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—— (5S)-N-[2-(3-methoxyanilino)-2-oxoethyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide —— C20H24N2O3S
(5S)-N-[2-(3-methoxyanilino)-2-oxoethyl]-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
—— (5R)-5-[[(5S)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C16H22N2O2
(5R)-5-[[(5S)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— 5-(1,3-benzothiazol-2-yl)-N'-[2-(4-fluorophenyl)acetyl]pentanehydrazide —— C20H20FN3O2S
5-(1,3-benzothiazol-2-yl)-N'-[2-(4-fluorophenyl)acetyl]pentanehydrazide
—— (5R)-7-methoxy-N-[2-(5-methyl-1,3-thiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C17H22N2O2S
(5R)-7-methoxy-N-[2-(5-methyl-1,3-thiazol-2-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5S)-1-methyl-5-[[(2S)-1,1,1-trifluoro-3-phenylpropan-2-yl]amino]piperidin-2-one —— C15H19F3N2O
(5S)-1-methyl-5-[[(2S)-1,1,1-trifluoro-3-phenylpropan-2-yl]amino]piperidin-2-one
—— (5R)-1-methyl-5-[[(1S)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one —— C18H25N3O2
(5R)-1-methyl-5-[[(1S)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one
—— (5R)-5-[[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C15H20N2O2
(5R)-5-[[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5S)-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C15H20N2O2
(5S)-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5S)-5-[[(5S)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C16H22N2O2
(5S)-5-[[(5S)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7,9-dimethyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C18H24N2O2
(5R)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7,9-dimethyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5Z)-5-[[1-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-2,5-dimethylpyrrol-3-yl]methylidene]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C25H21Cl2N3O3S
(5Z)-5-[[1-[4-[(2,4-dichlorophenyl)methoxy]phenyl]-2,5-dimethylpyrrol-3-yl]methylidene]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)methylidene]-1-(3,5-dimethylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H23ClN2O4S
(5Z)-5-[(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)methylidene]-1-(3,5-dimethylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7,9-dimethyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C18H24N2O2
(5S)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-7,9-dimethyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5S)-5-[[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C15H20N2O2
(5S)-5-[[(5S)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5Z)-5-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1-(4-chlorophenyl)-3-ethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H16BrClN2O4S
(5Z)-5-[(3-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1-(4-chlorophenyl)-3-ethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[[5-(4-chlorophenyl)sulfanylthiophen-2-yl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C18H13ClN2O2S3
(5Z)-5-[[5-(4-chlorophenyl)sulfanylthiophen-2-yl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-1-methyl-5-[[(2R)-1,1,1-trifluoro-3-phenylpropan-2-yl]amino]piperidin-2-one —— C15H19F3N2O
(5R)-1-methyl-5-[[(2R)-1,1,1-trifluoro-3-phenylpropan-2-yl]amino]piperidin-2-one
—— (5E)-1-(2,3-dichlorophenyl)-5-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C26H23Cl2N3O2S
(5E)-1-(2,3-dichlorophenyl)-5-[[2,5-dimethyl-1-(4-propan-2-ylphenyl)pyrrol-3-yl]methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-5-[[(5R)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C16H22N2O2
(5R)-5-[[(5R)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5E)-1-(2-methylphenyl)-5-[(4-pyrrolidin-1-ylphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C22H21N3O2S
(5E)-1-(2-methylphenyl)-5-[(4-pyrrolidin-1-ylphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5E)-5-[[5-(3,4-dichlorophenyl)furan-2-yl]methylidene]-1-(2-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H11Cl2FN2O3S
(5E)-5-[[5-(3,4-dichlorophenyl)furan-2-yl]methylidene]-1-(2-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-1-methyl-5-[[(1S)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one —— C18H25N3O2
(5S)-1-methyl-5-[[(1S)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one
—— (5Z)-5-[[2-[(2S)-butan-2-yl]oxy-3-methoxyphenyl]methylidene]-1-(3-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C22H21FN2O4S
(5Z)-5-[[2-[(2S)-butan-2-yl]oxy-3-methoxyphenyl]methylidene]-1-(3-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-5-[[(5R)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C16H22N2O2
(5S)-5-[[(5R)-7-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5R)-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one —— C15H20N2O2
(5R)-5-[[(5R)-2,3,4,5-tetrahydro-1-benzoxepin-5-yl]amino]piperidin-2-one
—— (5Z)-5-[(3-bromo-4-ethoxy-5-methoxyphenyl)methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H19BrN2O4S
(5Z)-5-[(3-bromo-4-ethoxy-5-methoxyphenyl)methylidene]-1-(4-methylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H21FN2O4S
(5Z)-5-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H29N3S
(5S)-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5R)-1-methyl-5-[[(1R)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one —— C18H25N3O2
(5R)-1-methyl-5-[[(1R)-1-[4-(2-oxopyrrolidin-1-yl)phenyl]ethyl]amino]piperidin-2-one
—— (5Z)-5-[(2-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1-(3,5-dimethylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H17BrN2O4S
(5Z)-5-[(2-bromo-4-hydroxy-5-methoxyphenyl)methylidene]-1-(3,5-dimethylphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5R)-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H29N3S
(5R)-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5S)-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H29N3S
(5S)-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5S)-N-[(2-cyclopropyl-1,3-thiazol-4-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine —— C18H22N2OS
(5S)-N-[(2-cyclopropyl-1,3-thiazol-4-yl)methyl]-8-methyl-2,3,4,5-tetrahydro-1-benzoxepin-5-amine
—— (5R)-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine —— C18H29N3S
(5R)-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-1,2,4,5-tetrahydro-3-benzothiepin-5-amine
—— (5Z)-5-[[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C24H24N2O4S
(5Z)-5-[[3-ethoxy-4-[(3-methylphenyl)methoxy]phenyl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5S)-7-(5-bromo-2-nitrophenyl)-2-oxa-7-azaspiro[4.4]nonane —— C13H15BrN2O3
(5S)-7-(5-bromo-2-nitrophenyl)-2-oxa-7-azaspiro[4.4]nonane
—— (5Z)-5-[(3-fluoro-4-morpholin-4-ylphenyl)methylidene]-1-(4-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C22H20FN3O4S
(5Z)-5-[(3-fluoro-4-morpholin-4-ylphenyl)methylidene]-1-(4-methoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5,7-difluoro-N-[(3R)-1-methyl-6-oxopiperidin-3-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamide —— C16H19F2N3O2
5,7-difluoro-N-[(3R)-1-methyl-6-oxopiperidin-3-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamide
—— (5R)-7-(5-bromo-2-nitrophenyl)-2-oxa-7-azaspiro[4.4]nonane —— C13H15BrN2O3
(5R)-7-(5-bromo-2-nitrophenyl)-2-oxa-7-azaspiro[4.4]nonane
—— 5-nitro-2-N-[[(2R)-oxolan-2-yl]methyl]-2-N-(thiophen-2-ylmethyl)pyrimidine-2,4-diamine —— C14H17N5O3S
5-nitro-2-N-[[(2R)-oxolan-2-yl]methyl]-2-N-(thiophen-2-ylmethyl)pyrimidine-2,4-diamine
—— (5E)-5-[[1-(3,4-dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C20H17Cl2N3O2S
(5E)-5-[[1-(3,4-dichlorophenyl)-2,5-dimethylpyrrol-3-yl]methylidene]-1-prop-2-enyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-1-(2-methoxyphenyl)-5-[(1-prop-2-ynylindol-3-yl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C23H17N3O3S
(5Z)-1-(2-methoxyphenyl)-5-[(1-prop-2-ynylindol-3-yl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-{[5-(3-fluorophenyl)-2-furyl]methylene}-1-(4-methoxyphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione —— C22H15FN2O4S
5-{[5-(3-fluorophenyl)-2-furyl]methylene}-1-(4-methoxyphenyl)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione
—— (5Z)-5-[(5-chlorothiophen-2-yl)methylidene]-1-(4-ethoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H13ClN2O3S2
(5Z)-5-[(5-chlorothiophen-2-yl)methylidene]-1-(4-ethoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]methylidene]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H14Br2N2O3S
(5Z)-5-[[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]methylidene]-1-methyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-nitro-2-N-[[(2S)-oxolan-2-yl]methyl]-2-N-(thiophen-2-ylmethyl)pyrimidine-2,4-diamine —— C14H17N5O3S
5-nitro-2-N-[[(2S)-oxolan-2-yl]methyl]-2-N-(thiophen-2-ylmethyl)pyrimidine-2,4-diamine
—— (5E)-5-[(3,5-dichloro-4-hydroxyphenyl)methylidene]-1-(4-ethoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H14Cl2N2O4S
(5E)-5-[(3,5-dichloro-4-hydroxyphenyl)methylidene]-1-(4-ethoxyphenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-5-[(3,4-diethoxyphenyl)methylidene]-1-(3-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C21H19FN2O4S
(5Z)-5-[(3,4-diethoxyphenyl)methylidene]-1-(3-fluorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5Z)-1-(3-chloro-4-methylphenyl)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H15ClN2O4S
(5Z)-1-(3-chloro-4-methylphenyl)-5-[(4-hydroxy-3-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— (5E)-1-(3-fluorophenyl)-5-[(1-prop-2-enylindol-3-yl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C22H16FN3O2S
(5E)-1-(3-fluorophenyl)-5-[(1-prop-2-enylindol-3-yl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione