— ethyl 2-(2-(((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)amino)ethoxy)-3-bromo-6-methyl-5-((methylsulfonyl)oxy)benzoate 1616290-25-5 C28H33BrN2O7S
ethyl 2-(2-(((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)amino)ethoxy)-3-bromo-6-methyl-5-((methylsulfonyl)oxy)benzoate
—— 7-(4-fluorophenyl)-5-(methylselanyl)-8-phenyl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene 1264117-36-3 C20H17FOSe
7-(4-fluorophenyl)-5-(methylselanyl)-8-phenyl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene
—— 5-cyclopropyl-4-(2,2-difluoroethoxy)pyridine-2-carboxylic acid hydrochloride 1613239-43-2 C11H11F2NO3*ClH
5-cyclopropyl-4-(2,2-difluoroethoxy)pyridine-2-carboxylic acid hydrochloride
—— (5Z)-5-({1-[4-bromo-2-(trifluoromethyl)benzyl]piperidin-4-yl}methylidene)-4-(prop-2-yn-1-ylamino)-1,3-thiazol-2(5H)-one 1422127-29-4 C20H19BrF3N3OS
(5Z)-5-({1-[4-bromo-2-(trifluoromethyl)benzyl]piperidin-4-yl}methylidene)-4-(prop-2-yn-1-ylamino)-1,3-thiazol-2(5H)-one
—— 4-((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)-9-bromo-7-isopropoxy-6-methyl-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one 1616290-27-7 C28H31BrN2O4
4-((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)-9-bromo-7-isopropoxy-6-methyl-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-one
—— benzyl 3-(tert-butoxycarbonylamino)-3-(2-ethoxy-2-oxoethyl)pyrrolidine-1-carboxylate 1613298-64-8 C21H30N2O6
benzyl 3-(tert-butoxycarbonylamino)-3-(2-ethoxy-2-oxoethyl)pyrrolidine-1-carboxylate
—— 4-{[2-(benzyloxy)-4,6-dimethylpyridin-3-yl]methyl}-6-methyl-9-[2-(methylamino)pyrimidin-5-yl]-7-(propan-2-yloxy)-3,4-dihydro-1,4-benzoxazepin-5(2H)-one 1616290-50-6 C33H37N5O4
4-{[2-(benzyloxy)-4,6-dimethylpyridin-3-yl]methyl}-6-methyl-9-[2-(methylamino)pyrimidin-5-yl]-7-(propan-2-yloxy)-3,4-dihydro-1,4-benzoxazepin-5(2H)-one
—— 3-benzoyloxetan-2-one 1403871-75-9 C10H8O3
3-benzoyloxetan-2-one
—— 4-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-6-methyl-5-oxo-7-(propan-2-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine-9-carbonitrile 1616286-79-3 C22H25N3O4
4-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-6-methyl-5-oxo-7-(propan-2-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine-9-carbonitrile
—— tert-butyl 3-(benzyloxycarbonylamino)-4-(4-methylpiperazin-1-yl)benzoate 1613475-25-4 C24H31N3O4
tert-butyl 3-(benzyloxycarbonylamino)-4-(4-methylpiperazin-1-yl)benzoate
—— 7-(4-bromophenyl)-5-(methylthio)-8-phenyl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene 1264117-34-1 C20H17BrOS
7-(4-bromophenyl)-5-(methylthio)-8-phenyl-3-oxa-bicyclo[4.2.0]octa-1(8),5-diene
—— 3-(2,2-dimethylpropanoyl)-4-hydroxy-2-(4-methoxyphenyl)-1-[4-(1,2-oxazol-3-yl)phenyl]-2H-pyrrol-5-one 1067183-14-5 C25H24N2O5
3-(2,2-dimethylpropanoyl)-4-hydroxy-2-(4-methoxyphenyl)-1-[4-(1,2-oxazol-3-yl)phenyl]-2H-pyrrol-5-one
—— ethyl 2-(2-(((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)((tert-butoxy)carbonyl)amino)ethoxy)-3-bromo-6-methyl-5-((methylsulfonyl)oxy)benzoate 1616290-23-3 C33H41BrN2O9S
ethyl 2-(2-(((2-(benzyloxy)-4,6-dimethylpyridin-3-yl)methyl)((tert-butoxy)carbonyl)amino)ethoxy)-3-bromo-6-methyl-5-((methylsulfonyl)oxy)benzoate
—— (3-(2-methoxyethoxy)-2-methylphenyl)methanol 1296309-22-2 C11H16O3
(3-(2-methoxyethoxy)-2-methylphenyl)methanol
—— 2-(2-chloro-6-fluorophenyl)-5-(4-methyl-6-(trifluoromethyl)pyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine 1612288-95-5 C20H12ClF4N3
2-(2-chloro-6-fluorophenyl)-5-(4-methyl-6-(trifluoromethyl)pyridin-3-yl)-1H-pyrrolo[2,3-b]pyridine
—— ethyl (Z)-2-[[(2S)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-3-methylbutanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-3-phenylprop-2-enoate 1050655-36-1 C33H44N4O8
ethyl (Z)-2-[[(2S)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-3-methylbutanoyl]amino]propanoyl]amino]-4-methylpentanoyl]amino]-3-phenylprop-2-enoate
—— [4-[4-[3-[[(2-Methylpropan-2-yl)oxycarbonylamino]methyl]phenyl]piperidine-1-carbonyl]-1-benzothiophen-2-yl]boronic acid 1411992-68-1 C26H31BN2O5S
[4-[4-[3-[[(2-Methylpropan-2-yl)oxycarbonylamino]methyl]phenyl]piperidine-1-carbonyl]-1-benzothiophen-2-yl]boronic acid
—— ethyl (Z)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-3-phenylprop-2-enoate 1050655-38-3 C37H52N4O7
ethyl (Z)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]-3-phenylprop-2-enoate
—— 5-bromo-4-(cyclopropylmethoxy)picolinic acid 1613238-35-9 C10H10BrNO3
5-bromo-4-(cyclopropylmethoxy)picolinic acid
—— allyl 5-[(4,6-dimethoxypyrimidin-2-yl)oxy]-2-methylindol-4-carboxylate 155012-63-8 C19H19N3O5
allyl 5-[(4,6-dimethoxypyrimidin-2-yl)oxy]-2-methylindol-4-carboxylate
—— [4-[N-(3-methylphenyl)-4-[4-(N-(3-methylphenyl)anilino)phenyl]anilino]phenyl]methanol 1429193-85-0 C39H34N2O
[4-[N-(3-methylphenyl)-4-[4-(N-(3-methylphenyl)anilino)phenyl]anilino]phenyl]methanol
—— 4-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyridine 1612287-99-6 C13H17BF3NO2
4-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)pyridine
—— ethyl 6-hydroxy-2-methyl-3-[(methylsulfonyl)oxy]benzoate 1616290-21-1 C11H14O6S
ethyl 6-hydroxy-2-methyl-3-[(methylsulfonyl)oxy]benzoate
—— phenyl 2,4-di-O-benzyl-3,6-O-(di-tert-butylsilylene)-1-thio-α-D-mannopyranoside 1447727-62-9 C34H44O5SSi
phenyl 2,4-di-O-benzyl-3,6-O-(di-tert-butylsilylene)-1-thio-α-D-mannopyranoside
—— 2-(Acetylmethylamino)-5-phenyl-Δ<sup>2</sup>-1,3,4-thiadiazole 14537-59-8 C11H11N3OS
2-(Acetylmethylamino)-5-phenyl-Δ<sup>2</sup>-1,3,4-thiadiazole
—— 4-[(cyclopropylmethyl)amino]-3-nitropyridin-2(1H)-one 1031340-04-1 C9H11N3O3
4-[(cyclopropylmethyl)amino]-3-nitropyridin-2(1H)-one
—— Ethyl 3-(2-benzoyl-4-bromophenyl)-2-diazo-3-oxopropanoate 1373347-21-7 C18H13BrN2O4
Ethyl 3-(2-benzoyl-4-bromophenyl)-2-diazo-3-oxopropanoate
—— 5-chloro-2,3-dihydro-[1,4]dioxino[2,3-d]pyridazine 1313733-62-8 C6H5ClN2O2
5-chloro-2,3-dihydro-[1,4]dioxino[2,3-d]pyridazine
—— sodium 3-(2-(2,3,4-trimethoxybenzamido)ethyl)-1H-1,2,4-triazole-5-carboxylate 1613253-85-2 C15H17N4O6*Na
sodium 3-(2-(2,3,4-trimethoxybenzamido)ethyl)-1H-1,2,4-triazole-5-carboxylate
—— 2-methylpropyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-cyano-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate 1491026-71-1 C24H32N5O8P
