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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-(3-isopropyl-1-methyl-1H-pyrazol-5-yl)-2-(3-methyl-1-tosyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-ol 1421253-83-9 C30H32N6O3S
6-(3-isopropyl-1-methyl-1H-pyrazol-5-yl)-2-(3-methyl-1-tosyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-ol
—— (2S)-1-({3-[4-(cyclobutyloxy)furo[3,2-c]pyridin-2-yl]imidazo[1,2-b]pyridazin-6-yl}oxy)propan-2-amine 1443500-08-0 C20H21N5O3
(2S)-1-({3-[4-(cyclobutyloxy)furo[3,2-c]pyridin-2-yl]imidazo[1,2-b]pyridazin-6-yl}oxy)propan-2-amine
—— 7-Oxa-10,13,18,20,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(19),2(22),3,5,14(21),15,17-heptaen-9-one 1429323-41-0 C16H15N5O2
7-Oxa-10,13,18,20,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(19),2(22),3,5,14(21),15,17-heptaen-9-one
—— 3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-tosyl-1H-indole 1421252-96-1 C22H26BNO4S
3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1-tosyl-1H-indole
—— 2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-3-(morpholin-4-yl)-propan-1-amine 1426928-40-6 C21H23N5O3
2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-3-(morpholin-4-yl)-propan-1-amine
—— tert-butyl [2-(6-{[(2S)-2-aminopropyl]oxy}imidazo[1,2-b]pyridazin-3-yl)-furo[3,2-c]pyridin-4-yl]ethylcarbamate 1443500-06-8 C23H28N6O4
tert-butyl [2-(6-{[(2S)-2-aminopropyl]oxy}imidazo[1,2-b]pyridazin-3-yl)-furo[3,2-c]pyridin-4-yl]ethylcarbamate
—— 2-hydroxy-1-(1-p-tolyl-cyclopropyl)ethanone 1067187-86-3 C12H14O2
2-hydroxy-1-(1-p-tolyl-cyclopropyl)ethanone
—— 5-(4-fluorobenzyl)-1-methyl-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid 1706456-27-0 C16H17FN2O2
5-(4-fluorobenzyl)-1-methyl-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid
—— 7-[4-(2-aminopropan-2-yl)phenyl]-5-(ethylamino)-3-methyl-3H,4H-pyrido[4,3-d]pyrimidin-4-one 1263076-97-6 C19H23N5O
7-[4-(2-aminopropan-2-yl)phenyl]-5-(ethylamino)-3-methyl-3H,4H-pyrido[4,3-d]pyrimidin-4-one
—— (R)-1-(4-(6-benzyl-2-(3-methyl-1-tosyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-3-methylpiperazin-1-yl)ethanone 1421253-53-3 C37H40N6O3S
(R)-1-(4-(6-benzyl-2-(3-methyl-1-tosyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-3-methylpiperazin-1-yl)ethanone
—— 2-(1-(4-fluorophenyl)cyclopropyl)-3-hydroxy-6,8-dimethylquinoline-4-carboxylic acid 1067186-88-2 C21H18FNO3
2-(1-(4-fluorophenyl)cyclopropyl)-3-hydroxy-6,8-dimethylquinoline-4-carboxylic acid
—— methyl 3-(6-phenylindolizin-8-yl)benzoate 1418760-48-1 C22H17NO2
methyl 3-(6-phenylindolizin-8-yl)benzoate
—— 3-methyl-1H-indole-4-carbonitrile 1425933-49-8 C10H8N2
3-methyl-1H-indole-4-carbonitrile
—— N-(3-methylbutyl)-4-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide 1330594-15-4 C24H32N6O
N-(3-methylbutyl)-4-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide
—— tert-butyl 4-((2-chloro-4-morpholinofuro[3,2-d]pyrimidin-6-yl)methyl) piperazine-1-carboxylate 1093066-87-5 C20H28ClN5O4
tert-butyl 4-((2-chloro-4-morpholinofuro[3,2-d]pyrimidin-6-yl)methyl) piperazine-1-carboxylate
—— (R)-1-(3-methyl-4-(2-(3-methyl-1-tosyl-1H-indol-4-yl)-6-(2-methyl-5-(3-methyloxetan-3-yl)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl)ethanone 1421253-56-6 C41H46N6O4S
(R)-1-(3-methyl-4-(2-(3-methyl-1-tosyl-1H-indol-4-yl)-6-(2-methyl-5-(3-methyloxetan-3-yl)phenyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)piperazin-1-yl)ethanone
—— 2-(1-(4-chlorophenyl)cyclopropyl)-3-hydroxy-6,8-dimethylquinoline-4-carboxylic acid 1067186-26-8 C21H18ClNO3
2-(1-(4-chlorophenyl)cyclopropyl)-3-hydroxy-6,8-dimethylquinoline-4-carboxylic acid
—— (2S)-1-{[3-(4-ethoxyfuro[3,2-c]pyridin-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-propan-2-amine 1443499-99-7 C18H19N5O3
(2S)-1-{[3-(4-ethoxyfuro[3,2-c]pyridin-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-propan-2-amine
—— 1-benzo[b]thiophen-3-yl-3-[4-(4-trifluoromethylbenzenesulfonyl)piperazin-1-yl]propan-1-one 1291057-95-8 C22H21F3N2O3S2
1-benzo[b]thiophen-3-yl-3-[4-(4-trifluoromethylbenzenesulfonyl)piperazin-1-yl]propan-1-one
—— 2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-cyclopropylethanamine 1426928-39-3 C19H18N4O2
2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-cyclopropylethanamine
—— 4-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-methylbutan-2-amine 1426928-21-3 C19H20N4O2
4-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-methylbutan-2-amine
—— (1S)-2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-1-phenylethanamine 1426928-24-6 C22H18N4O2
(1S)-2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-1-phenylethanamine
—— 3-(1-benzofuran-2-yl)-6-[3-(methylsulfonyl)propoxy]imidazolo[1,2-b]pyridazine 1428346-82-0 C18H17N3O4S
3-(1-benzofuran-2-yl)-6-[3-(methylsulfonyl)propoxy]imidazolo[1,2-b]pyridazine
—— 4-[2-(2,3-difluorophenyl)pyrimidin-4-yl]-N-pyridin-3-ylpiperazine-1-carboxamide 1143576-94-6 C20H18F2N6O
4-[2-(2,3-difluorophenyl)pyrimidin-4-yl]-N-pyridin-3-ylpiperazine-1-carboxamide
—— {3-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}carbamic acid methyl ester 1330594-45-0 C20H24N6O2
{3-[6-(1-methylpiperidin-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}carbamic acid methyl ester
—— 2,6-bis(6-monoamino-β-cyclodextrinmethyl)pyridine 1238398-19-0 C91H147N3O68
2,6-bis(6-monoamino-β-cyclodextrinmethyl)pyridine
—— 3-[2-(isopentylamino)-4-pyridyl]-N-(1-methyl-4-piperidyl)imidazo[1,2-b]pyridazin-6-amine 1432056-60-4 C22H31N7
3-[2-(isopentylamino)-4-pyridyl]-N-(1-methyl-4-piperidyl)imidazo[1,2-b]pyridazin-6-amine
—— (1S)-2-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-1-(4-fluorophenyl)ethanamine 1426928-71-3 C22H17FN4O2
(1S)-2-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-1-(4-fluorophenyl)ethanamine
—— N-(2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-phenylethyl)-2,2-dimethylpropan-1-amine 1460197-50-5 C27H28N4O2
N-(2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-2-phenylethyl)-2,2-dimethylpropan-1-amine
—— 2-(6-{[(2S)-2-aminopropyl]oxy}imidazo[1,2-b]pyridazin-3-yl)-N-ethylfuro[3,2-c]pyridin-4-amine 1443500-07-9 C18H20N6O2
2-(6-{[(2S)-2-aminopropyl]oxy}imidazo[1,2-b]pyridazin-3-yl)-N-ethylfuro[3,2-c]pyridin-4-amine
—— 3,11-bis-(2-nitrobenzenesulfonyl)-7-tert-butyloxycarbonyl-3,7,11,17-tetraazabicyclo[11.3.1]heptadeca-1(16),13(17),14-triene 1191071-98-3 C30H36N6O10S2
3,11-bis-(2-nitrobenzenesulfonyl)-7-tert-butyloxycarbonyl-3,7,11,17-tetraazabicyclo[11.3.1]heptadeca-1(16),13(17),14-triene
—— (1R)-2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-1-phenylethanamine 1426928-25-7 C22H18N4O2
(1R)-2-{[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-1-phenylethanamine
—— US9320737, III.7 1428346-88-6 C19H19N3O4S
US9320737, III.7
—— 3-hydroxy-2-phenyl-1,3-azaphosphorinane-3-oxide 1075800-02-0 C10H14NO2P
3-hydroxy-2-phenyl-1,3-azaphosphorinane-3-oxide
—— 3-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-3-(4-fluorophenyl)propan-1-amine 1426928-74-6 C23H19FN4O2
3-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-3-(4-fluorophenyl)propan-1-amine
—— {3-[6-(cyclopropylmethylamino)pyridin-3-yl]imidazo[1,2-b]pyridazin-6-yl}-(1-methylpiperidin-4-yl)amine 1330593-83-3 C21H27N7
{3-[6-(cyclopropylmethylamino)pyridin-3-yl]imidazo[1,2-b]pyridazin-6-yl}-(1-methylpiperidin-4-yl)amine
—— (2S)-1-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-3-phenylpropan-2-amine 1426928-60-0 C23H20N4O2
(2S)-1-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-3-phenylpropan-2-amine
—— (1S)-2-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-1-(4-chlorophenyl)ethanamine 1426928-72-4 C22H17ClN4O2
(1S)-2-[3-(1-benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-1-(4-chlorophenyl)ethanamine
—— 4-bromo-3-methyl-1-tosyl-1H-indole 1421254-71-8 C16H14BrNO2S
4-bromo-3-methyl-1-tosyl-1H-indole
—— 3-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-2-phenylpropan-1-amine 1426928-62-2 C23H20N4O2
3-[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy-2-phenylpropan-1-amine
—— N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(4-methylsulfonylphenyl)-1,2,4-triazole-3-carboxamide trifluoroacetate 1613021-36-5 C2HF3O2*C20H20N8O3S
N-[(3S)-1-imidazo[1,2-a]pyrazin-8-ylpyrrolidin-3-yl]-1-(4-methylsulfonylphenyl)-1,2,4-triazole-3-carboxamide trifluoroacetate
—— (R)-2-[[7-(3-aminopyrrolidin-1-yl)-3-methyl-2-oxo-2,3-dihydroimidazo[4,5-b] pyridin-1-yl]methyl]benzonitrile trifluoroacetate 1314943-93-5 C2HF3O2*C19H20N6O
(R)-2-[[7-(3-aminopyrrolidin-1-yl)-3-methyl-2-oxo-2,3-dihydroimidazo[4,5-b] pyridin-1-yl]methyl]benzonitrile trifluoroacetate
—— 2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-3-(pyridin-4-yl)-propan-1-amine 1426928-64-4 C22H19N5O2
2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}-3-(pyridin-4-yl)-propan-1-amine
—— (1R,2R)-2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}cyclohexanamine 1426928-30-4 C20H20N4O2
(1R,2R)-2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}cyclohexanamine
—— 2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}hex-5-en-1-amine 1426928-37-1 C20H20N4O2
2-{[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}hex-5-en-1-amine
—— 4-[6-(cyclopentylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide 1330075-48-3 C23H26F2N6O
4-[6-(cyclopentylamino)imidazo[1,2-b]pyridazin-3-yl]-2-fluoro-N-[[(2S,4R)-4-fluoropyrrolidin-2-yl]methyl]benzamide
—— 1-[[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxymethyl]cyclopropan-1-amine 1426928-61-1 C18H16N4O2
1-[[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxymethyl]cyclopropan-1-amine
—— 1-({[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}methyl)cyclobutanamine 1426928-36-0 C19H18N4O2
1-({[3-(1-Benzofuran-2-yl)imidazo[1,2-b]pyridazin-6-yl]oxy}methyl)cyclobutanamine
—— 3-{methyl[4-(1-phenylpiperazin-4-yl)butyl]amino}phenol 1610999-04-6 C21H29N3O
3-{methyl[4-(1-phenylpiperazin-4-yl)butyl]amino}phenol
—— [3-(6-butylaminopyridin-3-yl)imidazo[1,2-b]pyridazin-6-yl]-(1-methylpiperidin-4-yl)amine 1330593-89-9 C21H29N7
[3-(6-butylaminopyridin-3-yl)imidazo[1,2-b]pyridazin-6-yl]-(1-methylpiperidin-4-yl)amine