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中文名称 英文名称 CAS号 化学式 结构式图片
—— acetylamino-(2-acetylamino-4-methyl-thiazol-5-ylmethyl)-malonic acid diethyl ester 101437-42-7 C16H23N3O6S
acetylamino-(2-acetylamino-4-methyl-thiazol-5-ylmethyl)-malonic acid diethyl ester
—— phenyl-acetic acid-[2-(2-oxo-pyrrolidin-3-yl)-anilide] 101792-87-4 C18H18N2O2
phenyl-acetic acid-[2-(2-oxo-pyrrolidin-3-yl)-anilide]
—— methyl 4-hydroxy-1-(4-methoxyphenyl)-5-oxo-2-phenyl-4-(trifluoromethyl)-4,5-dihydro-1H-pyrrole-3-carboxylate 1616563-16-6 C20H16F3NO5
methyl 4-hydroxy-1-(4-methoxyphenyl)-5-oxo-2-phenyl-4-(trifluoromethyl)-4,5-dihydro-1H-pyrrole-3-carboxylate
—— 6-Methoxy-4-oxo-tetrahydro-pyran-2-carboxylic acid butyl ester 105896-29-5 C11H18O5
6-Methoxy-4-oxo-tetrahydro-pyran-2-carboxylic acid butyl ester
—— ethyl 2-(2-chloro-5-([(1-trifluoromethylcyclopropanecarbonyl)amino]methyl)phenylamino)-6-(2,2-difluoroethoxy)-1H-benzimidazole-5-carboxylate 1242269-51-7 C24H22ClF5N4O4
ethyl 2-(2-chloro-5-([(1-trifluoromethylcyclopropanecarbonyl)amino]methyl)phenylamino)-6-(2,2-difluoroethoxy)-1H-benzimidazole-5-carboxylate
—— methyl 3α-acetoxy-7α-hydroxy-19-trimethylacetoxy-5β-cholan-24-oate 171524-63-3 C32H52O7
methyl 3α-acetoxy-7α-hydroxy-19-trimethylacetoxy-5β-cholan-24-oate
—— 1-(4-(5-(4-cyclopropoxyphenyl)thiazol-2-yl)benzyl)azetidine-3-carboxylic acid 1444255-77-9 C23H22N2O3S
1-(4-(5-(4-cyclopropoxyphenyl)thiazol-2-yl)benzyl)azetidine-3-carboxylic acid
—— (3S)-7-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]-3-[5-(2-methoxyphenyl)-1H-imidazol-2-yl]-2,3-dihydro-5(1H)-indolizinone 1445864-53-8 C25H20ClN7O2
(3S)-7-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]-3-[5-(2-methoxyphenyl)-1H-imidazol-2-yl]-2,3-dihydro-5(1H)-indolizinone
—— 2-([1,4]dioxan-2-ylmethoxy)-9-(1-methyl-1H-indol-5-yl)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one 1445846-56-9 C26H25N3O4
2-([1,4]dioxan-2-ylmethoxy)-9-(1-methyl-1H-indol-5-yl)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one
—— 3-methyl-2-(4-phenyl-6-(phenylamino)-1,3,5-triazin-2-ylamino)butan-1-ol 1446502-72-2 C20H23N5O
3-methyl-2-(4-phenyl-6-(phenylamino)-1,3,5-triazin-2-ylamino)butan-1-ol
—— tert-butyl N-[8-tert-butyl-2-[(8,8-dioxo-1,4-dioxa-8lambda6-thiaspiro[4.5]decan-6-yl)methylcarbamoyl]-4-methylquinolin-6-yl]-N-(2,2,2-trifluoroethyl)carbamate 1443929-33-6 C30H40F3N3O7S
tert-butyl N-[8-tert-butyl-2-[(8,8-dioxo-1,4-dioxa-8lambda6-thiaspiro[4.5]decan-6-yl)methylcarbamoyl]-4-methylquinolin-6-yl]-N-(2,2,2-trifluoroethyl)carbamate
—— N-[(2S)-6-[[(1S,4S)-5-acetyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-4-[[(2S)-oxolan-2-yl]methoxy]benzamide 1119257-76-9 C30H37N3O4
N-[(2S)-6-[[(1S,4S)-5-acetyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl]-1,2,3,4-tetrahydronaphthalen-2-yl]-4-[[(2S)-oxolan-2-yl]methoxy]benzamide
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[[5-(difluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229657-16-2 C22H17ClF2N10O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-5-[[5-(difluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
—— 2-(heptoxymethyl)-3-methyl-1H-quinolin-4-one 1135025-76-1 C18H25NO2
2-(heptoxymethyl)-3-methyl-1H-quinolin-4-one
—— 4-hexyl-2-phenethyl-1,2,3,4-tetrahydroisoquinoline 1312343-61-5 C23H31N
4-hexyl-2-phenethyl-1,2,3,4-tetrahydroisoquinoline
—— 2-(thiophen-2-ylmethylene)-1-oxaspiro[3.5]nonan-3-one 1396787-24-8 C13H14O2S
2-(thiophen-2-ylmethylene)-1-oxaspiro[3.5]nonan-3-one
—— 1-(1-(1H-benzimidazol-2-yl)ethylideneamino)-6-(benzylideneamino)-4-(2-hydroxyphenyl)-2-oxo-1,2-dihydropyridine-3,5-dicarbonitrile 1338245-67-2 C29H19N7O2
1-(1-(1H-benzimidazol-2-yl)ethylideneamino)-6-(benzylideneamino)-4-(2-hydroxyphenyl)-2-oxo-1,2-dihydropyridine-3,5-dicarbonitrile
—— N3-(3-(dimethylamino)phenyl)-1H-1,2,4-triazole-3,5-diamine 1261496-31-4 C10H14N6
N3-(3-(dimethylamino)phenyl)-1H-1,2,4-triazole-3,5-diamine
—— 2-(4-chlorobutyl)tetrahydrothiophene 133387-61-8 C8H15ClS
2-(4-chlorobutyl)tetrahydrothiophene
—— 6-Ethoxy-8-phenyl-1,3,4,10a-tetrahydro-9H-2-oxa-4a,5-diaza-phenanthrene-7,10,10-tricarbonitrile 143815-82-1 C22H19N5O2
6-Ethoxy-8-phenyl-1,3,4,10a-tetrahydro-9H-2-oxa-4a,5-diaza-phenanthrene-7,10,10-tricarbonitrile
—— 2,5-dichloro-N-[3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl) phenyl]benzenesulfonamide 1314069-71-0 C18H19BCl3NO4S
2,5-dichloro-N-[3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl) phenyl]benzenesulfonamide
—— 3-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]sulfonyl-N-(4-fluoro-3-methylphenyl)benzamide 1445786-61-7 C27H29FN2O4S
3-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]sulfonyl-N-(4-fluoro-3-methylphenyl)benzamide
—— (R)-(2-(1-methyl-1H-indazol-5-yl)-1-(3-(2-oxobenzo[d]thiazol-3(2H)-yl)propanamido)ethyl)boronic acid 1444010-51-8 C21H23BN6O3
(R)-(2-(1-methyl-1H-indazol-5-yl)-1-(3-(2-oxobenzo[d]thiazol-3(2H)-yl)propanamido)ethyl)boronic acid
—— 2-[[(2R)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-heptoxyphenyl)pyrimidin-2-yl]phenyl]propanoyl]amino]acetic acid 1443791-78-3 C39H46N4O5
2-[[(2R)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-heptoxyphenyl)pyrimidin-2-yl]phenyl]propanoyl]amino]acetic acid
—— (±)-(3-{5-fluoro-2-[3-(6-methylpyridin-2-yl)butyryl]-1,2,3,4-tetrahydroisoquinolin-8-yl}-4-isopropoxyphenyl)acetic acid 1445887-95-5 C30H33FN2O4
(±)-(3-{5-fluoro-2-[3-(6-methylpyridin-2-yl)butyryl]-1,2,3,4-tetrahydroisoquinolin-8-yl}-4-isopropoxyphenyl)acetic acid
—— US9598416, Example 55 1443617-14-8 C22H24N6O2S
US9598416, Example 55
—— [(2S)-1-[7-(3-fluorophenyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidin-2-yl]methanol 1363283-67-3 C24H23FN4O
[(2S)-1-[7-(3-fluorophenyl)-2-methyl-3-phenylpyrazolo[1,5-a]pyrimidin-5-yl]pyrrolidin-2-yl]methanol
—— {(S)-3-[4-(6-methanesulfonyl-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-oxazol-4-yl-methanone 1445999-39-2 C23H24N4O6S
{(S)-3-[4-(6-methanesulfonyl-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-oxazol-4-yl-methanone
—— 1-[(2S,4R)-2-(fluoromethyl)-2-methyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-5-yl)urea 1444793-41-2 C21H23FN4O3
1-[(2S,4R)-2-(fluoromethyl)-2-methyl-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-5-yl)urea
—— 5-((2-phenyl-2-(piperazin-1-yl)ethyl)amino)quinazoline-8-carboxamide 1445782-58-0 C21H24N6O
5-((2-phenyl-2-(piperazin-1-yl)ethyl)amino)quinazoline-8-carboxamide
—— (R)-N-((1-(2-acetyl-9-cyclopropyl-6-fluoro-3-hydroxy-8-methoxy-4-oxo-4,9-dihydrothieno[2,3-b]quinolin-7-yl) pyrrolidin-3-yl)methyl)-5-fluoro-2-methylbenzenesulfonamide 1445534-50-8 C29H29F2N3O6S2
(R)-N-((1-(2-acetyl-9-cyclopropyl-6-fluoro-3-hydroxy-8-methoxy-4-oxo-4,9-dihydrothieno[2,3-b]quinolin-7-yl) pyrrolidin-3-yl)methyl)-5-fluoro-2-methylbenzenesulfonamide
—— {4-[5-fluoro-2-((R)-3-phenylbutyryl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-3-isopropoxyphenyl}acetic acid 1445888-96-9 C30H32FNO4
{4-[5-fluoro-2-((R)-3-phenylbutyryl)-1,2,3,4-tetrahydroisoquinolin-8-yl]-3-isopropoxyphenyl}acetic acid
—— 3-[2-[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]ethoxy]-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde 1444767-52-5 C20H29BO6
3-[2-[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]ethoxy]-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzaldehyde
—— adamantan-1-yl-(5-bromo-thiazol-2-ylmethyl)amine 1443122-49-3 C14H19BrN2S
adamantan-1-yl-(5-bromo-thiazol-2-ylmethyl)amine
—— ethyl α-[4-[2-[(4-amidinophenyl)aminocarbonyl]ethyl]-1-piperidinyl]-(3-pyridyl)acetate 1230638-08-0 C24H31N5O3
ethyl α-[4-[2-[(4-amidinophenyl)aminocarbonyl]ethyl]-1-piperidinyl]-(3-pyridyl)acetate
—— 3-methoxy-1-(4-oxo-cyclohexyl)-1H-pyridin-2-one 1252607-22-9 C12H15NO3
3-methoxy-1-(4-oxo-cyclohexyl)-1H-pyridin-2-one
—— (2S,4R)-1-benzoyl-4-(2-chloro-benzenesulfonyl)-pyrrolidine-2-carboxylic acid cyanomethyl-amide 1252632-58-8 C20H18ClN3O4S
(2S,4R)-1-benzoyl-4-(2-chloro-benzenesulfonyl)-pyrrolidine-2-carboxylic acid cyanomethyl-amide
—— 5-(4-oxo-cyclohex-1-enyl)-3H-benzothiazol-2-one 1252615-71-6 C13H11NO2S