2-methylpropyl (2S)-2-[[[(2R,3S,4R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-4-cyano-3-hydroxy-4-methyloxolan-2-yl]methoxy-phenoxyphosphoryl]amino]propanoate
—— cyclopropylmethyl-(2,3-dihydro-[1,4]dioxino[2,3-d]pyridazin-5-yl)-amine 1313733-65-1 C10H13N3O2
cyclopropylmethyl-(2,3-dihydro-[1,4]dioxino[2,3-d]pyridazin-5-yl)-amine
—— 3-cyclopropyl-2-{6-[(4-fluorophenyl)(4-methylpiperidin-1-yl)methyl]-4'-(trifluoromethyl)biphenyl-3-yl}propanoic acid 1257397-19-5 C32H33F4NO2
3-cyclopropyl-2-{6-[(4-fluorophenyl)(4-methylpiperidin-1-yl)methyl]-4'-(trifluoromethyl)biphenyl-3-yl}propanoic acid
—— (E)-N-(cyclopropylmethyl)-2-(1-(4-(trifluoromethoxy)phenylsulfonyl)piperidin-3-ylidene)acetamide 1246449-18-2 C18H21F3N2O4S
(E)-N-(cyclopropylmethyl)-2-(1-(4-(trifluoromethoxy)phenylsulfonyl)piperidin-3-ylidene)acetamide
—— N-(tert-butyl)-N,N'-dimethylguanidine 1189055-86-4 C7H17N3
N-(tert-butyl)-N,N'-dimethylguanidine
—— [4-Oxo-3-(3-pyridin-2-yl-[1,2,4]oxadiazol-5-ylmethyl)-3,4-dihydro-phthalazin-1-yl]-acetic acid 110703-54-3 C18H13N5O4
[4-Oxo-3-(3-pyridin-2-yl-[1,2,4]oxadiazol-5-ylmethyl)-3,4-dihydro-phthalazin-1-yl]-acetic acid
—— ethyl 1-formyl-5-hydroxy-5-(1,1-dimethylethyl)-4,5-dihydro-1H-pyrazole-3-carboxylate 1447673-57-5 C11H18N2O4
ethyl 1-formyl-5-hydroxy-5-(1,1-dimethylethyl)-4,5-dihydro-1H-pyrazole-3-carboxylate
—— (2E,6E,10E)-3,7,11-(15-d<sub>3</sub>)-tetramethylhexadeca-(14-d<sub>3</sub>)-2,6,10,14-tetraen-1-ol 1448620-49-2 C20H34O
(2E,6E,10E)-3,7,11-(15-d<sub>3</sub>)-tetramethylhexadeca-(14-d<sub>3</sub>)-2,6,10,14-tetraen-1-ol
—— ethyl (E)-3-[(3S)-2-[(2S)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-3-methylbutanoyl]amino]propanoyl]amino]-4-methylpentanoyl]-3,4-dihydro-1H-isoquinolin-3-yl]prop-2-enoate 1050655-55-4 C36H48N4O8
ethyl (E)-3-[(3S)-2-[(2S)-2-[[(2S)-3-hydroxy-2-[[(2S)-2-[(3-hydroxy-2-methylbenzoyl)amino]-3-methylbutanoyl]amino]propanoyl]amino]-4-methylpentanoyl]-3,4-dihydro-1H-isoquinolin-3-yl]prop-2-enoate
—— 3-Tert-butyl-4-(2-methoxyphenyl)-5-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-2,4-dihydropyrrolo[3,4-c]pyrazol-6-one 1067183-32-7 C25H25N5O3
3-Tert-butyl-4-(2-methoxyphenyl)-5-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-2,4-dihydropyrrolo[3,4-c]pyrazol-6-one
—— 5-benzyloxy-1-cyclopropylmethyl-2-difluoromethyl-1H-pyridin-4-one 1064076-93-2 C17H17F2NO2
5-benzyloxy-1-cyclopropylmethyl-2-difluoromethyl-1H-pyridin-4-one
—— N-(cyclopropylmethyl)pivalamide 1090891-87-4 C9H17NO
N-(cyclopropylmethyl)pivalamide
—— 2-{[1-(4-{[3-({3-[(DOTA-Ahx)-methyl-amino]-propyl}-methyl-amino)-propyl]-methyl-carbamoyl}-2-isopropyl-phenyl)-5-(2,6-dimethoxy-phenyl)-1H-pyrazole-3-carbonyl]-amino}-adamantane-2-carboxylic acid 1613332-64-1 C64H95N11O14
2-{[1-(4-{[3-({3-[(DOTA-Ahx)-methyl-amino]-propyl}-methyl-amino)-propyl]-methyl-carbamoyl}-2-isopropyl-phenyl)-5-(2,6-dimethoxy-phenyl)-1H-pyrazole-3-carbonyl]-amino}-adamantane-2-carboxylic acid
—— 2-{6-[(4-fluorophenyl)(4-methylpiperidin-1-yl)methyl]-4'-(trifluoromethyl)biphenyl-3-yl}-3-methylbutanoic acid 1257395-34-8 C31H33F4NO2
2-{6-[(4-fluorophenyl)(4-methylpiperidin-1-yl)methyl]-4'-(trifluoromethyl)biphenyl-3-yl}-3-methylbutanoic acid