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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[5-fluoro-4-(2-methoxyphenyl)-2-oxopyridin-1(2H)-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide 1398502-94-7 C18H21FN2O6S
4-[5-fluoro-4-(2-methoxyphenyl)-2-oxopyridin-1(2H)-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide
—— 4-amino-6-({1-[5-chloro-6-fluoro-2-methoxy-4'-(methylsulfonyl)biphenyl-3-yl]ethyl}amino)pyrimidine-5-carbonitrile 1402000-18-3 C21H19ClFN5O3S
4-amino-6-({1-[5-chloro-6-fluoro-2-methoxy-4'-(methylsulfonyl)biphenyl-3-yl]ethyl}amino)pyrimidine-5-carbonitrile
—— (4S,5R,6R)-4-Azido-5-(6-benzyloxycarbonylamino-hexanoylamino)-6-((1S,2R)-1,2,3-triacetoxy-propyl)-5,6-dihydro-4H-pyran-2-carboxylic acid ethyl ester 184643-33-2 C31H41N5O12
(4S,5R,6R)-4-Azido-5-(6-benzyloxycarbonylamino-hexanoylamino)-6-((1S,2R)-1,2,3-triacetoxy-propyl)-5,6-dihydro-4H-pyran-2-carboxylic acid ethyl ester
—— 4-(2-Diethylamino-ethylamino)-3-nitro-benzonitrile 15452-10-5 C13H18N4O2
4-(2-Diethylamino-ethylamino)-3-nitro-benzonitrile
—— Methyl 1-butyl-5-ethyl-3-[[2'-(1H-tetrazol-5-yl)-1,1'-biphenyl-4-yl]methyl]-1H-pyrazole-4-carboxylate 177846-20-7 C25H28N6O2
Methyl 1-butyl-5-ethyl-3-[[2'-(1H-tetrazol-5-yl)-1,1'-biphenyl-4-yl]methyl]-1H-pyrazole-4-carboxylate
—— (R,S)-(+)-N-(3-(1H-Imidazol-4-yl)propyl)-3-phenylbutanamide 163632-28-8 C16H21N3O
(R,S)-(+)-N-(3-(1H-Imidazol-4-yl)propyl)-3-phenylbutanamide
—— US10138229, Example 149 1558037-78-7 C22H21F4N5O3
US10138229, Example 149
—— 3-(1,3-benzothiazol-2-yl)-4-phenyl-1H-pyrrol-2-amine 1429046-80-9 C17H13N3S
3-(1,3-benzothiazol-2-yl)-4-phenyl-1H-pyrrol-2-amine
—— benzyl N-[1-[5-(1,3-benzothiazol-2-yl)-6-oxo-4-[[(3R)-piperidin-3-yl]amino]-1,6-dihydropyrimidin-2-yl]piperidin-4-yl]carbamate 1433165-25-3 C29H33N7O3S
benzyl N-[1-[5-(1,3-benzothiazol-2-yl)-6-oxo-4-[[(3R)-piperidin-3-yl]amino]-1,6-dihydropyrimidin-2-yl]piperidin-4-yl]carbamate
—— 1-[6-[3,5-dimethyl-2-[[5-methyl-2-(oxan-4-yl)-3,4-dihydro-1H-isoquinolin-6-yl]methoxy]phenyl]pyridin-2-yl]-5-methoxypyrazole-4-carboxylic acid 1579515-32-4 C34H38N4O5
1-[6-[3,5-dimethyl-2-[[5-methyl-2-(oxan-4-yl)-3,4-dihydro-1H-isoquinolin-6-yl]methoxy]phenyl]pyridin-2-yl]-5-methoxypyrazole-4-carboxylic acid
—— N-((S)-1-(3-chloro-4-cyanophenyl)-2-hydroxyethyl)-3-(tetrahydrofuran-3-ylamino)isoquinoline-6-carboxamide 1574396-29-4 C23H21ClN4O3
N-((S)-1-(3-chloro-4-cyanophenyl)-2-hydroxyethyl)-3-(tetrahydrofuran-3-ylamino)isoquinoline-6-carboxamide
—— (2S,4R)-2-((tert-butyldimethylsilyloxy)methyl)tetrahydro-2H-pyran-4-amine 1395080-67-7 C12H27NO2Si
(2S,4R)-2-((tert-butyldimethylsilyloxy)methyl)tetrahydro-2H-pyran-4-amine
—— methyl (2S)-2-(tert-butoxy)-2-[(22S)-4,18,22,28-tetramethyl-21,27-dioxa-1,5,7,8-tetraazahexacyclo[26.2.2.1<sup>(6,9)</sup>.1<sup>(10,14)</sup>.0<sup>(2,7)</sup>.0<sup>(15,20)</sup>]tetratriaconta-2,4,6(34),8,10(33),11,13,15(20),16,18-decaen-3-yl]acetate 1567218-23-8 C39H50N4O5
methyl (2S)-2-(tert-butoxy)-2-[(22S)-4,18,22,28-tetramethyl-21,27-dioxa-1,5,7,8-tetraazahexacyclo[26.2.2.1<sup>(6,9)</sup>.1<sup>(10,14)</sup>.0<sup>(2,7)</sup>.0<sup>(15,20)</sup>]tetratriaconta-2,4,6(34),8,10(33),11,13,15(20),16,18-decaen-3-yl]acetate
—— 5-Isopropylpyridine-2,3-diamine 1256820-19-5 C8H13N3
5-Isopropylpyridine-2,3-diamine
—— Methoxy-N-(2-methoxyethyl)-2-methylleucine 1250074-06-6 C11H23NO4
Methoxy-N-(2-methoxyethyl)-2-methylleucine
—— 2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-N-(1-methylimidazol-4-yl)sulfonyl-1,3-thiazole-4-carboxamide 1282545-09-8 C28H31N5O6S2
2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-N-(1-methylimidazol-4-yl)sulfonyl-1,3-thiazole-4-carboxamide
—— N-[6-(1H-indol-4-yl)-1H-indazol-4-yl]-2-({3-[(phenylmethyl)oxy]-1-piperidinyl}methyl)-1,3-thiazole-4-carboxamide formate 1198435-82-3 CH2O2*C32H30N6O2S
N-[6-(1H-indol-4-yl)-1H-indazol-4-yl]-2-({3-[(phenylmethyl)oxy]-1-piperidinyl}methyl)-1,3-thiazole-4-carboxamide formate
—— (5R)-3-bromo-7-(3-pyridinyl)-spiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-2'-amine 1215866-68-4 C19H13BrN4O2
(5R)-3-bromo-7-(3-pyridinyl)-spiro[chromeno[2,3-b]pyridine-5,4'-[1,3]oxazol]-2'-amine
—— (2R,6S,12Z,13aS,14aR,16aS)-5'-methyl-N-[(1-methylcyclopropyl)sulfonyl]-5,16-dioxo-6-[(3,3,3-trifluoropropanoyl)amino]-1,1',2',6,7,8,9,10,11,13a,14,15,16,16a-tetradecahydrospiro[cyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-2,3'-pyrano[2,3-c]quinoline]-14a-carboxamide 1565772-53-3 C37H44F3N5O7S
(2R,6S,12Z,13aS,14aR,16aS)-5'-methyl-N-[(1-methylcyclopropyl)sulfonyl]-5,16-dioxo-6-[(3,3,3-trifluoropropanoyl)amino]-1,1',2',6,7,8,9,10,11,13a,14,15,16,16a-tetradecahydrospiro[cyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-2,3'-pyrano[2,3-c]quinoline]-14a-carboxamide
—— 5-(3-(difluoromethyl)phenyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ethylamide 1571135-56-2 C16H16F2N2O2
5-(3-(difluoromethyl)phenyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxylic acid ethylamide
