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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(2-phenyl-thiazolidin-3-yl)-benzoic acid methyl ester 107919-56-2 C17H17NO2S
3-(2-phenyl-thiazolidin-3-yl)-benzoic acid methyl ester
—— <i>N</i>,<i>N</i>-dimethyl-<i>N</i>'-[1,2,3,4]thiatriazol-5-yl-<i>p</i>-phenylenediamine 119247-77-7 C9H11N5S
<i>N</i>,<i>N</i>-dimethyl-<i>N</i>'-[1,2,3,4]thiatriazol-5-yl-<i>p</i>-phenylenediamine
—— N-[3-((R)-Pyrrolidin-2-ylmethoxy)-4-methoxyphenyl]-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-2'-methylbiphenyl-4-carboxamide hydrochloride 174346-56-6 C29H30N4O4*ClH
N-[3-((R)-Pyrrolidin-2-ylmethoxy)-4-methoxyphenyl]-4'-(5-methyl-1,2,4-oxadiazol-3-yl)-2'-methylbiphenyl-4-carboxamide hydrochloride
—— 2,2-difluoro-8-(1-hydroxyethyl)-4-[(1-methyl-1H-benzimidazol-2-yl)methyl]-2H-1,4-benzoxazin-3(4H)-one 1263411-22-8 C19H17F2N3O3
2,2-difluoro-8-(1-hydroxyethyl)-4-[(1-methyl-1H-benzimidazol-2-yl)methyl]-2H-1,4-benzoxazin-3(4H)-one
—— 2,2-difluoro-4-[(6-fluoro-3-methyl-4-oxo-3,4-dihydro-2-quinazolinyl)methyl]-8-[(1S)-1-hydroxyethyl]-2H-1,4-benzoxazin-3(4H)-one 1263412-19-6 C20H16F3N3O4
2,2-difluoro-4-[(6-fluoro-3-methyl-4-oxo-3,4-dihydro-2-quinazolinyl)methyl]-8-[(1S)-1-hydroxyethyl]-2H-1,4-benzoxazin-3(4H)-one
—— Methyl 6-amino-3-cyclopropyl-4-oxoquinazoline-7-carboxylate 1039454-97-1 C13H13N3O3
Methyl 6-amino-3-cyclopropyl-4-oxoquinazoline-7-carboxylate
—— 1,4-bis[5-cyano-2-(cyanomethyl)-4-oxo-6-(methylthio)-4,5-dihydro-3H-pyrrolo[2,3-d]pyrimidin-3-yl]butane 1393649-89-2 C24H20N10O2S2
1,4-bis[5-cyano-2-(cyanomethyl)-4-oxo-6-(methylthio)-4,5-dihydro-3H-pyrrolo[2,3-d]pyrimidin-3-yl]butane
—— 8-(2-bromo-5-methylphenyl)-6-phenyl-2H-pyrimido[2,1-c][1,2,4]triazin-3-one 1202877-82-4 C19H15BrN4O
8-(2-bromo-5-methylphenyl)-6-phenyl-2H-pyrimido[2,1-c][1,2,4]triazin-3-one
—— 1-(5-methoxy-indol-3-yl)carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan] 1347066-23-2 C23H27N3O3
1-(5-methoxy-indol-3-yl)carbonyl-5'-aminomethyl-spiro[piperidine-4,3'-(2H)-benzo[b]furan]
—— 4'-methyl-5-(5-trifluoromethyl-[1,2,4]triazol-1-yl)-biphenyl-3-carboxylic acid (1-pyrazin-2-yl-ethyl)-amide 1161870-14-9 C23H19F3N6O
4'-methyl-5-(5-trifluoromethyl-[1,2,4]triazol-1-yl)-biphenyl-3-carboxylic acid (1-pyrazin-2-yl-ethyl)-amide
—— (6S)-6-((R)-2,3-dihydroxypropyl)-6-(4-fluorophenyl)-3-((1S)-1-(4-methoxyphenyl)ethyl)-1,3-oxazinan-2-one 1114084-61-5 C22H26FNO5
(6S)-6-((R)-2,3-dihydroxypropyl)-6-(4-fluorophenyl)-3-((1S)-1-(4-methoxyphenyl)ethyl)-1,3-oxazinan-2-one
—— 6-(pyridin-2-yl)-2-[(1,2,5,6-tetrahydropyridin-1-yl)carbonyl]imidazo[1,2-a]pyridine 1187162-67-9 C18H16N4O
6-(pyridin-2-yl)-2-[(1,2,5,6-tetrahydropyridin-1-yl)carbonyl]imidazo[1,2-a]pyridine
—— 7-[2-(2-thienyl)vinyl]-6H-pyrrolo[2,3-e][1,2,4]triazolo[1,5-a]pyrimidine 1101866-52-7 C13H9N5S
7-[2-(2-thienyl)vinyl]-6H-pyrrolo[2,3-e][1,2,4]triazolo[1,5-a]pyrimidine
—— 7,7-Dimethyl-6,8-dioxa-2-azaspiro[3.5]nonane 156720-75-1 C8H15NO2
7,7-Dimethyl-6,8-dioxa-2-azaspiro[3.5]nonane
—— (R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-chloro-phenyl)-ethyl]-3-(4-fluoro-phenyl)-2-hydroxy-propionamide 1300007-33-3 C24H24ClFN4O3
(R)-N-[(S)-1-[(6-amino-pyridin-3-ylmethyl)-carbamoyl]-2-(4-chloro-phenyl)-ethyl]-3-(4-fluoro-phenyl)-2-hydroxy-propionamide
—— 1-[3-(3-methylbenzyl)[1,2,4]thiadiazol-5-yl]piperazine 1029718-77-1 C14H18N4S
1-[3-(3-methylbenzyl)[1,2,4]thiadiazol-5-yl]piperazine
—— 5,7-dichloro-4-[(6-ethoxycarbonylmethyl-pyridin-3-ylcarbamoyl)-methoxy]-naphthalene-2-carboxylic methyl ester 1257342-98-5 C23H20Cl2N2O6
5,7-dichloro-4-[(6-ethoxycarbonylmethyl-pyridin-3-ylcarbamoyl)-methoxy]-naphthalene-2-carboxylic methyl ester
—— 2-[3-(isopropylamino)propylamino]-4-{3-methyl-4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-1-yl}benzamide 1260532-52-2 C30H32N6O
2-[3-(isopropylamino)propylamino]-4-{3-methyl-4-(quinolin-3-yl)-1H-pyrrolo[2,3-b]pyridin-1-yl}benzamide
—— (R)-methyl 5-(2-(5-fluoro-2-(2-methoxyethoxy)phenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate 1260846-96-5 C21H23FN4O4
(R)-methyl 5-(2-(5-fluoro-2-(2-methoxyethoxy)phenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxylate
—— (R)-N-tert-butyl-5-(2-(5-fluoropyridin-3-yl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1260841-24-4 C20H23FN6O
(R)-N-tert-butyl-5-(2-(5-fluoropyridin-3-yl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 3-isopropyl-4-(6-methoxypyridin-3-yl)-1H-pyrazolo[3,4-b]pyridine 1260536-78-4 C15H16N4O
3-isopropyl-4-(6-methoxypyridin-3-yl)-1H-pyrazolo[3,4-b]pyridine
—— (1S,2S)-2-(4-(5-((5-chloropyridin-2-yl)thio)-1-methyl-1H-imidazol-4-yl)phenyl)cyclopropanecarbontrile 1242441-59-3 C19H15ClN4S
(1S,2S)-2-(4-(5-((5-chloropyridin-2-yl)thio)-1-methyl-1H-imidazol-4-yl)phenyl)cyclopropanecarbontrile
—— 1-[(3,4-difluorophenyl)methyl]-N-[3-[4-(4-methyl-1,4-diazepan-1-yl)quinazolin-6-yl]prop-2-ynyl]-2-oxopyridine-3-carboxamide 1345441-23-7 C30H28F2N6O2
1-[(3,4-difluorophenyl)methyl]-N-[3-[4-(4-methyl-1,4-diazepan-1-yl)quinazolin-6-yl]prop-2-ynyl]-2-oxopyridine-3-carboxamide
—— 6-bromo-4-[[(3S)-1-methylpyrrolidin-3-yl]methoxy]quinoline 1345446-79-8 C15H17BrN2O
6-bromo-4-[[(3S)-1-methylpyrrolidin-3-yl]methoxy]quinoline
—— 2,5-dimethoxy-3-(trimethylstannyl)pyridine 1093951-74-6 C10H17NO2Sn
2,5-dimethoxy-3-(trimethylstannyl)pyridine
—— 8-(4-methanesulfonylmethyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine 1257704-73-6 C14H14N4O2S
8-(4-methanesulfonylmethyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamine
—— 2-(3-(3-(6-methoxypyridin-3-yl)pyrazin-2-yl)azetidin-1-yl)quinoline 2,2,2-trifluoroacetate 1349864-88-5 C2HF3O2*C22H19N5O
2-(3-(3-(6-methoxypyridin-3-yl)pyrazin-2-yl)azetidin-1-yl)quinoline 2,2,2-trifluoroacetate
—— N-(5-cyclopentyl-2,7-dioxo-1,2,4,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)acetamide 1257440-47-3 C13H16N4O3
N-(5-cyclopentyl-2,7-dioxo-1,2,4,7-tetrahydropyrazolo[1,5-a]pyrimidin-3-yl)acetamide
—— N-(3-((3-bromopyridin-2-yl)oxy)cyclobutyl)-4-methylbenzenesulfonamide 1349185-40-5 C16H17BrN2O3S
N-(3-((3-bromopyridin-2-yl)oxy)cyclobutyl)-4-methylbenzenesulfonamide
—— methyl 2-(5-([1,2,4]triazolo[1,5-a]pyridin-8-yloxy)-6-(3-(1-acetylpyridin-4-yl)-1,2,4-thiadiazol-5-ylamino)pyridin-3-ylthio)acetate 1065608-49-2 C23H24N8O4S2
methyl 2-(5-([1,2,4]triazolo[1,5-a]pyridin-8-yloxy)-6-(3-(1-acetylpyridin-4-yl)-1,2,4-thiadiazol-5-ylamino)pyridin-3-ylthio)acetate
—— 1-acetyl-4-[2-cyclohexyl-2-(2-methylamino-propionylamino)-acetyl]-octahydro-pyrrolo[3,2-b]pyrrole-3-carboxylic acid (1,2,3,4-tetrahydro-naphthalen-1-yl)-amide 1257312-81-4 C31H45N5O4
1-acetyl-4-[2-cyclohexyl-2-(2-methylamino-propionylamino)-acetyl]-octahydro-pyrrolo[3,2-b]pyrrole-3-carboxylic acid (1,2,3,4-tetrahydro-naphthalen-1-yl)-amide
—— 3-(3-furan-3-yl)-2-methoxy-6-(pyrid-3-ylsulphonylmethyl)benzoic acid 1286177-35-2 C18H15NO6S
3-(3-furan-3-yl)-2-methoxy-6-(pyrid-3-ylsulphonylmethyl)benzoic acid
—— N-[4-methyl-5-[3-(2-pyridin-3-ylethyl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-yl]acetamide 1292299-91-2 C15H15N5O2S
N-[4-methyl-5-[3-(2-pyridin-3-ylethyl)-1,2,4-oxadiazol-5-yl]-1,3-thiazol-2-yl]acetamide
—— 2,4,6-Trimethylphenylcarbamoylchlorid 121513-36-8 C10H12ClNO
2,4,6-Trimethylphenylcarbamoylchlorid
—— methyl 3-[6-(methanesulfonamido)-3,4-dihydro-1H-quinazolin-2-ylidene]-2-oxo-1H-indole-5-carboxylate 1092932-22-3 C19H18N4O5S
methyl 3-[6-(methanesulfonamido)-3,4-dihydro-1H-quinazolin-2-ylidene]-2-oxo-1H-indole-5-carboxylate
—— N-(4-chlorobenzyl)-4-(6-fluoro-2-oxo-1,2-dihydro-1'H-spiro[3,1-benzoxazine-4,4'-piperidin]-1'-yl)-2-(4-fluorophenyl)butanamide 1036924-01-2 C29H28ClF2N3O3
N-(4-chlorobenzyl)-4-(6-fluoro-2-oxo-1,2-dihydro-1'H-spiro[3,1-benzoxazine-4,4'-piperidin]-1'-yl)-2-(4-fluorophenyl)butanamide
—— d13-(S)-N-[3-(3,5-difluoro-4-thiomorpholin-4-yl-phenyl)-2-oxo-oxazolidin-5-ylmethyl]-acetamide 1032183-73-5 C16H19F2N3O3S
d13-(S)-N-[3-(3,5-difluoro-4-thiomorpholin-4-yl-phenyl)-2-oxo-oxazolidin-5-ylmethyl]-acetamide
—— N-(4-piperazin-1-ylpyridin-3-yl)-6-thiophen-2-ylpyridine-2-carboxamide 1107624-05-4 C19H19N5OS
N-(4-piperazin-1-ylpyridin-3-yl)-6-thiophen-2-ylpyridine-2-carboxamide
—— 2-[1-(4-tert-Butyl-phenyl)-3-(3,4-dichloro-phenyl)-1H-pyrazol-4-yl]-acetamide 1026671-75-9 C21H21Cl2N3O
2-[1-(4-tert-Butyl-phenyl)-3-(3,4-dichloro-phenyl)-1H-pyrazol-4-yl]-acetamide
—— 4-(methoxycarbonyl)-5-(4-chlorophenyl)-2-oxazoline 141366-83-8 C11H10ClNO3
4-(methoxycarbonyl)-5-(4-chlorophenyl)-2-oxazoline
—— N-ethyl-N-[2-(5-{[3-(pyrrolidin-1-ylcarbonyl)piperidino]methyl}-1,3-thiazol-2-yl)-1H-indol-7-yl]thiophene-2-sulfonamide trifluoroacetate 1020356-00-6 C2HF3O2*C28H33N5O3S3
N-ethyl-N-[2-(5-{[3-(pyrrolidin-1-ylcarbonyl)piperidino]methyl}-1,3-thiazol-2-yl)-1H-indol-7-yl]thiophene-2-sulfonamide trifluoroacetate
—— (S)-5-fluoro-1-(pyrrolidin-3-yl)-1H-benzo[d]imidazol-2(3H)-one 1257521-87-1 C11H12FN3O
(S)-5-fluoro-1-(pyrrolidin-3-yl)-1H-benzo[d]imidazol-2(3H)-one
—— (2S)-2-amino-N-[(3S)-1-[(2S)-1-amino-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl]propanamide 1246295-21-5 C10H18N4O3
(2S)-2-amino-N-[(3S)-1-[(2S)-1-amino-1-oxopropan-2-yl]-2-oxopyrrolidin-3-yl]propanamide
—— 1-cyclopropyl-N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-6-[6-(1-piperazinyl)-3-pyridinyl]-1H-indole-4-carboxamide 1346573-11-2 C30H34N6O2
1-cyclopropyl-N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-6-[6-(1-piperazinyl)-3-pyridinyl]-1H-indole-4-carboxamide
—— 7-bromo-N-(1-methylpiperidin-4-yl)quinoxalin-2-amine 1345445-03-5 C14H17BrN4
7-bromo-N-(1-methylpiperidin-4-yl)quinoxalin-2-amine
—— methyl (2S)-2-(4-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy}phenoxy)propanoate 116661-27-9 C16H13ClF3NO4
methyl (2S)-2-(4-{[3-chloro-5-(trifluoromethyl)pyridin-2-yl]oxy}phenoxy)propanoate
—— ethyl 6-[(4-methylphenyl)sulfonylhydrazinylidene]-2,3,4,5-tetrahydro-1H-indene-3a-carboxylate 144343-84-0 C19H24N2O4S
ethyl 6-[(4-methylphenyl)sulfonylhydrazinylidene]-2,3,4,5-tetrahydro-1H-indene-3a-carboxylate
—— N,N'-bis((S)-1-ethoxycarbonylethyl)-2-((R)-(6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl)amino)-3-oxo-3-(4-butoxycarbonylpiperazin-1-yl)propylphosphonic acid diamide 1159501-16-2 C38H57N8O10P
N,N'-bis((S)-1-ethoxycarbonylethyl)-2-((R)-(6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl)amino)-3-oxo-3-(4-butoxycarbonylpiperazin-1-yl)propylphosphonic acid diamide
—— [4-({[tert-butyl(dimethyl)silyl]oxy}methyl)-2-fluoro-5-methoxyphenyl]amine 1346763-82-3 C14H24FNO2Si
[4-({[tert-butyl(dimethyl)silyl]oxy}methyl)-2-fluoro-5-methoxyphenyl]amine
—— 3-methyl-[(3',4'-dichloro)-2-phenyl]morpholine hydrochloride 1350768-44-3 C11H13Cl2NO*ClH
3-methyl-[(3',4'-dichloro)-2-phenyl]morpholine hydrochloride