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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(3R,4R)-4-(18F)fluoranyl-3-[(2-methylpropan-2-yl)oxycarbonyl]oxolan-3-yl]-[(2-methylpropan-2-yl)oxycarbonyl]sulfamic acid 1351450-90-2 C14H24FNO8S
[(3R,4R)-4-(18F)fluoranyl-3-[(2-methylpropan-2-yl)oxycarbonyl]oxolan-3-yl]-[(2-methylpropan-2-yl)oxycarbonyl]sulfamic acid
—— US10485800, Cmpd ID FP 1351476-57-7 C26H25F3N4
US10485800, Cmpd ID FP
—— 9-[(1-acryloyl-4-piperidinyl)methyl]-6-amino-7-(4-phenoxyphenyl)-7,9-dihydro-8H-purin-8-one 1351635-76-1 C26H26N6O3
9-[(1-acryloyl-4-piperidinyl)methyl]-6-amino-7-(4-phenoxyphenyl)-7,9-dihydro-8H-purin-8-one
—— (4E,6E,8R)-N-[(3S,4S)-1,4-dimethyl-2,5-dioxopyrrolidin-3-yl]-8-[(1R,3R,4S,5R,8R)-1,4-dimethylspiro[2,9-dioxabicyclo[3.3.1]non-6-ene-8,2'-oxirane]-3-yl]-6-methyl-3-oxonona-4,6-dienamide 1319647-35-2 C26H34N2O7
(4E,6E,8R)-N-[(3S,4S)-1,4-dimethyl-2,5-dioxopyrrolidin-3-yl]-8-[(1R,3R,4S,5R,8R)-1,4-dimethylspiro[2,9-dioxabicyclo[3.3.1]non-6-ene-8,2'-oxirane]-3-yl]-6-methyl-3-oxonona-4,6-dienamide
—— PHD Inhibitor, 8{2} 1241877-24-6 C25H26N4O7
PHD Inhibitor, 8{2}
—— 4-(5-Chlorothiophen-2-yl)-2-hydroxybenzoic acid 1349846-95-2 C11H7ClO3S
4-(5-Chlorothiophen-2-yl)-2-hydroxybenzoic acid
—— 1-[(1-benzyl-4-hydroxy-2-oxo-1,2-dihydropyridazino[1,6-a]benzimidazol-3-yl)carbonyl]piperidine-4-carboxylic acid 1296651-97-2 C24H22N4O5
1-[(1-benzyl-4-hydroxy-2-oxo-1,2-dihydropyridazino[1,6-a]benzimidazol-3-yl)carbonyl]piperidine-4-carboxylic acid
—— 3-Benzofuranacetamide, 6-methoxy-N-[3-[[(phenylamino)carbonyl]amino]phenyl]- 1385677-95-1 C24H21N3O4
3-Benzofuranacetamide, 6-methoxy-N-[3-[[(phenylamino)carbonyl]amino]phenyl]-
—— (1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-9-(4-(methylsulfonyl)phenyl)-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysene-3a-carboxylic acid 1350914-91-8 C37H52O4S
(1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-9-(4-(methylsulfonyl)phenyl)-1-(prop-1-en-2-yl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysene-3a-carboxylic acid
—— 2-bromo-4-nitro-1-{(2S)-2-{[4'-(trifluoromethoxy)[1,1'-biphenyl]-4-yl]oxy}-3-[triisopropylsilyloxy]propyl}-1H-imidazole 1263417-25-9 C28H35BrF3N3O5Si
2-bromo-4-nitro-1-{(2S)-2-{[4'-(trifluoromethoxy)[1,1'-biphenyl]-4-yl]oxy}-3-[triisopropylsilyloxy]propyl}-1H-imidazole
—— N-[(4-hydroxy-1-{[6-(2-methylphenyl)pyridin-3-yl]methyl}-2-oxo-1,2,5,7-tetrahydrothieno[3,4-b]pyridin-3-yl)carbonyl]glycine trifluoroacetate 1186091-60-0 C2HF3O2*C23H21N3O5S
N-[(4-hydroxy-1-{[6-(2-methylphenyl)pyridin-3-yl]methyl}-2-oxo-1,2,5,7-tetrahydrothieno[3,4-b]pyridin-3-yl)carbonyl]glycine trifluoroacetate
—— 6-cyclopropyl-3-(pyrimidin-5-ylamino)pyrazine-2-carboxylic acid [5-(3-fluoro-azetidine-1-carbonyl)-1-methyl-1H-pyrazol-4-yl]amide 1352197-64-8 C20H20FN9O2
6-cyclopropyl-3-(pyrimidin-5-ylamino)pyrazine-2-carboxylic acid [5-(3-fluoro-azetidine-1-carbonyl)-1-methyl-1H-pyrazol-4-yl]amide
—— N-(4-(3-(5-tert-butylisoxazol-3-yl)ureido)phenyl)-5-(1,2,2,4,6,6-hexamethylpiperidin-4-yloxy)picolinamide 1351522-20-7 C31H42N6O4
N-(4-(3-(5-tert-butylisoxazol-3-yl)ureido)phenyl)-5-(1,2,2,4,6,6-hexamethylpiperidin-4-yloxy)picolinamide
—— 2-((4-chlorobenzyl)(methyl)amino)-5-fluoro-N-(2-oxo-5-(2,4,6-trichlorophenyl)-2,3-dihydro1H-benzo[e][1,4]diazepin-3-yl)nicotinamide 1351764-35-6 C29H20Cl4FN5O2
2-((4-chlorobenzyl)(methyl)amino)-5-fluoro-N-(2-oxo-5-(2,4,6-trichlorophenyl)-2,3-dihydro1H-benzo[e][1,4]diazepin-3-yl)nicotinamide
—— 4-((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-1-(prop-1-en-2-yl)-3a-(pyridin-3-ylmethylcarbamoyl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysen-9-yl)benzoic acid 1351277-71-8 C43H56N2O3
4-((1R,3aS,5aR,5bR,7aR,11aS,11bR,13aR,13bR)-5a,5b,8,8,11a-pentamethyl-1-(prop-1-en-2-yl)-3a-(pyridin-3-ylmethylcarbamoyl)-2,3,3a,4,5,5a,5b,6,7,7a,8,11,11a,11b,12,13,13a,13b-octadecahydro-1H-cyclopenta[a]chrysen-9-yl)benzoic acid
—— 5-[(2-chloropyridin-4-yl)thio]-4-(2-fluoropyridin-3-yl)thiophene-2-carbaldehyde 1138034-36-2 C15H8ClFN2OS2
5-[(2-chloropyridin-4-yl)thio]-4-(2-fluoropyridin-3-yl)thiophene-2-carbaldehyde
—— (3'S,4'S)-di-O-p-methoxybenzoyl-4-methyl-(-)-cis-khellactone 1440881-72-0 C31H28O9
(3'S,4'S)-di-O-p-methoxybenzoyl-4-methyl-(-)-cis-khellactone
—— —— 1161075-22-4 C20H22ClN5
—— (S)-2-Phenyl-propionic acid (1R,2R)-2-fluoro-1-p-tolylsulfanylmethyl-pent-4-enyl ester 142793-65-5 C22H25FO2S
(S)-2-Phenyl-propionic acid (1R,2R)-2-fluoro-1-p-tolylsulfanylmethyl-pent-4-enyl ester
—— 1-[(2S,8S,8aR)-8,8a-dimethyl-2,3,5,6,7,8-hexahydro-1H-naphthalen-2-yl](214C)ethanone 123331-97-5 C14H22O
1-[(2S,8S,8aR)-8,8a-dimethyl-2,3,5,6,7,8-hexahydro-1H-naphthalen-2-yl](214C)ethanone
—— 4-tert-butyldimethylsilyloxy-3-methoxyphenyl 2-thiazolyl ketone 131610-18-9 C17H23NO3SSi
4-tert-butyldimethylsilyloxy-3-methoxyphenyl 2-thiazolyl ketone
—— 4.4-Diaethoxy-3-imino-buttersaeure-aethylester 10495-10-0 C10H19NO4
4.4-Diaethoxy-3-imino-buttersaeure-aethylester
—— (2'R,4'S,5'R,6'S)-4'-hydroxy-5'-methyl-2',6'-bis(3-nitrophenyl)dispiro[indene-2,1'-cyclohexane-3',2''-indene]-1,1'',3,3''-tetraone 1438626-00-6 C35H24N2O9
(2'R,4'S,5'R,6'S)-4'-hydroxy-5'-methyl-2',6'-bis(3-nitrophenyl)dispiro[indene-2,1'-cyclohexane-3',2''-indene]-1,1'',3,3''-tetraone
—— 1-(((carbomethoxymethyl)carbamido)ethyl)-o-carborane 196314-90-6 C8H22B10N2O3
1-(((carbomethoxymethyl)carbamido)ethyl)-o-carborane
—— 2-(3-(tert-butoxycarbonyl)oxazolidin-2-yl)acetic acid 1265900-25-1 C10H17NO5
2-(3-(tert-butoxycarbonyl)oxazolidin-2-yl)acetic acid
—— methyl 1-amino-6-methyl-4-phenyl-2-naphthoate 1434590-53-0 C19H17NO2
methyl 1-amino-6-methyl-4-phenyl-2-naphthoate
—— 6-(2,2-dihydroxyacetyl)-5-(trifluoromethyl)nicotinonitrile 1245522-99-9 C9H5F3N2O3
6-(2,2-dihydroxyacetyl)-5-(trifluoromethyl)nicotinonitrile
—— (3-chloro-2-morpholino-1-cyclohexen-1-yl)-(4-methyl-phenyl)-methanone 133147-54-3 C18H22ClNO2
(3-chloro-2-morpholino-1-cyclohexen-1-yl)-(4-methyl-phenyl)-methanone
—— 5-[[(4,5-dihydro-5,5-dimethyl-3-isoxazolyl)sulfonyl]methyl]-2,3-dimethyl-6-(trifluoromethyl)-4(3H)-pyrimidinone 1202471-27-9 C13H16F3N3O4S
5-[[(4,5-dihydro-5,5-dimethyl-3-isoxazolyl)sulfonyl]methyl]-2,3-dimethyl-6-(trifluoromethyl)-4(3H)-pyrimidinone
—— 2-((4-nitrophenyl)(pyrimidin-2-ylamino)methyl)-1H-indene-1,3(2H)-dione 1058667-75-6 C20H14N4O4
2-((4-nitrophenyl)(pyrimidin-2-ylamino)methyl)-1H-indene-1,3(2H)-dione
—— 7-<(4-methylphenyl)sulphonyl>-8-phenyl-bicyclo<4.2.0>octa-2,7-diene 115843-48-6 C21H20O2S
7-<(4-methylphenyl)sulphonyl>-8-phenyl-bicyclo<4.2.0>octa-2,7-diene
—— 2-(3-(4-(4-(3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureido)naphthalen-1-yloxy)pyridin-2-yl)ureido)-N-(2-(pyridin-4-yl)ethyl)acetamide 1229607-24-2 C40H41N9O4
2-(3-(4-(4-(3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureido)naphthalen-1-yloxy)pyridin-2-yl)ureido)-N-(2-(pyridin-4-yl)ethyl)acetamide
—— 3-(8-chloro-1-iodoimidazo[1,5-a]pyrazin-3-yl)propanoic acid 1083164-28-6 C9H7ClIN3O2
3-(8-chloro-1-iodoimidazo[1,5-a]pyrazin-3-yl)propanoic acid
—— 1-(2-fluoro-5-nitro-phenyl)-ethanol 150295-21-9 C8H8FNO3
1-(2-fluoro-5-nitro-phenyl)-ethanol
—— Diethyl 2-benzamido-2-(3-oxo-1,3-diphenylpropyl)propanedioate 1228562-55-7 C29H29NO6
Diethyl 2-benzamido-2-(3-oxo-1,3-diphenylpropyl)propanedioate
—— —— 1205535-58-5 C19H24O2
—— 6-(((1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl)amino)-2-(pyridin-4-ylamino)-5-(thiazol-2-yl)pyrimidine hydrochloride 1596365-32-0 C18H20N6O3S*ClH
6-(((1R,2S,3R,4R)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl)amino)-2-(pyridin-4-ylamino)-5-(thiazol-2-yl)pyrimidine hydrochloride
—— —— 1176049-36-7 C18H11BrF6N2O3
—— 1-(2-{[4-oxo-3-(3-pyridin-3-ylphenyl)-3,4-dihydroquinazolin-2-yl]thio}hexanoyl)piperidine-4-carboxamide trifluoroacetate 1181221-51-1 C2HF3O2*C31H33N5O3S
1-(2-{[4-oxo-3-(3-pyridin-3-ylphenyl)-3,4-dihydroquinazolin-2-yl]thio}hexanoyl)piperidine-4-carboxamide trifluoroacetate
—— —— 1176076-00-8 C22H18ClN3O3
—— (2S,3R)-1,4-bis(benzyloxy)-3-chloro-2-butanol 123125-16-6 C18H21ClO3
(2S,3R)-1,4-bis(benzyloxy)-3-chloro-2-butanol
—— diethyl 1-benzyl-5-methyl-2-oxoindolin-3-yl phosphate 1399215-26-9 C20H24NO5P
diethyl 1-benzyl-5-methyl-2-oxoindolin-3-yl phosphate
—— [MoH(η2-peroxo)((Ph2PCH2CH2P(Ph)C6H4-o)2(C6F5)Si-P,P,P,P,Si)] 1384897-46-4 C58H47F5MoO2P4Si
[MoH(η2-peroxo)((Ph2PCH2CH2P(Ph)C6H4-o)2(C6F5)Si-P,P,P,P,Si)]
—— N'-(1-(4-chlorophenyl)-2,2-difluoro-3-oxo-3-phenylpropyl)benzohydrazide 1259388-04-9 C22H17ClF2N2O2
N'-(1-(4-chlorophenyl)-2,2-difluoro-3-oxo-3-phenylpropyl)benzohydrazide
—— (8S)-1'-{[5-(benzyloxy)pyridine-2-yl]methyl}-2,3-dihydrospyro[furo[2,3-g][1,4]benzodioxine-8,3'-indol]-2'(1'H)-one 1222556-70-8 C30H24N2O5
(8S)-1'-{[5-(benzyloxy)pyridine-2-yl]methyl}-2,3-dihydrospyro[furo[2,3-g][1,4]benzodioxine-8,3'-indol]-2'(1'H)-one
—— benziloyl-imidophosphoric acid tri-[1]naphthyl ester 121426-26-4 C44H32NO5P
benziloyl-imidophosphoric acid tri-[1]naphthyl ester
—— 1,2-bis(7-[(Z)-ethoxycarbonylmethylene]-5,6-dihydro-5H-6-one[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl)ethane-1,2-diol 1370705-20-6 C18H18N8O8S2
1,2-bis(7-[(Z)-ethoxycarbonylmethylene]-5,6-dihydro-5H-6-one[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-3-yl)ethane-1,2-diol
—— 2-(deuteriomethyl)-1,3-dimethylindole 132205-56-2 C11H13N
2-(deuteriomethyl)-1,3-dimethylindole
—— 2-(((2,6-dichloroquinolin-3-yl)methylene)amino)phenol 1236132-84-5 C16H10Cl2N2O
2-(((2,6-dichloroquinolin-3-yl)methylene)amino)phenol
—— (R)-1-(1-(6-chloroquinolin-2-yl)-5,6-dimethyl-1H-benzo[d]imidazol-2-yl)-N-(tetrahydrofuran-3-yl)piperidine-4-carboxamide 1395033-76-7 C28H30ClN5O2
(R)-1-(1-(6-chloroquinolin-2-yl)-5,6-dimethyl-1H-benzo[d]imidazol-2-yl)-N-(tetrahydrofuran-3-yl)piperidine-4-carboxamide