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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-[(2S)-2-(benzyloxy)propyl]-1-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-N-[3-methyl-4-(methylsulfonyl)phenyl]-1H-pyrrole-3-carboxamide 1221425-45-1 C31H30F4N2O4S
5-[(2S)-2-(benzyloxy)propyl]-1-[4-fluoro-2-(trifluoromethyl)phenyl]-2-methyl-N-[3-methyl-4-(methylsulfonyl)phenyl]-1H-pyrrole-3-carboxamide
—— N-{2-fluoro-3-[5-{2-[(2-hydroxyethyl)amino]-4-pyrimidinyl}-2-(tetrahydro-2H-pyran-4-yl)-1,3-thiazol-4-yl]prienyl}-1-propanesulfonamide 1307270-56-9 C23H28FN5O4S2
N-{2-fluoro-3-[5-{2-[(2-hydroxyethyl)amino]-4-pyrimidinyl}-2-(tetrahydro-2H-pyran-4-yl)-1,3-thiazol-4-yl]prienyl}-1-propanesulfonamide
—— (E,R)-4-(4-bromophenyl)-1-(pyridin-2-yl)-4-o-tolylbutan-2-one oxime 1354812-96-6 C22H21BrN2O
(E,R)-4-(4-bromophenyl)-1-(pyridin-2-yl)-4-o-tolylbutan-2-one oxime
—— 5-{5-[(4-chloro-benzyl)-methyl-amino]-pyridine-2-carbonyl}-2-(3-methoxy-benzoylamino)-benzoic acid 1245734-48-8 C29H24ClN3O5
5-{5-[(4-chloro-benzyl)-methyl-amino]-pyridine-2-carbonyl}-2-(3-methoxy-benzoylamino)-benzoic acid
—— (2R)-3-[4-(2-cyclopropylethynyl)-3-fluorophenyl]-2-[(3-fluoro-4-methylbenzoyl)amino]propanoic acid 1323994-63-3 C22H19F2NO3
(2R)-3-[4-(2-cyclopropylethynyl)-3-fluorophenyl]-2-[(3-fluoro-4-methylbenzoyl)amino]propanoic acid
—— [6-[6-(Trifluoromethyl)pyridin-3-yl]oxan-2-yl]methanamine 1312780-43-0 C12H15F3N2O
[6-[6-(Trifluoromethyl)pyridin-3-yl]oxan-2-yl]methanamine
—— 4',6'-O-o-nitrobenzylideneparomomycin 1043874-57-2 C30H48N6O16
4',6'-O-o-nitrobenzylideneparomomycin
—— 2-[[2-Bromo-4-(trifluoromethyl)phenyl]sulfonylamino]-3-[4-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)-3-fluorophenyl]propanoic acid 1323993-96-9 C24H22BrF4N3O5S
2-[[2-Bromo-4-(trifluoromethyl)phenyl]sulfonylamino]-3-[4-(5-cyclohexyl-1,2,4-oxadiazol-3-yl)-3-fluorophenyl]propanoic acid
—— 4-hydroxy-6-oxo-2-phenyl-6,7-dihydro-thieno[2,3-b]pyridine-5-carboxylic acid [4-(hexyloxy)phenyl]amide 1005331-62-3 C26H26N2O4S
4-hydroxy-6-oxo-2-phenyl-6,7-dihydro-thieno[2,3-b]pyridine-5-carboxylic acid [4-(hexyloxy)phenyl]amide
—— 2-((5-(chloromethyl)-1,2,4-oxadiazol-3-yl)methyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one 1354200-14-8 C17H11ClF3N5O3
2-((5-(chloromethyl)-1,2,4-oxadiazol-3-yl)methyl)-6-(4-(trifluoromethoxy)phenyl)-[1,2,4]triazolo[4,3-a]pyridin-3(2H)-one
—— 5-methyl-5-[4-(3-(2-propyl-4-pyrazinyloxyphenoxy)propoxy)phenyl]-2,4-thiazolidinedione 1100807-07-5 C26H27N3O5S
5-methyl-5-[4-(3-(2-propyl-4-pyrazinyloxyphenoxy)propoxy)phenyl]-2,4-thiazolidinedione
—— 6-{4-[4-amino-5-methylpyrimidin-2-yl]-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}[1,3]thiazolo[5,4-b]pyridin-2-amine 1379578-80-9 C21H21N7OS
6-{4-[4-amino-5-methylpyrimidin-2-yl]-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}[1,3]thiazolo[5,4-b]pyridin-2-amine
—— tert-butyl 4-(4-cyclopropyl-1-(2-hydroxyethyl)-1H-imidazol-2-yl)piperidine-1-carboxylate 1295518-73-8 C18H29N3O3
tert-butyl 4-(4-cyclopropyl-1-(2-hydroxyethyl)-1H-imidazol-2-yl)piperidine-1-carboxylate
—— 2-bromo-1,3-dipyridin-2-yl-1,3,2-diazaborolidine 1244036-79-0 C12H12BBrN4
2-bromo-1,3-dipyridin-2-yl-1,3,2-diazaborolidine
—— [8-methoxy-2-oxo-3-(2,4,6-trimethylphenyl)-1,8-diazaspiro[4.5]dec-3-en-4-yl] N-(2-cyanoethyl)-N-methylcarbamate 1145783-54-5 C23H30N4O4
[8-methoxy-2-oxo-3-(2,4,6-trimethylphenyl)-1,8-diazaspiro[4.5]dec-3-en-4-yl] N-(2-cyanoethyl)-N-methylcarbamate
—— 1-[(5-Bromopyridin-2-yl)methyl]-4-pyridin-4-ylpiperazine 1226985-79-0 C15H17BrN4
1-[(5-Bromopyridin-2-yl)methyl]-4-pyridin-4-ylpiperazine
—— 5-{5-[(4-chloro-phenyl)-cyclopropylmethyl-amino]picolinoyl}-2-[2-(pyridin-2-yloxy)-phenoxy]-benzoic acid 1245733-85-0 C34H26ClN3O5
5-{5-[(4-chloro-phenyl)-cyclopropylmethyl-amino]picolinoyl}-2-[2-(pyridin-2-yloxy)-phenoxy]-benzoic acid
—— 5-{5-[(4-chlorophenyl)(methyl)amino]picolinoyl}-2-(2,2-dimethylpropionyl)benzoic acid 1245734-69-3 C25H23ClN2O4
5-{5-[(4-chlorophenyl)(methyl)amino]picolinoyl}-2-(2,2-dimethylpropionyl)benzoic acid
—— 1,1-difluoro-3-iodomethylcyclopentane 1042153-28-5 C6H9F2I
1,1-difluoro-3-iodomethylcyclopentane
—— (5R)-5-[(5-methoxy-3-oxo-1H-isoindol-2-yl)methyl]-5-[2-[4-(1,2,4-triazol-1-yl)phenyl]ethynyl]imidazolidine-2,4-dione 1226988-15-3 C23H18N6O4
(5R)-5-[(5-methoxy-3-oxo-1H-isoindol-2-yl)methyl]-5-[2-[4-(1,2,4-triazol-1-yl)phenyl]ethynyl]imidazolidine-2,4-dione
—— 3-{5-[(4-chlorophenyl)(methyl)amino]picolinoyl}-5-(3-methoxybenzamido)-benzoic acid 1245701-99-8 C28H22ClN3O5
3-{5-[(4-chlorophenyl)(methyl)amino]picolinoyl}-5-(3-methoxybenzamido)-benzoic acid
—— 2-[5-[2-[2-(2-Chloro-3-fluorophenyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-1,3-thiazol-5-yl]tetrazol-2-yl]acetic acid 1246749-04-1 C18H17ClFN7O2S
2-[5-[2-[2-(2-Chloro-3-fluorophenyl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-1,3-thiazol-5-yl]tetrazol-2-yl]acetic acid
—— N-(5-(4-(4-amino-5-(trifluoromethyl)pyrimidin-2-yl)-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-chloropyridin-3-yl)methanesulfonamide 1379580-12-7 C21H20ClF3N6O3S
N-(5-(4-(4-amino-5-(trifluoromethyl)pyrimidin-2-yl)-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-chloropyridin-3-yl)methanesulfonamide
—— 4-chloro-1,1,1-trifluoro-5-methylhex-3-en-2-one 1442648-39-6 C7H8ClF3O
4-chloro-1,1,1-trifluoro-5-methylhex-3-en-2-one
—— 3-[2-(2,6-Dimethylpiperidin-1-yl)ethyl]-2-(4-phenylphenyl)thieno[3,2-d]pyrimidin-4-one 1004785-65-2 C27H29N3OS
3-[2-(2,6-Dimethylpiperidin-1-yl)ethyl]-2-(4-phenylphenyl)thieno[3,2-d]pyrimidin-4-one
—— tert-butyl (2S)-4-methyl-2-[[(1R,4S)-4-[4-[(1-methyl-2-oxopyridine-3-carbonyl)amino]piperidine-1-carbonyl]-1-phenyl-3,4-dihydro-2H-naphthalene-1-carbonyl]amino]pentanoate 1021900-43-5 C40H50N4O6
tert-butyl (2S)-4-methyl-2-[[(1R,4S)-4-[4-[(1-methyl-2-oxopyridine-3-carbonyl)amino]piperidine-1-carbonyl]-1-phenyl-3,4-dihydro-2H-naphthalene-1-carbonyl]amino]pentanoate
—— (R)-2-chloro-N-[1-cyclopentyl-2-(3-hydroxyazetidin-1-yl)ethyl]-4-fluoro-N-methylbenzamide 1380102-46-4 C18H24ClFN2O2
(R)-2-chloro-N-[1-cyclopentyl-2-(3-hydroxyazetidin-1-yl)ethyl]-4-fluoro-N-methylbenzamide
—— N-[(1S)-2-({5-[6-(cyclopropylmethoxy)-1,3-benzoxazol-2-yl]-4-methylisoxazol-3-yl}oxy)-1-methylethyl]acetamide 1380067-10-6 C20H23N3O5
N-[(1S)-2-({5-[6-(cyclopropylmethoxy)-1,3-benzoxazol-2-yl]-4-methylisoxazol-3-yl}oxy)-1-methylethyl]acetamide
—— (3-{4-[3-(3-chloro-phenyl)-4-(3,4-dimethyl-phenyl)-but-1-ynyl]-benzylamino}-propyl)-phosphonic acid 1379928-59-2 C28H31ClNO3P
(3-{4-[3-(3-chloro-phenyl)-4-(3,4-dimethyl-phenyl)-but-1-ynyl]-benzylamino}-propyl)-phosphonic acid
—— {(S)-2-[3-(2-methoxymethylphenyl)-[1,2,4]oxadiazol-5-yl]pyrrolidin-1-yl}-(5-methyl-2-[1,2,3]triazol-2-ylphenyl)methanone 1597517-51-5 C24H24N6O3
{(S)-2-[3-(2-methoxymethylphenyl)-[1,2,4]oxadiazol-5-yl]pyrrolidin-1-yl}-(5-methyl-2-[1,2,3]triazol-2-ylphenyl)methanone
—— 3-{4-[2-m-tolyloxyethoxy]phenyl}hex-4-ynoic acid 1354027-50-1 C21H22O4
3-{4-[2-m-tolyloxyethoxy]phenyl}hex-4-ynoic acid
—— [(2-Chlorophenyl)methyl]boronic acid 1350512-46-7 C7H8BClO2
[(2-Chlorophenyl)methyl]boronic acid
—— 6-chloro-2-[2-(3-chloropyridin-4-yl)pyridin-3-yl]-1H-benzimidazole 1228267-39-7 C17H10Cl2N4
6-chloro-2-[2-(3-chloropyridin-4-yl)pyridin-3-yl]-1H-benzimidazole
—— (S)-4-fluoro-3-methoxy-N-methyl-N-(3-methyl-1-(pyrrolidin-1-yl)butan-2-yl)benzamide 1380101-52-9 C18H27FN2O2
(S)-4-fluoro-3-methoxy-N-methyl-N-(3-methyl-1-(pyrrolidin-1-yl)butan-2-yl)benzamide
—— N5-(2-(3-fluorophenyl)-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N4,N4,1-trimethyl-1H-pyrazole-4,5-dicarboxamide 1380330-82-4 C20H18FN7O2
N5-(2-(3-fluorophenyl)-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N4,N4,1-trimethyl-1H-pyrazole-4,5-dicarboxamide
—— N-(1-acetylpiperidin-4-yl)-7-[2-(cyclopropylmethoxy)-4-fluoro-5-methoxyphenyl]-2-methyl-1H-pyrrolo[3,2-b]pyridine-3-carboxamide 1269236-64-7 C27H31FN4O4
N-(1-acetylpiperidin-4-yl)-7-[2-(cyclopropylmethoxy)-4-fluoro-5-methoxyphenyl]-2-methyl-1H-pyrrolo[3,2-b]pyridine-3-carboxamide
—— 3-[1-(3'-fluoro-4'-methoxy-biphenyl-3-sulfonyl)-5-methoxy-1H-indol-3-yl]-propionic acid 1055291-63-8 C25H22FNO6S
3-[1-(3'-fluoro-4'-methoxy-biphenyl-3-sulfonyl)-5-methoxy-1H-indol-3-yl]-propionic acid
