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中文名称 英文名称 CAS号 化学式 结构式图片
—— 8-hydroxy-6-(imidazo[1,2-a]pyridin-3-yl)quinazolin-4(3H)-one 1616830-04-6 C15H10N4O2
8-hydroxy-6-(imidazo[1,2-a]pyridin-3-yl)quinazolin-4(3H)-one
—— 8-hydroxy-6-(1-methyl-1H-imidazol-2-yl)quinazolin-4(3H)-one 1616829-77-6 C12H10N4O2
8-hydroxy-6-(1-methyl-1H-imidazol-2-yl)quinazolin-4(3H)-one
—— 8-hydroxy-6-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-4(3H)-one 1616829-98-1 C11H8N4O2S
8-hydroxy-6-(5-methyl-1,3,4-thiadiazol-2-yl)quinazolin-4(3H)-one
—— 8-hydroxy-6-(tetrahydro-2H-pyran-4-yl)quinazolin-4(3H)-one 2,2,2-trifluoroacetate 1616829-68-5 C2HF3O2*C13H14N2O3
8-hydroxy-6-(tetrahydro-2H-pyran-4-yl)quinazolin-4(3H)-one 2,2,2-trifluoroacetate
—— 8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine 616201-55-9 C12H16BrNO
8-Bromo-7-methoxy-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine
—— 8-hydroxy-6-(morpholine-4-carbonyl)quinazolin-4(3H)-one 1616828-55-7 C13H13N3O4
8-hydroxy-6-(morpholine-4-carbonyl)quinazolin-4(3H)-one
—— 8-acetyl-3,7-dihydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one 1532528-17-8 C22H14O7
8-acetyl-3,7-dihydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one
—— 8-acetyl-4,7-dihydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one 1532528-18-9 C22H14O7
8-acetyl-4,7-dihydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one
—— 8-acetyl-7-hydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one 1532528-16-7 C22H14O6
8-acetyl-7-hydroxy-10-(2-hydroxybenzoyl)-6H-benzo[c]chromen-6-one
—— 8-ethoxy-4-methyl-quinoline 61704-08-3 C12H13NO
8-ethoxy-4-methyl-quinoline
—— 8-phenyl-3-(phenylsulfonyl)-1,2-octadien-7-yne 502176-50-3 C20H18O2S
8-phenyl-3-(phenylsulfonyl)-1,2-octadien-7-yne
—— 8-(Furan-2-yl)octan-2-ol 126680-21-5 C12H20O2
8-(Furan-2-yl)octan-2-ol
—— 8-(6-methoxy-1-oxo-1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one 62620-38-6 C25H29N3O3
8-(6-methoxy-1-oxo-1,2,3,4-tetrahydro-naphthalen-2-ylmethyl)-1-phenyl-1,3,8-triaza-spiro[4.5]decan-4-one
—— [8-(4-methylbenzyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrazolo[1,5-a][1,3,5]triazin-7-yl]thiourea 1607831-18-4 C14H14N6OS2
[8-(4-methylbenzyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrazolo[1,5-a][1,3,5]triazin-7-yl]thiourea
—— {(8R)-8-methyl-3-{1-[4-(1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol 1403395-77-6 C20H23N5OS
{(8R)-8-methyl-3-{1-[4-(1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(1-isopropyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-86-0 C29H43N5OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(1-isopropyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— (8-methyl-3-{1-[4-(1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol 1403395-88-9 C20H23N5OS
(8-methyl-3-{1-[4-(1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-93-9 C26H36N4O2SSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— {8-methyl-3-{1-[4-(6-methylpyridin-3-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol 1403395-23-2 C23H26N4OS
{8-methyl-3-{1-[4-(6-methylpyridin-3-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol
—— (8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol 1403395-89-0 C20H22N4O2S
(8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol
—— [8-methyl-3-(1-{4-[5-(piperidin-1-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-91-4 C28H33N5O2S
[8-methyl-3-(1-{4-[5-(piperidin-1-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— 8,11-bis-(2-pyridylmethyl)5,6,7,8,9,10,16,17-octahydrodibenzo[e,m][1,4]dithia[8,11]diazacyclotetradecine 169476-59-9 C30H32N4S2
8,11-bis-(2-pyridylmethyl)5,6,7,8,9,10,16,17-octahydrodibenzo[e,m][1,4]dithia[8,11]diazacyclotetradecine
—— (8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(5-methylpyrazin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-95-1 C28H39N5OSSi
(8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(5-methylpyrazin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 8,11-dimethyl-5,6,7,8,9,10,16,17-octahydrodibenzo(e,m)-1,4-dithia-8,11,-diazacyclotetradecane 1006885-82-0 C20H26N2S2
8,11-dimethyl-5,6,7,8,9,10,16,17-octahydrodibenzo(e,m)-1,4-dithia-8,11,-diazacyclotetradecane
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(2-methoxypyridin-3-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-52-0 C29H40N4O2SSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(2-methoxypyridin-3-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— [(8R)-8-methyl-3-{1-[4-(2-methylpyrimidin-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-93-6 C22H25N5OS
[(8R)-8-methyl-3-{1-[4-(2-methylpyrimidin-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-[1-(4-isoxazol-4-ylphenyl)cyclopropyl]-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-85-9 C26H36N4O2SSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-[1-(4-isoxazol-4-ylphenyl)cyclopropyl]-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— {(8R)-8-methyl-3-{1-[4-(5-methylpyrimidin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol 1403395-57-2 C22H25N5OS
{(8R)-8-methyl-3-{1-[4-(5-methylpyrimidin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-87-1 C27H39N5OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— [8-(4-methoxybenzyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrazolo[1,5-a][1,3,5]triazin-7-yl]thiourea 1607831-20-8 C14H14N6O2S2
[8-(4-methoxybenzyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydropyrazolo[1,5-a][1,3,5]triazin-7-yl]thiourea
—— (8R)-4'-{1-[8-(hydroxymethyl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-3-yl]cyclopropyl}-N,N-dimethylbiphenyl-4-carboxamide 1403395-12-9 C26H30N4O2S
(8R)-4'-{1-[8-(hydroxymethyl)-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-3-yl]cyclopropyl}-N,N-dimethylbiphenyl-4-carboxamide
—— (8-methyl-3-{1-[4-(1-methyl-1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol 1403395-61-8 C21H25N5OS
(8-methyl-3-{1-[4-(1-methyl-1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol
—— [(8R)-(3-{1-[4-(1-ethyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)]methanol 1403396-83-7 C22H27N5OS
[(8R)-(3-{1-[4-(1-ethyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)]methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(5-methylpyridin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-29-1 C29H40N4OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(5-methylpyridin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— [8-methyl-3-(1-{4-[5-(trifluoromethyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-47-0 C23H23F3N4OS
[8-methyl-3-(1-{4-[5-(trifluoromethyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— [(8R)-8-methyl-3-{1-[4-(5-methylpyrazin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-92-5 C22H25N5OS
[(8R)-8-methyl-3-{1-[4-(5-methylpyrazin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-41-7 C27H39N5OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-[1-(4-pyridazin-3-ylphenyl)cyclopropyl]-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-59-7 C27H37N5OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-[1-(4-pyridazin-3-ylphenyl)cyclopropyl]-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-92-8 C26H37N5OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(1H-pyrazol-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— {(8R)-8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol 1403395-90-3 C20H22N4O2S
{(8R)-8-methyl-3-{1-[4-(1,3-oxazol-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol
—— (8-methyl-3-{1-[4-(6-methylpyridazin-3-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol 1403395-69-6 C22H25N5OS
(8-methyl-3-{1-[4-(6-methylpyridazin-3-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol
—— {8-methyl-3-{1-[4-(6-methylpyridin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol 1403395-26-5 C23H26N4OS
{8-methyl-3-{1-[4-(6-methylpyridin-2-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl}methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(4-methoxypyridin-3-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-68-8 C29H40N4O2SSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(4-methoxypyridin-3-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— [8-methyl-3-(1-{4-[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-84-5 C27H31N5O3S
[8-methyl-3-(1-{4-[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— (8-methyl-3-{1-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol 1403395-81-2 C21H25N5OS
(8-methyl-3-{1-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl)methanol
—— [8-methyl-3-(1-{4-[5-(pyrrolidin-1-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-83-4 C27H31N5O2S
[8-methyl-3-(1-{4-[5-(pyrrolidin-1-ylcarbonyl)pyridin-2-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— 8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(5-chloropyridin-2-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-64-4 C28H37ClN4OSSi
8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(5-chloropyridin-2-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— (8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(2-methylpyrimidin-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-98-4 C28H39N5OSSi
(8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-8-methyl-3-{1-[4-(2-methylpyrimidin-5-yl)phenyl]cyclopropyl}-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine
—— [8-methyl-3-(1-{4-[2-(trifluoromethyl)pyridin-3-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol 1403395-54-9 C23H23F3N4OS
[8-methyl-3-(1-{4-[2-(trifluoromethyl)pyridin-3-yl]phenyl}cyclopropyl)-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepin-8-yl]methanol
—— (8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(1-ethyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine 1403396-84-8 C28H41N5OSSi
(8R)-8-({[tert-butyl(dimethyl)silyl]oxy}methyl)-3-{1-[4-(1-ethyl-1H-pyrazol-4-yl)phenyl]cyclopropyl}-8-methyl-5,6,8,9-tetrahydro[1,2,4]triazolo[4,3-d][1,4]thiazepine