5-(4-oxo-cyclohex-1-enyl)-3H-benzothiazol-2-one
—— 1-(1H-imidazol-2-ylmethyl)-5-methoxy-2-methyl-2,3-dihydro-1H-indole 1023913-29-2 C14H17N3O
1-(1H-imidazol-2-ylmethyl)-5-methoxy-2-methyl-2,3-dihydro-1H-indole
—— 6-methyl-3-(propan-2-yl)-1H-indazole 1415740-56-5 C11H14N2
6-methyl-3-(propan-2-yl)-1H-indazole
—— 2-(3-aminomethyl-azetidin-3-yl)-8-[6-(2,4-difluoro-phenoxy)-pyridin-3-yl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam 1105658-80-7 C27H21F2N5O2
2-(3-aminomethyl-azetidin-3-yl)-8-[6-(2,4-difluoro-phenoxy)-pyridin-3-yl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam
—— 2-(7-(5-(3-(2-methylpyridin-4-yl)-5-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid 1163140-95-1 C28H21F3N4O4
2-(7-(5-(3-(2-methylpyridin-4-yl)-5-(trifluoromethoxy)phenyl)-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
—— 6-chloro-2-(4,4-difluorobut-3-enylthio)-pyrazine 172935-41-0 C8H7ClF2N2S
6-chloro-2-(4,4-difluorobut-3-enylthio)-pyrazine
—— 5-(3-amino-3-((3,4-difluorophenyl)carbamoyl)pyrrolidin-1-yl)quinazoline-8-carboxamide 1445782-27-3 C20H18F2N6O2
5-(3-amino-3-((3,4-difluorophenyl)carbamoyl)pyrrolidin-1-yl)quinazoline-8-carboxamide
—— (2S)-neopentyl 2-((((2R,3R,4R,5R)-5-(2-amino-6-(methylthio)-9H-purin-9-yl)-3,4-dihydroxy-4-methyltetrahydrofuran-2-yl)methoxy)(quinolin-6-yloxy)phosphorylamino)propanoate 1234491-53-2 C29H38N7O8PS
(2S)-neopentyl 2-((((2R,3R,4R,5R)-5-(2-amino-6-(methylthio)-9H-purin-9-yl)-3,4-dihydroxy-4-methyltetrahydrofuran-2-yl)methoxy)(quinolin-6-yloxy)phosphorylamino)propanoate
—— 1-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)-3-[(4R)-7-(trifluoromethoxy)-3,4-dihydro-2H-chromen-4-yl]urea 1444796-81-9 C20H18F3N3O4
1-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)-3-[(4R)-7-(trifluoromethoxy)-3,4-dihydro-2H-chromen-4-yl]urea
—— 6-chloro-2-(fluoromethyl)-N-[[(2R,6S)-6-(4-methylsulfanylphenyl)oxan-2-yl]methyl]pyrimidin-4-amine 1420297-80-8 C18H21ClFN3OS
6-chloro-2-(fluoromethyl)-N-[[(2R,6S)-6-(4-methylsulfanylphenyl)oxan-2-yl]methyl]pyrimidin-4-amine
—— 4-[5-(cyclopropylsulfonyl)-2-(2,4-difluorophenoxy)phenyl]-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1446235-22-8 C23H18F2N2O4S
4-[5-(cyclopropylsulfonyl)-2-(2,4-difluorophenoxy)phenyl]-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— 1-[4-((S)-cycloheptylamino-cyclohexyl-methyl)-[1,2,3]triazol-1-yl]-cyclopropanecarbonitrile 1333425-59-4 C20H31N5
1-[4-((S)-cycloheptylamino-cyclohexyl-methyl)-[1,2,3]triazol-1-yl]-cyclopropanecarbonitrile
—— N-[(1S)-1-[4-[1-(4-ethoxyphenyl)azetidin-3-yl]oxyphenyl]ethyl]-2-fluoroacetamide 1443669-89-3 C21H25FN2O3
N-[(1S)-1-[4-[1-(4-ethoxyphenyl)azetidin-3-yl]oxyphenyl]ethyl]-2-fluoroacetamide