—— (2R,11S,19aS)-15-fluoro-7,12-dimethyl-2-{[2-(2-naphthyl)acetyl]amino}-5,8,13-trioxo-N-(4-pyridinylmethyl)-2,3,6,7,8,9,10,11,12,13,19,19a-dodecahydro-1H,5H-pyrrolo[2,1-c][1,4,7,12]benzoxatriazacyclopentadecine-11-carboxamide trifluoroacetate 1264228-48-9 C2HF3O2*C39H41FN6O6
(2R,11S,19aS)-15-fluoro-7,12-dimethyl-2-{[2-(2-naphthyl)acetyl]amino}-5,8,13-trioxo-N-(4-pyridinylmethyl)-2,3,6,7,8,9,10,11,12,13,19,19a-dodecahydro-1H,5H-pyrrolo[2,1-c][1,4,7,12]benzoxatriazacyclopentadecine-11-carboxamide trifluoroacetate
—— —— 1637357-54-0 C12H24B10
—— 1-(2-fluoro-4-{4-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yloxyimino]cyclohexyl}phenyl)-3-methylurea 1393685-52-3 C24H33FN6O3
1-(2-fluoro-4-{4-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yloxyimino]cyclohexyl}phenyl)-3-methylurea
—— N-(cyclopropylsulfamoyl)-2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-4-carboxamide 1282545-27-0 C27H32N4O6S2
N-(cyclopropylsulfamoyl)-2-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-4-carboxamide
—— Potassium 6-beta-[S-1-Hydroxy-2-(4-hydroxyphenyl)-2-oxoethyl]penicillanate 109990-55-8 C16H16NO6S*K
Potassium 6-beta-[S-1-Hydroxy-2-(4-hydroxyphenyl)-2-oxoethyl]penicillanate
—— (R)-6-((1-(cyclopropanecarbonyl)pyrrolidin-3-yl)methyl)-5-(4'-(pyridin-4-yl)-[1,1'-biphenyl]-4-yl)-4,6-diazaspiro[2.4]hept-4-en-7-one 1579516-95-2 C31H30N4O2
(R)-6-((1-(cyclopropanecarbonyl)pyrrolidin-3-yl)methyl)-5-(4'-(pyridin-4-yl)-[1,1'-biphenyl]-4-yl)-4,6-diazaspiro[2.4]hept-4-en-7-one
—— (1S)-1-amino-1-(4-chloro-3-fluorophenyl)propan-2-ol 1336831-53-8 C9H11ClFNO
(1S)-1-amino-1-(4-chloro-3-fluorophenyl)propan-2-ol
—— 5-(4-cyclopropyl-[1,3]thiazolo[4,5-c]pyridin-2-yl)-2-morpholin-4-yl-4-[[(3R)-piperidin-3-yl]amino]-1H-pyrimidin-6-one;hydrochloride 1433153-28-6 C22H27N7O2S*ClH
5-(4-cyclopropyl-[1,3]thiazolo[4,5-c]pyridin-2-yl)-2-morpholin-4-yl-4-[[(3R)-piperidin-3-yl]amino]-1H-pyrimidin-6-one;hydrochloride
—— (3S,5S)-N-{1-[(4-hydroxypiperidin-1-yl)carbonyl]-5-[4-(trifluoromethyl)phenyl]piperidin-3-yl}benzenecarboxamide 1246028-70-5 C25H28F3N3O3
(3S,5S)-N-{1-[(4-hydroxypiperidin-1-yl)carbonyl]-5-[4-(trifluoromethyl)phenyl]piperidin-3-yl}benzenecarboxamide
—— —— 1390624-58-4 C14H12ClN5O2S
—— (3S,5R,8S)-3,8-bis(bromomethyl)-3-(tert-butyl)-8-phenyl-2,7-dioxaspiro[4.4]nonane 1643718-49-3 C19H26Br2O2
(3S,5R,8S)-3,8-bis(bromomethyl)-3-(tert-butyl)-8-phenyl-2,7-dioxaspiro[4.4]nonane
—— (2S,3S,6'S)-5-chloro-4',6,6'-trimethoxy-1'-methyl-3-sulfanylspiro[3H-1-benzofuran-2,3'-piperazine]-2',5'-dione 112875-52-2 C15H17ClN2O6S
