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吖庚因类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-6,7,8,9-tetrahydro-5H-pyrimido[1,6-a]azepin-2-yl]acetamide —— C15H19N5O4
2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-6,7,8,9-tetrahydro-5H-pyrimido[1,6-a]azepin-2-yl]acetamide
—— 3-(2-bromophenyl)-1,2,4,5,6,7-hexahydropyrazolo[3,4-b]azepine —— C13H14BrN3
3-(2-bromophenyl)-1,2,4,5,6,7-hexahydropyrazolo[3,4-b]azepine
—— 2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-benzyl-N-(2-furylmethyl)acetamide —— C21H25N5O3
2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-benzyl-N-(2-furylmethyl)acetamide
—— 7-[(3-furylmethyl)(methyl)amino]-2-methyl-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-3-one —— C14H20N4O2
7-[(3-furylmethyl)(methyl)amino]-2-methyl-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-3-one
—— (4-fluorophenyl)-N-(3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)methanesulfonamide —— C14H17FN4O3S
(4-fluorophenyl)-N-(3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)methanesulfonamide
—— 2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-methyl-N-[(3-methyl-1-propyl-1H-pyrazol-5-yl)methyl]acetamide —— C18H29N7O2
2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-methyl-N-[(3-methyl-1-propyl-1H-pyrazol-5-yl)methyl]acetamide
—— 5-chloro-N-(3-oxo-2,5,6,7,8,9-hexahydro-[1,2,4]triazolo[4,3-a]azepin-7-yl)thiophene-2-sulfonamide —— C11H13ClN4O3S2
5-chloro-N-(3-oxo-2,5,6,7,8,9-hexahydro-[1,2,4]triazolo[4,3-a]azepin-7-yl)thiophene-2-sulfonamide
—— 2-(3,5-dimethyl-4-isoxazolyl)-N-(2-methyl-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)acetamide —— C15H21N5O3
2-(3,5-dimethyl-4-isoxazolyl)-N-(2-methyl-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)acetamide
—— 2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-ethyl-N-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]acetamide —— C19H31N7O2
2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-ethyl-N-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]acetamide
—— 2-{7-Amino-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-2-YL}-N-[(1,3-dimethyl-1H-pyrazol-4-YL)methyl]-N-methylacetamide —— C16H25N7O2
2-{7-Amino-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-2-YL}-N-[(1,3-dimethyl-1H-pyrazol-4-YL)methyl]-N-methylacetamide
—— N,3,5-Trimethyl-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-1,2-oxazole-4-carboxamide —— C15H21N5O2
N,3,5-Trimethyl-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-1,2-oxazole-4-carboxamide
—— 2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-methyl-N-(pyridin-3-ylmethyl)acetamide —— C16H22N6O2
2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-methyl-N-(pyridin-3-ylmethyl)acetamide
—— 3-(4-Methyl-1H-pyrazol-1-YL)-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}propanamide —— C15H22N6O
3-(4-Methyl-1H-pyrazol-1-YL)-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}propanamide
—— 3-cyclohexyl-N-(2-methyl-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)propanamide —— C17H28N4O2
3-cyclohexyl-N-(2-methyl-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)propanamide
—— N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-3-(3,5-dimethyl-1,2-oxazol-4-YL)propanamide —— C19H27N5O3
N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-3-(3,5-dimethyl-1,2-oxazol-4-YL)propanamide
—— 7-{[(1,3-Dimethyl-1H-pyrazol-5-YL)methyl](methyl)amino}-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-3-one —— C15H24N6O
7-{[(1,3-Dimethyl-1H-pyrazol-5-YL)methyl](methyl)amino}-2-methyl-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-3-one
—— 1-(3-Fluorophenyl)-N-{3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}methanesulfonamide —— C14H17FN4O3S
1-(3-Fluorophenyl)-N-{3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}methanesulfonamide
—— N-{2-Methyl-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}cyclohex-3-ene-1-carboxamide —— C15H22N4O2
N-{2-Methyl-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}cyclohex-3-ene-1-carboxamide
—— 2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide —— C19H31N7O2
2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylacetamide
—— N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]thiophene-2-sulfonamide —— C15H20N4O3S2
N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]thiophene-2-sulfonamide
—— N-[3-(methoxymethyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl]-3-(1H-pyrazol-1-yl)propanamide —— C15H22N6O2
N-[3-(methoxymethyl)-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl]-3-(1H-pyrazol-1-yl)propanamide
—— N-cyclohexyl-N'-[2-(cyclopropylmethyl)-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl]urea —— C18H29N5O2
N-cyclohexyl-N'-[2-(cyclopropylmethyl)-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl]urea
—— N-{3-Cyclopropyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-2-methoxyacetamide —— C13H20N4O2
N-{3-Cyclopropyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-2-methoxyacetamide
—— 1-Benzyl-3-[2-(cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]urea —— C19H25N5O2
1-Benzyl-3-[2-(cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]urea
—— N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-1-ethyl-N-methyl-1H-pyrazole-4-sulfonamide —— C17H26N6O3S
N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-1-ethyl-N-methyl-1H-pyrazole-4-sulfonamide
—— 2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-(4-methylphenethyl)acetamide —— C18H25N5O2
2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-(4-methylphenethyl)acetamide
—— N-[3-(Methoxymethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-YL]acetamide —— C16H21F3N6O2
N-[3-(Methoxymethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-YL]acetamide
—— N,3-Dimethyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-amine —— C9H16N4
N,3-Dimethyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-amine
—— N-[2-(cyclopropylmethyl)-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl]-N,1-dimethyl-1H-imidazole-4-sulfonamide —— C16H24N6O3S
N-[2-(cyclopropylmethyl)-3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl]-N,1-dimethyl-1H-imidazole-4-sulfonamide
—— 2-(3,5-Dimethyl-1,2-oxazol-4-YL)-N-[3-(methoxymethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]acetamide —— C16H23N5O3
2-(3,5-Dimethyl-1,2-oxazol-4-YL)-N-[3-(methoxymethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]acetamide
—— 3-(3,5-Dimethyl-1,2-oxazol-4-YL)-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}propanamide —— C16H23N5O2
3-(3,5-Dimethyl-1,2-oxazol-4-YL)-N-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}propanamide
—— N-(2-furylmethyl)-N'-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)urea —— C14H19N5O2
N-(2-furylmethyl)-N'-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)urea
—— 7-[(2-furylmethyl)(methyl)amino]-2-methyl-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-3-one —— C14H20N4O2
7-[(2-furylmethyl)(methyl)amino]-2-methyl-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-3-one
—— N'-cyclopentyl-N-methyl-N-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)urea —— C15H25N5O
N'-cyclopentyl-N-methyl-N-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)urea
—— 2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-(furan-2-ylmethyl)-N-(3-methylbutyl)acetamide —— C19H29N5O3
2-(7-amino-3-oxo-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-2-yl)-N-(furan-2-ylmethyl)-N-(3-methylbutyl)acetamide
—— N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-N-methylpropane-1-sulfonamide —— C15H26N4O3S
N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-N-methylpropane-1-sulfonamide
—— 3-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-1-(2-phenylethyl)urea —— C20H27N5O2
3-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-1-(2-phenylethyl)urea
—— 7-Amino-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-3-one —— C7H12N4O
7-Amino-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-3-one
—— 2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-(2-chloro-4-fluorobenzyl)acetamide —— C16H19ClFN5O2
2-[7-amino-3-oxo-6,7,8,9-tetrahydro-3H-[1,2,4]triazolo[4,3-a]azepin-2(5H)-yl]-N-(2-chloro-4-fluorobenzyl)acetamide
—— 1-[(4-Fluorophenyl)methyl]-3-{3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}urea —— C15H18FN5O2
1-[(4-Fluorophenyl)methyl]-3-{3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}urea
—— 5-Chloro-N-methyl-N-{2-methyl-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}thiophene-2-sulfonamide —— C13H17ClN4O3S2
5-Chloro-N-methyl-N-{2-methyl-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}thiophene-2-sulfonamide
—— N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-N-methylmethanesulfonamide —— C13H22N4O3S
N-[2-(Cyclopropylmethyl)-3-oxo-2H,3H,5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL]-N-methylmethanesulfonamide
—— N-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)-N'-phenethylurea —— C17H23N5O
N-(3-methyl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-7-yl)-N'-phenethylurea
—— 3-Methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-amine —— C8H14N4
3-Methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-amine
—— N-{3-Cyclopropyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-2-(thiophen-2-YL)acetamide —— C16H20N4OS
N-{3-Cyclopropyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-A]azepin-7-YL}-2-(thiophen-2-YL)acetamide
—— N-[(2-Chlorophenyl)methyl]-2-[4-(5-methyl-1,2,4-oxadiazol-3-YL)-1,3-dioxo-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepin-2-YL]acetamide —— C21H22ClN5O4
N-[(2-Chlorophenyl)methyl]-2-[4-(5-methyl-1,2,4-oxadiazol-3-YL)-1,3-dioxo-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepin-2-YL]acetamide
—— 2-[(4-Bromophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione —— C19H19BrN4O3
2-[(4-Bromophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione
—— 2-[(4-Chlorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione —— C19H19ClN4O3
2-[(4-Chlorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione
—— 2-[(3,4-Difluorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione —— C19H18F2N4O3
2-[(3,4-Difluorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione
—— 2-[(3,5-Difluorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione —— C19H18F2N4O3
2-[(3,5-Difluorophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione