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中文名称 英文名称 CAS号 化学式 结构式图片
—— N4-(4-fluorophenyl)-N2-(4-{4-[(2-methylaminopyridin-3-ylmethyl)amino]piperidine-1-sulphonyl}-phenyl)pyrimidine-2,4-diamine 1049667-16-4 C28H31FN8O2S
N4-(4-fluorophenyl)-N2-(4-{4-[(2-methylaminopyridin-3-ylmethyl)amino]piperidine-1-sulphonyl}-phenyl)pyrimidine-2,4-diamine
—— 5-(5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-yloxymethyl)-isophthalic acid 1219739-34-0 C28H19ClN2O5
5-(5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-yloxymethyl)-isophthalic acid
—— 1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [2-(methanesulfonyl-methyl-amino)-pyrimidin-4-ylmethyl]-amide 1220168-08-0 C20H18FN7O3S
1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carboxylic acid [2-(methanesulfonyl-methyl-amino)-pyrimidin-4-ylmethyl]-amide
—— 8-fluoro-3-methyl-1-oxo-(S)-2-pyrrolidin-3-yl-1,2-dihydro-isoquinoline-4-carboxylic acid [(S)-cyclopropyl-(3-fluoro-phenyl)-methyl]-amide 1215094-11-3 C25H25F2N3O2
8-fluoro-3-methyl-1-oxo-(S)-2-pyrrolidin-3-yl-1,2-dihydro-isoquinoline-4-carboxylic acid [(S)-cyclopropyl-(3-fluoro-phenyl)-methyl]-amide
—— 8-(2,6-dichloro-3,5-dimethoxy-phenyl)-quinoxaline-5-carboxylic acid (4-diethylaminomethyl-1H-imidazol-2-yl)-amide 1197330-10-1 C25H26Cl2N6O3
8-(2,6-dichloro-3,5-dimethoxy-phenyl)-quinoxaline-5-carboxylic acid (4-diethylaminomethyl-1H-imidazol-2-yl)-amide
—— 5-(Benzo[d]thiazol-2-yl)-6-((1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)-cyclopentylamino)-2-(4-(pyridin-4-yl)piperidin-1-yl)pyrimidin-4(3H)-on 1433151-55-3 C27H30N6O4S
5-(Benzo[d]thiazol-2-yl)-6-((1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)-cyclopentylamino)-2-(4-(pyridin-4-yl)piperidin-1-yl)pyrimidin-4(3H)-on
—— 2-amino-4-methyl-6-(1H-pyrazol-4-yl)-8-((tetrahydrofuran-3-yl)methyl)pyrido[2,3-d]pyrimidin-7(8H)one 1013100-81-6 C16H18N6O2
2-amino-4-methyl-6-(1H-pyrazol-4-yl)-8-((tetrahydrofuran-3-yl)methyl)pyrido[2,3-d]pyrimidin-7(8H)one
—— 5-(3-(cyanomethoxy)-5-(isobutylcarbamoyl)phenyl)-2-(4-fluorophenyl)-N-methylbenzofuran-3-carboxamide 1217338-49-2 C29H26FN3O4
5-(3-(cyanomethoxy)-5-(isobutylcarbamoyl)phenyl)-2-(4-fluorophenyl)-N-methylbenzofuran-3-carboxamide
—— 5-[6-chloro-5-(3-methoxy-phenylethynyl)-1H-benzoimidazol-2-yloxy]-2-methyl-benzoic acid methyl ester 1219738-20-1 C25H19ClN2O4
5-[6-chloro-5-(3-methoxy-phenylethynyl)-1H-benzoimidazol-2-yloxy]-2-methyl-benzoic acid methyl ester
—— 5-(3,4,5-trimethoxyphenyl)-5-(2-carboxyprop-2-enyl)-3-methylene-2-pyrrolidinone 154188-13-3 C18H21NO6
