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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[1-(3,4-dichlorobenzyl)-2,3-dihydro-1H-indol-6-yl]benzoic acid 1202502-61-1 C22H17Cl2NO2
3-[1-(3,4-dichlorobenzyl)-2,3-dihydro-1H-indol-6-yl]benzoic acid
—— 4-[(3,4-dimethoxycinnamoyl)aminomethyl]benzoic acid 1053978-67-8 C19H19NO5
4-[(3,4-dimethoxycinnamoyl)aminomethyl]benzoic acid
—— 2-[4-(1-fluoro-ethyl)-3-(2-m-tolyl-ethoxy)-benzoylamino]-indane-2-carboxylic acid 1195941-35-5 C28H28FNO4
2-[4-(1-fluoro-ethyl)-3-(2-m-tolyl-ethoxy)-benzoylamino]-indane-2-carboxylic acid
—— trans-(2S,3R,4S,6R)-4-(dimethylamino)-2-(7-hydroxycyclotridecyloxy)-6-methyltetrahydro-2H-pyran-3-ol 1283116-36-8 C21H41NO4
trans-(2S,3R,4S,6R)-4-(dimethylamino)-2-(7-hydroxycyclotridecyloxy)-6-methyltetrahydro-2H-pyran-3-ol
—— 3-[(3-chloro-4-trifluoromethyl-phenyl)-methoxycarbonylmethyl-amino]-propionic acid tert-butyl ester 1290050-41-7 C17H21ClF3NO4
3-[(3-chloro-4-trifluoromethyl-phenyl)-methoxycarbonylmethyl-amino]-propionic acid tert-butyl ester
—— 6-(3-chloro-4-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-3-cyclohex-1-en-1-yl-1-[(2S)-1,4-dioxan-2-ylmethyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1207626-33-2 C25H26ClN5O3
6-(3-chloro-4-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-3-cyclohex-1-en-1-yl-1-[(2S)-1,4-dioxan-2-ylmethyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— rac-imidazo[1,2-a]pyridine-3-carboxylic acid [3-(2-methyl-5-m-tolyl-oxazole-4-carbonyl)-thiazolidin-2-ylmethyl]-amide 1204584-24-6 C24H23N5O3S
rac-imidazo[1,2-a]pyridine-3-carboxylic acid [3-(2-methyl-5-m-tolyl-oxazole-4-carbonyl)-thiazolidin-2-ylmethyl]-amide
—— 1-{4-[7-(2-{[2-(1H-imidazol-5-yl)ethyl]amino}ethyl)-4-morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-yl]phenyl}-3-pyridin-4-ylurea 1202884-73-8 C29H32N10O2
1-{4-[7-(2-{[2-(1H-imidazol-5-yl)ethyl]amino}ethyl)-4-morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-yl]phenyl}-3-pyridin-4-ylurea
—— (Z)-8-(2-cyclopropyl-7-methyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl-11-[1-(1H-tetrazol-5-yl)ethylidene]-6,11-dihydrodibenzo[b,e]oxepine 1046822-49-4 C28H25N7O
(Z)-8-(2-cyclopropyl-7-methyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl-11-[1-(1H-tetrazol-5-yl)ethylidene]-6,11-dihydrodibenzo[b,e]oxepine
—— 1,1-dimethylethyl 4-[(5'-{[({1-[({[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}amino)carbonyl]cyclopropyl}carbonyl)amino]methyl}-2'-fluoro-3-biphenylyl)methyl]-1-piperidinecarboxylate 1181078-82-9 C45H58FN7O5
1,1-dimethylethyl 4-[(5'-{[({1-[({[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}amino)carbonyl]cyclopropyl}carbonyl)amino]methyl}-2'-fluoro-3-biphenylyl)methyl]-1-piperidinecarboxylate
—— 1-(4-bromo-5-chloro-2-thienyl)-2-chloroethanol 1148011-97-5 C6H5BrCl2OS
1-(4-bromo-5-chloro-2-thienyl)-2-chloroethanol
—— 3-cyclopropyl-8-[2-(4-difluoromethoxy-3-fluoro-phenyl)-ethyl]-1-iodo-5,6-dihydro-8H-imidazo[1,5-a]pyrazine-7-carboxylic acid tert-butyl ester 1202690-59-2 C23H27F3IN3O3
3-cyclopropyl-8-[2-(4-difluoromethoxy-3-fluoro-phenyl)-ethyl]-1-iodo-5,6-dihydro-8H-imidazo[1,5-a]pyrazine-7-carboxylic acid tert-butyl ester
—— 4-{8-(4-((1S,4S)-5-tert-butyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)-phenyl-amino)imidazo[1,2-a]pyrazin-5-yl}-furan-2-carboxylic acid amide 1195065-43-0 C26H29N7O2
4-{8-(4-((1S,4S)-5-tert-butyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)-phenyl-amino)imidazo[1,2-a]pyrazin-5-yl}-furan-2-carboxylic acid amide
—— 8-{[4-({[tert-butyl(dimethyl)silyl]oxy}methyl)-2-methoxyphenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid 1202057-02-0 C25H33N5O4Si
8-{[4-({[tert-butyl(dimethyl)silyl]oxy}methyl)-2-methoxyphenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid
—— Pyrazolo[1,5-a]pyrimidine-3-carboxamide, N-[2-(dimethylamino)ethyl]-4,7-dihydro-5-methyl-7-oxo- 1788960-00-8 C12H17N5O2
Pyrazolo[1,5-a]pyrimidine-3-carboxamide, N-[2-(dimethylamino)ethyl]-4,7-dihydro-5-methyl-7-oxo-
—— 2-(1,3-benzothiazol-2-ylsulfanyl)-2-fluoroethyl acetate 1200123-12-1 C11H10FNO2S2
2-(1,3-benzothiazol-2-ylsulfanyl)-2-fluoroethyl acetate
—— 1-(3-chlorophenyl)-3-({[(1S,2R,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate 1039349-95-5 C2HF3O2*C24H26ClN3O
1-(3-chlorophenyl)-3-({[(1S,2R,4R)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate
—— (S)-N-(1-azabicyclo[2.2.2]oct-3-yl)-2-(1-methylcyclopropyl)benzoxazole-4-carboxamide 1006600-58-3 C19H23N3O2
(S)-N-(1-azabicyclo[2.2.2]oct-3-yl)-2-(1-methylcyclopropyl)benzoxazole-4-carboxamide
—— (E)-3-(4'-methanesulfonyl-biphenyl-3-yl)-3-phenyl-1-pyridin-4-yl-propan-1-one oxime 1354807-51-4 C27H24N2O3S
(E)-3-(4'-methanesulfonyl-biphenyl-3-yl)-3-phenyl-1-pyridin-4-yl-propan-1-one oxime
—— N-(2-{(E)-2-[3-tert-butyl-2-methoxy-5-(2-oxo-1,2-dihydro-pyridin-3-yl)-phenyl]-vinyl}-5-methanesulfonylamino-benzyl)-acetamide 1206772-60-2 C28H33N3O5S
N-(2-{(E)-2-[3-tert-butyl-2-methoxy-5-(2-oxo-1,2-dihydro-pyridin-3-yl)-phenyl]-vinyl}-5-methanesulfonylamino-benzyl)-acetamide
—— 6-(2,6-difluorobenzylamino)-8-amino-4-cyclopropyl-2-(3-fluorophenyl)pyrido[3,2-b]pyrazin-3(4H)-one 1205595-43-2 C23H18F3N5O
6-(2,6-difluorobenzylamino)-8-amino-4-cyclopropyl-2-(3-fluorophenyl)pyrido[3,2-b]pyrazin-3(4H)-one
—— (3-aminoazetidin-1-yl)-(2-fluoro-4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-phenyl)methanone 1204309-60-3 C23H32FN5O3
(3-aminoazetidin-1-yl)-(2-fluoro-4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-phenyl)methanone
—— 4-{3-[1-(5-chloropyrimidin-2-yl)piperidin-4-yl]propoxy}-2,6-dimethyl-N-(S)-1-pyrrolidin-3-ylmethylbenzamide 1204335-45-4 C26H36ClN5O2
4-{3-[1-(5-chloropyrimidin-2-yl)piperidin-4-yl]propoxy}-2,6-dimethyl-N-(S)-1-pyrrolidin-3-ylmethylbenzamide
—— 4-{3-[1-(3-ethyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-2-methyl-N-(R)-tetrahydro-furan-3-ylbenzamide 1204315-70-7 C24H34N4O4
4-{3-[1-(3-ethyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-2-methyl-N-(R)-tetrahydro-furan-3-ylbenzamide
—— 2,5-dimethyl-3-{4-[3-(pyridin-2-ylethynyl)benzoyl]piperazin-1-yl}pyrazine 1197354-15-6 C24H23N5O
2,5-dimethyl-3-{4-[3-(pyridin-2-ylethynyl)benzoyl]piperazin-1-yl}pyrazine
—— N-ethyl-1-(2-methyl-4-pyridinyl)-3-[[3-(trifluoromethyl)phenyl]amino]-1H-pyrazole-5-acetamide 1274885-81-2 C20H20F3N5O
N-ethyl-1-(2-methyl-4-pyridinyl)-3-[[3-(trifluoromethyl)phenyl]amino]-1H-pyrazole-5-acetamide
—— 3-{[(3-chlorophenyl)amino]methyl}-1-({3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]phenyl}carbonyl)azetidin-3-ol acetate salt 1035349-19-9 C2H4O2*C23H18ClF3IN3O2
3-{[(3-chlorophenyl)amino]methyl}-1-({3,4-difluoro-2-[(2-fluoro-4-iodophenyl)amino]phenyl}carbonyl)azetidin-3-ol acetate salt
—— N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-[2-(pyrrolidin-1-yl)ethyl]-3-(thiophen-3-yl)ureidomethyl]pyridine-2-carboxylic acid amide 1196983-67-1 C27H34N6O4S2
N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-[2-(pyrrolidin-1-yl)ethyl]-3-(thiophen-3-yl)ureidomethyl]pyridine-2-carboxylic acid amide
—— 4,5-dibromo-2-cyclopropyl-1H-imidazole 1269233-20-6 C6H6Br2N2
4,5-dibromo-2-cyclopropyl-1H-imidazole
—— (E)-3-{4-[4-(1-oxo-3,4-dihydro-1H-isoquinolin-2-yl)piperidin-1-ylmethyl]phenyl}acrylic acid methyl ester 1268716-74-0 C25H28N2O3
(E)-3-{4-[4-(1-oxo-3,4-dihydro-1H-isoquinolin-2-yl)piperidin-1-ylmethyl]phenyl}acrylic acid methyl ester
—— (R)-2-[(S)-4-(3-chloro-4-trifluoromethyl-phenylcarbamoyl)-3-methyl-2-oxo-piperazin-1-yl]-5-((S)-4-hydroxy-6-aza-spiro[2.5]oct-6-yl)-5-oxo-pentanoic acid methyl ester 1290050-68-8 C26H32ClF3N4O6
(R)-2-[(S)-4-(3-chloro-4-trifluoromethyl-phenylcarbamoyl)-3-methyl-2-oxo-piperazin-1-yl]-5-((S)-4-hydroxy-6-aza-spiro[2.5]oct-6-yl)-5-oxo-pentanoic acid methyl ester
—— (S)-1-[(S)-3-methyl-2-((S)-2-methylaminopropionylamino)butyryl]-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid (2-chloro-6-methylphenyl)amide 1595279-01-8 C24H30ClN5O3
(S)-1-[(S)-3-methyl-2-((S)-2-methylaminopropionylamino)butyryl]-2,3-dihydro-1H-pyrrolo[2,3-b]pyridine-2-carboxylic acid (2-chloro-6-methylphenyl)amide
—— 4-Amino-6-cyano-2-(1-(3-aminocarbinyl-1-methyl-1H-pyrrolo[2,3-c]pyridin-5-yl)ethyl)thio-pyrimidine 1102064-88-9 C16H17N7S
4-Amino-6-cyano-2-(1-(3-aminocarbinyl-1-methyl-1H-pyrrolo[2,3-c]pyridin-5-yl)ethyl)thio-pyrimidine
—— ethyl (R)-3-(5-(3-(N-(2-hydroxy-3-(2-methyl-5-phenylpentan-2-ylamino)propyl)-N-methylsulfamoyl)-5-(trifluoromethyl)phenyl)-4-methylthiophen-2-yl)propionate 1198615-25-6 C33H43F3N2O5S2
ethyl (R)-3-(5-(3-(N-(2-hydroxy-3-(2-methyl-5-phenylpentan-2-ylamino)propyl)-N-methylsulfamoyl)-5-(trifluoromethyl)phenyl)-4-methylthiophen-2-yl)propionate
—— 8-bromo-3-iodo-7-methoxy-2-phenyl-chromen-4-one 1279087-72-7 C16H10BrIO3
8-bromo-3-iodo-7-methoxy-2-phenyl-chromen-4-one
—— N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-(2-dimethylaminoethyl)-3-(pyridin-3-ylmethyl)ureidomethyl]pyridine-2-carboxylic acid amide 1196984-21-0 C27H35N7O4S
N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-(2-dimethylaminoethyl)-3-(pyridin-3-ylmethyl)ureidomethyl]pyridine-2-carboxylic acid amide
—— 1-(2,2-difluoro-1-phenylethyl)-3-(4-(2-methylpyridin-4-yl)phenyl)urea 1195172-59-8 C21H19F2N3O
1-(2,2-difluoro-1-phenylethyl)-3-(4-(2-methylpyridin-4-yl)phenyl)urea
—— 2-((1E,3E)-4-Phenyl-buta-1,3-dienyl)-1-(toluene-4-sulfonyl)-azetidine 124994-17-8 C20H21NO2S
2-((1E,3E)-4-Phenyl-buta-1,3-dienyl)-1-(toluene-4-sulfonyl)-azetidine
—— N-t-Butyl-tributyl-stannylamin 1067-30-7 C16H37NSn
N-t-Butyl-tributyl-stannylamin
—— 2-(2,4-difluoro-3-methoxy-benzyl)-2H-pyrazol-3-ylamine 1200440-05-6 C11H11F2N3O
2-(2,4-difluoro-3-methoxy-benzyl)-2H-pyrazol-3-ylamine
—— N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[3-phenethyl-1-[2-(pyrrolidin-1-yl)ethyl]ureidomethyl]pyridine-2-carboxylic acid amide 1196983-69-3 C31H40N6O4S
N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[3-phenethyl-1-[2-(pyrrolidin-1-yl)ethyl]ureidomethyl]pyridine-2-carboxylic acid amide
—— N-{(1S)-1-[((1S,4S)-5-{[5-(3-cyanophenyl)-2-pyridinyl]carbonyl}-2,5-diazabicyclo[2.2.1]hept-2-yl)carbonyl]-2,2-dimethylpropyl}-1H-indole-2-carboxamide 1206621-00-2 C33H32N6O3
N-{(1S)-1-[((1S,4S)-5-{[5-(3-cyanophenyl)-2-pyridinyl]carbonyl}-2,5-diazabicyclo[2.2.1]hept-2-yl)carbonyl]-2,2-dimethylpropyl}-1H-indole-2-carboxamide
—— 6A,6B,6D,6E-tetra-O-acetyl-β-cyclodextrin 1206782-72-0 C50H78O39
6A,6B,6D,6E-tetra-O-acetyl-β-cyclodextrin
—— N-cyclopentyl-5-(3,4-dihydroxyphenyl)furan-2-carboxamide 1141892-82-1 C16H17NO4
N-cyclopentyl-5-(3,4-dihydroxyphenyl)furan-2-carboxamide
—— [3,4-Dihydroxy-6-(5-methyl-1,2,4-oxadiazol-3-yl)-2-nitrophenyl]-(4-methylphenyl)methanone 1164106-59-5 C17H13N3O6
[3,4-Dihydroxy-6-(5-methyl-1,2,4-oxadiazol-3-yl)-2-nitrophenyl]-(4-methylphenyl)methanone
—— 3-((4-bromophenethylamino)methyl)-2-(thiophen-2-yl)quinolin-7-ol 1046138-64-0 C22H19BrN2OS
3-((4-bromophenethylamino)methyl)-2-(thiophen-2-yl)quinolin-7-ol
—— Cyclohexyl 3-hydroxy-4-methoxy-6-(5-methyl-1,2,4-oxadiazol-3-yl)-2-nitrobenzoate 1164108-46-6 C17H19N3O7
Cyclohexyl 3-hydroxy-4-methoxy-6-(5-methyl-1,2,4-oxadiazol-3-yl)-2-nitrobenzoate
—— 2-[4-[(2-hydroxy-3-naphthalen-1-yloxypropyl)amino]-2-oxo-1H-pyridin-3-yl]-6-(1-methylpiperidin-4-yl)-3H-pyrrolo[3,4-f]benzimidazole-5,7-dione 1008457-43-9 C33H32N6O5
2-[4-[(2-hydroxy-3-naphthalen-1-yloxypropyl)amino]-2-oxo-1H-pyridin-3-yl]-6-(1-methylpiperidin-4-yl)-3H-pyrrolo[3,4-f]benzimidazole-5,7-dione
—— 1-methyl-7-(((1-methyl-4-(4-fluorophenyl)piperidin-4-yl)methoxy)methyl)-5-(trifluoromethyl)-1H-indole 1100211-29-7 C24H26F4N2O
1-methyl-7-(((1-methyl-4-(4-fluorophenyl)piperidin-4-yl)methoxy)methyl)-5-(trifluoromethyl)-1H-indole
—— (S)-2-[4-[5-[3-(4-methyl-imidazol-1-yl)-5-trifluoromethyl-phenylcarbamoyl]-naphthalen-2-yloxy]-pyridin-2-ylcarbamoyl]-pyrrolidine-1-carboxylic acid 1,1-dimethylethyl ester 1072711-06-8 C37H35F3N6O5
(S)-2-[4-[5-[3-(4-methyl-imidazol-1-yl)-5-trifluoromethyl-phenylcarbamoyl]-naphthalen-2-yloxy]-pyridin-2-ylcarbamoyl]-pyrrolidine-1-carboxylic acid 1,1-dimethylethyl ester