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吖庚因类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-(Cyclopent-3-ene-1-carbonyl)-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C18H24N2O3
7-(Cyclopent-3-ene-1-carbonyl)-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— N,N-dimethyl-2-oxo-5,6,8,9-tetrahydro-1H-pyrido[2,3-d]azepine-7-carboxamide —— C12H17N3O2
N,N-dimethyl-2-oxo-5,6,8,9-tetrahydro-1H-pyrido[2,3-d]azepine-7-carboxamide
—— N-[(3-fluorophenyl)methyl]-4-methoxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxamide —— C17H19FN4O2
N-[(3-fluorophenyl)methyl]-4-methoxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxamide
—— 1-[4-(Cyclopropylamino)-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-3-hydroxypropan-1-one —— C15H22N4O2
1-[4-(Cyclopropylamino)-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-3-hydroxypropan-1-one
—— (5-Methyl-1,2-oxazol-4-yl)-[4-(1-methylpyrazol-4-yl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methanone —— C17H18N6O2
(5-Methyl-1,2-oxazol-4-yl)-[4-(1-methylpyrazol-4-yl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methanone
—— Cyclopent-3-en-1-yl-(4-pyridin-4-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methanone —— C19H20N4O
Cyclopent-3-en-1-yl-(4-pyridin-4-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methanone
—— 7-[(5-Ethylfuran-2-yl)methyl]-4-methoxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C16H21N3O2
7-[(5-Ethylfuran-2-yl)methyl]-4-methoxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— Cyclopropyl-[2-phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methanone —— C21H26N4O
Cyclopropyl-[2-phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methanone
—— 3-Oxo-3-[2-phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]propanenitrile —— C20H23N5O
3-Oxo-3-[2-phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]propanenitrile
—— 4-Ethyl-7-(2-methoxyethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C13H21N3O
4-Ethyl-7-(2-methoxyethyl)-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 2-Methyl-4-[(4-thiophen-3-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methyl]-1,3-thiazole —— C17H18N4S2
2-Methyl-4-[(4-thiophen-3-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methyl]-1,3-thiazole
—— 4-Methyl-7-[(1-methylimidazol-2-yl)methyl]-2-phenyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C20H23N5
4-Methyl-7-[(1-methylimidazol-2-yl)methyl]-2-phenyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 1-(2,4-Dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carbonyl)cyclopropane-1-carbonitrile —— C15H18N4O
1-(2,4-Dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carbonyl)cyclopropane-1-carbonitrile
—— 1-Methyl-7-(5-methyl-1,2-oxazole-4-carbonyl)-4,5,6,8-tetrahydropyrazolo[3,4-c]azepine-3-carbonitrile —— C14H15N5O2
1-Methyl-7-(5-methyl-1,2-oxazole-4-carbonyl)-4,5,6,8-tetrahydropyrazolo[3,4-c]azepine-3-carbonitrile
—— 2-Ethoxy-1-[2-methyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone —— C16H26N4O2
2-Ethoxy-1-[2-methyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone
—— 1-[2-(4-Fluorophenyl)-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone —— C19H23FN4O
1-[2-(4-Fluorophenyl)-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone
—— 1-[2-Phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone —— C19H24N4O
1-[2-Phenyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone
—— 1-[4-(Cyclopropylamino)-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-hydroxy-2-methylpropan-1-one —— C16H24N4O2
1-[4-(Cyclopropylamino)-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-2-hydroxy-2-methylpropan-1-one
—— 3-Hydroxy-1-[2-methyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]propan-1-one —— C15H24N4O2
3-Hydroxy-1-[2-methyl-4-(propan-2-ylamino)-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]propan-1-one
—— 2-(4-Fluorophenyl)-4-methyl-7-[(1-methylimidazol-2-yl)methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C20H22FN5
2-(4-Fluorophenyl)-4-methyl-7-[(1-methylimidazol-2-yl)methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 4-N-cyclopropyl-7-(oxan-4-yl)-2-N-propan-2-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine —— C19H31N5O
4-N-cyclopropyl-7-(oxan-4-yl)-2-N-propan-2-yl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-2,4-diamine
—— 1,2-Dimethyl-5-thiophen-2-ylsulfonyl-4,6,7,8-tetrahydropyrazolo[4,3-c]azepin-3-one —— C13H17N3O3S2
1,2-Dimethyl-5-thiophen-2-ylsulfonyl-4,6,7,8-tetrahydropyrazolo[4,3-c]azepin-3-one
—— 7-(2-Methoxyethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C17H23N3O2S
7-(2-Methoxyethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-Methylsulfonyl-1-(oxan-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C16H24N2O4S
