| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 3-(3-fluorophenyl)-N-[(1R)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]propanamide | —— | C18H23FN4O |
| —— | 3-(3-fluorophenyl)-N-[(1S)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]propanamide | —— | C18H23FN4O |
| —— | 3-[(3R)-1-prop-2-enylpiperidin-3-yl]-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepine | —— | C15H24N4 |
| —— | 1-[(1S)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)urea | —— | C14H22N8O |
| —— | 1-[(1R)-1-(4-methyl-1,2,4-triazol-3-yl)ethyl]-3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)urea | —— | C14H22N8O |
| —— | 3-(3-propyl-1,2,4-oxadiazol-5-yl)-N-[(1S)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]propanamide | —— | C17H26N6O2 |
| —— | 3-(3-propyl-1,2,4-oxadiazol-5-yl)-N-[(1R)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]propanamide | —— | C17H26N6O2 |
| —— | 2-methyl-N-[(2S)-1-(3-methylpyridin-2-yl)propan-2-yl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine | —— | C18H25N5 |
| —— | 2-methyl-N-[(2R)-1-(3-methylpyridin-2-yl)propan-2-yl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine | —— | C18H25N5 |
| —— | (2R)-3-cyclohexyl-3-oxo-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)propanenitrile | —— | C16H22N4O |
| —— | (2S)-3-cyclohexyl-3-oxo-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)propanenitrile | —— | C16H22N4O |
| —— | 2-[[(2R)-2-benzylbutyl]amino]-3,5,6,7,8,9-hexahydropyrimido[4,5-d]azepin-4-one | —— | C19H26N4O |
| —— | (13S)-13-(5-ethylfuran-2-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C15H15N3O2S |
| —— | (13R)-13-(5-ethylfuran-2-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C15H15N3O2S |
| —— | (13S)-13-[2-(propylamino)pyrimidin-5-yl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C16H18N6OS |
| —— | 2,7-dimethyl-N-[(2S)-1-thiophen-3-ylpropan-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine | —— | C17H24N4S |
| —— | (13R)-13-[2-(propylamino)pyrimidin-5-yl]-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C16H18N6OS |
| —— | 7-[(2R)-3-(1H-imidazol-5-yl)-2-pyrrol-1-ylpropanoyl]-2,3-dimethyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one | —— | C20H24N6O2 |
| —— | 2,7-dimethyl-N-[(2R)-1-thiophen-3-ylpropan-2-yl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine | —— | C17H24N4S |
| —— | 1-[4-[[(1R)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]amino]-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone | —— | C20H30N6O |
| —— | 1-[4-[[(1S)-1-(1-ethyl-3,5-dimethylpyrazol-4-yl)ethyl]amino]-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone | —— | C20H30N6O |
| —— | (8R)-2-amino-8-[2-(4-chlorophenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C17H14ClN5OS |
| —— | (8S)-2-amino-8-[2-(4-chlorophenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C17H14ClN5OS |
| —— | 1-[4-[[(2S)-2-hydroxy-3-methoxypropyl]amino]-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone | —— | C15H24N4O3 |
| —— | 1-[4-[[(2R)-2-hydroxy-3-methoxypropyl]amino]-2-methyl-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-7-yl]ethanone | —— | C15H24N4O3 |
| —— | (8R)-2-amino-8-(2-methoxypyridin-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C13H14N4O2S |
| —— | (8S)-2-amino-8-(2-methoxypyridin-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C13H14N4O2S |
| —— | 2,7-dimethyl-N-[(1R)-1-(1-methylpyrazol-4-yl)ethyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine | —— | C16H24N6 |
| —— | 2,7-dimethyl-N-[(1S)-1-(1-methylpyrazol-4-yl)ethyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-amine | —— | C16H24N6 |
| —— | 2-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-4-ylethyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine | —— | C20H28N6O |
| —— | (1S,2R)-2-(2-chlorophenyl)-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)cyclopropane-1-carboxamide | —— | C18H21ClN4O |
| —— | (1R,2R)-2-(2-chlorophenyl)-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)cyclopropane-1-carboxamide | —— | C18H21ClN4O |
| —— | (1R,2S)-2-(2-chlorophenyl)-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)cyclopropane-1-carboxamide | —— | C18H21ClN4O |
| —— | (8S)-2-amino-8-(2-ethyl-1,2,4-triazol-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C11H14N6OS |
| —— | (8R)-2-amino-8-(2-ethyl-1,2,4-triazol-3-yl)-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C11H14N6OS |
| —— | (8S)-2-amino-8-[2-(3-methylphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C18H17N5OS |
| —— | (8R)-2-amino-8-[2-(3-methylphenyl)pyrimidin-5-yl]-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-c]azepin-6-one | —— | C18H17N5OS |
| —— | 2-methyl-N-[(2R)-2-morpholin-4-yl-2-pyridin-2-ylethyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine | —— | C20H28N6O |
| —— | 2-methyl-N-[(2S)-2-morpholin-4-yl-2-pyridin-2-ylethyl]-6,7,8,9-tetrahydro-5H-pyrimido[4,5-d]azepin-4-amine | —— | C20H28N6O |
| —— | 2-[[(3R)-oxan-3-yl]amino]-1,5,6,7,8,9-hexahydropyrimido[4,5-d]azepin-4-one | —— | C13H20N4O2 |
| —— | 2,3-dimethyl-7-[(3S)-3-(2-methylimidazol-1-yl)butanoyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one | —— | C18H25N5O2 |
| —— | 2,3-dimethyl-7-[(3R)-3-(2-methylimidazol-1-yl)butanoyl]-5,6,8,9-tetrahydropyrimido[4,5-d]azepin-4-one | —— | C18H25N5O2 |
| —— | (13R)-4-methyl-13-(5-methyl-1-propylpyrazol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C17H21N5OS |
| —— | (13S)-4-methyl-13-(5-methyl-1-propylpyrazol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C17H21N5OS |
| —— | (13S)-4-methyl-13-(3,3,3-trifluoropropyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C13H14F3N3OS |
| —— | (13R)-4-methyl-13-(3,3,3-trifluoropropyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one | —— | C13H14F3N3OS |
| —— | N-[(1S)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]-3-thiophen-2-ylpropanamide | —— | C16H22N4OS |
| —— | 2-pyrazol-1-yl-N-[(1R)-1-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)ethyl]acetamide | —— | C14H20N6O |
| —— | (2R)-2-methyl-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)pentanamide | —— | C14H24N4O |
| —— | (2S)-2-ethoxy-N-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl)propanamide | —— | C13H22N4O2 |