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中文名称 英文名称 CAS号 化学式 结构式图片
—— [[(2R,3S,5R)-5-(6-aminopurin-9-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxyphosphinic acid 120152-59-2 C10H15N5O8P2
[[(2R,3S,5R)-5-(6-aminopurin-9-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxyphosphinic acid
—— ethyl 1-(fluoromethyl)-5-{2-[4-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-4-carboxylate 1359029-15-4 C16H16F4N2O2
ethyl 1-(fluoromethyl)-5-{2-[4-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-4-carboxylate
—— 5-((3-phenylazetidin-3-yl)amino)quinoline-8-carboxamide 1445781-94-1 C19H18N4O
5-((3-phenylazetidin-3-yl)amino)quinoline-8-carboxamide
—— 4-(3-(6-(1H-imidazol-2-yl)pyridin-3-yl)-7-(bis((2-(trimethylsilyl)ethoxy)methyl)amino)-6-(methylsulfonyl)pyrazolo[1,5-a]pyrimidin-5-yl)-1-(2-methoxyethoxy)cyclohexanecarboxamide 1361450-73-8 C37H58N8O7SSi2
4-(3-(6-(1H-imidazol-2-yl)pyridin-3-yl)-7-(bis((2-(trimethylsilyl)ethoxy)methyl)amino)-6-(methylsulfonyl)pyrazolo[1,5-a]pyrimidin-5-yl)-1-(2-methoxyethoxy)cyclohexanecarboxamide
—— N-[5-[4-[5-(oxolane-2-carbonylamino)-1,3,4-thiadiazol-2-yl]butyl]-1,3,4-thiadiazol-2-yl]oxolane-2-carboxamide 1439389-87-3 C18H24N6O4S2
N-[5-[4-[5-(oxolane-2-carbonylamino)-1,3,4-thiadiazol-2-yl]butyl]-1,3,4-thiadiazol-2-yl]oxolane-2-carboxamide
—— N1-(2-pyridin-4-yl-5,8-dihydro-6H-thiopyrano[4',3':4,5]thieno[2,3-d]pyrimidin-4-yl)ethane-1,2-diamine 1438880-74-0 C16H17N5S2
N1-(2-pyridin-4-yl-5,8-dihydro-6H-thiopyrano[4',3':4,5]thieno[2,3-d]pyrimidin-4-yl)ethane-1,2-diamine
—— 1-((4-cyclopropanemethylamino)-6-(2,6-dimethylphenoxy)-7-fluoroquinazolin-2-yl)-1H-pyrazole-4-carboxylic acid 1357482-00-8 C24H22FN5O3
1-((4-cyclopropanemethylamino)-6-(2,6-dimethylphenoxy)-7-fluoroquinazolin-2-yl)-1H-pyrazole-4-carboxylic acid
—— 2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(cyclohexylmethylcarbamoyl)-6-methylphenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229655-47-3 C28H26ClF3N10O2
2-(3-chloropyridin-2-yl)-N-[4-cyano-2-(cyclohexylmethylcarbamoyl)-6-methylphenyl]-5-[[5-(trifluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide
—— 1-(4'-fluoro-biphenyl-4-carbonyl)-4-(4-fluoro-phenyl)-piperidine-4-carboxylic acid 4-fluoro-benzylamide 1246387-73-4 C32H27F3N2O2
1-(4'-fluoro-biphenyl-4-carbonyl)-4-(4-fluoro-phenyl)-piperidine-4-carboxylic acid 4-fluoro-benzylamide
—— 4-Bromo-N-(5-chloro-2-{2-chloro-5-[(1-methylcyclohexylamido)methyl]phenylamino}-1-methyl-6-benzimidazolyl)benzamide 1242268-92-3 C30H30BrCl2N5O2
4-Bromo-N-(5-chloro-2-{2-chloro-5-[(1-methylcyclohexylamido)methyl]phenylamino}-1-methyl-6-benzimidazolyl)benzamide
—— N-(1-{[2-chloro-6-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-3-yl)-2,6-difluorobenzamide 1253186-75-2 C18H11ClF5N3O
N-(1-{[2-chloro-6-(trifluoromethyl)phenyl]methyl}-1H-pyrazol-3-yl)-2,6-difluorobenzamide
—— (R)-N-(pyridazin-3-yl)-1-(4-(trifluoromethyl)phenyl)-3,4-dihydroiso-quinoline-2(1H)-carboxamide 1159997-45-1 C21H17F3N4O
(R)-N-(pyridazin-3-yl)-1-(4-(trifluoromethyl)phenyl)-3,4-dihydroiso-quinoline-2(1H)-carboxamide
—— 3-({4-[(cyclohexyl{2-methyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methyl)amino]benzoyl}amino)propanoic acid 1150212-17-1 C29H31F3N2O4
3-({4-[(cyclohexyl{2-methyl-5-[4-(trifluoromethyl)phenyl]-3-furyl}methyl)amino]benzoyl}amino)propanoic acid
—— 5-(1,4-dioxa-spiro[4.5]dec-8-yl)-1H-pyridin-2-one 1252689-62-5 C13H17NO3
5-(1,4-dioxa-spiro[4.5]dec-8-yl)-1H-pyridin-2-one
—— (R)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-(4-(trifluoromethyl)phenyl)-3,4-dihydroisoquinoline-2(1H)-carboxamide 1159997-54-2 C27H25F3N2O
(R)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1-(4-(trifluoromethyl)phenyl)-3,4-dihydroisoquinoline-2(1H)-carboxamide
—— N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[[5-(1,1,2,2,2-pentafluoroethyl)tetrazol-1-yl]methyl]pyrazole-3-carboxamide 1229659-05-5 C26H22ClF5N10O2
N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[[5-(1,1,2,2,2-pentafluoroethyl)tetrazol-1-yl]methyl]pyrazole-3-carboxamide
—— Ethyl 2-[4-[3-[(4-formylphenoxy)methyl]-2-methylphenyl]-3,5-dimethylphenoxy]acetate 1148023-05-5 C27H28O5
Ethyl 2-[4-[3-[(4-formylphenoxy)methyl]-2-methylphenyl]-3,5-dimethylphenoxy]acetate
—— 4-((2-(dimethylamino)ethyl)(ethyl)amino)-6-phenyl-N-(2-(5-phenyloxazol-2-yl)phenyl)picolinamide 1148120-62-0 C33H33N5O2
4-((2-(dimethylamino)ethyl)(ethyl)amino)-6-phenyl-N-(2-(5-phenyloxazol-2-yl)phenyl)picolinamide
—— N-(7-hydroxynon-8-en-2-ynyl)-4-methyl-N-(3-phenylprop-2-ynyl)benzenesulfonamide 1140383-61-4 C25H27NO3S
N-(7-hydroxynon-8-en-2-ynyl)-4-methyl-N-(3-phenylprop-2-ynyl)benzenesulfonamide
—— 8-Methoxy-N-propyl-N-[3-(2,3-dihydro-1,1-dioxo-3-oxo-1,2-benzisothiazolyl)propyl]-2-aminotetralin 134466-13-0 C24H30N2O4S
8-Methoxy-N-propyl-N-[3-(2,3-dihydro-1,1-dioxo-3-oxo-1,2-benzisothiazolyl)propyl]-2-aminotetralin
—— tetraethyl-[2-(4,7-dimethyl-imidazo-[4,5-d]pyridazin-1-yl)-ethylidene]-bisphosphonate 1149342-10-8 C17H30N4O6P2
tetraethyl-[2-(4,7-dimethyl-imidazo-[4,5-d]pyridazin-1-yl)-ethylidene]-bisphosphonate
—— N-(6-{1-[2-(4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-4-yloxy}pyridin-3-yl)-4-trifluoromethylbenzamide 1150461-21-4 C35H32F3N5O5
N-(6-{1-[2-(4-benzo[1,3]dioxol-5-ylmethylpiperazin-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indol-4-yloxy}pyridin-3-yl)-4-trifluoromethylbenzamide
—— N-[4-bromo-2-(2H-tetrazol-5-yl)-phenyl]-3,5-bis-trifluoromethyl-benzamide 1159711-33-7 C16H8BrF6N5O
N-[4-bromo-2-(2H-tetrazol-5-yl)-phenyl]-3,5-bis-trifluoromethyl-benzamide
—— 9-[(1R)-1-[5-[3-(aminomethyl)phenyl]-2-(trifluoromethoxy)phenyl]ethyl]-2-[[(3R)-pyrrolidin-3-yl]methylamino]-7H-purin-8-one 1152086-40-2 C26H28F3N7O2
9-[(1R)-1-[5-[3-(aminomethyl)phenyl]-2-(trifluoromethoxy)phenyl]ethyl]-2-[[(3R)-pyrrolidin-3-yl]methylamino]-7H-purin-8-one
—— 6-(5-(trifluoromethyl)pyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1159823-19-4 C12H8F3N5
6-(5-(trifluoromethyl)pyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— 4-((S)-2-{[6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-5-phosphonopentanoyl)piperazine-1-carboxylic acid butyl ester 1159500-91-0 C30H43N6O8P
4-((S)-2-{[6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-5-phosphonopentanoyl)piperazine-1-carboxylic acid butyl ester
—— 2-(4-[5-(1-methyl-1H-pyrrole-3-sulfonyl)-hexahydro-pyrrolo[3,4-c]pyrrol-2-ylmethyl]-phenoxy)-benzothiazole 1146692-91-2 C25H26N4O3S2
2-(4-[5-(1-methyl-1H-pyrrole-3-sulfonyl)-hexahydro-pyrrolo[3,4-c]pyrrol-2-ylmethyl]-phenoxy)-benzothiazole
—— 1-(5-[4-(benzothiazol-2-yloxy)-benzyl]-hexahydro-pyrrolo[3,4-b]pyrrol-1-yl)-ethanone 1146692-49-0 C22H23N3O2S
1-(5-[4-(benzothiazol-2-yloxy)-benzyl]-hexahydro-pyrrolo[3,4-b]pyrrol-1-yl)-ethanone
—— 2-{[5-methyl-6-({4-[(2-methyl-2H-1,2,3-triazol-4-yl)amino]quinazolin-6-yl}oxy)pyridin-3-yl]oxy}ethanol 1154579-21-1 C19H19N7O3
2-{[5-methyl-6-({4-[(2-methyl-2H-1,2,3-triazol-4-yl)amino]quinazolin-6-yl}oxy)pyridin-3-yl]oxy}ethanol
—— N-[2-(dimethylamino)ethyl]-5-oxo-2,4,5,6-tetrahydro-1H-thiopyrano[3,4-c]quinoline-9-carboxamide hydrochloride 1151832-54-0 C17H21N3O2S*ClH
N-[2-(dimethylamino)ethyl]-5-oxo-2,4,5,6-tetrahydro-1H-thiopyrano[3,4-c]quinoline-9-carboxamide hydrochloride
—— 1-[(4-bromophenyl)methyl]-5-methyl-N-{4-[(3-methylbutyl)oxy]phenyl}-1H-1,2,3-triazole-4-carboxamide 1150701-47-5 C22H25BrN4O2
1-[(4-bromophenyl)methyl]-5-methyl-N-{4-[(3-methylbutyl)oxy]phenyl}-1H-1,2,3-triazole-4-carboxamide
—— 5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-N-(2-(trifluoromethyl)phenyl)pyridine-3-sulfonamide 1159823-10-5 C18H13F3N6O2S
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-6-yl)-N-(2-(trifluoromethyl)phenyl)pyridine-3-sulfonamide
—— 2-morpholin-4-yl-N-6-pyridin-4-ylmethyl-[4,5']bipyrimidinyl-6,2'-diamine 1155304-92-9 C18H20N8O
2-morpholin-4-yl-N-6-pyridin-4-ylmethyl-[4,5']bipyrimidinyl-6,2'-diamine
—— 1H-Pyrrole-3-acetic acid, 1-ethyl-4-(4-ethylbenzoyl)-2,5-dihydro-5-(methylthio)-2-oxo- 1269531-57-8 C18H21NO4S
1H-Pyrrole-3-acetic acid, 1-ethyl-4-(4-ethylbenzoyl)-2,5-dihydro-5-(methylthio)-2-oxo-
—— [(4R)-4-[tert-butyl(dimethyl)silyl]oxy-2-methylcyclohexa-1,5-dien-1-yl] acetate 1199941-02-0 C15H26O3Si
[(4R)-4-[tert-butyl(dimethyl)silyl]oxy-2-methylcyclohexa-1,5-dien-1-yl] acetate
—— 6,15,23,32-Tetrakis[2-(2,6-dioctoxyphenyl)ethynyl]-2,19-diazaheptacyclo[28.4.0.03,8.04,34.013,18.017,21.020,25]tetratriaconta-1(30),3(8),4,6,13(18),14,16,20(25),21,23,31,33-dodecaen-9,11,26,28-tetrayne 1444561-84-5 C128H158N2O8
6,15,23,32-Tetrakis[2-(2,6-dioctoxyphenyl)ethynyl]-2,19-diazaheptacyclo[28.4.0.03,8.04,34.013,18.017,21.020,25]tetratriaconta-1(30),3(8),4,6,13(18),14,16,20(25),21,23,31,33-dodecaen-9,11,26,28-tetrayne
—— 2-[[2-(6-Chloro-2,4-dioxoquinazolin-1-yl)acetyl]-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]acetic acid 1401247-33-3 C19H23ClN4O7
2-[[2-(6-Chloro-2,4-dioxoquinazolin-1-yl)acetyl]-[2-[(2-methylpropan-2-yl)oxycarbonylamino]ethyl]amino]acetic acid
—— 6-(2,6-dichlorobenzyl)imidazo[1,2-a]pyrimidin-7-ylamine 1072514-22-7 C13H10Cl2N4
6-(2,6-dichlorobenzyl)imidazo[1,2-a]pyrimidin-7-ylamine
—— 2-[5-bromo-3-(2,4-dichlorobenzoyl)-4-(2,2-dimethylpropyl)thiophen-2-yl]isoindol-ine-1,3-dione 1529778-32-2 C24H18BrCl2NO3S
2-[5-bromo-3-(2,4-dichlorobenzoyl)-4-(2,2-dimethylpropyl)thiophen-2-yl]isoindol-ine-1,3-dione
—— <(3,5-Di-tert-butylphenoxycarbonyl)methyl>triphenylphosphoniumbromid 119788-24-8 Br*C34H38O2P
<(3,5-Di-tert-butylphenoxycarbonyl)methyl>triphenylphosphoniumbromid
—— 16-[3-methoxy-4-{2-(piperidin-1-yl)ethoxy}-benzylidene]-5-androstene-3β,17β-diol 1151468-95-9 C34H49NO4
16-[3-methoxy-4-{2-(piperidin-1-yl)ethoxy}-benzylidene]-5-androstene-3β,17β-diol
—— 2-((7-(1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl)quinolin-5-yloxy)methyl)nicotinamide 1421340-21-7 C25H20N4O3
2-((7-(1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl)quinolin-5-yloxy)methyl)nicotinamide
—— N,N-dimethyl-5-[[4-[4-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-yl]amino]-1H-indole-2-carboxamide 1391601-22-1 C21H17F3N6O
N,N-dimethyl-5-[[4-[4-(trifluoromethyl)pyridin-2-yl]pyrimidin-2-yl]amino]-1H-indole-2-carboxamide
—— (S)-3-{[5-(2,3-difluoro-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-3-m-tolyl-propionic acid 1420833-44-8 C19H15F2N3O4
(S)-3-{[5-(2,3-difluoro-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-3-m-tolyl-propionic acid
—— 3-[(1S)-1-[(2-aminopyrido[3,2-d]pyrimidin-4-yl)amino]ethyl]-8-(2-methylpyrimidin-5-yl)-2-phenylisoquinolin-1-one 1420619-48-2 C29H24N8O
3-[(1S)-1-[(2-aminopyrido[3,2-d]pyrimidin-4-yl)amino]ethyl]-8-(2-methylpyrimidin-5-yl)-2-phenylisoquinolin-1-one
—— (R)-N-(1-cyclopropylethyl)-2-(4-(4-fluorobenzoyl)piperidin-1-yl)-N-((4-oxo-4,5,7,8-tetrahydro-3H-pyrano[4,3-d]pyrimidin-2-yl)methyl)ethanamide 1419950-65-4 C27H33FN4O4
(R)-N-(1-cyclopropylethyl)-2-(4-(4-fluorobenzoyl)piperidin-1-yl)-N-((4-oxo-4,5,7,8-tetrahydro-3H-pyrano[4,3-d]pyrimidin-2-yl)methyl)ethanamide
—— (2S,6R)-2-Morpholin-4-yl-1,8,11-triaza-tricyclo[5.2.2.02,6]undeca-8,10-diene-7,9,10-tricarboxylic acid triethyl ester 117663-63-5 C21H30N4O7
(2S,6R)-2-Morpholin-4-yl-1,8,11-triaza-tricyclo[5.2.2.02,6]undeca-8,10-diene-7,9,10-tricarboxylic acid triethyl ester
—— (4-Methoxy-2-oxocyclohex-3-en-1-yl) 2-methylpropanoate 132783-37-0 C11H16O4
(4-Methoxy-2-oxocyclohex-3-en-1-yl) 2-methylpropanoate
—— (N-((2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)-N-methylcarbamoyl)methyl acetate 1033742-99-2 C16H19ClN4O4S
(N-((2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)-N-methylcarbamoyl)methyl acetate
—— 4-iodo-1,3-diisopropylimidazol-2-ylidene borane 1338729-05-7 C9H18BIN2
4-iodo-1,3-diisopropylimidazol-2-ylidene borane