5-(3,4,5-trimethoxyphenyl)-5-(2-carboxyprop-2-enyl)-3-methylene-2-pyrrolidinone
—— 3,3-Diethyl-3,4,5,6-tetrahydro-5,6-dioxo-2H-naphth<2,1-e>-1,3-oxazinium-chlorid 130084-25-2 C16H18NO3*Cl
3,3-Diethyl-3,4,5,6-tetrahydro-5,6-dioxo-2H-naphth<2,1-e>-1,3-oxazinium-chlorid
—— 1-(4,4-Dimethyl-3-trimethylsilanyloxy-pent-1-ynyl)-1,1,2,2,2-pentamethyl-disilane 130995-05-0 C15H34OSi3
1-(4,4-Dimethyl-3-trimethylsilanyloxy-pent-1-ynyl)-1,1,2,2,2-pentamethyl-disilane
—— 4-amino-1-ethyl-7-methoxy-[1,2,4]triazolo[4,3-a]quinoxaline methanesulfonate 127710-50-3 CH4O3S*C12H13N5O
4-amino-1-ethyl-7-methoxy-[1,2,4]triazolo[4,3-a]quinoxaline methanesulfonate
—— N-(4-fluorophenyl)-7-methyl-5-(6-methyl-1H-1,3-benzodiazol-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 1266342-97-5 C21H17FN6
N-(4-fluorophenyl)-7-methyl-5-(6-methyl-1H-1,3-benzodiazol-2-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— 1-<i>p</i>-tolyl-1<i>H</i>-[1,2,4]triazole-3,5-diyldiamine 109442-43-5 C9H11N5
1-<i>p</i>-tolyl-1<i>H</i>-[1,2,4]triazole-3,5-diyldiamine
—— 2,6-Dichloro-4-[3-[[4-[[[6-(trifluoromethyl)pyridin-3-yl]methylamino]methyl]phenyl]methoxy]-1,2,4-triazin-6-yl]phenol 1191247-83-2 C24H18Cl2F3N5O2
2,6-Dichloro-4-[3-[[4-[[[6-(trifluoromethyl)pyridin-3-yl]methylamino]methyl]phenyl]methoxy]-1,2,4-triazin-6-yl]phenol
—— 2-(2-fluoro-4-hydroxyphenyl)thiazol-4-carboxylic acid [4-(5-amino-3,3-dimethylcyclohexyl)pyridin-3yl]amide 1187054-56-3 C23H25FN4O2S
2-(2-fluoro-4-hydroxyphenyl)thiazol-4-carboxylic acid [4-(5-amino-3,3-dimethylcyclohexyl)pyridin-3yl]amide
—— Methyl 5-[[5-amino-1-[6-[5-amino-4-[(4-methoxycarbonyl-2-methylpyrazol-3-yl)diazenyl]-3-methylpyrazol-1-yl]pyrimidin-4-yl]-3-methylpyrazol-4-yl]diazenyl]-1-methylpyrazole-4-carboxylate 1186407-33-9 C24H26N16O4
Methyl 5-[[5-amino-1-[6-[5-amino-4-[(4-methoxycarbonyl-2-methylpyrazol-3-yl)diazenyl]-3-methylpyrazol-1-yl]pyrimidin-4-yl]-3-methylpyrazol-4-yl]diazenyl]-1-methylpyrazole-4-carboxylate
—— 3-(4-(6-(6-(2-(3-fluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)pyridin-2-yl)piperazin-1-yl)propanenitrile 1196548-45-4 C28H29FN8
3-(4-(6-(6-(2-(3-fluorophenyl)pyrrolidin-1-yl)imidazo[1,2-b]pyridazin-3-yl)pyridin-2-yl)piperazin-1-yl)propanenitrile
—— N-(1-(3-(cyclopentyloxy)phenyl)ethyl)-3-((2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methoxy)propane-1-sulfonamide 1198221-48-5 C21H29N3O6S
N-(1-(3-(cyclopentyloxy)phenyl)ethyl)-3-((2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methoxy)propane-1-sulfonamide
—— (R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-fluoro-phenyl)-ethyl]-2-piperidin-1-yl-propionamide 1194095-88-9 C23H30FN5O2
