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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(4-chlorophenyl)-N-(2,2-diethoxyethyl)-N-(4-methoxyphenyl)propiolamide 1383129-43-8 C22H24ClNO4
3-(4-chlorophenyl)-N-(2,2-diethoxyethyl)-N-(4-methoxyphenyl)propiolamide
—— tert-butyl 4-hydroxy-2-hydroxymethyl-6-tetrahydropyranyloxyhexanoate 152010-78-1 C16H30O6
tert-butyl 4-hydroxy-2-hydroxymethyl-6-tetrahydropyranyloxyhexanoate
—— 4-methyl-1-phenylpent-1-yn-3-yl pent-2-ynoate 1001421-91-5 C17H18O2
4-methyl-1-phenylpent-1-yn-3-yl pent-2-ynoate
—— 4,6-O-benzylidene-α-D-glucopyranose 1,2-O-(methyl 2-phenylorthoacetate) 1344087-19-9 C21H22O7
4,6-O-benzylidene-α-D-glucopyranose 1,2-O-(methyl 2-phenylorthoacetate)
—— 1-Ethyl-3-[4-(2-methoxyethoxy)-3-(1-methylpyrazol-4-yl)phenyl]-5-phenyl-7-(trifluoromethyl)-1,5-benzodiazepine-2,4-dione 1329989-28-7 C31H29F3N4O4
1-Ethyl-3-[4-(2-methoxyethoxy)-3-(1-methylpyrazol-4-yl)phenyl]-5-phenyl-7-(trifluoromethyl)-1,5-benzodiazepine-2,4-dione
—— 5-(3-chloro-2-fluoro-phenyl)-4-(4-fluoro-phenyl)-3-isopropyl-4,5-dihydro-2H-pyrrolo[3,4-c]pyrazol-6-one 1441739-01-0 C20H16ClF2N3O
5-(3-chloro-2-fluoro-phenyl)-4-(4-fluoro-phenyl)-3-isopropyl-4,5-dihydro-2H-pyrrolo[3,4-c]pyrazol-6-one
—— 1-(7-amino-3-(6-fluoroquinolin-3-yl)-5-(4-hydroxy-4-(hydroxymethyl)cyclohexyl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone 1361449-80-0 C24H24FN5O3
1-(7-amino-3-(6-fluoroquinolin-3-yl)-5-(4-hydroxy-4-(hydroxymethyl)cyclohexyl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone
—— ethyl 2-(2-bromophenyl)-1H-indole-5-carboxylate 1379511-76-8 C17H14BrNO2
ethyl 2-(2-bromophenyl)-1H-indole-5-carboxylate
—— 4-{2-(2,4-difluorophenoxy)-5-[(phenylsulfonyl)methyl]phenyl}-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1446235-40-0 C27H20F2N2O4S
4-{2-(2,4-difluorophenoxy)-5-[(phenylsulfonyl)methyl]phenyl}-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— α-<1-Carboxy-ethyl>-γ-valerolacton 13555-68-5 C8H12O4
α-<1-Carboxy-ethyl>-γ-valerolacton
—— methyl 2-[4-[[(3R)-3-aminopyrrolidin-1-yl]methyl]phenoxy]acetate 1444123-67-4 C14H20N2O3
methyl 2-[4-[[(3R)-3-aminopyrrolidin-1-yl]methyl]phenoxy]acetate
—— 7-(4-ethylpiperazin-1-yl)-3-(5-methylpyrazolo[1,5-a]pyridin-2-yl)-2H-chromen-2-one 1446330-45-5 C23H24N4O2
7-(4-ethylpiperazin-1-yl)-3-(5-methylpyrazolo[1,5-a]pyridin-2-yl)-2H-chromen-2-one
—— 2-[[(2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-heptoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]propanoyl]amino]-2-methylpropanoic acid 1443788-92-8 C39H48N4O6
2-[[(2S)-2-[(4-tert-butylbenzoyl)amino]-3-[4-[5-(4-heptoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]propanoyl]amino]-2-methylpropanoic acid
—— Fmoc-Nle-ψ[PO(OAd)]-Gly-COOH 1261301-19-2 C32H40NO6P
Fmoc-Nle-ψ[PO(OAd)]-Gly-COOH
—— 3-(2,5-bis(chloromethyl)-4-methoxyphenoxy)propan-1-ol 1335100-08-7 C12H16Cl2O3
3-(2,5-bis(chloromethyl)-4-methoxyphenoxy)propan-1-ol
—— —— 198290-89-0 C30H48N4Si2Zr
—— 1-{5-[4-(3-acetyl-4-hydroxyphenoxy)-2,3,5,6-tetrafluorophenoxy]-2-hydroxyphenyl}ethan-1-one 1429063-84-2 C22H14F4O6
1-{5-[4-(3-acetyl-4-hydroxyphenoxy)-2,3,5,6-tetrafluorophenoxy]-2-hydroxyphenyl}ethan-1-one
—— (3aR,6aR)-2,2-dimethyl-3a,6a-dihydrofuro[2,3-d][1,3]dioxole 123487-69-4 C7H10O3
(3aR,6aR)-2,2-dimethyl-3a,6a-dihydrofuro[2,3-d][1,3]dioxole
—— 5-(3-cyclopropylmethoxy-4-methoxy-2-(3-methoxymethyloxetan-3-ylmethoxy)phenyl)-3H-isobenzofuran-1-one 1345880-58-1 C25H28O7
5-(3-cyclopropylmethoxy-4-methoxy-2-(3-methoxymethyloxetan-3-ylmethoxy)phenyl)-3H-isobenzofuran-1-one
—— (2S,3S,4R,5R)-2-allyltetrahydro-2H-pyran-3,4,5-triyl triacetate 1079109-82-2 C14H20O7
(2S,3S,4R,5R)-2-allyltetrahydro-2H-pyran-3,4,5-triyl triacetate
—— (1R,2R,4R)-4-(hydroxymethyl)-2-methoxy-1-<(triisopropylsilyl)oxy>cyclohexane 128684-91-3 C17H36O3Si
(1R,2R,4R)-4-(hydroxymethyl)-2-methoxy-1-<(triisopropylsilyl)oxy>cyclohexane
—— 5-[3,5-bis-(4-methoxyphenyl)-4,5-dihydropyrazol-1-ylmethylene]-2-thioxo-3-p-tolylthiazolidin-4-one 1621417-88-6 C28H25N3O3S2
5-[3,5-bis-(4-methoxyphenyl)-4,5-dihydropyrazol-1-ylmethylene]-2-thioxo-3-p-tolylthiazolidin-4-one
—— 3-[[5-Chloro-1-(3-methylsulfonylpropyl)pyrrolo[3,2-b]pyridin-2-yl]methyl]-1-(2,2,2-trifluoroethyl)imidazo[4,5-c]pyridin-2-one 1383252-71-8 C20H19ClF3N5O3S
3-[[5-Chloro-1-(3-methylsulfonylpropyl)pyrrolo[3,2-b]pyridin-2-yl]methyl]-1-(2,2,2-trifluoroethyl)imidazo[4,5-c]pyridin-2-one
—— US9598416, Example 66 1443617-25-1 C23H28N6OS
US9598416, Example 66
—— 2-(dimethylamino)-2-(2-chlorophenyl)acetic acid 1007878-92-3 C10H12ClNO2
2-(dimethylamino)-2-(2-chlorophenyl)acetic acid
—— 2-[(R)-2-(7-(tetrahydropyran-4-yl)amino-1H-indol-2-yl)-4,5-dihydrothiazol-4-yl]-1-methylaminoethanone 1172996-73-4 C19H24N4O2S
2-[(R)-2-(7-(tetrahydropyran-4-yl)amino-1H-indol-2-yl)-4,5-dihydrothiazol-4-yl]-1-methylaminoethanone
—— 5-bromo-N-[5-bromo-2-methyl-1,1-dioxo-7-(propan-2-ylcarbamoyl)-2,3-dihydro-1-benzothiophen-6-yl]-2-(3-chloropyridin-2-yl)pyrazole-3-carboxamide 1103246-29-2 C22H20Br2ClN5O4S
5-bromo-N-[5-bromo-2-methyl-1,1-dioxo-7-(propan-2-ylcarbamoyl)-2,3-dihydro-1-benzothiophen-6-yl]-2-(3-chloropyridin-2-yl)pyrazole-3-carboxamide
—— N-(4-cyclohexyl-thiazol-2-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide 1253381-80-4 C27H34N6O2S
N-(4-cyclohexyl-thiazol-2-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide
—— {1-[4-(4-oxo-3,4,5,6,7,8-hexahydro-quinazolin-2-yl)-cyclohexyl]-azetidin-3-yl}-carbamic acid tert-butyl ester 1252690-24-6 C22H34N4O3
{1-[4-(4-oxo-3,4,5,6,7,8-hexahydro-quinazolin-2-yl)-cyclohexyl]-azetidin-3-yl}-carbamic acid tert-butyl ester
—— 8-hydroxy-5-methyl-5,6,7,8,9,10-hexahydro-5,9-methano-benzocycloocten-11-one 110181-09-4 C14H16O2
8-hydroxy-5-methyl-5,6,7,8,9,10-hexahydro-5,9-methano-benzocycloocten-11-one
—— —— 1402571-28-1 C24H28BrNO6Si
—— methyl 2-chloromercurio-3-acetoxy-2,3-diphenylcyclopropane-1-carboxylate 104124-51-8 C19H17ClHgO4
methyl 2-chloromercurio-3-acetoxy-2,3-diphenylcyclopropane-1-carboxylate
—— 3-(3,4-Dichlorophenyl)-3-(2-hydroxyethoxy)-1-(3-isopropoxybenzylcarbonyl)piperidine 173086-70-9 C24H29Cl2NO4
3-(3,4-Dichlorophenyl)-3-(2-hydroxyethoxy)-1-(3-isopropoxybenzylcarbonyl)piperidine
—— methyl N-[5-[1-[5-[[2-methoxy-3-[(propan-2-ylamino)methyl]-5-(trifluoromethyl)phenyl]carbamoyl]-2-methylphenyl]triazol-4-yl]-1,3-thiazol-2-yl]carbamate 1096693-70-7 C27H28F3N7O4S
methyl N-[5-[1-[5-[[2-methoxy-3-[(propan-2-ylamino)methyl]-5-(trifluoromethyl)phenyl]carbamoyl]-2-methylphenyl]triazol-4-yl]-1,3-thiazol-2-yl]carbamate
—— 2-[2-(Methoxymethyl)-1,3-dioxan-2-yl]-6-(1-pyridin-3-ylpyrazol-4-yl)pyridine 1292295-06-7 C19H20N4O3
2-[2-(Methoxymethyl)-1,3-dioxan-2-yl]-6-(1-pyridin-3-ylpyrazol-4-yl)pyridine
—— 3-(2-chlorophenyl)-8-cyclopropyl-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1035927-54-8 C16H18ClN3S
3-(2-chlorophenyl)-8-cyclopropyl-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 5-chloro-3-(2,4-dioxo-1H-quinazolin-3-yl)-N-(4-fluorophenyl)sulfonyl-1-methylindole-2-carboxamide 1154600-55-1 C24H16ClFN4O5S
5-chloro-3-(2,4-dioxo-1H-quinazolin-3-yl)-N-(4-fluorophenyl)sulfonyl-1-methylindole-2-carboxamide
—— [(1E,5E)-1-(cyclopenten-1-yl)-6-iodo-3-methylhexa-1,5-dien-3-yl]oxy-trimethylsilane 131720-97-3 C15H25IOSi
[(1E,5E)-1-(cyclopenten-1-yl)-6-iodo-3-methylhexa-1,5-dien-3-yl]oxy-trimethylsilane
—— tricarbonyl(η6-o-tri-isopropylsilylbenzaldehyde)chromium(0) 126639-03-0 C19H26CrO4Si
