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—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(propanoylamino)phenoxy]-1-(2,5-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid —— C26H32N4O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(propanoylamino)phenoxy]-1-(2,5-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid
—— (5E)-5-[(1-phenyltriazol-4-yl)methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C15H12N4OS2
(5E)-5-[(1-phenyltriazol-4-yl)methylidene]-3-prop-2-enyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(3,4-dimethyl-1,2-oxazol-5-yl)-N,N-dimethyl-4-[(2S)-1-[(4-propan-2-ylphenyl)methyl]pyrrolidin-2-yl]pyrimidin-2-amine —— C25H33N5O
5-(3,4-dimethyl-1,2-oxazol-5-yl)-N,N-dimethyl-4-[(2S)-1-[(4-propan-2-ylphenyl)methyl]pyrrolidin-2-yl]pyrimidin-2-amine
—— (5E)-2-cyclopentylimino-5-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methylidene]-1,3-thiazolidin-4-one —— C14H15F3N4OS
(5E)-2-cyclopentylimino-5-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methylidene]-1,3-thiazolidin-4-one
—— 5-(3,4-dimethyl-1,2-oxazol-5-yl)-N,N-dimethyl-4-[(2R)-1-[(4-propan-2-ylphenyl)methyl]pyrrolidin-2-yl]pyrimidin-2-amine —— C25H33N5O
5-(3,4-dimethyl-1,2-oxazol-5-yl)-N,N-dimethyl-4-[(2R)-1-[(4-propan-2-ylphenyl)methyl]pyrrolidin-2-yl]pyrimidin-2-amine
—— 5-[(E)-1-chloro-2-(4-phenyl-1,3-thiazol-2-yl)ethenyl]-N-(4-fluorophenyl)-1,3,4-thiadiazole-2-carboxamide —— C20H12ClFN4OS2
5-[(E)-1-chloro-2-(4-phenyl-1,3-thiazol-2-yl)ethenyl]-N-(4-fluorophenyl)-1,3,4-thiadiazole-2-carboxamide
—— (5E)-5-[(6,8-dichloro-2H-chromen-3-yl)methylidene]-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H10Cl2N2O2S2
(5E)-5-[(6,8-dichloro-2H-chromen-3-yl)methylidene]-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-Bromo-1-(cyclopropylcarbonyl)-6-{[4-(2-fluorophenyl)piperazin-1-yl]sulfonyl}indoline —— C22H23BrFN3O3S
5-Bromo-1-(cyclopropylcarbonyl)-6-{[4-(2-fluorophenyl)piperazin-1-yl]sulfonyl}indoline
—— 5-[4-[(2R)-1-[(3,4-dichlorophenyl)methyl]pyrrolidin-2-yl]-2-methylpyrimidin-5-yl]-3,4-dimethyl-1,2-oxazole —— C21H22Cl2N4O
5-[4-[(2R)-1-[(3,4-dichlorophenyl)methyl]pyrrolidin-2-yl]-2-methylpyrimidin-5-yl]-3,4-dimethyl-1,2-oxazole
—— (5E)-2-(2,5-dimethylphenyl)imino-5-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methylidene]-1,3-thiazolidin-4-one —— C17H15F3N4OS
(5E)-2-(2,5-dimethylphenyl)imino-5-[[1-(2,2,2-trifluoroethyl)imidazol-2-yl]methylidene]-1,3-thiazolidin-4-one
—— 5-cyclopropyl-3-[1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one —— C18H22N6O2
5-cyclopropyl-3-[1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl]-2H-triazolo[4,5-d]pyrimidin-7-one
—— 5-chloro-6-[[(Z)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enoyl]amino]pyridine-3-carboxamide —— C19H18ClN3O4
5-chloro-6-[[(Z)-3-(3-methoxy-4-prop-2-enoxyphenyl)prop-2-enoyl]amino]pyridine-3-carboxamide
—— (5E)-1-methyl-5-[(Z)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one —— C17H16N2O
(5E)-1-methyl-5-[(Z)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one
—— 5-[(4Z)-4-benzylidene-2-methyl-5-oxoimidazol-1-yl]-1,3-dihydrobenzimidazol-2-one —— C18H14N4O2
5-[(4Z)-4-benzylidene-2-methyl-5-oxoimidazol-1-yl]-1,3-dihydrobenzimidazol-2-one
—— (5Z)-1-methyl-5-[(Z)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one —— C17H16N2O
(5Z)-1-methyl-5-[(Z)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 2-(2-oxo-1,3-thiazolidin-3-yl)acetate —— C15H14N2O4S
(5-Phenyl-1,3-oxazol-2-yl)methyl 2-(2-oxo-1,3-thiazolidin-3-yl)acetate
—— (5Z)-5-[(3-methoxy-4-methylsulfanylphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one —— C17H18N2O2S
(5Z)-5-[(3-methoxy-4-methylsulfanylphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one
—— 5-[(Z)-3-(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)prop-2-enoyl]-1,3-dihydroindol-2-one —— C21H19NO4
5-[(Z)-3-(4-hydroxy-3-methoxy-5-prop-2-enylphenyl)prop-2-enoyl]-1,3-dihydroindol-2-one
—— (5Z)-1-methyl-5-[(E)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one —— C17H16N2O
(5Z)-1-methyl-5-[(E)-3-phenylprop-2-enylidene]-6,7-dihydroindazol-4-one
—— 5-[(Z)-3-(3-methoxy-4-methylsulfanylphenyl)prop-2-enoyl]-1,3-dihydroindol-2-one —— C19H17NO3S
5-[(Z)-3-(3-methoxy-4-methylsulfanylphenyl)prop-2-enoyl]-1,3-dihydroindol-2-one
—— (5E)-3-methyl-4-oxo-5-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methylidene]-6,7-dihydro-1-benzofuran-2-carboxylic acid —— C19H14N2O4S
(5E)-3-methyl-4-oxo-5-[(2-pyridin-2-yl-1,3-thiazol-4-yl)methylidene]-6,7-dihydro-1-benzofuran-2-carboxylic acid
—— 5-methyl-N-[4-[[(Z)-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]phenyl]-1,2-oxazole-4-carboxamide —— C19H17N3O4
5-methyl-N-[4-[[(Z)-3-(5-methylfuran-2-yl)prop-2-enoyl]amino]phenyl]-1,2-oxazole-4-carboxamide
—— 5-cyclopropyl-3-[[5-[(Z)-2-(4-fluorophenyl)ethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C16H14FN5OS
5-cyclopropyl-3-[[5-[(Z)-2-(4-fluorophenyl)ethenyl]-1H-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— 5-methyl-N-[4-[[(Z)-3-thiophen-3-ylprop-2-enoyl]amino]phenyl]-1,2-oxazole-4-carboxamide —— C18H15N3O3S
5-methyl-N-[4-[[(Z)-3-thiophen-3-ylprop-2-enoyl]amino]phenyl]-1,2-oxazole-4-carboxamide
—— 5-(2-chlorophenyl)-12-[(2S)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H19ClN4O3
5-(2-chlorophenyl)-12-[(2S)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-(2-chlorophenyl)-12-[(2R)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H21ClN4O2
5-(2-chlorophenyl)-12-[(2R)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5-chlorothiophen-2-yl)-[(2R)-3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-piperidine]-1'-yl]methanone —— C21H24ClN5OS
(5-chlorothiophen-2-yl)-[(2R)-3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-piperidine]-1'-yl]methanone
—— (5-chlorothiophen-2-yl)-[(2S)-3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-piperidine]-1'-yl]methanone —— C21H24ClN5OS
(5-chlorothiophen-2-yl)-[(2S)-3-cyclopentyliminospiro[1,4-dihydropyrido[2,3-b]pyrazine-2,3'-piperidine]-1'-yl]methanone
—— 5-(2-chlorophenyl)-12-[(2S)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H21ClN4O2
5-(2-chlorophenyl)-12-[(2S)-2-methylbutanoyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— (5-chloro-2-methoxyphenyl)-[(2R)-3-(2-methoxyethylimino)spiro[1,4-dihydroquinoxaline-2,3'-piperidine]-1'-yl]methanone —— C23H27ClN4O3
(5-chloro-2-methoxyphenyl)-[(2R)-3-(2-methoxyethylimino)spiro[1,4-dihydroquinoxaline-2,3'-piperidine]-1'-yl]methanone
—— (5-chloro-2-methoxyphenyl)-[(2S)-3-(2-methoxyethylimino)spiro[1,4-dihydroquinoxaline-2,3'-piperidine]-1'-yl]methanone —— C23H27ClN4O3
(5-chloro-2-methoxyphenyl)-[(2S)-3-(2-methoxyethylimino)spiro[1,4-dihydroquinoxaline-2,3'-piperidine]-1'-yl]methanone
—— 5-(2-chlorophenyl)-12-[(2R)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one —— C20H19ClN4O3
5-(2-chlorophenyl)-12-[(2R)-oxolane-2-carbonyl]-2,6,7,12-tetrazatricyclo[7.4.0.03,7]trideca-1(9),2,4-trien-8-one
—— 5-[(Z)-3-[(2S)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxoprop-1-enyl]-1,3-dimethylpyrimidine-2,4-dione —— C20H22FN3O3
5-[(Z)-3-[(2S)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxoprop-1-enyl]-1,3-dimethylpyrimidine-2,4-dione
—— 5-[(Z)-3-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxoprop-1-enyl]-1,3-dimethylpyrimidine-2,4-dione —— C20H22FN3O3
5-[(Z)-3-[(2R)-2-[(3-fluorophenyl)methyl]pyrrolidin-1-yl]-3-oxoprop-1-enyl]-1,3-dimethylpyrimidine-2,4-dione
—— 5-chloro-N-methyl-2-[[(Z)-3-[4-(methylcarbamoyl)phenyl]prop-2-enoyl]amino]benzamide —— C19H18ClN3O3
5-chloro-N-methyl-2-[[(Z)-3-[4-(methylcarbamoyl)phenyl]prop-2-enoyl]amino]benzamide
—— 5-[(Z)-3-(2,3-dihydro-1-benzofuran-5-yl)prop-2-enoyl]-1,3-dihydroindol-2-one —— C19H15NO3
5-[(Z)-3-(2,3-dihydro-1-benzofuran-5-yl)prop-2-enoyl]-1,3-dihydroindol-2-one
—— 5-bromo-N-[(2R)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide —— C11H12BrF3N2O2
5-bromo-N-[(2R)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide
—— 5,6-dimethoxy-2-[(Z)-2-(thiadiazol-4-yl)ethenyl]-1,3-benzothiazole —— C13H11N3O2S2
5,6-dimethoxy-2-[(Z)-2-(thiadiazol-4-yl)ethenyl]-1,3-benzothiazole
—— 5-[[(Z)-but-2-enyl]sulfonylmethyl]-1-[4-(trifluoromethyl)phenyl]tetrazole —— C13H13F3N4O2S
5-[[(Z)-but-2-enyl]sulfonylmethyl]-1-[4-(trifluoromethyl)phenyl]tetrazole
—— 5-[(Z)-3-(3,4-dihydro-2H-1,5-benzodioxepin-6-yl)prop-2-enoyl]-1,3-dihydroindol-2-one —— C20H17NO4
5-[(Z)-3-(3,4-dihydro-2H-1,5-benzodioxepin-6-yl)prop-2-enoyl]-1,3-dihydroindol-2-one
—— 5-[(Z)-3-(2-phenylpyrimidin-5-yl)prop-2-enoyl]thiophene-2-carboxylic acid —— C18H12N2O3S
5-[(Z)-3-(2-phenylpyrimidin-5-yl)prop-2-enoyl]thiophene-2-carboxylic acid
—— (5Z)-5-[[3-(2-methoxyethoxy)phenyl]methylidene]-1-methyl-6,7-dihydroindazol-4-one —— C18H20N2O3
(5Z)-5-[[3-(2-methoxyethoxy)phenyl]methylidene]-1-methyl-6,7-dihydroindazol-4-one
—— (5Z)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one —— C16H16N2O3
(5Z)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one
—— (5Z)-5-[[3-methoxy-4-(2-methoxyethoxy)phenyl]methylidene]-1-methyl-6,7-dihydroindazol-4-one —— C19H22N2O4
(5Z)-5-[[3-methoxy-4-(2-methoxyethoxy)phenyl]methylidene]-1-methyl-6,7-dihydroindazol-4-one
—— 5-[(Z)-3-(2-pyrrolidin-1-ylpyrimidin-5-yl)prop-2-enoyl]thiophene-2-carboxylic acid —— C16H15N3O3S
5-[(Z)-3-(2-pyrrolidin-1-ylpyrimidin-5-yl)prop-2-enoyl]thiophene-2-carboxylic acid
—— 5-bromo-N-[(2S)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide —— C11H12BrF3N2O2
5-bromo-N-[(2S)-1-(trifluoromethoxy)butan-2-yl]pyridine-3-carboxamide
—— (5E)-5-[(1-methyl-3-propan-2-ylpyrazol-4-yl)methylidene]-2-piperidin-1-yl-1,3-thiazol-4-one —— C16H22N4OS
(5E)-5-[(1-methyl-3-propan-2-ylpyrazol-4-yl)methylidene]-2-piperidin-1-yl-1,3-thiazol-4-one
—— 5-(1,3,4-oxadiazol-2-yl)-1-[(Z)-3-phenylprop-2-enyl]pyridin-2-one —— C16H13N3O2
5-(1,3,4-oxadiazol-2-yl)-1-[(Z)-3-phenylprop-2-enyl]pyridin-2-one
—— 5-chloro-2-[(Z)-2-(thiadiazol-4-yl)ethenyl]-1,3-benzothiazole —— C11H6ClN3S2
5-chloro-2-[(Z)-2-(thiadiazol-4-yl)ethenyl]-1,3-benzothiazole
—— (5Z)-5-[(3-hydroxy-4-methoxyphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one —— C16H16N2O3
(5Z)-5-[(3-hydroxy-4-methoxyphenyl)methylidene]-1-methyl-6,7-dihydroindazol-4-one