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中文名称 英文名称 CAS号 化学式 结构式图片
—— (S)-2-({2-[3-(3-hydroxy-phenyl)propylamino]-4,6-dimethyl-pyrimidine-5-carbonyl}amino)-3-[(thiazole-4-carbonyl)amino]propionic acid 1400704-27-9 C23H26N6O5S
(S)-2-({2-[3-(3-hydroxy-phenyl)propylamino]-4,6-dimethyl-pyrimidine-5-carbonyl}amino)-3-[(thiazole-4-carbonyl)amino]propionic acid
—— N-[3-[(2,2-dimethylpropylamino)methyl]-4-methyl-5-(trifluoromethyl)phenyl]-3-[4-(5-methoxypyridin-3-yl)triazol-1-yl]-4-methylbenzamide 1096693-48-9 C30H33F3N6O2
N-[3-[(2,2-dimethylpropylamino)methyl]-4-methyl-5-(trifluoromethyl)phenyl]-3-[4-(5-methoxypyridin-3-yl)triazol-1-yl]-4-methylbenzamide
—— 3-(2-fluoro-4-iodo-phenylamino)-1-methyl-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid ((1R)-2,3-dihydroxy-propoxy)-amide 1030381-09-9 C18H18FIN4O4
3-(2-fluoro-4-iodo-phenylamino)-1-methyl-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid ((1R)-2,3-dihydroxy-propoxy)-amide
—— rac-1-{1-[6-chloro-3-(3-chloro-benzyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-piperidine-3-carbonyl}-piperidine-4-carboxylic acid amide 1015685-78-5 C27H30Cl2N4O3
rac-1-{1-[6-chloro-3-(3-chloro-benzyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-piperidine-3-carbonyl}-piperidine-4-carboxylic acid amide
—— 2-(2-methylammopyrimidin-5-yl)-morpholino-6-(4-N-methylsulfonyl(piperazin-1-yl)methyl)thieno[2,3-d]pyrimidine 1032756-02-7 C21H28N8O3S2
2-(2-methylammopyrimidin-5-yl)-morpholino-6-(4-N-methylsulfonyl(piperazin-1-yl)methyl)thieno[2,3-d]pyrimidine
—— (S)-3-(4-(4-chlorophenoxy)phenyl)-5,5-dimethyl-4-phenyloxazolidin-2-one 1035486-66-8 C23H20ClNO3
(S)-3-(4-(4-chlorophenoxy)phenyl)-5,5-dimethyl-4-phenyloxazolidin-2-one
—— 7-chloro-6-(2-chloropyridin-4-yl)-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinoline 1021911-34-1 C29H29Cl2N3O
7-chloro-6-(2-chloropyridin-4-yl)-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinoline
—— Drimenol 192724-27-9 C15H26O
Drimenol
—— (2S)-2-amino-1-{3-[(4-chlorophenyl)amino]-2-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}propan-1-one 1261114-32-2 C21H21ClFN5O
(2S)-2-amino-1-{3-[(4-chlorophenyl)amino]-2-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}propan-1-one
—— [5-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrimidin-2-yl]-(4-trifluoromethylbenzyl)amine 1029047-75-3 C20H16F3N5
[5-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)pyrimidin-2-yl]-(4-trifluoromethylbenzyl)amine
—— (E)-1-(4-bromophenyl)-2-(4-methoxyphenylsulfenyl)-3-(4-bromophenyl)prop-2-en-1-one 1035197-79-5 C22H16Br2O2S
(E)-1-(4-bromophenyl)-2-(4-methoxyphenylsulfenyl)-3-(4-bromophenyl)prop-2-en-1-one
—— (E)-1-(4-bromophenyl)-2-(4-methylphenylsulfenyl)-3-(5-bromo-3-indolyl)prop-2-en-1-one 1035198-21-0 C24H17Br2NOS
(E)-1-(4-bromophenyl)-2-(4-methylphenylsulfenyl)-3-(5-bromo-3-indolyl)prop-2-en-1-one
—— N-[[(2S,5R,6R)-5,6-dimethoxy-5,6-dimethyl-1,4-dioxan-2-yl]methyl]-4-methyl-N-[3-(4-methylphenyl)prop-2-ynyl]benzenesulfonamide 1006389-14-5 C26H33NO6S
N-[[(2S,5R,6R)-5,6-dimethoxy-5,6-dimethyl-1,4-dioxan-2-yl]methyl]-4-methyl-N-[3-(4-methylphenyl)prop-2-ynyl]benzenesulfonamide
—— [4-[3-(1,2-oxazol-4-yl)phenyl]-1-(7H-pyrrolo[3,2-e]pyrimidin-4-yl)piperidin-4-yl]methanamine 1035345-77-7 C21H22N6O
[4-[3-(1,2-oxazol-4-yl)phenyl]-1-(7H-pyrrolo[3,2-e]pyrimidin-4-yl)piperidin-4-yl]methanamine
—— [3-(7-piperidin-1-ylimidazo[1,2-a]pyridin-3-yl)-phenyl]-[1,3,4]thiadiazol-2-yl-amine 1036761-59-7 C20H20N6S
[3-(7-piperidin-1-ylimidazo[1,2-a]pyridin-3-yl)-phenyl]-[1,3,4]thiadiazol-2-yl-amine
—— 1-[2-methyl-4-(1-methyl-1H-pyrazolo[3,4-c]pyridin-4-yl)-phenyl]-3-(3-trifluoromethyl-phenyl)-urea 1032943-21-7 C22H18F3N5O
1-[2-methyl-4-(1-methyl-1H-pyrazolo[3,4-c]pyridin-4-yl)-phenyl]-3-(3-trifluoromethyl-phenyl)-urea
—— benzyl N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-(trifluoromethoxy)phenyl]carbamate 1035419-62-5 C28H24F3N3O4
benzyl N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-(trifluoromethoxy)phenyl]carbamate
—— (3E,9R)-9-hydroxy-1-(6-methoxy-2,8-dimethylchromen-2-yl)-4,8,12-trimethyltrideca-3,11-diene-2,10-dione 1033849-79-4 C28H38O5
(3E,9R)-9-hydroxy-1-(6-methoxy-2,8-dimethylchromen-2-yl)-4,8,12-trimethyltrideca-3,11-diene-2,10-dione
—— (3,4-difluoro-phenyl)-[6-(3,5-dimethyl-pyrazol-1-yl)-pyridin-2-yl]-amine 1043893-74-8 C16H14F2N4
(3,4-difluoro-phenyl)-[6-(3,5-dimethyl-pyrazol-1-yl)-pyridin-2-yl]-amine
—— 1-methyl-5-(methyl(4-morpholinobenzyl)amino)-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one 1033443-32-1 C21H28N6O2
1-methyl-5-(methyl(4-morpholinobenzyl)amino)-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one
—— methyl 2-[2-(4-bromo-phenylsulfanyl)-2-phenyl-acetylamino]-5-chloro-benzoate 1052073-85-4 C22H17BrClNO3S
methyl 2-[2-(4-bromo-phenylsulfanyl)-2-phenyl-acetylamino]-5-chloro-benzoate
—— 4-amino-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-piperidine-4-carboxylic acid (pyridin-2-ylmethyl)-amide hydrochloride 1035345-17-5 C18H21N7O*ClH
4-amino-1-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-piperidine-4-carboxylic acid (pyridin-2-ylmethyl)-amide hydrochloride
—— 4-[3-({2-[3-(diphenylmethyl)-6-oxopyridazin-1(6H)-yl]ethyl}sulfanyl)phenoxy]butanoic acid 1034017-04-3 C29H28N2O4S
4-[3-({2-[3-(diphenylmethyl)-6-oxopyridazin-1(6H)-yl]ethyl}sulfanyl)phenoxy]butanoic acid
—— N-{2-[2-(4-cyclopropyl-phenoxymethyl)-1H-benzoimidazol-5-yl]-phenyl}-methanesulfonamide 1033624-79-1 C24H23N3O3S
N-{2-[2-(4-cyclopropyl-phenoxymethyl)-1H-benzoimidazol-5-yl]-phenyl}-methanesulfonamide
—— (R)-2-(4-(cyclopropylsulfonyl)-2-oxopyridin-1(2H)-yl)-N-(5-fluorothiazol-2-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide 1036205-61-4 C19H22FN3O5S2
(R)-2-(4-(cyclopropylsulfonyl)-2-oxopyridin-1(2H)-yl)-N-(5-fluorothiazol-2-yl)-3-(tetrahydro-2H-pyran-4-yl)propanamide
—— (6R)-6-(2-aminoethyl)-4-{(1R)-1-[1-benzyl-4-(3-chlorophenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholin-3-one 1039747-01-7 C26H31ClN4O2
(6R)-6-(2-aminoethyl)-4-{(1R)-1-[1-benzyl-4-(3-chlorophenyl)-1H-imidazol-2-yl]-2-methylpropyl}morpholin-3-one
—— ethyl 3-[7-({4-[(3-methoxybenzoyl)amino]piperidin-1-yl}methyl)-2-naphthyl]propanoate 1018072-69-9 C29H34N2O4
ethyl 3-[7-({4-[(3-methoxybenzoyl)amino]piperidin-1-yl}methyl)-2-naphthyl]propanoate
—— 2,2,4,4-tetramethyl-6-(quinolin-5-yl)-1,2,3,4-tetrahydrofuro[2,3-h]quinolin-3-one 1040279-42-2 C24H22N2O2
2,2,4,4-tetramethyl-6-(quinolin-5-yl)-1,2,3,4-tetrahydrofuro[2,3-h]quinolin-3-one
—— 1-{5-[4-(4-chloro-phenyl)-5-phenyl-[1,2,3]triazol-2-yl]-pentyl}-piperidine 1025358-30-8 C24H29ClN4
1-{5-[4-(4-chloro-phenyl)-5-phenyl-[1,2,3]triazol-2-yl]-pentyl}-piperidine
—— 2-chloro-5-[(4-fluorophenyl)-methylsulfamoyl]-N-(6-methyl-2-pyridinyl)benzamide 1031073-17-2 C20H17ClFN3O3S
2-chloro-5-[(4-fluorophenyl)-methylsulfamoyl]-N-(6-methyl-2-pyridinyl)benzamide
—— 1-phenyl-3-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]imidazolidin-2-one 1197337-94-2 C17H13F3N4O
1-phenyl-3-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]imidazolidin-2-one
—— 3-Benzhydryl-6-bromoquinazolin-4-one 1197004-90-2 C21H15BrN2O
3-Benzhydryl-6-bromoquinazolin-4-one
—— 2-[4-(4,6-dimethoxypyrimidin-2-yloxy)phenoxy]propionic acid 1260249-24-8 C15H16N2O6
2-[4-(4,6-dimethoxypyrimidin-2-yloxy)phenoxy]propionic acid
—— (2R,3S,4R)-1,3,4-tris(phenylmethoxy)-4-(1-phenylpyrazol-4-yl)butan-2-ol 1055327-74-6 C34H34N2O4
(2R,3S,4R)-1,3,4-tris(phenylmethoxy)-4-(1-phenylpyrazol-4-yl)butan-2-ol
—— ethyl 2,4-dihydroxy-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydroquinoline-3-carboxylate 1332486-06-2 C14H17NO5
ethyl 2,4-dihydroxy-7,7-dimethyl-5-oxo-5,6,7,8-tetrahydroquinoline-3-carboxylate
—— —— 1370708-19-2 C19H13NOS2
—— (3-hydroxy-phenylthiocarbamoyl)-amidophosphoric acid diethyl ester 108629-77-2 C11H17N2O4PS
(3-hydroxy-phenylthiocarbamoyl)-amidophosphoric acid diethyl ester
—— 2-(2-phenylethylamino)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide 1023652-44-9 C22H25N5OS
2-(2-phenylethylamino)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
—— 2-(4-tert-butyl-phenoxymethyl)-5-(2-methanesulfonyl-phenyl)-1H-benzoimidazole 1033623-85-6 C25H26N2O3S
2-(4-tert-butyl-phenoxymethyl)-5-(2-methanesulfonyl-phenyl)-1H-benzoimidazole
—— 3-(cyclohexylmethyl)-N-[2-(diethylamino)-1-methylethyl]-2-oxo-2,3-dihydro-1H-benzimidazole-1-carboxamide 1012880-99-7 C22H34N4O2
3-(cyclohexylmethyl)-N-[2-(diethylamino)-1-methylethyl]-2-oxo-2,3-dihydro-1H-benzimidazole-1-carboxamide
—— (S)-4-[2-(4-trifluoromethylphenyl)ethyl]-4,5-dihydrooxazol-2-ylamine 1043492-33-6 C12H13F3N2O
(S)-4-[2-(4-trifluoromethylphenyl)ethyl]-4,5-dihydrooxazol-2-ylamine
—— (3R,4S)-4-[4-[3,4-dihydroxy-3-(hydroxymethyl)butyl]phenyl]-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-1-[4-[2-[4-(2-hydroxyethyl)-1,3-thiazol-2-yl]ethyl]phenyl]azetidin-2-one 1025467-54-2 C36H41FN2O6S
(3R,4S)-4-[4-[3,4-dihydroxy-3-(hydroxymethyl)butyl]phenyl]-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-1-[4-[2-[4-(2-hydroxyethyl)-1,3-thiazol-2-yl]ethyl]phenyl]azetidin-2-one
—— (3-{[1-(5-chloro-2-methoxy-benzenesulfonyl)-2,3-dihydro-1H-indole-6-carbonyl]-amino}-pyrazol-1-yl)-acetic acid 1034775-87-5 C21H19ClN4O6S
(3-{[1-(5-chloro-2-methoxy-benzenesulfonyl)-2,3-dihydro-1H-indole-6-carbonyl]-amino}-pyrazol-1-yl)-acetic acid
—— (2S)-N-[1-[6-[2-(difluoromethyl)benzoimidazol-1-yl]-2-morpholin-4-yl-pyrimidin-4-yl]-4-piperidyl]pyrrolidine-2-carboxamide 1013424-58-2 C26H32F2N8O2
(2S)-N-[1-[6-[2-(difluoromethyl)benzoimidazol-1-yl]-2-morpholin-4-yl-pyrimidin-4-yl]-4-piperidyl]pyrrolidine-2-carboxamide
—— N-(2-hydroxy-3-(pyrrolidin-1-yl)propyl)-2-methyl-7-[1,2-dihydro-5-fluoro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide 1032267-26-7 C25H29FN4O3
N-(2-hydroxy-3-(pyrrolidin-1-yl)propyl)-2-methyl-7-[1,2-dihydro-5-fluoro-2-oxo-3H-indol-(Z)-3-ylidene]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
—— 4-[2-(5-methyl-1-phenyl-1 H-1,2,4-triazol-3-yloxy)ethyl]morpholine 1025011-47-5 C15H20N4O2
4-[2-(5-methyl-1-phenyl-1 H-1,2,4-triazol-3-yloxy)ethyl]morpholine
—— 2-(5H-chromeno[2,3-b]pyridin-5-yl)-2-methyl-N-1,2,4-thiadiazol-5-ylpropanamide 1008113-86-7 C18H16N4O2S
2-(5H-chromeno[2,3-b]pyridin-5-yl)-2-methyl-N-1,2,4-thiadiazol-5-ylpropanamide
—— 1-butanoyl-3-{5-[3-(cyclopentyloxy)-4-methoxyphenyl]pyrimidin-2-yl}-1,3-dihydro-2H-benzimidazol-2-one 1048378-85-3 C27H28N4O4
1-butanoyl-3-{5-[3-(cyclopentyloxy)-4-methoxyphenyl]pyrimidin-2-yl}-1,3-dihydro-2H-benzimidazol-2-one
—— 8-(tert-butylamino)-6-({4-[(3-hydroxy-3-methylazetidin-1-yl)methyl]pyridin-2-yl}amino)-2-(2-hydroxyethyl)-1,2-dihydro-2,7-naphthyridin-1-one 1263394-98-4 C24H32N6O3
8-(tert-butylamino)-6-({4-[(3-hydroxy-3-methylazetidin-1-yl)methyl]pyridin-2-yl}amino)-2-(2-hydroxyethyl)-1,2-dihydro-2,7-naphthyridin-1-one
—— (2S)-2-amino-1-{3-[(4-chloro-3-fluorophenyl)amino]-2-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}propan-1-one 1261112-98-4 C21H20ClF2N5O
(2S)-2-amino-1-{3-[(4-chloro-3-fluorophenyl)amino]-2-(4-fluorophenyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazin-7-yl}propan-1-one