tricarbonyl(η6-o-tri-isopropylsilylbenzaldehyde)chromium(0)
—— (S)-(9H-fluoren-9-yl)methyl 1-((2,2-diethoxyethyl)(quinolin-8-ylmethyl)amino)-1,4-dioxo-4-(tritylamino)butan-2-ylcarbamate 1222066-72-9 C54H52N4O6
(S)-(9H-fluoren-9-yl)methyl 1-((2,2-diethoxyethyl)(quinolin-8-ylmethyl)amino)-1,4-dioxo-4-(tritylamino)butan-2-ylcarbamate
—— (S)-tert-butyl 5-amino-6-((2,2-diethoxyethyl)(3,3-diphenylpropyl)amino)-6-oxohexylcarbamate 1222068-86-1 C32H49N3O5
(S)-tert-butyl 5-amino-6-((2,2-diethoxyethyl)(3,3-diphenylpropyl)amino)-6-oxohexylcarbamate
—— 3-(2-Cyanophenyl)-1,2-oxazole-5-carboxylicacid 1695964-04-5 C11H6N2O3
3-(2-Cyanophenyl)-1,2-oxazole-5-carboxylicacid
—— 4-(4-(4-(trifluoromethyl)phenyl)-1H-imidazol-2-yl)piperidine 1082950-13-7 C15H16F3N3
4-(4-(4-(trifluoromethyl)phenyl)-1H-imidazol-2-yl)piperidine
—— (7R,8S)-8-ethyl-7-hydroxy-2,3,8-trimethyl-5,6,7,8-tetrahydro-4H-chromen-4-one 152764-77-7 C14H20O3
(7R,8S)-8-ethyl-7-hydroxy-2,3,8-trimethyl-5,6,7,8-tetrahydro-4H-chromen-4-one
—— N-benzyloxycarbonyl-3-amino-4-oxo-5-(5-(piperidin-1-yl)tetrazol-2-yl)pentanoic acid 188890-97-3 C19H24N6O5
N-benzyloxycarbonyl-3-amino-4-oxo-5-(5-(piperidin-1-yl)tetrazol-2-yl)pentanoic acid
—— N-phenyl-6-(pyridin-3-ylamino)-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214929-21-1 C19H17N5O2
N-phenyl-6-(pyridin-3-ylamino)-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— 2-hydroxy-N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-acetamide 1215221-73-0 C19H22F3N7O3S
2-hydroxy-N-{2-[6-propyl-4-(3-trifluoromethyl-5,6-dihydro-8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl)-thieno[2,3-d]pyrimidin-2-yloxy]-ethyl}-acetamide
—— 3-[(5-benzoyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-N-(4-chlorophenyl)benzamide 1313038-69-5 C26H18ClN5O2
3-[(5-benzoyl-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-N-(4-chlorophenyl)benzamide
—— (S)-3-(4'-cyano-biphenyl-4-yl)-2-({(S)-7-cyclobutanecarbonyl-3-[4-(3,4-dichloro-benzyloxy)-phenyl]-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline-8-carbonyl}-amino)-propionic acid 1246824-36-1 C46H39Cl2N3O7
(S)-3-(4'-cyano-biphenyl-4-yl)-2-({(S)-7-cyclobutanecarbonyl-3-[4-(3,4-dichloro-benzyloxy)-phenyl]-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline-8-carbonyl}-amino)-propionic acid
—— 2-[Dimethyl(4,4,5,5,6,6,7,7,8,8,8-undecafluorooctyl)azaniumyl]acetate 171184-14-8 C12H14F11NO2
2-[Dimethyl(4,4,5,5,6,6,7,7,8,8,8-undecafluorooctyl)azaniumyl]acetate