—— 6-(N-(2-(2-bromoethoxy)ethyl)methylsulfonamido)-5-cyclopropyl-N-methyl-2-p-tolylfuro[2,3-b]pyridine-3-carboxamide 1345182-48-0 C24H28BrN3O5S
6-(N-(2-(2-bromoethoxy)ethyl)methylsulfonamido)-5-cyclopropyl-N-methyl-2-p-tolylfuro[2,3-b]pyridine-3-carboxamide
—— 6-ethoxy-N-(4-methoxy-phenyl)-N'-(1-methyl-piperidin-4-yl)-[1,3,5]triazine-2,4-diamine 1174126-18-1 C18H26N6O2
6-ethoxy-N-(4-methoxy-phenyl)-N'-(1-methyl-piperidin-4-yl)-[1,3,5]triazine-2,4-diamine
—— N-cyclopropyl-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1224939-95-0 C16H16N6O
N-cyclopropyl-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 4-[[[4-[2-[2-(2-Benzamidoethoxy)ethoxy]ethylamino]-6-[4-(benzylcarbamoyl)anilino]-1,3,5-triazin-2-yl]amino]methyl]benzoic acid 1282038-31-6 C38H40N8O6
4-[[[4-[2-[2-(2-Benzamidoethoxy)ethoxy]ethylamino]-6-[4-(benzylcarbamoyl)anilino]-1,3,5-triazin-2-yl]amino]methyl]benzoic acid
—— 4-((3,4-dichlorophenyl)(hydroxy)methyl)-3-methoxybenzamide 1354962-83-6 C15H13Cl2NO3
4-((3,4-dichlorophenyl)(hydroxy)methyl)-3-methoxybenzamide
—— 4-(1-cyano-8-methoxyindolizine-3-yl)benzoic acid 1246844-79-0 C17H12N2O3
4-(1-cyano-8-methoxyindolizine-3-yl)benzoic acid
—— N-[4-(dimethylamino)phenyl]-3-{4-[(4-fluorobenzyl)amino]-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl}benzamide 1174125-42-8 C27H24F4N6O2
N-[4-(dimethylamino)phenyl]-3-{4-[(4-fluorobenzyl)amino]-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl}benzamide
—— 4-[2-Ethyl-5-(3,5,6-trichloropyridin-2-yl)oxyphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1235557-17-1 C22H22Cl3NO4
4-[2-Ethyl-5-(3,5,6-trichloropyridin-2-yl)oxyphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— 3-[7-chloro-1-(4'-trifluoromethyl-biphenyl-3-sulfonyl)-1H-indol-3-yl]-propionic acid 1055293-28-1 C24H17ClF3NO4S
3-[7-chloro-1-(4'-trifluoromethyl-biphenyl-3-sulfonyl)-1H-indol-3-yl]-propionic acid
—— 6-((1R,2S)-2-aminocyclohexylamino)-2-(3,5-dimethylphenylamino)-5-fluoronicotinamide 1374972-89-0 C20H26FN5O
6-((1R,2S)-2-aminocyclohexylamino)-2-(3,5-dimethylphenylamino)-5-fluoronicotinamide
—— 5-[(2S)-2-(benzyloxy)propyl]-1-[2-(difluoromethyl)-4-fluorophenyl]-2-methyl-N-[3-methyl-4-(methylsulfonyl)phenyl]-1H-pyrrole-3-carboxamide 1221425-43-9 C31H31F3N2O4S
5-[(2S)-2-(benzyloxy)propyl]-1-[2-(difluoromethyl)-4-fluorophenyl]-2-methyl-N-[3-methyl-4-(methylsulfonyl)phenyl]-1H-pyrrole-3-carboxamide
—— 3-((R)-2-amino-2-phenyl-ethyl)-5-(4-benzo[1,3]dioxol-5-ylmethyl-piperazin-1-yl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione 1308375-16-7 C32H33F2N5O4
3-((R)-2-amino-2-phenyl-ethyl)-5-(4-benzo[1,3]dioxol-5-ylmethyl-piperazin-1-yl)-1-(2,6-difluoro-benzyl)-6-methyl-1H-pyrimidine-2,4-dione
—— 4-(4-Ethylthiophen-2-yl)phenol 1261951-61-4 C12H12OS
4-(4-Ethylthiophen-2-yl)phenol