(R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-fluoro-phenyl)-ethyl]-2-piperidin-1-yl-propionamide
—— N-methyl-3-(3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl)benzenesulfonamide 1033724-46-7 C14H12N4O3S
N-methyl-3-(3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl)benzenesulfonamide
—— N-[7-(5-bromo-2-chlorophenyl)-6-(4-chlorophenyl)-2,2-dimethyl-3,4-dihydro-2H-pyrano[2,3-b]pyridin-4-yl]-2-hydroxy-2-methylpropanamide 1044586-02-8 C26H25BrCl2N2O3
N-[7-(5-bromo-2-chlorophenyl)-6-(4-chlorophenyl)-2,2-dimethyl-3,4-dihydro-2H-pyrano[2,3-b]pyridin-4-yl]-2-hydroxy-2-methylpropanamide
—— 4-(1,3-benzothiazol-2-ylmethyl)-2,2-difluoro-8(1-hydroxyethyl)-2H-1,4-benzoxazin-3(4H)-one 1263411-23-9 C18H14F2N2O3S
4-(1,3-benzothiazol-2-ylmethyl)-2,2-difluoro-8(1-hydroxyethyl)-2H-1,4-benzoxazin-3(4H)-one
—— N-[[1-[5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]piperidin-4-yl]methyl]hexanamide 1321872-21-2 C24H32N6O
N-[[1-[5-[2-(6-aminopyridin-3-yl)ethynyl]-6-methylpyrimidin-4-yl]piperidin-4-yl]methyl]hexanamide
—— N-Hexyl-2-(6-methoxy-1,3,4,5-tetrahydro-3-acenaphthylenyl)-acetamide 1139164-52-5 C21H29NO2
N-Hexyl-2-(6-methoxy-1,3,4,5-tetrahydro-3-acenaphthylenyl)-acetamide
—— [Cd(homophthalate)(1,3-bis(4-pyridyl)propane)] 1335033-41-4 C9H6O4*C13H14N2*Cd
[Cd(homophthalate)(1,3-bis(4-pyridyl)propane)]
—— (4Z)-4-(2-(imidazolidin-2-ylidene)-3-(4-methoxyphenyl)-3-oxopropylidene)-3-methyl-1-phenyl-1H-pyrazol-5(4H)-one 1463517-80-7 C23H22N4O3
(4Z)-4-(2-(imidazolidin-2-ylidene)-3-(4-methoxyphenyl)-3-oxopropylidene)-3-methyl-1-phenyl-1H-pyrazol-5(4H)-one
—— 2-(3-chloro-5-methylphenyl)-4,4,6-trimethyl-1,3,2-dioxaborinane 1451144-86-7 C13H18BClO2
2-(3-chloro-5-methylphenyl)-4,4,6-trimethyl-1,3,2-dioxaborinane
—— —— 1146347-26-3 C49H41FeIN4O6
—— 12-(2,5-dibromothiophene-3-yl)dodecyl acetate 1548449-58-6 C18H28Br2O2S
12-(2,5-dibromothiophene-3-yl)dodecyl acetate
—— (E)-2-cinnamyl-4-fluoroaniline 1310708-03-2 C15H14FN
(E)-2-cinnamyl-4-fluoroaniline
—— diethyl 5-bromo-3-(4-chlorophenylamino)-2-oxoindolin-3-ylphosphonate 1210948-96-1 C18H19BrClN2O4P
diethyl 5-bromo-3-(4-chlorophenylamino)-2-oxoindolin-3-ylphosphonate
—— (2R,16R)-16-(tert-butyldimethylsilyloxy)-2-(4-methoxybenzyloxy)heptadecan-1-ol 1587697-43-5 C31H58O4Si
(2R,16R)-16-(tert-butyldimethylsilyloxy)-2-(4-methoxybenzyloxy)heptadecan-1-ol
—— 5'-methyl-1,3-diphenyl-4,5-dihydrospiro[furo[3,4-e]pyrazolo[4,3-b]pyridine-8,3'-indoline]-2',7(1H)-dione 1310545-66-4 C28H20N4O3
5'-methyl-1,3-diphenyl-4,5-dihydrospiro[furo[3,4-e]pyrazolo[4,3-b]pyridine-8,3'-indoline]-2',7(1H)-dione
—— —— 1620645-43-3 C19H33NO3SSi
—— US10202379, Reference Example 317 1370240-49-5 C25H25N3O4S
US10202379, Reference Example 317
—— 5-ethyl-6-{2-[4-(1-isopropyl-R-pyrrolidin-2-yl-methoxy)phenyl]benzoxazol-6-yl}-4,5-dihydro-2H-pyridazin-3-one 1346700-94-4 C27H32N4O3
5-ethyl-6-{2-[4-(1-isopropyl-R-pyrrolidin-2-yl-methoxy)phenyl]benzoxazol-6-yl}-4,5-dihydro-2H-pyridazin-3-one
—— 3-[1-(2-methoxyethyl)-1H-pyrazol-4-yl]-2-methyl-8-(4-morpholinyl)-6-(trifluoromethyl)-imidazo[1,2-b]pyridazine 1298031-66-9 C18H21F3N6O2
3-[1-(2-methoxyethyl)-1H-pyrazol-4-yl]-2-methyl-8-(4-morpholinyl)-6-(trifluoromethyl)-imidazo[1,2-b]pyridazine
—— 5-[2-(3-hydroxymethyloxetan-3-ylmethoxy)-3,4-dimethoxyphenyl]indan-1-one 1345878-56-9 C22H24O6
5-[2-(3-hydroxymethyloxetan-3-ylmethoxy)-3,4-dimethoxyphenyl]indan-1-one
—— 2-(3-(4-(7-(1-methyl-1H-pyrazol-4-yl)imidazo[1,2-c]pyrimidin-5-yl)-1H-pyrazol-1-yl)-1-((1-trifluoromethyl)cyclopropanecarbonyl)azetidin-3-yl)acetonitrile 1339888-80-0 C23H20F3N9O
2-(3-(4-(7-(1-methyl-1H-pyrazol-4-yl)imidazo[1,2-c]pyrimidin-5-yl)-1H-pyrazol-1-yl)-1-((1-trifluoromethyl)cyclopropanecarbonyl)azetidin-3-yl)acetonitrile
—— 3-(4-bromobenzyl)-8-chloro-5-hydroxy-4-methyl-1H-quinolin-2-one 1071497-10-3 C17H13BrClNO2
3-(4-bromobenzyl)-8-chloro-5-hydroxy-4-methyl-1H-quinolin-2-one
—— 2-(4-bromophenyl)-4-methyl[1]benzothiopyrano[4,3-c ]pyrazol-3(2 H)-one 128789-94-6 C17H11BrN2OS
2-(4-bromophenyl)-4-methyl[1]benzothiopyrano[4,3-c ]pyrazol-3(2 H)-one
—— 2-(thiophen-2-yl)-2-(4-fluorophenylamino)acetonitrile 1249139-69-2 C12H9FN2S
2-(thiophen-2-yl)-2-(4-fluorophenylamino)acetonitrile
—— (E)-methyl 5-{2-sec-butyl-5-[2-(furan-2-yl)ethyl]-5-methyl-1,3,2-dioxaborolan-4-yl}pent-2-enoate 1314866-94-8 C19H29BO5
(E)-methyl 5-{2-sec-butyl-5-[2-(furan-2-yl)ethyl]-5-methyl-1,3,2-dioxaborolan-4-yl}pent-2-enoate
—— —— 1333503-46-0 C40H65O7P
—— 4-butyl-3-methyl-1-phenyl-1,7-dihydro-5H-furo[3,4-b]pyrazolo[4,3-e]pyridine-5-one 1049682-38-3 C19H19N3O2
4-butyl-3-methyl-1-phenyl-1,7-dihydro-5H-furo[3,4-b]pyrazolo[4,3-e]pyridine-5-one
—— (R,E)-ethyl 5-(hydroxymethyl)-8-phenyloct-6-enoate 1449246-12-1 C17H24O3
(R,E)-ethyl 5-(hydroxymethyl)-8-phenyloct-6-enoate
—— 5-[4-(3-chloropropoxy)phenyl]-2-isopropyl-2H-pyridazin-3-one 1353387-78-6 C16H19ClN2O2
5-[4-(3-chloropropoxy)phenyl]-2-isopropyl-2H-pyridazin-3-one
—— 6-amino-3-(6-((4-(dimethylamino)benzylidene)amino)-5-nitropyridin-3-yl)-4-methyl-2H-chromen-2-one 1145997-02-9 C24H21N5O4
6-amino-3-(6-((4-(dimethylamino)benzylidene)amino)-5-nitropyridin-3-yl)-4-methyl-2H-chromen-2-one