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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methoxy-5-(3-(piperidin-1-yl)propoxy)aniline 1258492-32-8 C15H24N2O2
2-methoxy-5-(3-(piperidin-1-yl)propoxy)aniline
—— Trifluoro-methanesulfonic acid 3-biphenyl-4-ylmethyl-4-oxo-chroman-7-yl ester 179107-69-8 C23H17F3O5S
Trifluoro-methanesulfonic acid 3-biphenyl-4-ylmethyl-4-oxo-chroman-7-yl ester
—— 4-(4-aminopiperidin-1-yl)-2,2-diphenylbutanenitrile 1412903-11-7 C21H25N3
4-(4-aminopiperidin-1-yl)-2,2-diphenylbutanenitrile
—— ethyl {3-chloro-4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetate 1004513-88-5 C26H22ClF2NO6
ethyl {3-chloro-4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]phenyl}acetate
—— 6-(4-nitrophenyl)-1-tosylpiperidine-2,4-dione 1186526-43-1 C18H16N2O6S
6-(4-nitrophenyl)-1-tosylpiperidine-2,4-dione
—— 4-(4-phenylpiperazin-1-yl)isoquinoline-6-carboxamide 1235380-73-0 C20H20N4O
4-(4-phenylpiperazin-1-yl)isoquinoline-6-carboxamide
—— N<sup>3</sup>-(4-methoxyfumaroyl)-L-2,3-diaminopropanoyl-UPOC 130905-37-2 C18H23N5O11
N<sup>3</sup>-(4-methoxyfumaroyl)-L-2,3-diaminopropanoyl-UPOC
—— methyl 1-amino-3-(4-methylphenyl)-2-naphthoate 1581713-36-1 C19H17NO2
methyl 1-amino-3-(4-methylphenyl)-2-naphthoate
—— 2-benzyl-5-methoxy-4-[4-(trifluoromethyl)phenyl]-pyridazin-3(2H)-one 1345839-36-2 C19H15F3N2O2
2-benzyl-5-methoxy-4-[4-(trifluoromethyl)phenyl]-pyridazin-3(2H)-one
—— 4-(2-hydroxyethyl)-5-methyl-2-(3-methylphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-one 1001077-44-6 C12H15N3O2
4-(2-hydroxyethyl)-5-methyl-2-(3-methylphenyl)-2,4-dihydro-3H-1,2,4-triazol-3-one
—— (1S,3S,5R)-2-(tert-butoxycarbonyl)-6,6-difluoro-2-azabicyclo[3.1.0]hexane-3-carboxylic acid 1400990-36-4 C11H15F2NO4
(1S,3S,5R)-2-(tert-butoxycarbonyl)-6,6-difluoro-2-azabicyclo[3.1.0]hexane-3-carboxylic acid
—— bis-(fluorodiphenylsilyl)mercury 104925-64-6 C24H20F2HgSi2
bis-(fluorodiphenylsilyl)mercury
—— Eptastigmine tartrate 121652-76-4 C25H39N3O8
Eptastigmine tartrate
—— (8S)-2-(morpholin-4-yl)-8-(trifluoromethyl)-9-[4-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one 1260585-58-7 C19H18F6N4O2
(8S)-2-(morpholin-4-yl)-8-(trifluoromethyl)-9-[4-(trifluoromethyl)phenyl]-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one
—— N-((R)-((S)-3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide 1398511-76-6 C18H14Cl2N2O6S
N-((R)-((S)-3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide
—— ethyl {4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-3-fluorophenyl}acetate 1004513-80-7 C26H22F3NO6
ethyl {4-[4-[(2,2-difluoroethyl)oxy]-9-(ethyloxy)-1,3-dioxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-3-fluorophenyl}acetate
—— 6-Bromo-2-(phenylsulfonyl)-2,3-dihydroisoquinoline-4(1H)-one 1235382-79-2 C15H12BrNO3S
6-Bromo-2-(phenylsulfonyl)-2,3-dihydroisoquinoline-4(1H)-one
—— 2-(4-nitrophenyl)-4-phenylsulfonyl-1-tosyl-2,5-dihydro-1H-pyrrole 1192593-18-2 C23H20N2O6S2
2-(4-nitrophenyl)-4-phenylsulfonyl-1-tosyl-2,5-dihydro-1H-pyrrole
—— ethyl (3-chloro-4-{4-(ethyloxy)-3-hydroxy-1-oxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetate 1004514-44-6 C26H23ClF3NO6
ethyl (3-chloro-4-{4-(ethyloxy)-3-hydroxy-1-oxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetate
—— (Z,Z)-5-(3-chloro-4-hydroxybenzylidene)-2-isopropylimino-3-m-tolyl-thiazolidin-4-one 1228116-92-4 C20H19ClN2O2S
(Z,Z)-5-(3-chloro-4-hydroxybenzylidene)-2-isopropylimino-3-m-tolyl-thiazolidin-4-one
—— Example 41 1347434-80-3 C26H28ClF3N2O3S
Example 41
—— 2-cyclopropyl-propane-1,2-diamine 1021392-54-0 C6H14N2
2-cyclopropyl-propane-1,2-diamine
—— methyl 1-amino-3-(2-methylphenyl)-2-naphthoate 1581713-37-2 C19H17NO2
methyl 1-amino-3-(2-methylphenyl)-2-naphthoate
—— 6-(furan-2-yl)-1-tosylpiperidine-2,4-dione 1186526-48-6 C16H15NO5S
6-(furan-2-yl)-1-tosylpiperidine-2,4-dione
—— (3-chloro-4-{1,3-dioxo-4,9-bis[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid 1004514-36-6 C24H14ClF6NO6
(3-chloro-4-{1,3-dioxo-4,9-bis[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid
—— 1-{5-[2-oxo-2-(4-trifluoromethylphenyl)ethyl]furan-2-yl}propan-2-one 1195869-76-1 C16H13F3O3
1-{5-[2-oxo-2-(4-trifluoromethylphenyl)ethyl]furan-2-yl}propan-2-one
—— (4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}-3-fluorophenyl)acetic acid 1004514-40-2 C24H17F4NO6
(4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}-3-fluorophenyl)acetic acid
—— methyl 3-((tert-butyldimethylsilyl)oxy)-2-(N-(prop-2-yn-1-yl)vinylsulfonamido)propanoate 1357283-08-9 C15H27NO5SSi
methyl 3-((tert-butyldimethylsilyl)oxy)-2-(N-(prop-2-yn-1-yl)vinylsulfonamido)propanoate
—— (4R,5S)-4-(methoxycarbonyl)-5-(4-nitrophenyl)-N-tosyl-2-imidazoline 1245746-93-3 C18H17N3O6S
(4R,5S)-4-(methoxycarbonyl)-5-(4-nitrophenyl)-N-tosyl-2-imidazoline
—— 3-(2-(2,2,2-trifluoroethoxy)-phenyl)-4-fluorobenzoic acid 1055983-96-4 C15H10F4O3
3-(2-(2,2,2-trifluoroethoxy)-phenyl)-4-fluorobenzoic acid
—— (S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-diphenylcyclopent-1-enyl)methyl)benzenesulfonamide 1397711-83-9 C31H26N2O5S
(S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-diphenylcyclopent-1-enyl)methyl)benzenesulfonamide
—— 4-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole 1257078-38-8 C9H14N4O2
4-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-pyrazole
—— (S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-bis(4-(trifluoromethyl)phenyl)cyclopent-1-enyl)methyl)benzenesulfonamide 1397711-97-5 C33H24F6N2O5S
(S)-4-methyl-N-((4-nitrophenyl)(5-oxo-4,4-bis(4-(trifluoromethyl)phenyl)cyclopent-1-enyl)methyl)benzenesulfonamide
—— ethyl 6-methyl-5-{[(4-methylphenyl)sulfonyl]amino}-4-oxo-5-azaspiro[2.4]hept-6-ene-7-carboxylate 1177445-87-2 C17H20N2O5S
ethyl 6-methyl-5-{[(4-methylphenyl)sulfonyl]amino}-4-oxo-5-azaspiro[2.4]hept-6-ene-7-carboxylate
—— 4-[(4-nitro-1H-pyrazol-1-yl)methyl]pyridine 1006571-33-0 C9H8N4O2
4-[(4-nitro-1H-pyrazol-1-yl)methyl]pyridine
—— (3-chloro-4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid 1004514-42-4 C24H17ClF3NO6
(3-chloro-4-{4-(ethyloxy)-1,3-dioxo-9-[(2,2,2-trifluoroethyl)oxy]-1,3-dihydro-2H-benzo[f]isoindol-2-yl}phenyl)acetic acid
—— 4-(2-fluorophenyl)-2-phenyl-5-(phenyl(tosyl)methyl)oxazole 1432969-19-1 C29H22FNO3S
4-(2-fluorophenyl)-2-phenyl-5-(phenyl(tosyl)methyl)oxazole
—— Example 36 1347137-33-0 C32H33ClF3N3O3
Example 36
—— dimethyl 2-(furan-2-yl)-1-tosyl-5-(trifluoromethyl)-1H-pyrrole-3,4-dicarboxylate 1619266-88-4 C20H16F3NO7S
dimethyl 2-(furan-2-yl)-1-tosyl-5-(trifluoromethyl)-1H-pyrrole-3,4-dicarboxylate
—— N-((3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(2-fluorophenyl)methyl)-4-methylbenzenesulfonamide 1398511-77-7 C18H14Cl2FNO4S
N-((3,4-dichloro-5-oxo-2,5-dihydrofuran-2-yl)(2-fluorophenyl)methyl)-4-methylbenzenesulfonamide
—— 5-[3-chloro-4-(2-cyclohexylethoxy)benzylidene]-1,3-thiazolidine-2,4-dione 1239610-72-0 C18H20ClNO3S
5-[3-chloro-4-(2-cyclohexylethoxy)benzylidene]-1,3-thiazolidine-2,4-dione
—— N-((S)-((R)-4-isopropyl-5-oxo-2-phenyl-4,5-dihydrooxazol-4-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide 1207097-64-0 C26H25N3O6S
N-((S)-((R)-4-isopropyl-5-oxo-2-phenyl-4,5-dihydrooxazol-4-yl)(4-nitrophenyl)methyl)-4-methylbenzenesulfonamide
—— methyl 4-({2-[(2-hydroxypropyl)(pyridin-2-ylsulfonyl)amino]-4,5-dimethylphenoxy}methyl)benzoate 1202394-18-0 C25H28N2O6S
methyl 4-({2-[(2-hydroxypropyl)(pyridin-2-ylsulfonyl)amino]-4,5-dimethylphenoxy}methyl)benzoate
—— 4-(adamantan-1-ylaminomethyl)-2-chlorophenol 1304584-74-4 C17H22ClNO
4-(adamantan-1-ylaminomethyl)-2-chlorophenol
—— [4-(4-Acryloylamino-piperidin-1-ylmethyl)-phenyl]carbamic acid benzyl ester 1392490-92-4 C23H27N3O3
[4-(4-Acryloylamino-piperidin-1-ylmethyl)-phenyl]carbamic acid benzyl ester
—— (5R)-5-(4-nitropyrazol-1-yl)piperidin-2-one 1201935-66-1 C8H10N4O3
(5R)-5-(4-nitropyrazol-1-yl)piperidin-2-one
—— 15,24-Dioxa-3,7,18,21-tetraaza-tricyclo[23.4.0.0<sup>9,14</sup>]nonacosa-1(25),9(14),10,12,26,28-hexaene-17,22-dione 141944-94-7 C23H30N4O4
15,24-Dioxa-3,7,18,21-tetraaza-tricyclo[23.4.0.0<sup>9,14</sup>]nonacosa-1(25),9(14),10,12,26,28-hexaene-17,22-dione
—— (3,4-dihydro-2H-1,5-benzodioxepin-2-yl)methylamine 1022974-16-8 C9H11NO2
(3,4-dihydro-2H-1,5-benzodioxepin-2-yl)methylamine
—— 2-[(Z)-2-(4-Methoxy-phenylamino)-1-nitro-vinyl]-benzene-1,4-diol 134387-68-1 C15H14N2O5
2-[(Z)-2-(4-Methoxy-phenylamino)-1-nitro-vinyl]-benzene-1,4-diol
—— —— 1198424-80-4 C23H43ClSi2