7-Methylsulfonyl-1-(oxan-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 1-(2-Methoxyethyl)-7-(2-thiophen-3-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C18H22N2O3S
1-(2-Methoxyethyl)-7-(2-thiophen-3-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— N,N-dimethyl-2-[7-[(1-methylpyrazol-4-yl)methyl]-2-oxo-5,6,8,9-tetrahydropyrido[2,3-d]azepin-1-yl]acetamide —— C18H25N5O2
N,N-dimethyl-2-[7-[(1-methylpyrazol-4-yl)methyl]-2-oxo-5,6,8,9-tetrahydropyrido[2,3-d]azepin-1-yl]acetamide
—— N-cyclopropyl-2-oxo-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-7-carboxamide —— C19H28N4O2
N-cyclopropyl-2-oxo-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepine-7-carboxamide
—— 7-(Furan-3-ylmethyl)-1-(oxan-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C20H26N2O3
7-(Furan-3-ylmethyl)-1-(oxan-4-ylmethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(2-Cyclopropylacetyl)-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C17H24N2O3
7-(2-Cyclopropylacetyl)-1-(2-methoxyethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 1-(Cyclopropylmethyl)-7-(2-thiophen-3-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C19H22N2O2S
1-(Cyclopropylmethyl)-7-(2-thiophen-3-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(Cyclopropylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C18H23N3OS
7-(Cyclopropylmethyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 1-(Cyclopropylmethyl)-7-[(1-methylpyrazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C18H24N4O
1-(Cyclopropylmethyl)-7-[(1-methylpyrazol-4-yl)methyl]-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 1-(Cyclopropylmethyl)-7-ethylsulfonyl-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C15H22N2O3S
1-(Cyclopropylmethyl)-7-ethylsulfonyl-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-Methylsulfonyl-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C16H25N3O3S
7-Methylsulfonyl-1-(2-pyrrolidin-1-ylethyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— N-cyclopropyl-1-(2-methoxyethyl)-2-oxo-5,6,8,9-tetrahydropyrido[2,3-d]azepine-7-carboxamide —— C16H23N3O3
N-cyclopropyl-1-(2-methoxyethyl)-2-oxo-5,6,8,9-tetrahydropyrido[2,3-d]azepine-7-carboxamide
—— 1-(2-Methoxyethyl)-7-(2-thiophen-2-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one —— C18H22N2O3S
1-(2-Methoxyethyl)-7-(2-thiophen-2-ylacetyl)-5,6,8,9-tetrahydropyrido[2,3-d]azepin-2-one
—— 7-(Furan-2-ylmethyl)-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C16H21N3O2
7-(Furan-2-ylmethyl)-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 4-Methoxy-7-[(2-methoxypyridin-3-yl)methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C16H20N4O2
4-Methoxy-7-[(2-methoxypyridin-3-yl)methyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— [4-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-pyridazin-4-ylmethanone —— C17H19N5O2
[4-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]-pyridazin-4-ylmethanone
—— 7-(Furan-3-ylmethyl)-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C16H21N3O2
7-(Furan-3-ylmethyl)-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 7-[(5-Methylthiophen-2-yl)methyl]-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C17H23N3OS
7-[(5-Methylthiophen-2-yl)methyl]-4-propan-2-yloxy-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 7-Cyclopropylsulfonyl-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C12H17N3O2S
7-Cyclopropylsulfonyl-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 7-Ethylsulfonyl-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C11H17N3O2S
7-Ethylsulfonyl-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 4-Ethyl-7-ethylsulfonyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C12H19N3O2S
4-Ethyl-7-ethylsulfonyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— N,N,4-trimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxamide —— C12H18N4O
N,N,4-trimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine-7-carboxamide
—— 2-[[4-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methyl]-1,3-thiazole —— C16H20N4OS
2-[[4-[(3R)-oxolan-3-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]methyl]-1,3-thiazole
—— 7-(Furan-2-ylmethyl)-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine —— C14H17N3O
7-(Furan-2-ylmethyl)-4-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepine
—— 2-[(4-Ethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methyl]-1,3-thiazole —— C14H18N4S
2-[(4-Ethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl)methyl]-1,3-thiazole
—— (E)-3-(2,6-difluorophenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C16H14F2N4
(E)-3-(2,6-difluorophenyl)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-3-[5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C21H20ClFN6
(E)-3-[5-chloro-1-[(4-fluorophenyl)methyl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile