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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-((R)-5-{[(S)-1-(3-fluoro-6-methoxy-[1,5]naphthyridin-4-yl)-pyrrolidin-3-ylamino]-methyl}-2-oxo-oxazolidin-3-yl)-4H-benzo[1,4]thiazin-3-one 1072825-81-0 C25H25FN6O4S
6-((R)-5-{[(S)-1-(3-fluoro-6-methoxy-[1,5]naphthyridin-4-yl)-pyrrolidin-3-ylamino]-methyl}-2-oxo-oxazolidin-3-yl)-4H-benzo[1,4]thiazin-3-one
—— (1R,2S,5S)-3-[(2S)-2-[[(2S)-1-(4,4-dimethyl-2,6-dioxopiperidin-1-yl)-3,3-dimethylbutan-2-yl]carbamoylamino]-3,3-dimethylbutanoyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxylic acid 1063968-44-4 C28H46N4O6
(1R,2S,5S)-3-[(2S)-2-[[(2S)-1-(4,4-dimethyl-2,6-dioxopiperidin-1-yl)-3,3-dimethylbutan-2-yl]carbamoylamino]-3,3-dimethylbutanoyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxylic acid
—— N-(3-chlorobenzyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)pentyl]-2H-indazole-6-carboxamide 1002110-36-2 C23H25ClN4O3
N-(3-chlorobenzyl)-2-[2-(2-oxo-1,3-oxazolidin-3-yl)pentyl]-2H-indazole-6-carboxamide
—— 6-amino-2-butoxy-9-{6-[2-(4-methylpiperazin-1-yl)ethoxy]pyridin-3-ylmethyl}-7,9-dihydropurin-8-one 1059071-72-5 C22H32N8O3
6-amino-2-butoxy-9-{6-[2-(4-methylpiperazin-1-yl)ethoxy]pyridin-3-ylmethyl}-7,9-dihydropurin-8-one
—— N-((1S,5S)-1-ethyl-6-hydroxy-5-((4-hydroxymethylphenylsulfonyl)(isopropyl)amino)hexyl)-β-phenyl-L-phenylalaninamide 1138084-55-5 C33H45N3O5S
N-((1S,5S)-1-ethyl-6-hydroxy-5-((4-hydroxymethylphenylsulfonyl)(isopropyl)amino)hexyl)-β-phenyl-L-phenylalaninamide
—— 2-(4-fluorophenyl)-5-(4-methoxy-2-methyl-5-(1-(3-methyl-1,2,4-oxadiazol-5-yl)cyclopropylcarbamoyl)phenyl)-N-methylbenzofuran-3-carboxamide 1217338-12-9 C31H27FN4O5
2-(4-fluorophenyl)-5-(4-methoxy-2-methyl-5-(1-(3-methyl-1,2,4-oxadiazol-5-yl)cyclopropylcarbamoyl)phenyl)-N-methylbenzofuran-3-carboxamide
—— N-(2-acetylaminocyclohexyl)-3,5-difluoro-4-(2-propynyloxy)benzamide 1078725-99-1 C18H20F2N2O3
N-(2-acetylaminocyclohexyl)-3,5-difluoro-4-(2-propynyloxy)benzamide
—— tert-butyl 2-{[2-(5-{2-[5-(4-acetylpiperazin-1-yl)pyridin-2-yl]ethyl}thiophen-2-yl)ethyl]carbamoyl}-hydrazinecarboxylate 1197295-40-1 C25H36N6O4S
tert-butyl 2-{[2-(5-{2-[5-(4-acetylpiperazin-1-yl)pyridin-2-yl]ethyl}thiophen-2-yl)ethyl]carbamoyl}-hydrazinecarboxylate
—— 4-{3-[1-(3-chloro-benzyl)-5,6-difluoro-1H-benzoimidazol-2-yl]-pyridin-2-yloxymethyl}-benzoic acid methyl ester 1281980-40-2 C28H20ClF2N3O3
4-{3-[1-(3-chloro-benzyl)-5,6-difluoro-1H-benzoimidazol-2-yl]-pyridin-2-yloxymethyl}-benzoic acid methyl ester
—— (S)-N-{2-[di(5-indanyl)-phosphonomethylamino]-3-(4-biphenylyl)-propionyl}-3-aminopropionic acid 147862-15-5 C37H39N2O6P
(S)-N-{2-[di(5-indanyl)-phosphonomethylamino]-3-(4-biphenylyl)-propionyl}-3-aminopropionic acid
—— 1-((3-(2-chlorophenyl)-5-methylquinoxalin-2-yl)methyl)-3-(1H-pyrazol-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine 1064136-10-2 C24H18ClN9
1-((3-(2-chlorophenyl)-5-methylquinoxalin-2-yl)methyl)-3-(1H-pyrazol-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
—— 1-naphthalen-1-yl-3-[5-(3-thioureido-phenoxy)-pentyl]-urea 1092450-02-6 C23H26N4O2S
1-naphthalen-1-yl-3-[5-(3-thioureido-phenoxy)-pentyl]-urea
—— 4-(4-cyanophenyl)-N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2-methyl-1H-pyrrole-3-carboxamide 1089145-24-3 C28H28FN5O2
4-(4-cyanophenyl)-N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fluoro-2-oxo-1,2-dihydro-3H-indol-3-ylidene)methyl]-2-methyl-1H-pyrrole-3-carboxamide
—— 7-chloro-1-prop-2-enyl-9H-carbazol-2-ol 1094084-39-5 C15H12ClNO
7-chloro-1-prop-2-enyl-9H-carbazol-2-ol
—— β-D-2',3'-dideoxy-4'-selenocytidine 1100358-60-8 C9H13N3O2Se
β-D-2',3'-dideoxy-4'-selenocytidine
—— 7-bromo-2-(5-chloro-2-methoxyphenylamino)-4,5,6,7-tetrahydrocyclohepta[d]thiazol-8-one 1067637-99-3 C15H14BrClN2O2S
7-bromo-2-(5-chloro-2-methoxyphenylamino)-4,5,6,7-tetrahydrocyclohepta[d]thiazol-8-one
—— 4-(2-{3,5-dichloro-6-[(3-isopropylphenoxy)methyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoic acid 1091595-75-3 C24H23Cl2NO4
4-(2-{3,5-dichloro-6-[(3-isopropylphenoxy)methyl]-2-oxopyridin-1(2H)-yl}ethyl)benzoic acid
—— 2-(benzofuran-5-yl)-N-(5-methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-4-amine 1093108-92-9 C21H23N7O
2-(benzofuran-5-yl)-N-(5-methyl-1H-pyrazol-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-4-amine
—— 2-(3,4-dichloro-phenyl)-4-((R)-4-methanesulfonyl-3-methyl-piperazin-1-yl)-2-methyl-N-quinoxalin-6-ylmethylbutyramide 1093079-22-1 C26H31Cl2N5O3S
2-(3,4-dichloro-phenyl)-4-((R)-4-methanesulfonyl-3-methyl-piperazin-1-yl)-2-methyl-N-quinoxalin-6-ylmethylbutyramide
—— N-benzyl-6-phenyl-N'-((2-(trimethylsilyl)ethoxy)methyl)-3,3'-biindoline-2,2'-dione 1078598-98-7 C35H36N2O3Si
N-benzyl-6-phenyl-N'-((2-(trimethylsilyl)ethoxy)methyl)-3,3'-biindoline-2,2'-dione
—— N-(6-fluoro-4-oxo-2-pyrrolidin-1-yl-4H-quinazolin-3-yl)-2-(3-fluoro-4-trifluoromethylphenyl)acetamide 1086683-86-4 C21H17F5N4O2
N-(6-fluoro-4-oxo-2-pyrrolidin-1-yl-4H-quinazolin-3-yl)-2-(3-fluoro-4-trifluoromethylphenyl)acetamide
—— 4-amino-2-(5-chloro-furan-2-yl)thieno[2,3-d]pyrimidine-6-carbaldehyde 1221434-83-8 C11H6ClN3O2S
4-amino-2-(5-chloro-furan-2-yl)thieno[2,3-d]pyrimidine-6-carbaldehyde
—— N-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)cyclohexanecarboxamide 1041395-75-8 C31H39N5O3
N-(3-(2-oxo-4-phenyl-5-(piperazine-1-carbonyl)-3-o-tolyl-2,3-dihydro-1H-imidazol-1-yl)propyl)cyclohexanecarboxamide
—— 4,6-dihydroxy-2-[(5-methoxy-2-phenyl-1H-indol-3-yl)methyl]-1-benzofuran-3(2H)-one 1200532-91-7 C24H19NO5
4,6-dihydroxy-2-[(5-methoxy-2-phenyl-1H-indol-3-yl)methyl]-1-benzofuran-3(2H)-one
—— 1-{3-[2-aminopyridin-4-yl]-[2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid isobutylamide 1071133-65-7 C23H28N6O
1-{3-[2-aminopyridin-4-yl]-[2,6]naphthyridin-1-yl}piperidine-4-carboxylic acid isobutylamide
—— N-cyclopentyl-1-(1-(2-ethylbutyl)-5,6-dimethyl-1H-benzo[d]imidazol-2-yl)piperidine-4-carboxamide 1268710-34-4 C26H40N4O
N-cyclopentyl-1-(1-(2-ethylbutyl)-5,6-dimethyl-1H-benzo[d]imidazol-2-yl)piperidine-4-carboxamide
—— 1-(6-methyl-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-1H-imidazole-2-carboxylic acid ethyl ester 1197846-14-2 C22H22N4O2
1-(6-methyl-2-p-tolyl-imidazo[1,2-a]pyridin-3-ylmethyl)-1H-imidazole-2-carboxylic acid ethyl ester
—— [5-bromo-4-(1-piperazin-1-yl-[2,6]naphthyridin-3-yl)pyridin-2-yl]-cyclohexylamine 1071136-43-0 C23H27BrN6
[5-bromo-4-(1-piperazin-1-yl-[2,6]naphthyridin-3-yl)pyridin-2-yl]-cyclohexylamine
—— 1-cyclohexyl-3-[2-(2-oxo-1H-cyclohepta[b]pyrrol-3-yl)-3H-benzimidazol-5-yl]urea 1253838-14-0 C23H23N5O2
1-cyclohexyl-3-[2-(2-oxo-1H-cyclohepta[b]pyrrol-3-yl)-3H-benzimidazol-5-yl]urea
—— 2-(3-methylphenyl)-N-(4-{3-[4-(pyridin-4-yl)piperazin-1-yl]quinoxalin-6-yl}phenyl)acetamide 1271840-36-8 C32H30N6O
2-(3-methylphenyl)-N-(4-{3-[4-(pyridin-4-yl)piperazin-1-yl]quinoxalin-6-yl}phenyl)acetamide
—— N-[2-(6,6-dimethyl-1,4,5,7-tetrahydroindazol-3-yl)-1H-indol-6-yl]-2,3-dihydroxy-N-methylpropanamide 1309784-75-5 C21H26N4O3
N-[2-(6,6-dimethyl-1,4,5,7-tetrahydroindazol-3-yl)-1H-indol-6-yl]-2,3-dihydroxy-N-methylpropanamide
—— N-(Prop-2-yn-1-yl)piperidin-4-amine 1183805-43-7 C8H14N2
N-(Prop-2-yn-1-yl)piperidin-4-amine
—— 5-[4-(7-hydroxy-6-methyl-indan-4-ylmethyl)-3,5-dimethyl-pyrazol-1-ylmethyl]-1H-pyrazol-3-ol 1092552-21-0 C20H24N4O2
5-[4-(7-hydroxy-6-methyl-indan-4-ylmethyl)-3,5-dimethyl-pyrazol-1-ylmethyl]-1H-pyrazol-3-ol
—— N-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl]-N'-(1H-indazol-5-yl)pyrimidine-4,6-diamine 1093165-42-4 C23H22FN7
N-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethyl]-N'-(1H-indazol-5-yl)pyrimidine-4,6-diamine
—— N-(4-chloro-benzyl)-2-(3,4-dichloro-phenyl)-4-(4-methanesulfonyl-piperazin-1-yl)-2-methylbutyramide 1093078-13-7 C23H28Cl3N3O3S
N-(4-chloro-benzyl)-2-(3,4-dichloro-phenyl)-4-(4-methanesulfonyl-piperazin-1-yl)-2-methylbutyramide
—— (S)-N-(1-cyclohexylethyl)-6-(2-(pyridin-3-yl)pyrimidin-4-yloxy)benzo[d]thiazol-2-amine 1086108-74-8 C24H25N5OS
(S)-N-(1-cyclohexylethyl)-6-(2-(pyridin-3-yl)pyrimidin-4-yloxy)benzo[d]thiazol-2-amine
—— N-(3-{2-amino-4-[4-(difluoromethoxy)phenyl]-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl}phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide 1065165-79-8 C28H21F5N6O3
N-(3-{2-amino-4-[4-(difluoromethoxy)phenyl]-1-methyl-5-oxo-4,5-dihydro-1H-imidazol-4-yl}phenyl)-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
—— N-(1,3,4-thiadiazol-2-yl)-2-(1-(3-(trifluoromethyl)phenylsulfonyl)piperidin-4-ylideneaminooxy)acetamide 1092463-32-5 C16H16F3N5O4S2
N-(1,3,4-thiadiazol-2-yl)-2-(1-(3-(trifluoromethyl)phenylsulfonyl)piperidin-4-ylideneaminooxy)acetamide
—— 2-methoxy-N-[2-(1-methyl-6-oxo-1,6-dihydro-4,4'-bipyrimidinyl-2-yl)-ethyl]-4-trifluoromethyl-benzamide 1083007-57-1 C20H18F3N5O3
2-methoxy-N-[2-(1-methyl-6-oxo-1,6-dihydro-4,4'-bipyrimidinyl-2-yl)-ethyl]-4-trifluoromethyl-benzamide
—— N-(2-(1H-[1,2,3]triazolo[4,5-b]pyridin-1-yl)-4-chloro-5-fluorophenyl)-4-tert-butylbenzenesulfonamide 1094756-75-8 C21H19ClFN5O2S
N-(2-(1H-[1,2,3]triazolo[4,5-b]pyridin-1-yl)-4-chloro-5-fluorophenyl)-4-tert-butylbenzenesulfonamide
—— 2-[(3-fluoropyridin-2-yl)amino]-5-phenylthiophene-3-carboxamide 1093871-77-2 C16H12FN3OS
2-[(3-fluoropyridin-2-yl)amino]-5-phenylthiophene-3-carboxamide
—— N-(2,4-difluorophenyl)-5-[8-(1-methyl-1H-imidazol-5-yl)-1,5-naphthyridin-2-yl]-3-pyridinesulfonamide 1092565-63-3 C23H16F2N6O2S
N-(2,4-difluorophenyl)-5-[8-(1-methyl-1H-imidazol-5-yl)-1,5-naphthyridin-2-yl]-3-pyridinesulfonamide
—— 5-(1',7',7'-trimethylbicyclo[2.2.1]hept-2'-yl)resorcinol 1072783-06-2 C16H22O2
5-(1',7',7'-trimethylbicyclo[2.2.1]hept-2'-yl)resorcinol
—— (3-[6-(3-diethylaminomethyl-phenyl)-pyrimidin-4-ylamino]-phenyl)-methanesulfonamide 1073485-06-9 C22H27N5O2S
(3-[6-(3-diethylaminomethyl-phenyl)-pyrimidin-4-ylamino]-phenyl)-methanesulfonamide
—— 3-(2,3-dichlorophenyl)-1-ethylpyrrolidin-3-ol 1092572-26-3 C12H15Cl2NO
3-(2,3-dichlorophenyl)-1-ethylpyrrolidin-3-ol
—— 4,6-dihydroxy-2-[(1-methyl-5-nitro-1H-indol-3-yl)methylene]-1-benzofuran-3(2H)-one 1200532-05-3 C18H12N2O6
4,6-dihydroxy-2-[(1-methyl-5-nitro-1H-indol-3-yl)methylene]-1-benzofuran-3(2H)-one
—— 3-((1H-1,2,4-triazol-5-yl)methyl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridine 1197849-02-7 C16H12ClN5
3-((1H-1,2,4-triazol-5-yl)methyl)-2-(4-chlorophenyl)imidazo[1,2-a]pyridine
—— N-(11-Octylamino-10-hydroxyundecyl)-succinimide 170637-01-1 C23H44N2O3
N-(11-Octylamino-10-hydroxyundecyl)-succinimide
—— 1,4-Diaza-1-methyl-5-oxo-cycloundecen-(6-cis) 16620-88-5 C10H18N2O
1,4-Diaza-1-methyl-5-oxo-cycloundecen-(6-cis)
—— rac-N-{3-[1-(4-fluoro-benzyl)-4-hydroxy-5-isopropyl-2-oxo-1,2,5,6-tetrahydro-pyridin-3-yl]-1,1-dioxo-1,4-dihydro-1λ6-thieno[2,3-e][1,2,4]thiadiazin-7-ylmethyl}-methanesulfonamide 1198469-11-2 C22H25FN4O6S3
rac-N-{3-[1-(4-fluoro-benzyl)-4-hydroxy-5-isopropyl-2-oxo-1,2,5,6-tetrahydro-pyridin-3-yl]-1,1-dioxo-1,4-dihydro-1λ6-thieno[2,3-e][1,2,4]thiadiazin-7-ylmethyl}-methanesulfonamide