(2S,3S,6'S)-5-chloro-4',6,6'-trimethoxy-1'-methyl-3-sulfanylspiro[3H-1-benzofuran-2,3'-piperazine]-2',5'-dione
—— —— 119604-62-5 C16H13BF3NO7
—— 1-(4-{4-[1-(5-ethyl-pyrimidin-2-yl)piperidin-4-yloxyimino]cyclohexyl}-2,5-difluorophenyl)-3-isopropylurea 1393685-11-4 C27H36F2N6O2
1-(4-{4-[1-(5-ethyl-pyrimidin-2-yl)piperidin-4-yloxyimino]cyclohexyl}-2,5-difluorophenyl)-3-isopropylurea
—— 4-chloro-N-[1-(2-hydroxy-3-nitrophenyl)ethylideneamino]benzamide 1235578-11-6 C15H12ClN3O4
4-chloro-N-[1-(2-hydroxy-3-nitrophenyl)ethylideneamino]benzamide
—— 4,4'-(4-(furan-2-yl)pyridine-2,6-diyl)diphenol 1383781-95-0 C21H15NO3
4,4'-(4-(furan-2-yl)pyridine-2,6-diyl)diphenol
—— 2-propylsulfanyl-furan 16003-06-8 C7H10OS
2-propylsulfanyl-furan
—— 7a-Butyl-hexahydro-pyrrolo[1,2-a]imidazole 123414-20-0 C10H20N2
7a-Butyl-hexahydro-pyrrolo[1,2-a]imidazole
—— N,N-diethylethanamine;5-(5-methylsulfanyl-1,3,4-thiadiazol-2-yl)-1,3,4-thiadiazole-2-carbodithioic acid 114020-06-3 C6H4N4S5*C6H15N
N,N-diethylethanamine;5-(5-methylsulfanyl-1,3,4-thiadiazol-2-yl)-1,3,4-thiadiazole-2-carbodithioic acid
—— (5Z,7E)-isopropyl 7-acetyl-3,4-dihydro-4-oxo-2H-1,2-diazepine-3-carboxylate 1246011-28-8 C11H14N2O4
(5Z,7E)-isopropyl 7-acetyl-3,4-dihydro-4-oxo-2H-1,2-diazepine-3-carboxylate
—— [(η5-(H2CC(Me)CH2)2C8H8P)(C5H4CH2CHCH2)]Fe 1210109-77-5 C24H31FeP
[(η5-(H2CC(Me)CH2)2C8H8P)(C5H4CH2CHCH2)]Fe
—— —— 1456596-00-1 C22H16F3N5OS
—— 1-[5-tert-butyl-2-methoxy-3-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]phenyl]-3-[(1S,2R)-1-hydroxy-5-methoxy-2,3-dihydro-1H-inden-2-yl]urea 1283525-94-9 C24H29F3N2O5
1-[5-tert-butyl-2-methoxy-3-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]phenyl]-3-[(1S,2R)-1-hydroxy-5-methoxy-2,3-dihydro-1H-inden-2-yl]urea
—— —— 1446521-35-2 C21H28N2O5
—— —— 1374596-12-9 C18H20N2O4
—— 4-(4-amino-3,5-difluorophenyl)cyclohexanone O-[1-(5-methylpyrimidin-2-yl)piperidin-4-yl]oxime 1407965-86-9 C22H27F2N5O
4-(4-amino-3,5-difluorophenyl)cyclohexanone O-[1-(5-methylpyrimidin-2-yl)piperidin-4-yl]oxime
—— 1-(3,5-dideoxy-3,5-epithio-2-O-methylsulphonyl-β-D-xylofuranosyl)uracil 115195-76-1 C10H12N2O6S2
1-(3,5-dideoxy-3,5-epithio-2-O-methylsulphonyl-β-D-xylofuranosyl)uracil
—— —— 1440972-69-9 C11H19NO3
—— N-[1-(3,5-difluorophenyl)-3-(4-fluorophenylthio)-2-propenylidene]-4-methylaniline 1140915-19-0 C22H16F3NS
N-[1-(3,5-difluorophenyl)-3-(4-fluorophenylthio)-2-propenylidene]-4-methylaniline
—— N-[(4-chloro-2-hydroxyphenyl)methylideneamino]-3-nitrobenzamide 1235716-40-1 C14H10ClN3O4
N-[(4-chloro-2-hydroxyphenyl)methylideneamino]-3-nitrobenzamide